| 111-132 | Progress towards the Synthesis of Sordarin and its Analogs | Huan Liang; Marco Ciufolini |
| 133-141 | Regioselective Nucleophilic Aromatic Substitution of Benzo[c][2,7]naphthyridines | Charles F. Nutaitis; Katrin Przyuski; Vincent Ross |
| 143-150 | Synthesis of Various 2,8-Cyclooctadiene-1,2-dicarboxylates | Ayse Uzgoren-Baran; Nazan Tunoglu; Gurol Okay |
| 151-160 | An Improved Non-chromatographic Scale-up Synthesis of a New 1,6,7,8-Substituted-4-oxo-1,4-dihydroquinoline-3-carboxylic Acid as a Potent Bacterial Topoisomerase Inhibitor | Xun Li; Scott Youells; Ronald K. Russell; Armin Roessler; Tobias Schmid; Roger Faessler; Michele A. Weidner-Wells; Eugene B. Grant; Mark J. Macielag |
| 161-167 | Practical and Efficient Synthesis of 4,4′-Dihydroxy-3,3′-dinitrodiphenyl Ether and 1,3-bis(4-Hydroxy-3-nitrophenoxy)benzene in Aqueous Alkaline Medium | Mitsutaka Imoto; Motonori Takeda; Akihiro Tamaki; Hisaji Taniguchi; Kazuhiko Mizuno |
| 169-173 | Efficient Iodine-catalyzed Synthesis of 3-Aryl 4(3H)-quinazolinones | Min Wang; Zhi-Guo Song; Ting-Ting Zhang |
| 175-182 | Facile and Mild Synthesis of bis(3-Indolyl)methanes | R. Ghorbani-Vaghei; S. M. Malaekehpoor |
| 183-185 | A New Route for the Synthesis of Ozagrel Hydrochloride | Chenglong Yu; Baohai Zhao; Yihong Zhao; Jimao Lin |
| 187-190 | Expedient Preparation of 4,6-Dihalo-3-arylisobenzofuran-1(3H)-ones from 3,5-Dihalo-N-ethylbenzamides | Lynn M. Bradley; Carleton G. Collins; Erica R. Tabakin; David A. Hunt |
| C | Editorial Board Page | |
| 505-542 | α-, β-,γ- AND ω-CYCLOPROPYLPHOSPHONATES. PREPARATION AND BIOLOGICAL ACTIVITY | Abed Al Aziz Al Quntar; Valery M. Dembitsky; Morris Srebnik |
| 543-550 | A SIMPLE AND EFFICIENT PROCEDURE FOR THE BECKMANN REARRANGEMENT OF OXIME USING bis-(TRICHLOROMETHYL) CARBONATE/DMF | W. K. Su; Y. Zhang; J. J. Li; P. Li |
| 551-556 | SYNTHESIS OF 4-CYANO- AND 5-AMINOPYRAZOLES AND DEAMINATION OF 5-AMINOPYRAZOLES | R. B. Toche; M. A. Kazi; M. N. Jachak |
| 557-561 | 4-IODO-6-METHOXYQUINOLINE | Alex C. Bissember; Martin G. Banwell |
| 561-566 | A SHORT SYNTHESIS OF THE NATURALLY OCCURRING 2,3,3′,4,4′,5,5′-HEPTACHLORO- (“Q1”) AND HEPTABROMO-1′-METHYL-1,2′-BIPYRROLES | Liangfeng Fu; Gordon W. Gribble |
| 566-571 | SYNTHESIS OF SUBSTANCES RELATED TO FLUTICASONE PROPIONATE | Jin Zheng; Qinglin Lai; Yiru Dai; Qingjie Zhao; Jingshan Shen |
| 572-574 | AN EFFICIENT ONE-STEP METHOD FOR THE LARGE-SCALE SYNTHESIS OF 2,4-THIAZOLIDINEDIONE | Ge Meng; Zhen-Yu Li; Mei-Lin Zheng |
| 574-579 | AN IMPROVED APPROACH TO N-SUBSTITUTED MALEIMIDES AND PHTHALIMIDES BY MICROWAVE-PROMOTED MITSUNOBU REACTION | Christoph D. Mayer; Marcus Kehrel; Franz Bracher |
| 579-585 | A NOVEL ACCESS TO SOME 1,4-DICHLOROISOQUINOLINES FROM PHENACYL AZIDES | R. E. Chen; X. H. Zhou; W. H. Zhong; W. K. Su |
| 586-589 | SYNTHESIS OF ARYL 14H-DIBENZO[A,J]XANTHENES USING ZIRCONIUM(IV) OXIDE CHLORIDE AS A CATALYST | Elaheh Mosaddegh; Mohammad Reza Islami |
| 591-596 | INDEXES | |
| C | Editorial Board Page | |
| 513-538 | THE ASYMMETRIC AZA-MICHAEL REACTION. A REVIEW | Jose L. Vicario; Dolores Badía; Luisa Carrillo; Juan Etxebarria; Efraim Reyes; Nerea Ruiz |
| 539-546 | SYNTHESIS OF 2-MERCAPTOBENZOTHIAZOLE AND OF 2-MERCAPTO-BENZIMIDAZOLE DERIVATIVES USING POLYMER-SUPPORTED ANIONS | D. S. Dalal; N. S. Pawar; P. P. Mahulikar |
| 546-550 | AN EFFICIENT SYNTHESIS OF TRICYCLIC COMPOUNDS, (±)-(4aβ,8aβ,10aα)-1,2,3,4,4a,6,7,8,8a,9,10,10a-DODECAHYDRO-1,1,4a-TRIMETHYL-2-OXOPHENANTHRENE-8a-CARBOXYLIC ACID, ITS METHYL ESTER, AND (±)-(4aβ,8aβ,10aα)-3,4,4a,6,7,8,8a,9,10,10a-DECAHYDRO-8a-HYDROXYMETHYL-1,1,4a-TRIMETHYLPHENANTHREN-2(1H)-ONE | Tadashi Honda; Yukiko Honda; Hidenori Yoshizawa; Gordon W. Gribble |
| 550-555 | A SYNTHESIS OF SELECTED o,o'-DISUBSTITUTED DIARYLACETIC ESTERS AND DIARYLMETHANES | Richard A. Bunce; James E. Schammerhorn |
| 555-559 | A CONVENIENT SYNTHESIS OF 3-ETHOXYCARBONYLAMINO-2-HYDROXY-4-PHENYLBUTYRIC ACID | Li Jun Lei; Xu Chang He |
| 560-565 | SYNTHESIS OF 2,4(1H,3H)-QUINAZOLINEDIONE AND 3-SUBSTITUTED 2,4(1H,3H)-QUINAZOLINEDIONES | J. S. Petrov; G. N. Andreev |
| 566-569 | A NOVEL SYNTHESIS OF 2-CHLORO-4-FLUORO-5-NITROBENZENESULFONYL CHLORIDE | Xiao-Hua Du; Sheng Chen; Mei Zheng; Zhen-Yuan Xu |
| 569-574 | EFFICIENT AND COST-EFFECTIVE SYNTHESIS OF DIALKYL CHLOROPHOSPHATES | P. D. Shakya; D. K. Dubey; Deepak Pardasani; Meehir Palit; A. K. Gupta |
| 575-579 | REGIOSELECTIVE SYNTHESIS OF E-OXIMES CATALYZED BY FERRIC CHLORIDE UNDER SOLVENT-FREE CONDITIONS | Hossein Eshghi; Asadollah Hassankhani |
| 579-584 | TWO-STEP PROTIC SOLVENT-CATALYZED REACTION OF PHENYLETHYLAMINE WITH METHYL ACRYLATE | H. Fakhraian; M. Babaie Panbeh Riseh |
| 585-589 | NITRIC ACID AND PHOSPHORUS PENTOXIDE SUPPORTED ON SILICA GEL AS A MILD AND EFFICIENT SYSTEM FOR THE OXIDATION OF BENZYLIC ALCOHOLS UNDER SOLVENT-FREE CONDITIONS | Abdol R. Hajipour; Behzad Kooshki; Arnold E. Ruoho |
| 589-594 | ALTERNATE SYNTHESES OF PRODAN AND ACRYLODAN | Steven S. Silvonek; Carl B. Giller; Christopher J. Abelt |
| 595-602 | INDEXES | |
| C | Editorial Board Page | |
| 297-330 | DIBENZO[bf]OXEPINES: SYNTHESES AND APPLICATIONS. A REVIEW | Roberto Olivera; Raul Sanmartin; Fátima Churruca; Esther Domínguez |
| 331-335 | PRACTICAL ROUTE TO A β-KETOPHOSPHONATE, A KEY INTERMEDIATE FOR THE TOTAL SYNTHESIS OF 20(S)-CPT AND RELATED ANALOGUES | Ming Huo; Yun-Yan Kuang; Fen-Er Chen |
| 337-340 | VILSMEIER-HAACK SYNTHESIS OF AROMATIC ALDEHYDES USING bis-(TRICHLOROMETHYL) CARBONATE AND DIMETHYLFORMAMIDE | W. G. Shan; X. J. Shi; W. K. Su |
| 341-345 | AN EXPEDITIOUS, PRACTICAL LARGE SCALE SYNTHESIS OF 4-AMINO-2-CHLORO-6,7-DIMETHOXYQUINAZOLINAZOLINE | G. Kumaraswamy; Nivedita Jena; M. N. V. Sastry; B. Ashok Kumar |
| 347-351 | N-ALKYLATION OF N-MONOSUBSTITUTED SULFONAMTOES IN IONIC LIQUIDS | Yi Hu; Zhen-Chu Chen; Zhang-Goo Le; Qin-Guo Zheng |
| 353-359 | SYNTHESIS OF TETRAHEDRAL CARBOXAMIDE HYDROGEN BOND ACCEPTORS | Amy S. Cannon; Tianying Jian; Jun Wang; John C. Warner |
| 361-362 | IMPROVED SYNTHESIS OF 3-AMINOFURAZAN-4-CARBOXYLIC ACID | Kevin G. Meyer |
| 363-366 | HEXAMETHYL ENETETR AMMONIUM FLUOROCHROMATE. A NEW REAGENT FOR OXIDATION OF ORGANIC SUBSTRATES | Ersan Turunc; Fatma Aydin |
| 367-370 | PREPARATION OF TRIAZAPHENAN THRENES | Charles F. Nutaitis; Megan Brennan |
| 371-374 | A CONVERGENT SYNTHETIC ROUTE TO 2-OXOPYRIDO[2,3-a]CARBAZOLES via 2-OXOPYRANO[2,3-a]CARBAZOLES FROM 1-OXO-1,2,3,4-TETRAHYDROCARBAZOLES | I. Antony Danish; K. J. Rajendra Prasad |
| 375-379 | A CONVENIENT METHOD FOR THE PREPARATION OF 2,5-bis-(4-AMINOPHENYL)-1,3,4-OXADIAZOLE | Matthew C. Davis; Andrew P. Chafin |
| 380-383 | AN IMPROVED PROCEDURE FOR THE ETHERIFICATION OF α-HYDROXY ACID DERIVATIVES | Sanjeev Kumar; Uma Ramachandran |
| 383-386 | FACILE BECKMANN REARRANGEMENT OF KETOXIMES MEDIATED BY YTTRIUM TRIFLATE | Surya Kanta De |
| 386-390 | AN IMPROVED SYNTHESIS OF NEOCRYPTOLEPINE | Robert Engqvist; Jan Bergman |
| C | Editorial Board Page | |
| 99-120 | HOMOGENEOUS RHODIUM(I)-CATALYZED REDUCTIVE AMINATIONS | Vitali I. Tararov; Renat Kadyrov; Thomas H. Riermeier; Uwe Dingerdissen; Armin Börner |
| 121-127 | A NOVEL AND DIRECT METHOD FOR THE PREPARATION OF 4-AMINO-1,1,3,3-TETRASUBSTTTUTED GUANIDINES AND OF [1,2,4]TRIAZOLO-FUSED HETEROCYCLIC DERIVATIVES | M. Abdul-Ghan; Sh. N. Khattab; A. M. El-Massry; A. El-Faham; Adel Amer |
| 129-133 | PREPARATION OF METHYL 2-METHOXYCARBONYLMETHYL-6-OXO-1,6-DIHYDROPYRIDINE-3-CARBOXYLATE | Song Feng; Xuchang He; Gengli Yu; Yu Xia; Donglu Bai |
| 135-140 | AN ANOMALOUS HOUBEN-HOESCH REACTION AND SOME APPLICATIONS IN ARYLATION REACTIONS | F. Sánchez-Viesca; María R. Gómez; Martha Berros |
| 141-149 | SYNTHESIS OF URETHANES BY A MODIFIED CURTIUS REACTION WITH ALCOHOLS | Armandodoriano Bianco; Francesco Bonadies; Raffaella Napolitano; Giancarlo Ortaggi |
| 151-155 | SYNTHESIS OF 3-SUBSTITUTED-2-ACYLIMINO-4-THIAZOLIDONES UNDER MICROWAVE IRRADIATION | Yanqing Peng; Gonghua Song; Ling Liu |
| 156-161 | WILLIAMSON REACTION IN IONIC LIQUIDS | Zhen Yuan Xu; Dan Qian Xu; Bao You Liu |
| 161-163 | IMPROVED SYNTHESIS OF PHENYLSELENOGLYCOLIC ACIDS | Hamdi Özkan; Ali Disli; Yilmaz Yildirir |
| 164-166 | A NOVEL AND SIMPLE SYNTHESIS OF (1S, 2S)-2-AMINO-l-(p-NITROPHENYL)-3-TRITYLOXYPROPANOL | Jian-Li Yuan; Hui-Fen Dai; Fen-Er Chen |
| 166-170 | SYNTHESIS OF 2-SUBSTITUTED THIAZOLIDINE-4-CARBOXYLIC ACIDS | Elena Pini; Donatella Nava; Riccardo Stradi |
| 170-173 | FACILE ONE-POT SYNTHESIS OF FLUORESCENT BENZOTHIENO[2,3:c]QUINOLINE | Harjinder Singh Bhatti; Sambamurthy Seshadri |
| 173-177 | SYNTHESIS OF PHENYLENE 1,3- AND 1,44bis(METHYLENE)-3-CARBAMOYL PYRIDINIUM BROMIDES | Feng Zhou; Chi-Hua Wang; John C. Warner |
| 178-182 | THE STRUCTURE OF “ITCA”, A URINARY METABOLITE OF CYANIDE | Herbert T. Nagasawa; Steven E. Cummings; Steven I. Baskin |
| 182-185 | A PRACTICAL SYNTHESIS OF ETHYL L-GLUTAMINE (L-Theanine) | Haining Gu; Yongxiang Jiang; Jiong Wang |
| 185-187 | A FACILE AND DIRECT SYNTHESIS OF ALENDRONATE FROM PYRROLIDONE | Guangyu Xu; Yuyuan Xie; Xihan Wu |
| 188-191 | MODIFIED AND CONVENIENT METHODS FOR THE PREPARATION OF SOME NTTRO MUSKS | Javad Safaei-Ghomi; Abdolhamid Bamoniri |
| 192-194 | SYNTHESIS OF 2-CHLORO- AND 2,5-DICHLOROBENZOPHENONES | A. G. Pinkus; F. S. Y. Ma; L. Y. C. Meng; T. C. Chang |
| 195-199 | NEW AND IMPROVED SYNTHESIS OF (±)-4-BROMO-7,8-DIMETHOXY-ISOCHROMAN-3-ONE, A KEY INTERMEDIATE FOR THE ELABORATION OF (±)-cis-ALPININE AND (±)-cis-ALPINIGENINE | DaríO A. Bianchi; Teodoro S. Kaufman |
| C | Editorial Board Page | |
| 527-581 | REGENERATION OF CARBONYL COMPOUNDS FROM OXIMES, HYDRAZONES, SEMICARBAZONES, ACETALS, 1,1-DIACETATES, 1,3-DITHIOLANES, 1,3-DITHIANES AND 1,3-OXATHIOLANES | Abdol Reza Hajipour; Sepideh Khoee; Arnold E. Ruoho |
| 583-601 | o-DIACYLBENZENES IN ORGANIC SYNTHESIS. A REVIEW | Antigoni Kotali; Philip A. Harris |
| 603-608 | A RELIABLE MULTIGRAM SYNTHESIS OF (±) DOXAZOSIN | G. Kumaraswamy; A. K. Das; Nivedita Jena |
| 609-613 | A NEW SYNTHESIS OF FLUMAZENEL SUITABLE FOR FLUORINE-18 LABELING | Gianluigi Broggini; Marco Orlandi; Alberto Turconi; Caterina Zoni |
| 613-616 | A FACILE SYNTHESIS OF DISULFIDES BY OXIDATION OF THIOLS WITH bis(TRICHLOROMETHYL) CARBONATE AND TRIPHENYLPHOSPHINE OXIDE | Y. S. Li; X. R. Liang; W. K. Su |
| 616-619 | A MILD AND EFFICIENT METHOD FOR RACEMIZATION OF α-AMINO ESTERS | Uma Ramachandran; Sudhanshu Kumar; H. P. S. Chawla |
| 620-622 | CONVENIENT PREPARATION OF A NEW ZWITTERIONIC TOSYLATE | Mireia Condom; SebastiáN Ondoño; Joan Suades |
| 623-626 | A DIELS-ALDER SYNTHESIS OF PYRIDINES | J. B. Hendrickson; Jian Wang |
| 627-630 | A CONVENIENT PROCEDURE FOR INDIRECT OXIDATION OF AROMATIC METHYL GROUPS TO ALDEHYDES AND CARBOXYLIC ACIDS | Leslie W. Deady; Shane M. Devine; Michael L. Rogers |
| 631-637 | INDEXES | |
| C | Editorial Board Page | |
| 361-368 | EFFECT OF CATIONS, SUBSTRATES AND TEMPERATURE ON THE MICROWAVE-ASSISTED SAPONIFICATION OF BENZOIC AND MESITOIC ESTERS | Laurence Perreux; André Loupy |
| 369-374 | TFFH AS A USEFUL REAGENT FOR THE CONVERSION OF CARBOXYLIC ACIDS TO ANILIDES, HYDRAZIDES AND AZIDES | A. El-Fahm; M. Abdul-Ghani |
| 375-382 | SYNTHESIS OF S-ARYL-D,L-CYSTEINES AND INCORPORATION INTO KERATIN SEQUENCES | Avram Gold; Tae-Gyu Nam; K. Jayaraj; R. Sangaiah; David G. Happer; Louise M. Ball; John E. French; Leena A. Nylander-French |
| 383-387 | POLYMER-SUPPORTED 4-(PHENYLSELENO)MORPHOLINE AS A USEFUL α-SELENENYLATING AGENT FOR SATURATED ALDEHYDES. A HIGHLY EFFICIENT ROUTE TO α-HALOALDEHYDES ON SOLID PHASE | Shou-Ri Sheng; Xian Huang |
| 387-390 | EFFICIENT SYNTHESIS OF 4-ISOCYANO-2,2,6,6-TETRAMETHYLPIPERIDINE-1-OXYL | Jerzy Zakrzewski; Jaroslaw Hupko |
| 391-396 | NEW EFFICIENT SYNTHESIS OF 2-ALKYLTHIO-5-BENZYLJDENE-4H-IMIDAZOLIN-4-ONES | Ming-Wu Ding; Yong Sun; Xiao-Peng Liu; Zhao-Jie Liu |
| 397-400 | SYNTHESIS OF THE DASYCARPIDONE SKELETON | Nesimi Uludag; Tahsin Uyar; Süleyman Patir |
| 401-408 | SOLVENT-FREE SYNTHESIS OF SPIRO[3H-INDOLE-3,2′-THIAZOLIDINES] | Anshu Dandia; Ruby Singh; Kapil Arya |
| 409-411 | ALTERNATIVE SYNTHESIS OF N,N′-DJPHENYLTHIOUREA AND ITS ANALYSIS BY LC-MS | Yu-Chun Xiong; Zhi-Min Zong; Fa-Qin Jiang; Xin-Hua Yuan; Xiao-Hua Wang; Ya-Fei Ji; Li Xu; Hong-Zhan Xiao; Lin-Tao He; Chun-Qi Li; Xian-Yong Wei |
| 412-414 | CHLOROMETHYL METHYL SULFONE BY OXIDATION OF CHLOROMETHYL METHYL SULFIDE | Mieczyslaw Makosza; Marek Surowiec |
| 414-417 | SIMPLE METHODOLOGY FOR THE PURIFICATION OF AMINO ACIDS | Antonio José Mota; Elena Castellanos; Eusebio Juaristi |
| 418-420 | A SHORT SYNTHESIS OF ar-TODOMATUIC ACID AND DIHYDRO-ar-TURMERONE BY THE HECK REACTION | S. B. Solabannavar; P. P. Wadgaonkar; U. V. Desai; R. B. Mane |
| 420-422 | A CONVENIENT SYNTHESIS OF 1,1′- and 1,2′-DINAPHTHYLMETHANONES | L. Wu; Z. M. Zong; X. Y. Wei; Y. M. Qin; G. L. Zou |
| 422-425 | SYNTHESIS OF 2,5- AND 2,6-DINITROFLUOROBENZENES AND RELATED HYDROQUINONES | E. J. Behrman; Ssuhen Chen |
| 426-429 | SYNTHESIS OF 2,5-DISUBSTITUTED 1,3,4-OXADIAZOLES USING DRY MEDIA | M. Kidwai; R. Mohan |
| 429-432 | A NEW APPROACH TO THE SYNTHESIS OF 1,3-AMINOALCOHOLS FROM MESO CYCLIC ACID ANHYDRIDE | Jia-Hai Ye; You Huang; Ru-Yu Chen |
| 433-438 | REACTIONS OF INDOLE-2,3-DIONES WITH 3-AMINOPROPANOL | Anshu Dandia; Meha Sati; Sangeeta Sanan; R. Joshi |
| 439-443 | METHYL 2-CHLORO-4-FLUOROPHENYLTRIOACETATE AS A NEW INTERMEDIATE IN THE SYNTHESIS OF PESTICIDES | Zhenyuan Xu; Xiaohua Du; Jianbo Gu |
| C | Editorial Board Page | |
| 559-583 | SYNTHETIC APPROACHES TOWARD THE BENGAMIDE FAMILY OF ANTITUMOR MARINE NATURAL PRODUCTS. A REVIEW | Frederick R. Kinder Jr |
| 585-608 | THE ZINCKE REACTION. A REVIEW | Wei-Chieh Cheng; Mark J. Kurth |
| 609-642 | THE BIRCH REDUCTION OF STEROIDS. A REVIEW | Hélène Pellissier; Maurice Santelli |
| 643-646 | CONVENIENT SYNTHESIS OF DI(n-OCTADECYL)AMINE AND DI(n-HEXADECYL)AMINE | Luciano Lattuada; Fulvio Uberti |
| 647-651 | IODINATION OF AROMATIC COMPOUNDS UNDER MILD AND SOLVENT-FREE CONDITIONS | Abdol R. Hajipour; Arnold E. Ruoho |
| 652-655 | PREPARATION OF 5,10,11,11a-TETRAHYDRO-1H, 3H-THIAZOLO[2,3-c]-AND 5,10,11,11a-TETRAHYDRO-1H, 3H-THIAZOLO[4,3-c]-[1,4]BENZODIAZEPINES | Alexey B. Dyatkin; Bruce E. Maryanoff |
| 655-657 | FACILE PREPARATION OF trans-2,3-bis(-tert-BUTYLAMINOMETHYL) NORBORNENE | J. H. Wynne; W. M. Stalick |
| 658-664 | SYNTHESIS OF 1-[4-(1,5-DIALKYL-1H-1,2,4-TRIAZOL-3-YL)]BENZYL-1H-INDOLES AND 5,6-DIHALOQUINOLONES | Yaseen A. Al-Soud; Rana F. Halah; Najim A. Al-Masoudi |
| 665-670 | A CONVENIENT REDUCTION OF HIGHLY FUNCTIONALIZED AROMATIC CARBOXYLIC ACIDS TO ALCOHOLS WITH BORANE-THF AND BORON TRIFLUORIDE-ETHERATE | M. H. Chen; E. Iakovleva; S. Kesten; J. Magano; D. Rodriguez; K. E. Sexton; J. Zhang; H. T. Lee |
| 671-680 | INDEXES | |
| C | Editorial Board Page | |
| 205-234 | AMINES via NUCLEOPHJLIC 1,2-ADDITION TO KETIMINES. CONSTRUCTION OF NITROGEN-SUBSTITUTED QUATERNARY CARBON ATOMS. A REVIEW | Arno G. Steinig; Denice M. Spero |
| 235-264 | RECENT ADVANCES IN THE CHEMISTRY OF OXIMES | Edgars Ãbele; Edmunds Lukevics |
| 265-269 | SYNTHESIS OF (S)-(-)-1-[(9-FLUORENYLMETHOXYCARBONYL)AMINO-5-CARBOXYPENTYL]-3-HYDROXYPYRIDINIUM TRIFLUOROACETATE | Maciej Adamczyk; Rajarathnam E. Reddy |
| 269-271 | MICROWAVE-ASSISTED SYNTHESIS OF TRIARYL PHOSPHATES | A. D. Sagar; N. A. Shinde; B. P. Bandgar |
| 272-275 | SIMPLE AND PRACTICAL SYNTHESES OF DIBENZYL, BENZYL ETHYL AND BENZYL METHYL MALONATES | Ana Luisa Silva; Adrián Covarrubias-zúñiga; Luis Angel Maldonado |
| 276-279 | A ONE-POT SYNTHESIS OF PYRAZOLO [3,4-b][1,4]OXAZINES | M. A. Raslan; F. M. Abd El-Latif; H. H. Otto; K. U. Sadek |
| 280-283 | A RAPID METHOD FOR THE CYCLIZATION OF 2′-HYDROXYCHALCONES INTO FLAVONES | Mukta Gupta; Satya Paul; Rajive Gupta; Andre Loupy |
| 284-287 | RAPID N-ALKYLATION OF CARBAZOLE, PHENOTHIAZLNE AND ACRIDONE UNDER MICROWAVE IRRADIATION | Xingjun Fan; Jinmao You; Tianquan Jiao; Ganzu Tan; Xianda Yu |
| 287-290 | ESTERIFICATION BY MICROWAVE IRRADIATION ON ACTIVATED CARBON | Xingjun Fan; Keguo Yuant; Caili Hao; Nan Li; Ganzu Tan; Xianda Yu |
| 290-293 | SYNTHESIS OF 4-BORONO-2-FLUOROPHENYLALANINE | G. W. Kabalka; N. K. Reddy; L. Wang; R. R. Malladi |
| 293-297 | PREPARATION OF bis-[SPIROFLUORENE-9,4′-(1-AZA-2-CYCLOPENTENE)[1,5-a]INDOLINE-8′-YL]SULFONE | E. O. Gogritchiani; H. Dürr; Sh. A. Samsoniya |
| 298-301 | AN OPTIMIZED PREPARATION OF 2,3-DIHYDRO-1-METHYL-4-OXONAPHTHALENE-1-CARBOXYLIC ACID | A. G. Lo Cascio; G. R. Labadie; M. Gonzalez Sierra; R. M. Cravero |
| 302-306 | FACILE AND EFFICIENT SYNTHESIS OF α-AMINOPHOSPHONATE DERIVATIVES OF 1,3,4-OXADIAZOLE AND 1,3,4-THIADIAZOLE | Shui-Ming Lu; Ru-Yu Chen |
| C | Editorial Board Page | |
| 359-377 | REACTIONS OF CARBON TETRACHLORIDE AND CARBON TETRABROMIDE WITH ANIONS AND CARBANIONS. A REVIEW | Edgars Abele; Edmunds Lukevics |
| 379-397 | THE CHEMISTRY OF 4′,5′-UNSATURATED NUCLEOSIDES. A REVIEW | Clemens Lamberth |
| 399-405 | A COMPARISON OF IMINE FORMING METHODOLOGIES | Brian E. Love; Tavia S. Boston; Binh T. Nguyen; Jeffrey R. Rorer |
| 407-412 | ACYLATION AND ALKYLATION OF 2- AND 4-METHYLBENZONITRILE | Richard A. Bunce; Lara B. Johnson |
| 413-421 | N-SUBSTITUTED 3-OXA- AND 3-THIA-7-AZABICYCLO[3.3.1]NONANES AS POTENTIAL PRECURSORS OF ANTIARRHYTHMICS | Sameer Tyagi; Kevin M. Couch; Gregory L. Garrison; K. Darrell Berlin; Benajmin J. Scherlag; Eugene Patterson; Ralph Lazzara |
| 423-425 | SYNTHESIS OF N-(5-AMINO-2-PYRIMIDn)-N′-[4-(p-FLUOROPHENYL)-4-OXOBUTYL]PIPERAZINE, A USEFUL INTERMEDIATE TO ANTIPSYCHOTIC AGENTS | Gianluigi Broggini; Gaetano Zecchi |
| 425-429 | SYNTHESIS OF N-(3-MERCAPTOPROPANOYL)-AZA-18-CROWN-6, N-(4-MERCAPTOBUTANOYL)-AZA-18-CROWN-6 AND THEIR DIMERS | Xinhao Yang; J. Justin Gooding; D. Brynn Hibbert; Naresh Kumar |
| 429-433 | NEW N,N′-bis (SUBSTITUTED PHENYLAZO) PIPERAZINES AND THEIR CLEAVAGE REACTIONS IN ACETIC ACID | Erkan Yanarates; Ali Disli; Yilmaz Yildirir |
| 433-439 | PHASE-TRANSFER CATALYZED ALKYLATION OF HYDROXY 9,10-ANTHRAQUINONES | Douglas R. Robello; Teresa D. Eldridge; Edward J. Urankar |
| 440-442 | MULTI-GRAM SYNTHESIS OF DIMYRISTOYL PENTAERYTHRITOL | Mike E. Lizarzaburu; Ryan M. Jones; Michael H. Nantz; Mark J. Kurth |
| 442-447 | IMPROVED SYNTHESIS OF cis-9,10-DIHYDRO-9,10,-PHENANTHRENEDICARBOXIMIDES AND 9,10-PHENANTHRENEDICARBOXIMIDES | Piotr Grycz; Jacek Gawroński |
| 447-450 | PREPARATION OF 3-TETRADECYLINDOLE | James H. Wynne; George W. Mushrush; Wayne M. Stalick |
| 450-453 | A NOVEL METHOD FOR THE SYNTHESIS OF TELLUROESTERS | Songlin Zhang; Yongmin Zhang |
| 453-456 | AN EFFICIENT ONE-POT SYNTHESIS OF α-PHENYLSELENO-α,β-UNSATURATED NITRILES via ARSONIUM SALTS | Gui-Sheng Deng; Zhi-Zhen Huang; Xian Huang |
| 456-459 | AN IMPROVED SYNTHESIS OF Nα-BENZYLOXYCARBONYL-L-LYSINE | Ełżbieta Masiukiewicz; Stanislaw Wiejak; Barbara Rzeszotarska |
| 460-462 | IMPROVED PREPARATION OF METHYL 4,6-O-BENZYLIDENE-α-D-GLUCOPYRANOSIDE | Rolando A. Spanevello; Damiáh D. Saavedra |
| 462-465 | A NEW AND EFFICIENT SOLVENT-FREE SYNTHESIS OF bis-ARYL CARBODIAZONES | Hong Wang; Yulu Wang; Jianping Li; Xiaoyang Wang |
| C | Editorial Board Page | |
| 373-400 | APPLICATIONS OF TRIMETHYLSILYL HALIDES-OXIDANTS COMBINATIONS IN ORGANIC SYNTHESIS. A REVIEW | Padma S. Vankar; M. Venkat Ram Reddy; Yashwant D. Vankar |
| 401-425 | PHOTOCHEMICAL TRANSFORMATIONS OF 2(5H)-FURANONES. A REVIEW | Ahmed I. Hashem; Alexander Senning; Abdel-Sattar S. Hamad |
| 427-432 | A RAPID WILLIAMSON SYNTHESIS UNDER MICROWAVE IRRADIATION IN DRY MEDIUM | Dariusz Bogdal; Jan Pielichowski; Krzysztof Jaskot |
| 433-437 | FACILE SYNTHESIS OF 5-(DIHYDROXYBORYL)-2,4-bis(ALKOXY)PYRIMIDINES AND N(1)-SUBSTITUTED 5-(DIHYDROXYBORYL)URACILS | Hanna Wojtowicz-Rajchel; Krzysztof Golankiewicz |
| 439-446 | SYNTHESIS AND SPECTRAL DATA OF SOME NEW N-NITROSO-N-PHENYLHYDROXYLAMINE (CUPFERRON) DERIVATIVES | Alexandru T. Balaban; Robert E. Garfield; Melanie J. Lesko; William A. Seitz |
| 447-451 | A FACILE SYNTHESIS OF o-, m-, p-(TRIMETHYLSTANNYL)BENZYL CHLORIDES AND AMINES | A. B. Koldobsky; V. E. Vakhmistrov; O. S. Shilova; V. N. Kalinin; K. Abbaspour Tehrani; N. De Kimpe |
| 451-453 | A NOVEL ROUTE TO 4-ARYLIDENE-2-PHENYL-5(4H)-OXAZOLONES | M. Kidwai; R. Kumar |
| 453-455 | IMPROVED PREPARATION OF FLURBIPROFEN | M. N. Deshmukh; V. Lakshminarayana |
| 455-460 | EFFICIENCY OF THE VILSMEIER-HAACK METHOD IN THE SYNTHESIS OF p-AMINOBENZALDEHYDES | Ryszard Gawinecki; Sylwia Andrzejak; Agnieszka Puchala |
| 460-463 | IMPROVED PREPARATION OF SURFACTANTS DERIVED FROM SUCROSE WITH ULTRASOUND | Jacques Besson; Catherine Fayet; J. Gelas; Christelle Lamazzi |
| 463-466 | AN EFFICIENT AND FACILE PROCEDURE FOR DEPROTECTION OF 1,1-DIACETATES USING ANHYDROUS FERROUS SULFATE | T. S. Jin; Y. R. Ma; Z. H. Zhang; T. S. Li |
| 467-469 | A HIGH YIELDING PREPARATION OF 2,2′-BIPYRIDINE-1-OXIDE | F. W. Joachim Demnitz; Maria Betânia D'heni |
| 469-472 | SURFACE MEDIATED SYNTHESIS OF O-PHOSPHOROTHIOATES | K. Ramadas; N. Janarthanan; D. Meera Rani |
| 473-476 | AN IMPROVED PREPARATION OF S,S'-DIMETHYL N-CYANODITHIOIMINOCARBONATE | Lyndon K. Marble |
| 477-481 | NEW SYNTHESES OF bis(TETRAMETHYLENE)FLUOROFORMAMIDINIUM HEXAFLUOROPHOSPHATE (BTFFH) AND 1,3-DIMETHYL-2-FLUORO-4,5-DIHYDRO-1H-IMIDAZOLIUM HEXAFLUOROPHOSPHATE (DFIH). UTILITY IN PEPTIDE COUPLING REACTIONS | Ayman El-Faham |
| 481-484 | SYNTHESIS OF BENZO[c][2,7]NAPHTHYRIDINES AND 2,13-DIAZABENZO[b]CHRYSENE | Charles F. Nutaitis; Matthew L. Crawley; Judy Obaza-Nutaitis |
| 485-488 | PREPARATION OF O-(3,3,8,10,10-PENTAMETHYL-1,2-DITHIA-5,8-DIAZACYCLODECAN-5-YL)ETHYL O-PIVALOYLOXYMETHYL PHENYLPHOSPHONATE | Nicholas Bodor; Katalin Prokai-Tatrai; Emo Koltai; Laszlo Prokai |
| C | Editorial Board Page | |
| 1-51 | BIOMIMETIC AND SYNTHETIC APPROACHES TO MARINE SPONGE ALKALOIDS DERIVED FROM BIS-PYRIDINE MACROCYCLES. A REVIEW | Norbert Matzanke; Robert J. Gregg; Steven M. Weinreb |
| 53-61 | 2-SUBSTITUTED HEXAHYDROPYRIMIDINES AND THEIR TAUTOMERISM | Kirill N. Zelenin; Valeriy V. Alekseyev; Ilya V. Ukraintsev; Igor V. Tselinsky |
| 63-70 | REDUCTION OF ORGANIC COMPOUNDS WITH THEXYL-S-BUTOXYBORANE | Jin Soon Cha; Seok Won Chang; Jong Mi Kim; Oh Oun Kwon; Joong Hyun Chun; Sung Dong Cho; Hyung Soo Lee |
| 71-78 | SYNTHESIS OF (1R,3S)-3-AMINO-1,2,2-TRIMETHYLCYCLOPENTYLMETHANOL | José M. Blanco; Olga Caamaño; Franco Fernández; Xerardo García-Mera; José E. Rodríguez |
| 79-85 | IMPROVED SYNTHESIS OF 7,7-DIMETHYL-1,4-DIOXO-2,3,4,5,6,7-HEXAHYDROINDEN-2-YL-ACETIC AND PROPIONIC ACID FROM CITRAL | István Kádas; Géza Árvai; Gabriella Horváth |
| 87-90 | MICROWAVE-PROMOTED SYNTHESIS OF 1-ARYLOXY-3-ALKYLAMINO-2-PROPANOLS | Beata Pchelka; Jan Plenkiewicz |
| 90-93 | FACILE SYNTHESES OF P-(DICYANOMETHYLENE)BENZOQUINONES | Masato Nanasawa; Hiroshi Takahashi; Tetsuo Kuwabara |
| 93-96 | SYNTHESIS AND CYCLIZATION OF 1-(N-NITROAMIDINO)THIOUREAS TO 2,4-DIAMINOTHIAZOLES | R. Binu; K. K. Thomas; G. C. Jenardanan; K. N. Rajasekharan |
| 97-99 | AN EFFICIENT OXIDATION ARYLSEMICARBAZIDES TO THE AZO UREAS | Cailan Wang; Yulu Wang; Xiaoyang Wang; Jianping Li; Hong Wang; Shensong Zhang |
| 100-103 | A SIMPLE, ONE-POT PROCEDURE FOR THE PREPARATION OF DOPAMINERGIC ALKYLTHIOAPOMORPHINES | Sándor Berényi; Csaba Csutorás; Susanna Gyulai; Sándor Makleit |
| 103-106 | REGIOSELECTIVE EPOXIDE RING-OPENING TO THE ENANTIOMERICALLY PURE α-HYDROXY ANALOGUE OF S-TERT-BUTYL CYSTEINE | Florine Cavelier; Anne-Marie Yim |
| 107-109 | IMPROVED SYNTHESIS OF O-BENZENEDISULFONIMIDE | Franklin A. Davis; Gajendran Sundarababu; Hongyan Qi |
| 109-114 | 1-ALKYLIDENE(ARYLIDENE)AMINO-2-AMINOETHANES AND THEIR TAUTOMERIZATION TO IMIDAZOLIDINES | Kirill N. Zelenin; Ilya V. Ukraintzev |
| 115-116 | IMPROVED PREPARATION OF 5,6-DICHLOROCYCLOHEX-2-ENE-1,4-DIONE | Vitor Francisco Ferreira; Francis J. Schmitz |
| 117-120 | A CONVENIENT SYNTHESIS OF (E)-(1-PROPENYLSULFONYL)BENZENE | L. M. Finkielsztein; E. N. Alesso; B. Lantaño; J. M. Aguirre; G. Y. Moltrasio Iglesias |
| C | Editorial Board Page | |
| 603-629 | OPTICALLY ACTIVE SELENIUM AND TELLURIUM COMPOUNDS. SYNTHESIS AND APPLICATION FOR ASYMMETRIC SYNTHESIS. A REVIEW | Toshio Shimizu; Nobumasa Kamigata |
| 631-664 | THE SYNTHESIS OF ISOCOUMARINS OVER THE LAST DECADE. A REVIEW | Elio Napolitano |
| 665-669 | REDUCTION OF CARBOXYLIC ACIDS TO ALDEHYDES BY THEXYLALKOXYBORANES | Jin Soon Cha; Seok Won Chang; Jong Mi Kim; Oh Oun Kwon; Jae Cheol Lee |
| 671-677 | SYNTHESIS OF AMINOTOLUENESULFONAMIDE DERIVATIVES USING CONVENTIONAL HEATING OR MICROWAVE-ASSISTED METHODS | Rolando Pérez; Eduardo R. Pérez; Margarita Suárez; Leandro González; André Loupy; María Luisa Jimeno; Carmen Ochoa |
| 679-685 | IMPROVED SYNTHESES OF 2,2',3,3',6,6'-HEXACHLOROBIPHENYL | Stephen C. Waller; Eugene A. Mash |
| 687-689 | CONDENSATION REACTION OF ACYLOINS WITH UREA WITHOUT SOLVENT UNDER MICROWAVE IRRADIATION | Jun-Cai Feng; Qing-Hua Meng; Yang Liu; Li Dai |
| 689-696 | CHEMICAL TRANSFORMATION OF DIHYDRO- AND TETRAHYDRO-1,5-BENZODIAZEPIN-2-ONES INTO AMIDINES | Benedikta Dale Puodziunaite; Lina Vertelyte; Regina Janciene; Zita Stumbreviciute |
| 696-701 | N-ACETYL-α,β-DEHYDROAMINO ACID N'-METHYLAMIDES AND N',N'-DIMETHYLAMIDES | Leszek Smelka; Barbara Rzeszotarska; Malgorzata A. Broda; Zbigniew Kubica |
| 701-706 | A FACILE SYNTHESIS FOR RACEMIC AND OPTICALLY ACTIVE 1-AMINOINDANS | Ramy Lidor; Eliezer Bahar; Ora Zairi; Gasan Atili; Dora Amster |
| 707-710 | SYNTHESIS OF HEXASUBSTITUTED NITROBENZENE DERIVATIVESvia VICARIOUS NUCLEOPHILIC SUBSTITUTION OF HYDROGEN | M. Makosza; S. Nizamov |
| 711-715 | A NOVEL ROUTE TO NEW DIBENZO[b,f][1,5]DIAZOCINE DERIVATIVES AS CHEMOSENSITIZERS | E. Nonnenmacher; A. Hever; A. Mahamoud; C. Aubert; J. Molnar; J. Barbe |
| 715-719 | N-BROMOSUCCINIMIDE-CHLOROFORM, A MORE CONVENIENT METHOD TO NUCLEAR BROMINATE REACTIVE AROMATIC HYDROCARBONS | Reginald H. Mitchell; Yongsheng Chen; Ji Zhang |
| 721-734 | INDEXES | |
| C | Editorial Board Page | |
| 365-407 | REDUCTIVE CLAISEN REARRANGEMENTS OF ALLYLOXYANTHRAQUINONES. A REVIEW | Richard C. Cambie; Jared B. J. Milbank; Peter S. Rutledge |
| 409-458 | RECENT PROGRESS IN THE USE OF HYPERVALENT IODINE REAGENTS IN ORGANIC SYNTHESIS. A REVIEW | Tsugio Kitamura; Yuzo Fujiwara |
| 459-464 | p-CHLOROPHENOL AS A SOLVENT FOR CYCLOADDITION OF CYCLOPENTADIENONES WITH NON-ACTIVATED OLEFINS | Tamaki Jikyo; Masashi Eto; Toshikazu Matsuoka; Kazunobu Harano |
| 465-470 | SYNTHESIS OF 6-HYDROXY-3,4,5,6-TETRAHYDRO-2-PYRIDONES AND 3,4-DIHYDRO-2-PYRIDONES BY H2O2/DMSO HYDRATION OF Δ-KETONITRILES | Attilio Citterio; Elena Carnevali; Alessandra Farina; Valdo Meille; Stefano Alini; Livius Cotarca |
| 471-473 | AN IMPROVED ROUTE TO CYCLOALKA[b]PYRROLE 2-CARBOXYLATES | C. Balsamini; A. Bedini; G. Tarzia; A. Tontini |
| 473-476 | SYNTHESES AND STEREOCHEMISTRY OF TETRAHYDROFURAN DERIVATIVES FROM α-PINENE | Fu-Chu Liu; Zhen-Qi Mei; You-Chu Wang; Jun Lin |
| 477-480 | SYNTHESIS OF SUBSTITUTED 1-TETRALONES | Punit Kumar |
| 480-484 | DETHIOACETALIZATION OF DITHIOLANES WITH FERRIC NITRATE AND SILICA GEL IN HEXANE | Masao Hirano; Ken Ukawa; Shigetaka Yakabe; Takashi Morimoto |
| 485-488 | SYNTHESIS OF 3-O-BENZYL-3,7-IMINO-1,3,6,7-TETRADEOXY-L-MANNO-HEPTITOL AND OF 3-O-BENZYL-3,7-IMINO-1,3,6,7-TETRADEOXY-D-GLUCO-HEPTITOL | Fabio Degiorgis; Marco Lombardo; Claudio Trombini |
| 488-494 | A CONVENIENT SYNTHESIS OF NEW HALOTHIENYL β-AMINOACIDS AS VERSATILE BUILDING BLOCKS | Olivier Renault; Patrick Dallemagne; Sylvain Rault |
| 494-496 | NEW SIMPLE SYNTHESIS OF THE HOUSEFLY SEX ATTRACTANT | Yao-Pin Yen; Fey-Long Wang |
| 497-498 | IMPROVED ONE-POT PREPARATION OF TETRAMETHYLFLUOROFORMAMIDINIUM HEXAFLUOROPHOSPHATE | Tomas Vojkovsky; Brian Drake |
| C | Editorial Board Page | |
| 243-283 | BRIDGED POLYCYCLIC AROMATIC HYDROCARBONS. A REVIEW | Ronald G. Harvey |
| 285-292 | SYNTHESIS OF NEW ARYL AND HETEROAROMATIC SUBSTITUTED PYRIDINES, PYRAZOLES, PYRIMIDINES AND PYRAZOLO[3,4-D]PYRIDAZINES | Fatima Al-Omran; Nouria Al-Awadi; Adel Abou El-Khair; Mohammed Hilmy Elnagdi |
| 293-299 | TETRAHYDROPYRANYLOXY-DIRECTED ortho LITHIATION OF AROMATIC SYSTEMS. SYNTHESIS OF o-HYDROXYCINNAMATE ESTERS FROM PHENOLS | Richard A. Bunce; Joel D. Moore |
| 300-303 | A NEW ROUTE FOR THE PREPARATION OF XANTHENE DERIVATIVES USING FRIEDEL-CRAFTS INTRAMOLECULAR CYCLOBENZYLATION | Takehiko Yamato; Masayasu Komine; Yoshiaki Nagano |
| 303-308 | SYNTHESIS OF (1R,cis)-2-(3-AMINO-2,2-DIMETHYLCYCLOBUTYL)ETHANOL, A PRECURSOR OF CYCLOBUTANE CARBOCYCLIC NUCLEOSIDES | José E. R. Borges; Franco Fernández; Xerardo García; Antonio R. Hergueta; Carmen López |
| 308-311 | AN IMPROVED PROCEDURE FOR THE SYNTHESIS OF ANHYDROECGONINE METHYL ESTER | C. R. Holmquist; K. R. Parham; J. A. Holleman; F. I. Carroll |
| 311-314 | SYNTHESIS OF UNSYMMETRICAL α-(N-ARYLCARBONYL)AMINO DIORGANYL SELENIDES via BENZOTRIAZOLE INTERMEDIATES PROMOTED BY SmI2 | Weiliang Bao; Yongmin Zhang; Yunfa Zheng |
| 315-321 | REDUCTION OF 1,3-AZOLE AND 1,3-BENZAZOLE CARBINOLS WITH SODIUM BOROHYDRIDE-TRIFLUOROACETIC ACID | Charles F. Nutaitis; Judy Obaza-Nutaitis |
| 321-330 | ELECTROPHILIC SUBSTITUTION OF 7-tert-BUTYL-1-SUBSTITUTED PYRENES. A NEW ROUTE FOR THE PREPARATION OF 1,3-DISUBSTITUTED PYRENES | Takehiko Yamato; Masakazu Fujimoto; Yoshiaki Nagano; Akira Miyazawa; Masashi Tashiro |
| 330-335 | EFFICIENT SYNTHESIS OF EXO-1-AZABICYCLO[2.2.1]HEPTAN-3-OL | Stephen D. Barrett; Juan C. Jaen; Bradley W. Caprathe; Anthony J. Thomas; Haile Tecle |
| 335-337 | TETRAHYDROFURAN RING-OPENING WITH ACID ANHYDRIDES CATALYZED BY SAMARIUM TRIIODIDE | Weiliang Bao; Taokai Ying; Yongmin Zhang; Mingxin Yu |
| 338-341 | THE EFFICIENT SYNTHESIS OF FMOC-L-HOMOGLUTAMINE | Kazimierz Wiśniewski; Aleksandra S. Kolodziejczyk |
| 341-347 | ALLYLIC AND PHENOLIC PHOSPHATE ESTERS OF DEXANABINOL | Emil Pop; Ferenc Soti; Anat Biegon; Marcus E. Brewster |
| 347-352 | SYNTHESIS OF 4H-CYCLOPENTA[def]CHRYSENE AND OTHER METHYLENE-BRIDGED POLYCYCLIC HYDROCARBONS | Wei Dai; Ronald G. Harvey |
| 352-355 | N-PERFLUOROALKANESULFONYLPHOSPHORAMIDES via AN IMPROVED ATHERTON-TODD REACTION | Shizheng Zhu; Jie Zhang; Bin Xu; Chaoyue Qin |
| 355-357 | A NOVEL SYNTHESIS OF 4-CYANO-2-(2-HYDROXYBENZOYL)PYRIDO[1,2-α]-BENZIMIDAZOLES FROM 3-FORMYLCHROMONE | Kusukuntla Venkat Reddy; A. V. Subba Rao |
| 358-361 | AN EFFICIENT SYNTHESIS OF 3-BROMO-2-(BROMOMETHYL)-1-PROPENE | Theodore Axenrod; Kajal K. Das; Hamid Yazdekhasti; Paritosh R. Dave; Alfred G. Stern |
| 361-364 | A CONCISE SYNTHESIS OF SYMMETRIC 1,3,5-C3-TRISUBSTITUTED BENZENES | M. W. Majchrzak; J. N. Zobel; D. J. Obradovich; G. A. Peterson |
| C | Editorial Board Page | |
| 137-176 | SELECTIVE TRANSITION METAL-PROMOTED CARBON-CARBON AND CARBON-HETEROATOM BOND FORMATION. A REVIEW | Renzo Rossi; Fabio Bellina |
| 177-183 | A PRACTICAL PREPARATION OF L-ASPARTYL-D-2-AMINOBUTYRIC ACID (S)-α-PHENYLPROPYLAMIDE, A NEW HIGH-POTENCY SWEETENER | George A. King III; James G. Sweeny |
| 185-194 | SYNTHESIS OF NITRONES FROM 3,4-DIHYDROISOQUINOLINE DERIVATIVES BY OXIDATION WITH m-CHLOROPEROXYBENZOIC ACID | Bao-Xiang Zhao; Yang Yu; Shoji Eguchi |
| 195-199 | AN ALTERNATIVE STRATEGY FOR THE PURIFICATION OF meso-2,4-PENTANEDIOL | Barbara Gordillo; Javier Hernández |
| 201-205 | ADIPOYLATION OF 2-METHOXYNAPHTHALENE | C. Balo; F. Fernández; E. Lens; C. López |
| 207-210 | NEWER ROUTE FOR THE SYNTHESIS OF β-PHENYLTHIO, β-PHENYLSULFINYL AND β-PHENYLSULFONYL NITROETHYLENES | V. Ramamoorthy; S. Sivasubramanian; S. Muthusubramanian |
| 211-214 | A CONVENIENT SYNTHESIS OF OXAZOLO[3,2-a]QUINOLONES | Hisham A. Abd El-Nabi |
| 214-218 | SYNTHESIS OF DIETHYL 3-ARYL-3-OXOPROPYLPHOSPHONATES | Jen-Wen Yu; Steve K. Huang |
| 218-221 | ASYMMETRIC SYNTHESIS OF (R)-N-(t-BUTOXYCARBONYL)-4-CYANOPHENYLALANINE METHYL ESTER | Angelo Pecunioso; Damiano Papini; Bruno Tamburini; Francesco Tinazzi |
| 221-223 | A FACILE SYNTHESIS OF 3-FLUOROTHIOPHENE-2-CARBOXYLIC ACID | Edward C. Taylor; Ping Zhou |
| 223-226 | THE ALKYLATION OF COUMARIN AT C-3 OF 4-HYDROXYCOUMARIN | Ibro Tabakovic; Katmerka Tabakovic; Igor Gaon |
| 226-230 | AN IMPROVED GENERAL METHOD FOR THE PREPARATION OF 4-ARYL SUBSTITUTED bisPYRAZOLO[3,4-b;4,3'-e]PYRIDINES | Agnieszka Puchala; Danuta Rasala; Erkki Kolehmainen; Monika Prokesová |
| 231-234 | AN ALTERNATIVE SYNTHESIS OF ETHYL 3-(2-CHLORO-4,5-DIFLUOROPHENYL)-3-OXOPROPIONATE AND ETHYL 3-(2,6-DICHLORO-5-FLUOROPYRIDIN-3-YL)-3-OXOPROPIONATE | Frank J. Urban; Bernard S. Moore; Peter L. Spargo |
| 234-236 | AN IMPROVED SYNTHESIS OF bis(p-PHENYLENE)-32-CROWN-4 | Devdatt S. Nagvekar; Harry W. Gibson |
| 237-240 | IMPROVED SYNTHESES OF 20- AND 26-MEMBERED bis(5-CARBOMETHOXY-1,3-PHENYLENE) CROWN ETHERS | Devdatt S. Nagvekar; Harry W. Gibson |
| 240-242 | 5-BENZYLOXYRESORCINOL, A MONOPROTECTED PHLOROGLUCINOL | Devdatt S. Nagvekar; Harry W. Gibson |
| C | Editorial Board Page | |
| 249-288 | bis-PROTECTED HYDROXYLAMINES AS REAGENTS IN ORGANIC SYNTHESIS. A REVIEW | Jeffrey L. Romine |
| 289-318 | THE TRIFLUOROMETHYL GROUP IN ORGANIC SYNTHESIS. A REVIEW | Alexander S. Kiselyov; Lucjan Strekowski |
| 319-324 | SIMPLE PROCEDURES FOR THE PREPARATION OF α,ω-HYDROXYALKANETHIOLS | Luis E. Iglesias; Alicia Baldessari; Eduardo G. Gros |
| 325-332 | SYNTHESIS OF 6H-bis-[1]-BENZOPYRANO[2,3-b:3′,4′-e]PYRIDIN-8(8H)ONES AND 3-(2′-HYDROXYBENZOYL)-5H-[1]BENZOPYRANO[4,3-b]PYRIDINES AND THEIR DERIVATIVES | K. Venkat Reddy; G. Sabitha; A. V. Subba Rao |
| 333-338 | STEREOSPECIFIC ONE-POT SYNTHESIS OF 5-CARBOXY-3,4-DIPHENYLIMIDAZOLIDIN-2-ONE, A USEFUL PRECURSOR TO THE CORRESPONDING 2,3-DIAMINOPROPANOIC ACID | Ivanka K. Kavrakova; Maria J. Lyapova |
| 339-344 | AN UNUSUAL EPIMERIZATION IN THE OXIDATION OF A 4C-(HYDROXYMETHYL)-2,3,4-TRIDEOXY-2-HEXENOPYRANOSIDE USING FETIZON'S REAGENT | Andrew G. H. Wee; Lin Zhang |
| 345-347 | CONVENIENT AND EFFICIENT SYNTHESIS OF IMIDAZOLIUM CYCLOPHANES | Cheng-He Zhou; Ru-Gang Xie; Hua-Ming Zhao |
| 348-351 | EFFICIENT PREPARATION OF 4-SUBSTITUTED-6-ACYL-7-METHOXYCOUMARINS | M. V. Paradkar; M. S. Kulkarni; S. A. Kulkarni; H. M. Godbole |
| 352-355 | A COMPARATIVE STUDY OF OXIDANTS ON THIOLS | K. Ramadas; N. Srinivasan; N. Janarthanan; R. Pritha |
| 355-359 | SELECTIVE REDUCTION OF α,β-UNSATURATED ALDEHYDES AND KETONES TO ALLYLIC ALCOHOLS WITH DHSOBUTYLALKOXYALANES | Jin Soon Cha; Oh Oun Kwon; Sang Yong Kwon |
| 360-361 | 4-CARBOMETHOXYNICOTINIC ACID | B. S. Moore; R. W. McLaughlin; F. J. Urban; G. R. Young |
| 362-365 | SYNTHESIS OF 2-ARYL[1,2,4]-TRIAZOLO[5,1-b]BENZOTHIAZOLES | Huey-Min Wang; Ling-Ching Chen |
| 366-369 | AN OLIGO VICINAL DIIMINE BY THE EHRLICH-SACHS REACTION OF A β-IMINOKETONE WITH NITROSOBENZENE | Frank Millich; Modasser T. El-Shoubary |
| C | Editorial Board Page | |
| 127-164 | PROGRESS IN THE MITSUNOBU REACTION. A REVIEW | David L. Hughes |
| 165-171 | TOTAL SYNTHESIS OF (±)-SIGMOIDIN-A [3′,4′,5,7-TETRAHYDROXY-2-(γ,γ-DIMETHYLALLYL)FLAVANONE] AND OF ANTIARONEF | Lianyun Zhao; Yulin Li |
| 173-177 | AN EFFICIENT ONE POT SYNTHESIS OF N,N-DISUBSTITUTED UNSYMMETRICAL UREAS AND CARBAMATES | N. Choy; K. Y. Moon; C. Park; Y. C. Son; W. H. Jung; Ho-Il Choi; C. S. Lee; C. R. Kim; S. C. Kim; H. Yoon |
| 179-183 | REDUCTIVE ALKYLATION OF α-AMINOAMIDES | Paolo Pevarello; Raffaella Amici; Vittorio Pinciroli; Mario Varasi |
| 185-192 | CONDENSATION OF FORMALDEHYDE WITH PHLOROGLUCINOL AND ITS MONOMETHYL ETHER | E. Kiehlmann; E. C. Lathioor; K. W. Lai |
| 193-201 | SYNTHESIS AND ENZYMATIC RESOLUTION OF A CARBOCYCLIC ANALOGUE OF RIBOFURANOSYLAMINE | Michael L. Edwards; James E. Matt Jr.; David L. Wenstrup; Christopher A. Kemper; Rose A. Persichetti; Alexey L. Margolin |
| 203-209 | SYNTHESES OF α- AND β-DIMERS OF LITHOCHOLIC ACID ESTERS | Yuexian Li; Jerry Ray Dias |
| 211-214 | SYNTHESIS OF cis-[4-(AMINOMETHYL)-2-CYCLOPENTENYL]METHANOL FROM NORBORNADIENE | Carmen Balo; Belen Dominguez; Franco Fernandez; Evangelina Lens; Carmen Lopez |
| 215-216 | A CONVENIENT SYNTHESIS OF 2(5H)-FURANONE | Ruzhen Cao; Chong Liu; Lunzu Liu |
| 217-221 | SYNTHESIS OF 7-DESOXY-8-ALLYLCOUMARINS | Raghao S. Mali; Ashok S. Walture; Kantipudi N. Babu |
| 221-225 | EXPEDIENT SYNTHESES OF ESPINTANOL, p-METHOXYCARVACROL AND THYMOQUTNOL DIMETHYL ETHER | Bjora C. Soderberg; Shari L. Fields |
| 226-230 | CONDENSATION OF 1,4-DIACETYL-2,5-PIPERAZINEDIONE WITH ALDEHYDES PROMOTED BY ULTRASONICALLY DISPERSED POTASSIUM | Li Xin Wang; Yao Zeng Shi; Ming Hua Xu; Hong Wen Hu |
| 230-234 | SYNTHESIS OF 1,3,6,8-TETRAMETHOXY-cis-4b,5,9b,10-TETRAHYDROINDENO[2,1-a]INDENE-5,10-DIONE | D. E. Bianchi; E. N. Alesso; G. Y. Moltrasio Iglesias |
| 234-237 | RAPID OXIDATION OF SULFIDES AND SULFOXIDES WITH SODIUM HYPOCHLORITE | Jitender M. Khurana; Atulya K. Panda; Abhijit Ray; Amita Gogia |
| 237-241 | MIXED DISULFIDES OF L-CYSTEINE AND ITS DERIVATIVES WITH 2-MERCAPTOETHANOL | Herbert T. Nagasawa; Jonathan F. Cohen; William B. Rathbun |
| 242-244 | 6,6-bis(CARBOXY-2-OXABUTYL)-4,8-DIOXAUNDECANE-I,II-DICARBOXYLIC ACID | George R. Newkome; Claus D. Weis |
| 245-246 | SYNTHESES OF 2-CHLORO-4,5-DIFLUOROBENZOIC ACID | Zhibin Li; Naihua Huang |
| 247 | CORRIGENDUM | |
| C | Editorial Board Page | |
| 603-612 | CYCLOADDITIONS OF AZIDOALKYLCARBOXYLATES TO ACETYLENES AND ENAMINES. REGIOSELECTIVE SYNTHESIS OF SUBSTITUTED TRIAZOLES | F. Palacios; A. M. Ochoa de Retana; J. Pagalday; J. M. Sánchez |
| 613-619 | NOVEL SYNTHESIS OF SOME PYRIDINETHIONE NUCLEOSIDES RELATED TO 3-DEAZAUREDINE | Adel M. E. Attia; Elsayed I. Ibrahim; Fouad E. A. Hay; Mohammed M. A. Abbasi; Hanaa A. E. Mansour |
| 621-624 | PRACTICAL SYNTHESIS AND CHARACTERIZATION OF 7-BENZYLIDENENALTREXONE (BNTX) | Anita H. Lewin; Melanie R. Nilsson; Jason P. Burgess; F. Ivy Carroll |
| 625-635 | 1,3-DIPOLAR CYCLOADDITION OF AZIDOALKYLPHOSPHONATES AND CARBOXYLATES TO MALEIMIDE AND NAPHTHOQUINONE | F. Palacios; A. M. Ochoa de Retana; J. Pagalday |
| 637-644 | A SYNTHESIS OF 4-α-GUANIDINO-2-DEOXY-2,3-DIDEHYDRO N-ACETYLNEURAMINIC ACID | John Scheigetz; Robert Zamboni; Michael A. Bernstein; Bruno Roy |
| 645-650 | REGIOSELECTIVE BROMINATION OF CARDANOL DERIVATIVES | O. A. Attanasi; S. Buratti; P. Filippone |
| 651-652 | IMPROVED SYNTHESIS OF 2H-1,3(3H)-OXAZINE-2,6-DIONE (OXAURACIL) | Gretchen M. Rehberg; Brian M. Glass |
| 652-656 | DIBROMANTIN AS A REAGENT FOR THE AROMATIC BROMINATION OF POLYALKYLBENZENES | Xavier Herault; Pakorn Bovonsombat; Edward Mc Nelis |
| 657-659 | AN IMPROVED SYNTHESIS OF 1-(2-HYDROXYETHYL)URACIL | Baijayantimala Garnaik |
| 660-663 | SRN1 REACTIONS IN LIQUID AMMONIA AT ROOM TEMPERATURE | P. G. Manzo; S. M. Palacios; R. A. Alonso; R. A. Rossi |
| 663-667 | FACILE SYNTHESIS OF 3-CHLOROCOUMARINS | Raghao S. Mali; Jyoti V. Deshpande |
| 668-670 | PREPARATION OF NEW 4′,5′-DISUBSTITUTED BENZOCROWN ETHERS | Haluk Akkus; Ahmet Gül |
| 671-674 | PREPARATION OF 2(2-HYDROXYMETHYL-6-METHYL)PHENYLETHANOL | D. G. Tombari; A. G. Moglioni; G. Y. Moltrasio Iglesias |
| 674-678 | A CONVENIENT SYNTHESIS OF δ-CONICEINE | Norbert De Kimpe; Elena Stanoeva; Angelina Georgieva; Marian Keppens; Oleg Kulinkovich |
| 678-682 | SYNTHESIS OF PYRAZINO(3,2,1-J,K)CARBAZOLE DERIVATIVES | K. J. Rajendra Prasad; C. S. Vijayalakshmi; D. Sowmithran |
| 682-684 | AN EFFICIENT SYNTHESIS OF (S)-(+)-2-TRIDECANOL ACETATE, AN AGGREGATION PHEROMONE OF DROSOPHILA MULLERI | Franz Bracher; Brigitte Schulte |
| 685-690 | SYNTHESES OF 3-AND 3,3′-SUBSTITUTED 1,1′-BI-2-NAPHTHOLS | Jing Li; Weidong Li; Ying Li; Yulin Li; Shiyan Yang |
| 691-694 | SYNTHESIS OF A SPIROCYCLIC OXENDOLE ANALOGUE AS A PUTATIVE REPLACEMENT FOR PR02-PRO3-GLY4-PHE5 IN BRADYKININ ANTAGONISTS | R. Richard Goehring |
| C | Editorial Board Page | |
| 393-420 | SYNTHESIS OF CARCINOGENIC OXYGENATED DERIVATIVES OF BENZ[c]ACRIDINES. A REVIEW | Noboru Motohashi; Masami Kawase; Jahangir Emrani |
| 421-428 | SYNTHESIS OF 4-(NITROBENZYL- AND BENZOYL)PIPERIDINE DERIVATIVES BY NITRATION OF ARYLALKYLPIPERIDINES | Siya Ram |
| 429-438 | SYNTHESIS OF IMIDAZOQUINOLINES AND IMIDAZOISOQUINOLINES FROM AZANAPHTHALENE CARBOXYLIC ACIDS | Kevin C. Langry |
| 439-444 | AN ALTERNATIVE SYNTHESIS OF ARYL AND HETEROARYL BROMIDES FROM ACTIVATED ARYL HYDROXY COMPOUNDS | Alan R. Katritzky; Jianqing Li; Christian V. Stevens; David J. Ager |
| 445-457 | A CONVERGENT SYNTHESIS OF (±)-SARCOPHYTOL-A BENZYL ETHER | Weidong Li; Jianmin Mao; Ying Li; Yulin Li |
| 459-464 | REDUCTION OF ORGANIC COMPOUNDS WITH SODIUM ALUMINUM HYDRIDE IN THEORETICAL AMOUNT | Jin Soon Cha; Herbert C. Brown |
| 465-468 | SYNTHESIS OF SEVERAL N-SUBSTITUTED AMINO-2-PYRIDONES | Galal E. H. Elgemeie; Samia R. El-Ezbawy; Hosny A. Ali; Abdel-Kader Mansour |
| 469-471 | IMPROVED ALKYLATION OF ETHYL ACETOACETATE AND DIETHYL MALONATE | Didier Barbry; Catherine Faven; Aziz Ajana |
| 471-472 | IMPROVED PREPARATION OF 4-CHLOROMETHYLPHENYL ACETATE | Jørn B. Christensen |
| 473-476 | SYNTHESIS AND COMPETITIVE N- AND O-ALKYLATION OF 10-METHYLPYRIDO[3,2-g]QUINOLINE-4,6-DIONE | A. Mahamoud; J. -P. Galy; J. Barbe |
| 476-478 | A CONVENIENT PREPARATION OF 9H-FLUORENE-9-ACETIC ACID | R. Richard Goehring |
| 479-482 | REGIOSELECTIVE SYNTHESIS OF 10-HYDROXY-11-METHOXYAPORPHINE FROM (RS)-10,11-DIHYDROXYAPORPHINE | Jack C. Kim; Won-Woo Park |
| 482-484 | A SHORT SYNTHESIS OF TRIDEC-12-EN-2-ONE, THE MINOR CONSTITUENT OF THE BARK OF LITSEA ELLIPTICA (LAURACEAE) | S. Mithran; A. S. Subbaraman; V. R. Mamdapur |
| 485-488 | TREATMENT OF CONJUGATED AZOALKENES WITH N-ACYL-N'-TOSYLHYDRAZIDES. A USEFUL ENTRY TO ASYMMETRIC bis-ACYLHYDRAZONES | Orazio A. Attanasi; Stefania Santeusanio; Franco Serra-Zanetti |
| 488-491 | A HIGHLY STEREOSELECTIVE TRANSFORMATION OF β-SANTALENE TO (E)-β-SANTALOL | P. A. Unnikrishnan |
| 491-494 | A SUPERIOR METHOD FOR THE SYNTHESIS OF 7a-METHYL-2,3,7,7a-TETRAHYDRINDEN-5(6H)-ONE | H. Surya Prakash Rao; K. Subba Reddy |
| 494-497 | A SIMPLE AND SHORT SYNTHESIS OF 2(2′-AMINOBENZYLAMINO)BENZYL ALCOHOL, A CONSTITUENT OF JUSTICIA GENDARUSSA BURM LEAVES | Vijayendra P. Kamat; Janardan K. Kirtany |
| 498 | ADDENDUM. A SIMPLE, EFFICIENT PREPARATION OF 1,1-bis(TRIMETHYLSILOXY)-1,3-BUTADIENE | |
| C | Editorial Board Page | |
| 257-290 | RECENT PROGRESS IN THE USE OF SULFONYL RADICALS IN ORGANIC SYNTHESIS. A REVIEW | Michèle P. Bertrand |
| 291-320 | THE SYNTHESIS AND REACTIONS OF PRISMANES. RECENT DEVELOPMENTS | Mark A. Forman; William P. Dailey |
| 321-326 | FACILE AND HIGH-YIELD SYNTHESIS OF NEW 4-PHOSPHORANYLIDENE-4,5-DIHYDROPYRAZOL-5-ONES BY REACTION OF CONJUGATED AZOALKENES WITH PHOSPHINES | Orazio A. Attanasi; Paolino Filippone; Daniela Giovagnoli |
| 327-330 | A SIMPLE AND EFFICIENT PREPARATION OF METHOXYMETHYL ESTERS OF PENICILLINS AND CEPHALOSPORINS | Jacek Pankowski; Jerzy Winiarski |
| 331-335 | A SIMPLE SYNTHESIS OF THE HETEROCYCLIC S,S-DIPHENYLSULFILIMINES | Olga G. Vlasova; Oleg A. Rakitin; Lenor I. Khmelnitski |
| 337-341 | AN ALTERNATE METHOD FOR THE SYNTHESIS OF SECONDARY NITRAMINES | Z. Daszkiewicz; A. Domański; J. B. Kyziol |
| 343-346 | AN EFFICIENT, LARGE-SCALE SYNTHESIS OF IDOXIFENE {(E)-1-[4-[2-(N-PYRROLIDINO)ETHOXY]PHENYL]-1-(4-IODOPHENYL)-2-PHENYL-1-BUTENE} | Raymond McCague; Gerard A. Potter; Michael Jarman |
| 347-349 | SINGLE-STEP SYNTHESIS OF 2,3-DIHYDRO-2,2DIMETHYL-1H-PHENOTHIAZIN-4(10H)-ONES | V. Gupta; A. Gupta; R. S. Rathore; R. R. Gupta |
| 349-352 | AN IMPROVED SYNTHESIS OF THIENO(2,3-B)QUINOLINES via S-OXIDES | S. P. Rajendran; P. Shanmugam |
| 353-355 | OXIDATIVE REARRANGEMENT OF THE PURINE RING USING MAGNESIUM MONOPERPHTHALATE | Adel Amer |
| 355-357 | AN ECONOMICAL PREPARATION OF 2-(2-BROMOETHYL)-1,3-DIOXANE | Jorn B. Christensen; Anne Schluter |
| 357-360 | SYNTHESIS OF N-PHOSPHORYLUREAS BY REACTION OF PHOSPHORYLAMIDES WITH N-SUBSTITUTED TRICHLOROACETAMIDES | Jan Petrov; I. Atanassova; V. Ognyanova |
| 360-362 | SYNTHESIS OF 3-ACETOACETYL-7-METHYL-2H,5H-PYRANO[4,3-B]PYRAN-2,5-DIONE | B. Boutemeur-Kheddis; A. Bendaas; M. Hamdi; R. Sakellariou; V. Spéziale |
| 362-366 | A NEW APPROACH TO ALKYL 2-OXOQUINOLINE-3-ACETATES BY TRIPHENYLPHOSPHINE-INDUCED CYCLIZATION OF ALKYL O-FORMYLMALEANILATES | N. P. Argade; S. M. Babar; V. Balasubramaniyan |
| 366-370 | EFFICIENT REGIOSELECTIVE ALKYLATION OF 2-CARBOXAMIDOPIPERAZINE. APPLICATION TO THE SYNTHESIS OF THE NMDA COMPETITIVE ANTAGONIST ()-CPP | P. Pevarello; G. Scappi; M. Varasi |
| 370-373 | PURIFICATION OF 1,2-DIHYDRONAPHTHALENE- AN IMPORTANT INTERMEDIATE IN THE HYDROPROCESSING OF NAPHTHALENE | Mike D. Cagle; Sharbil J. Firsan; E. J. Eisenbraun |
| C | Editorial Board Page | |
| 607-632 | PROGRESS IN THE FISCHER INDOLE REACTION. A REVIEW | David L. Hughes |
| 633-637 | SYNTHESIS OF DIMETHYL 1,4-DIHYDROXY-5,6,8-TRIMETHOXYNAPHTHALENE-2,3-DICARBOXYLATE, A KEY INTERMEDIATE FOR FREDERICAMYCIN A | Raghao S. Mali; Prakash G. Jagtap |
| 639-647 | SYNTHESIS OF 2-0-PROTECTED GLYCEROL DERIVATIVES | J. Michael Chong; Kenneth K. Sokoll |
| 649-657 | SYNTHESIS OF FUNCTIONALIZED ACRYLATES | Michele Curci; Jean-Luc Mieloszynski; Daniel Paquer |
| 659-663 | ONE-POT SYNTHESIS PF NOVEL 10-ARYL[1,2,4]TRIAZOLO[3′,4′:2,3][1,3,4]-THIADIAZEPINO[6,7-c]QUINOLIN-6(5H)-ONES | A. Jayashree; Malleshwar Darbarwar |
| 665-671 | PREPARATIVE SYNTHESIS OF RL-252 VANADYL COMPLEX | Michael W. Wilson; John C. Hodges |
| 673-679 | PREPARATION OF OPTICALLY ACTIVE NEW MERCAPTO CHIRAL AUXILIARIES DERIVED FROM CAMPHOR | Dong-Sheng Lee; Shung-Ming Hung; Ming-Chun Lai; Han-Yang Chu; Teng-Kuei Yang |
| 681-683 | A NEW METHOD FOR THE SYNTHESIS OF DIACYL SELENIDES | Yongmin Zhang; Xueshun Jia; Xunjun Zhou |
| 683-686 | SYNTHESIS OF N-METHYLATED QUINOLONES | J. N. Domínguez; J. Charris |
| 687-689 | A FACILE SYNTHESIS OF β-DAMASCONE | P. A. Unnikrishnan |
| 690-693 | A SIMPLE PROCEDURE FOR THE PREPARATION OF (METHYL- AND PHENYLTHIO)ARYLOXYACETONITRILES | Andrzej Jończyk; Essa-Hassan Muttar |
| 693-695 | A CONVENIENT METHOD FOR THE SYNTHESIS OF FLAVANONES BY THE SELECTIVE OXIDATION OF FLAVAN-4-OLS WITH HYPERVALENT IODINE | Om V. Singh |
| 696-698 | CHLOROFORM-MEDIATED DDQ OXIDATION OF N-METHOXYSEPTORINOL, A SUBSTANCE ISOLATED FROM THE FUNGUS SEPTORIA NODORUM BERK | M. Devys; M. Barbier; J. F. Bousquet; A. Kollmann |
| 698-703 | SYNTHESIS OF CARBENOXOLONE ANALOGS FROM ARGENTATIN B | Roberto Martínez; Ma. del Rosario Arellano-García; Mariano Martínez-Vazquéz; A. Gallegos Julian |
| 703-704 | SIMPLE AND CONVENIENT PROCEDURE FOR THE PREPARATION OF 1-METHYL-4-NITROBENZIMIDAZOLE | Viktor Milata; Dusan Ilavský |
| 705-706 | PREPARATION OF SOME 2,3-DIHYDROBENZOTHIAZOLE-2-CARBOXAMIDES | H. P. Penner; Racine Gamer; Edgar L. Scott III |
| 707-708 | AN IMPROVEMENT IN THE SYNTHESIS OF 1,2,4,9-TETRAHYDROCARBAZOL-3-ONE | William A. Boulanger; Victoria Dolsen |
| 708-710 | A SIMPLE PREPARATION OF 4-AMINO-5-ARYL-2H-IMIDAZOL-2-ONES | Madhu Srivastava; Ram Lakhan |
| 711 | CORRIGENDUM | |
| 713-727 | INDEXES | |
| C | Editorial Board Page | |
| 481-513 | PREPARATION AND REACTIONS OF INDOLIN-2(3H)-ONES. A REVIEW | Gary M. Karp |
| 515-556 | THE LATERAL METALATION OF ISOXAZOLES. A REVIEW | Nicholas R. Natale; Yousef R. Mirzaei |
| 557-562 | PREPARATION OF PHENYLGLYCOLIC ACIDS AND SODIUM p-(N,N-DIALKYLAMINO)PHENYLGLYCOLATES | Alan R. Katritzky; Barbara Galuszka; Stanislaw Rachwal; Doreen Lynch |
| 563-568 | FACILE LARGE SCALE SYNTHESIS OF 5-ALKYLURACILS | Henryk Koroniak; Aleksander Jankowski; Miroslaw Krasnowski |
| 569-575 | SYNTHESIS OF 2-ARYL-4,5,6,7-TETRAHYDRO-6,6-DIMETHYL-2 H-BENZO[D][1,2,3]TRIAZOL-4-ONES | H. Abdel Hamid; A. Mousaad; M. Sayed; E. S. H. El Ashry |
| 577-579 | AN IMPROVED SYNTHESIS OF 5-(3,4-DIMETHOXYPHENYL)-3-HYDROXY-4-NITROCYCLOHEXENE | A. F. Ibañez; A. R. Martinez; G. Y. Moltrasio Iglesias |
| 579-581 | AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1,6-DICARBOXYHEX-3-ENE | Pradeep T. Deota; Sugra Abid |
| 581-583 | A FACILE SYNTHESIS OF bis(3-ARYL-3-OXO-1-PROPENYL)BENZENES | Jian-Guo Shao; Jing-Feng Zhou; Chang-Qing Liu; Qi Zhong |
| 583-585 | AN IMPROVED SYNTHESIS OF 2-METHALLYLOXYPHENOL | V. B. Deodhar; V. S. Dalavoy; U. R. Nayak |
| 585-587 | SYNTHESIS OF 1-HYDROXY-7-PHENOXYNAPHTHALENE | Alan R. Katritzky; Marudai Balasubramanian; Michael Siskin |
| 588-590 | FACILE SYNTHESIS OF 2-ARYL-4H-3,1-BENZOXAZIN-4-ONES | D. V. Ramana; E. Kantharaj |
| 590-592 | PREPARATION OF bis(2,2,2-TRIFLUOROETHYL)SELENIDE AND TELLURIDE AND OF BIS(2,2,2-TRIFLUOROETHYL)DISELENIDE AND DITELLURIDE | K. K. Bhasin; Vijay Gupta; R. Khajuria; R. P. Sharma |
| 592-594 | SYNTHESIS OF PENTAFLUOROPHENYL-4-(N-MALEIMIDOMETHYL) CYCLOHEXANE-1-CARBOXYLATE (FMCC) | Maciej Adamczyk; Donald Johnson |
| 595-597 | A SIMPLE, EFFICIENT PREPARATION OF 1,1-BIS(TRIMETHYLSILOXY)-1,3-BUTADIENE | Gregory S. Welmaker |
| 597-599 | A ONE-STEP PREPARATION AND HETERO-DIELS-ALDER DIMERIZATION OF 2-PHENYLPROPENAL | Tarja Laitalainen; Pirjo Kuronen; Antti Hesso |
| 600-601 | A SIMPLE AND PRACTICAL APPROACH TO UNSYMMETRICAL PHENYLUREAS | Krishnamurthy Ramadas; Natarajan Srinivasan |
| 602-606 | THIOPHENO[3,2][1]BENZAZEPINE, BENZO[3,4]CYCLOHEPTA[2,1-b]THIOPHENES, THIAZOLO[5,4-d][1]BENZAZEPINE AND BENZO[3,4]CYCLOHEPTA[2,1-d]THIAZOLES | V. Peesapati; N. Lingaiah |
| C | Editorial Board Page | |
| 141-208 | THE USE OF ISOCYANIDES IN HETEROCYCLIC SYNTHESIS. A REVIEW | Stefano Marcaccini; Tomás Torroba |
| 209-213 | AN EFFICIENT, LARGE-SCALE SYNTHESIS OF TRIISOPENTADECANOIN | Thomas A. Foglia; Peter D. Vail |
| 215-222 | SELENIUM OXIDE OXIDATION OF ABIETA-7,13-DIENES IN METHANOL | A. San Feliciano; J. M. Miguel del Corral; M. Gordaliza; M. A. Salinero |
| 223-228 | CONVENIENT SYNTHESIS OF 6-METHYL, 8-METHYL AND 6,8-DIMETHYL DERIVATIVES OF 5-HYDROXY-1,2,3,4-TETRAHYDRO-2-QUINOLINONE | Dominique Blondet; Francette Laure; Jean-Claude Pascal |
| 229-231 | IMPROVED PREPARATION OF AMINOMETHYLENEMALONIC ACID DERIVATIVES BY TIN-PROMOTED ADDITION OF DIETHYL MALONATES TO NITRILES | Marco Nicolini; Attilio Citterio |
| 232-233 | IMPROVED AND CONVENIENT SYNTHESIS OF DISULFIDES IN THE ABSENCE OF SOLVENT CATALYZED BY CLAYFEN | Harshadas M. Meshram |
| 234-237 | SYNTHESIS OF 2-DIMETHYLAMINO-5-(α-CHLOROALKENYL)-13-OXAZIN-6-ONES | Egle M. Beccalli; Alessandro Marchesini |
| 237-240 | THE SYNTHESIS OF TWO BICYCLO[4.3.0]NONANE DERIVATIVES | C. W. Bird; R. Cooper |
| 241-243 | MICHAEL REACTION OF FLUORENE AND INDENE BY PHASE-TRANSFER CATALYSIS | Yan Chaoguo; Lu Wenxing; Wu Jitao |
| 243-246 | PREPARATION OF THE RACEMATE AND ENANTIOMERS OF 3-HYDROXY-5,5-DIMETHYLHEXANOIC ACID | Wayne J. Brouillette; Ahmed S. Abuelyaman; Carla A. Hosmer; Robert N. Comber; Ashraf Saeed |
| 247-249 | AN EFFICIENT PREPARATION OF 2H-[5,4-b]-PYRIDOISOTHIAZOLONE | Stephen W. Wright; Ronald L. Corbett |
| 249-251 | AN IMPROVED SYNTHESIS OF 1-(t-BUTYLOXYCARBONYL)-3-(BROMOMETHYL)INDOLE | T. K. Venkatachalam; S. Mzengeza; M. Diksic |
| 252-255 | SYNTHESIS OF 3,6-DIMETHOXY-2-NAPHTHALDEHYDE | Adel M. Moussa; Jun-Rui Yang; Margaret E. Langmuir |
| 255-258 | A PRACTICAL PROCEDURE FOR THE SYNTHESIS OF 5-SUBSTITUTED γ-LACTAMS | Z. Y. Wei; E. E. Knaus |
| C | Editorial Board Page | |
| 623-647 | SYNTHETIC OXIDATIONS WITH HYPOCHLORITES. A REVIEW | Jacek Skarzewski; Renata Siedlecka |
| 649-654 | SYNTHESES OF 2,3-DIHALO-1-(PHENYLSULFONYL)INDOLES | Gordon W. Gribble; Brett D. Allison; Samuel C. Conway; Mark G. Saulnier |
| 655-659 | SELECTIVE NITROSATION OF DIALKYLUREAS CONTAINING A BASIC β-NITROGEN | Joseph E. Saavedra; David W. Farnsworth |
| 661-665 | CONVENIENT PREPARATION OF 1-ADAMANTANOL FROM ADAMANTANE INDUCED BY A HYDRIDE TRANSFER | M. Gami; R. Jalal; R. Gallo |
| 665-669 | FORMATION OF A 1,2-DIHYDROPYRAZINE USING AN AMINO ACID AND D-GLUCOSE | C. W. Yuan; J. Beauhaire; C. Marty; J. L. Fourrey; H. Richard |
| 670-672 | AN IMPROVED SYNTHESIS OF 2,3,4,6,7,8-HEXAHYDROQUINOLINES | Elmar Schuster; Gerhard Jas; Dieter Schumann |
| 673-675 | A FACILE PREPARATION OF 2,3,4,4a,5-6-HEXAHYDROQUINOLINE | Bodo Juhnke; Gerhard Jas; Dieter Schumann |
| 675-678 | A CONVENIENT SYNTHESIS OF SOME NEW PYRANO[2,3-d]PYRIMIDINES | V. K. Ahluwalia; Rakesh Kumar; Renu Aggarwal |
| 679-681 | SYNTHESIS OF 2(N-ALKYLAMINO)ISOBUTYRALDEHYDES | Norbert De Kimpe; Marc Boeykens; Mark Boelens; Kurt De Buck; Johan Cornelis |
| 682-684 | SIMPLE SYNTHESIS OF ARYLALIPHATIC DIKETONES | Adama Saba; Faustin Sié Sib; Jean-Pierre Aycard |
| 685-687 | A CONVENIENT SYNTHESIS OF cis-(1R)-N-BENZYL-(2S)-(HYDROXYMETHYL)CYCLOHEXYLAMINE | B. Vanderplas; C. W. Murtiashaw; T. Sinay; F. J. Urban |
| 687-690 | STUDY IN CROSSOVER FRIES MIGRATION | R. N. Khanna; K. P. Singh; Jyotsana Sharma |
| 690-692 | AN IMPROVED SYNTHESIS OF 2,4-DIMETHOXYPHENYLACETIC ACID | E. N. Alesso; J. M. Aguirre; G. Y. Moltrasio Lglesias |
| 692-694 | A CONVENIENT SYNTHESIS OF (4-NITROPHENYL) (4-PIPERIDINYL) KETONE | Michel Monclus; André Luxen |
| 695-696 | A CONVENIENT PROCEDURE FOR THE PREPARATION OF 2-BROMO-1-PHENYLETHANOL | S. S. Bhosale; P. L. Joshi; A. S. Rae |
| 696-698 | A CONVENIENT PREPARATION OF 4-CYCLOPROPYLPHENOL | Bruce W. Horrom; H. Mazdiyasni |
| 698-701 | A NEW SYNTHESIS OF 3-AMINO-1-IMIDAZOLIN-4-ONES BY THE HYDRAZINOLYSIS OF 5-OXAZOLONES | Vinod K. Ahluwalia; Mukesh K. Sharma; Rashmi Sharma |
| 701-704 | IMPROVED PREPARATION OF WHYDROXYPROGESTERONE | M. O. Violeta Benedetti; Gerardo Burton |
| 705-717 | INDEXES | |
| C | Editorial Board Page | |
| 501-507 | PREPARATION OF NOVEL 2-AMINOADAMANTYL- AND 4-AMINOPROTOADAMANTYLCARBONITRILES | Kata Mlinaríc-Majerski; Mira Kaselj; Danko Škare |
| 509-516 | IMPROVED SYNTHESIS OF 3-HALO- AND 3-METHOXYPHENANTHRENES | Ana Eirín; Franco Fernández; Carmen González; Carmen López |
| 517-520 | METHYL CYCLOPROPENE-3-CARBOXYLATES BY DIRECT CATALYTIC CYCLOPROPENATION OF ACETYLENES WITH METHYL DIAZOACETATE | E. A. Shapiro; A. V. Kalinin; O. M. Nefedov |
| 520-522 | A FACILE SYNTHESIS OF 2-(2′-SUBSTITUTED VINYL)BENZOXAZOLES | Jian-Guo Shao; Qi Zhong; Hai-Ping Liao; Chang-Qing Liu; Jing-Feng Zhou |
| 523-525 | FACILE SYNTHESIS AND AANTIMICROBIAL ACTIVITY OF SPIROBICYCLO[3.2.1]OCTANE-2′,3-(4H)-[2H]-THIAZOLO[3,2-B]-s-TETRAZINES | Jag Mohan |
| 525-527 | SYNTHESIS OF EVERNIPENTANONE BY ADDITION OF n-BUTYLLITHIUM ON ETHYL EVERNINATE | M. Devys; E. Desnoës; M. Barbier |
| 527-532 | SYNTHESIS OF β- AND γ-ALKOXY AND β-DIMETHYLAMINO 1- AND 2-SUBSTITUTED-1,3-CYCLOPENTADIENES | William S. Rees Jr.; Kerstin A. Dippel |
| 532-536 | SYNTHESIS OF MODELS RELATED TO TASPINE | M. L. Scarpati; A. Bianco; R. Lo Scalzo |
| 536-539 | A CONVENIENT METHOD FOR THE PREPARATION OF cis-3,4,8,8a-TETRAHYDRO-6H-[1,3]-DIOXEPINO[5,6-d]OXAZOLES | Miljenko Dumć; Ivan Butula; Mladen Vinković; Boris Kamenar |
| 540-543 | FORMATION OF 1-CHLORO-1-ALKYNES FROM 1,1-DICHLORO-1-ALKENES UNDER PHASE-TRANSFER CONDITIONS WITHOUT SOLVENT | Peter Vinczer; Szilvia Sztruhar; Lajos Novak; Csaba Szantay |
| 543-546 | SYNTHESIS OF TWO METHYLBENZOSUBERONES AND A DIMETHYLBENZOCYCLOHEPTENE | Arthur G. Anderson Jr; Harry F. Richards |
| 546-548 | SYNTHESIS OF ESTRIOL 16α-4′,5′-DEHYDROGLUCURONIDE | Maciek Adamczyk; Yon-Yih Chen; Jeffrey R. Fishpaugh |
| 548-551 | SYNTHESIS OF CYCLOPROPANES USING S-ETHENYLSULFILIMINES | Katsuya Ikeda; Hiroshi Satoh; Tamotsu Yamamoto |
| 553-582 | RECENT PROGRESS IN THE CHEMISTRY OF ACYLSILANES. A REVIEW | Pier F. Cirillo; James S. Panek |
| 583-621 | RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF SUBSTITUTED PIPERIDINES. A REVIEW | Chia-Lin J. Wang; Mark A. Wuonola |
| C | Editorial Board Page | |
| 245-284 | BIOSYNTHETIC, BIOMIMETIC AND RELATED EPOXIDE CYCLIZATIONS. A REVIEW | Stephen K. Taylor |
| 285-307 | “CESIUM ION EFFECT” AND MACROCYCLIZATION. A CRITICAL REVIEW | Carlo Galli |
| 309-325 | ELECTROCATALYTIC HYDROGENATION ON HYDROGEN-ACTIVE ELECTRODES. A REVIEW | Jean-Claude Moutet |
| 327-330 | ONE-POT CONVERSION OF CARBOXYLIC ACIDS TO ALDEHYDES BY TREATMENT OF ACYLOXY-9-BORABICYCLO[3,3,1]NONANES WITH LITHIUM tris(DIETHYLAMINO)ALUMINUM HYDRIDE | Jin Soon Cha; Jae Cheol Lee; Heung Soo Lee; Sung Eun Lee |
| 331-334 | SELECTIVE CONVERSION OF AROMATIC NITRILES TO ALDEHYDES BY LITHIUM tris(DIHEXYLAMINO)ALUMINUM HYDRIDE | Jin Soon Cha; Sung Eun Lse; Heung Soo Lee |
| 335-337 | TRANSFORMATION OF CARBOXYLIC ESTERS TO ALDEHYDES WITH LITHIUM tris(DIETHYLAMINO)ALUMINUM HYDRIDE | Jin Soon Cha; Soo Jin Min; Jae Cheol Lee; Heung Soo Lee; Sung Eun Lee |
| 338-339 | AN IMPROVED PROCEDURE FOR THE ISOLATION OF 2-(N,N-DIETHYJAMINOMETHYL)-4-NITROPHENOL | M. C. B. V. de Souza; A. M. R. Bernardino; M. C. Soares; M. G. Retzlaff |
| 339-342 | SYNTHESIS OF 4-trans-[1-[4-[2-(5-CHLORO-2-METHOXYBENZAMIDO)ETHYL] BENZENESULFONYL]UREIDO]CYCLOHEXANOL HEMISUCCINATE ESTER | Robert L. Stephont; R. Sam Niedbala; Keith J. Schrayt; Ned D. Heindel |
| 342-345 | SYNTHESIS OF 1-(2-(2,4-DICHLOROPHENYL)-2-[(2-THIENYL)METHOXY]ETHYL]-lH-IMIDAZOLE AND 1-[2-(2,4-DICHLOROPHEL)-2-[(2-FURYL)METHOXY]ETHYL]-1H-IMIDAZOLE, TWO NEW MICONAZOLE ANALOGUES | Raymundo Cruz-Almanza; Teresa Hemández; Francisco Pérez; Cristina Lemini |
| 346-349 | ONE-POT SYNTHESIS OF ISOTHIOCYANATES FROM PRIMARY AMINES SYNTHESIS USING CYANAMIDE? | Tamotsu Yamamoto; Susumu Sugiyama; Kenji Akimoto; Kiyoshi Hayashi |
| 349-351 | AN IMPROVED SYNTHESIS OF 2,4-HEXADIEN-l-OL | Peter Vinczer; Lajos Novak; Csaba Szantay |
| 352-354 | CONSTRUCTION OF THE PYRAZOLO[1,5-a] [4,1]BENZOTHIAZEPINE SYSTEM BY INTRAMOLECULAR NITRILIMINE CYCLOADDITION | Gianluigi Broggini; Luca Bruché; Gaetano Zecchi |
| 355-358 | SYNTHESIS OF STEROIDAL HETEROCYCLIC COMPOUNDS FROM A CLAISEN CONDENSATION PRODUCT OF A 6-KETO STEROL | A. U. Siddiqui; U. M. Rao; M. Srinivas; A. H. Siddiqui |
| 358-362 | NEW HETEROCYCLES FORMING REACTIONS OF ACYL THIOFORMANILIDES | Zhong E. Lu; Da Qing Sun; Tian Lin Xu; Jun Wan; Le Cun Xu; Ke Qian Chen |
| 363-365 | OXIDATION OF ALCOHOLS USING TRIPHOSGENE | I. A. Rivero; R. Somanathan; L. H. Hellberg |
| 365-368 | A STUDY ON CYANOACETIC ACID HYDRAZIDE | A. Aykut Ikizler; Aysun Lkizler; Neslihan Uzunismail |
| C | Editorial Board Page | |
| i | IMPORTANT NOTICE TO AUTHORS | |
| 1-5 | SYNTHESIS OF SOME TETRAHYDRO-3,3′-BISQUNAZOLIN-4,4′-DIONES | A. K. D. Bhavani; P. S. N. Reddy |
| 7-12 | REDUCTIVE DECYANATION vs ADDITION OF GRIGNARD REAGENTS WITH HINDERED NITRILES | Stuart S. Kulp; Anthony Romanelli |
| 13-20 | RING OPENING OF SOME SUBSTITUTED STYRENE OXIDES | Ulhas P. Dhokte; A. Somasekar Rao |
| 21-26 | SYNTHESIS OF SOME SPIRO-ISOXAZOLIDINE-3,5-DIONES | D. Bhaskar Reddy; V. Padmavathi; B. Seenaiah; M. V. Ramana Reddy |
| 27-32 | SYNTHESIS OF FURANO BENZOSUBERONES AND FURANO TETRALONES via CLAISEN REARRANGEMENT | V. Peesapati; N. Lingaiah |
| 33-37 | SYNTHESIS OF NEW SUBSTITUTED PYRIDINES, PYRANO[2,3-d]IMIDAZOLES AND PYRROLO[2,1-b]QUINAZOLINES | O. H. Hishmat; A. A. Magd El Din; N. A. Ismail |
| 39-43 | AN IMPROVED PROCEDURE FOR THE PREPARATION AND RESOLUTION OF dl-2,3-DIMETHYLSUCCINIC ACID | Scott C. Sutton; Michael H. Nantz; Shawn R. Hitchcock |
| 45-48 | PREPARATION OF N-BENZOYL-1-(5,6-DIMETHOXYINDANYLMETHYLAMINE) FROM 5,6-DIMETHOXYINDANONE | D. G. Tombari; A. G. Moglioni; F. P. Dominici; G. Y. Moltrasio de Iglesias |
| 48-51 | STEREOSELECTIVE REDUCTION OF PIVALOYLOXYMETHYL (2S,5R,6S)-6-ACETYL-3,3-DIMETHYL-7-OXO-4-THIA-1-AZABICYCLO[3.2.0]HEPTANE-2-CARBOXYLATE WITH SODIUM BOROHYDRIDE | Daniele Donati; Carla Marchioro; Bruno Tamburini; Antonella Ursini |
| 52-54 | CONVENIENT SYNTHESIS OF NIESHOUTIN (CYCLOOBLZQUETIN), A FUROCOUMARIN ISOLATED FROM THE HEARTWOOD OF Ptaeroxylon obliquum | R. S. Mali; Anita R. Manekar; S. G. Tilve |
| 55-57 | A NEW, MILD PREPARATION OF 2,4,6-TRINITROFLUOROBENZENE | Julian M. Dust; Richard A. Mandeville |
| 57-60 | AN IMPROVED SYNTHESIS OF MONOESTERS OF PHOSPHORIC ACID | Agnes M. Modro; Tomasz A. Modro |
| 60-63 | REACTION OF THIONYL BROMIDE WITH KETONES | S. M. Al-Mousawi; I. Bhatti; S. D. Saraf |
| 64-66 | A CONVENIENT SYNTHESIS OF METHYL 4-AMINO-5-CHLORO-2-MTHOXYBENZOATE | Richard L. Ehrenkaufer; James G. Scripko; Patricia L. Hoffman |
| 66-67 | IMPROVED SYNTHESIS OF DIMETHYLAMINOTHIOACETAMIDE | Kenneth P. Moder; Frank R. Busch; David C. Richter |
| 67-70 | A NEW ROUTE FOR SYNTHESIS OF 1-TRIACONTANOL | B. V. S. K. Rao; R. Supharao |
| 71-73 | SYNTHESIS OF NOVEL 9-ARYL-2,8-DIMETHYL-9H-PURIN-6-AMINES BASED ON STERICALLY HINDERED o-BROMOANILINES | S. V. Eswaran; S. K. Sajadian |
| C | Editorial Board Page | |
| 571-592 | 1,2-bis(ARYLSULFONYL)ALKENES. A REVIEW | Sergio Cossu; Ottorino De Lucchi; Davide Fabbri; Giulia Licini; Lucia Pasquato |
| 593-610 | THE CHEMISTRY OF 1,3-DIOXIMES. A BRIEF REVIEW | Antigoni Kotali; Vassilios P. Papageorgiou |
| 611-616 | A ONE-POT PREPARATION OF DIMETHYL N-ALKYLIMINODITHIOCARBONATES | C. Alvarez-Ibarra; M. L. Quiroga; E. Martinez-Santos; E. Toledano |
| 617-620 | A CONVENIENT PREPARATION OF DIPHENYLMETHANES FROM BROMOBENZENES USING THE GRIGNARD CROSS-COUPLING REACTION | Takehiko Yamato; Naozumi Sakaue; Kazuaki Suehiro; Masashi Tashiro |
| 621-626 | NITRO DERIVATIVES OF BENZOCOUMARINS. KEY INTERMEDIATES IN THE SYNTHESIS OF BENZOCOUMARIN-BASED FLUORESCENT REAGENTS FOR BIOLOGICAL APPLICATIONS | Jun-Rui Yang; Carol A. Lambert; Margaret E. Langmuir; Richard Laura |
| 627-631 | AN ALTERNATE SYNTHESIS OF 3,4-DIAMINOBEZOPHENONE AND OF MEBENDAZOLE | N. R. Ayyangar; R. J. Lahoti; Thomas Daniel |
| 633-638 | SYNTHESIS OF (E,E)-BIS(ARYLCYCLOPROPYL) SULFONES FROM NOVEL (E,E)-BIS(STYRYL) SULFONES | M. V. Ramana Reddy; D. Bhaskar Reddy; P. V. Ramana Reddy; S. Vijayalakshmi |
| 639-643 | SYNTHESIS OF PRIMIN AND MICONIDIN AND THEIR 3-METHOXY ISOMERS | Sunday S. Arogba |
| 645-650 | NOVEL SYNTHESIS OF PYRIDINE-2(1H)THIONES, N-AMINO-2-PYRIDONES AND PYRIDAZINE DERIVATIVES | G. H. Elgemeie; S. R. El-Ezbawy; M. M. Ramiz; O. A. Mansour |
| 651-654 | OXIDATION OF ADAMANTANE TO 1-ADAMANTANOL USING TETRA-N-BUTYLAMMONIUM OXONE | Rajkumar Kumarathasan; Norman R. Hunter |
| 655-658 | SYNTHESIS OF 2-HALO-4,5-DIFLUOROBENZOIC ACIDS | Tamim F. Braish; Darrell E. Fox |
| 658-660 | AN IMPROVED PREPARATION OF QUINUCLIDIN-3-THIOL | S. D. Aster; S. S. Yang; G. D. Berger |
| 660-665 | THE REACTION OF NINHYDRIN WITH ACETIC ACID | Jack B. Campbell; Edward R. Lavagnino; Charles W. Ryan |
| 665-667 | FACILE CHROMONE RING-OPENING OF KHELLIN | Emile Al-Farhan; Philip M. Keehn; Robert Stevenson |
| 667-670 | A NEW METHOD FOR THE SYNTHESIS OF 3β-HYDROXY-4α-BROMOCARANE AND OF cis-3-CARENE EPOXIDE | Milind D. Choubal; Joseph Y. Bassett |
| 670-672 | A NOVEL CLASS OF OXAZOLE DERIVATIVES. 4-ACYL-2-ARYLTHIO-5-ETHOXYOXAZOLES | Ricardo Bossio; Stefano Marcaccini; Roberto Pepino; Cecilia Polo; Tomás Torroba |
| 673-676 | THE MANNICH REACTION OF CYCLIC KETONES, AROMATIC ALDEHYDES AND AROMATIC AMINES | Yi Lin; Zou Junhua; Lei Huangshu; Lin Xiaomei; Zhang Mingxiao |
| 676-679 | IMPROVED SYNTHESIS OF A 2-ARYLBENZO[B]FURAN-3-CARBOXYLIC ACID | Michel Barbier |
| 679-682 | SYNTHESIS OF NOVEL TRIAZOLO[2,3,b]-1,3,4-THIADIAZOLIUM SALTS | Zhu Zheng-Hua; Chen Shu-Ling; Yao Zu-Guang |
| C | Editorial Board Page | |
| 399-402 | N-ALKYLATION OF HINDERED SECONDARY AROMATIC AMINES WITH 2-IODOBUTANE | Alan R. Katritzky; Jing Wu; Stanislaw Rachwal |
| 403-411 | REDUCTION OF HETEROCYCLIC ALCOHOLS WITH SODIUM BOROHYDRIDE-TRIFLUOROACETIC ACID. PREPARATION OF bis-HETEROCYCLIC METHANES | Charles F. Nutaitis; Richard Patragnoni; Greg Goodkin; Beth Neighbour; Judy Obaza-Nutaitis |
| 413-418 | SYNTHESIS OF THIENO[3,2-e]-1,2,4-TRIAZOLO[a]PYRIMIDINES | S. Tumkevicius; J. Mickiene |
| 419-424 | THE BROMINATION OF 2,5-DIMETHOXYBENZALDEHYDE. STRUCTURAL PROOF OF THE 6-BROMO ISOMER via 3,6-DIMETHOXYBENZOCYCLOBUTENE | Manik S. Sardessai; Hanley N. Abramson |
| 425-427 | 2,4-DI-t-BUTYLBROMOBENZENE BY SILVER ION-ASSISTED BROMINATION OF 1,3-DI-t-BUTYLBENZENE | Albeit J. Fry; Shastra Solomon |
| 427-431 | REDUCTION CLEAVAGE OF AROMATIC CYCLIC ACETALS WITH ZIRCONIUM CHLORIDE-LITHIUM ALUMINUM HYDRIDE | Wu Shaozu; Ren Tianhui; Chen Ning; Zhang Yulan |
| 432-434 | SYNTHESIS OF cis-Δ6-OCTALIN-1,4-DIONE bis-ACETALS | Stan V. D'Andrea; Jeremiah P. Freeman; Jacob Szmuszkovicz |
| 435-438 | PREPARATION OF N-UNSUBSTITUTED THIOAMIDES BY A MODIFIED WILLGERODT-KINDLER REACTION | Qi-Dong You; Hou-Yuan Zhou; Qi-Zhou Wang; Xing-Han Lei |
| 438-441 | SOLVENT EFFECT ON THE GOMBERG-BACHMANN-HEY ARYLAPON OF PYRIDINE | Marek Gurczynski; Piotr Tomasik |
| 441-442 | IMPROVED SYNTHESIS OF 2,4-HEXADIENOIC ACID | Péter Vinczer; Lajos Novák; Csaba Szántay |
| 443-447 | APPLICATION OF POTASSIUM t-BUTOXIDE IN TOLUENE AS A BASE IN THE WITTIG REACTION IN LARGE-SCALE PHEROMONE SYNTHESES | Péter Vinczer; Lajos Novák; Csaba Szántay |
| 447-450 | A CONVENIENT SYNTHESIS OF 2,5-DIAMINO-1,4-BENZENEDIOL | Muthiah Inbasekaran; Robert Strom |
| 450-455 | REACTION OF 4-[BIS(ALKYLTHIO)METHYLENE]-2-PHENYL-2-OXAZOLIN-5-ONES WITH AMBIDENT NUCLEOPHILES | Jalpana Roy; N. S. Rawat |
| 455-457 | A RAPID PREPARATION OF 2,2′-DIMERCAPTOBIPHENYL | Sergio Cossu; Giovanna Delogu; Davide Fabbri; Paola Maglioli |
| 458-459 | PREPARATION OF TETRAETHYL (OXYDI-2,1-ETHANEDIYL)BISPHOSPHONATE AND 1,2-BIS[2-(DIETHYLPHOSPHONO)ETHOXY]ETHANE | Balram Dhawan; Derek Redmore |
| 460-463 | SYNTHESIS OF A HEXAALKYNYLHEXAPHENYLBENZENE | John A. Hyatt |
| 465-543 | TAXANE DITERPENE SYNTHESIS STRATEGIES. A REVIEW | Charles S. Swindell |
| 545-568 | RECENT DEVELOPMENTS IN THE AREA OF ANNDLATED FURANS. A REVIEW | Albert Padwa; S. Shaun Murphree |
| 569 | CORRIGENDA | |
| C | Editorial Board Page | |
| 133-138 | AN EFFICIENT SYNTHESIS OF α-ASARONE | Francisco Díaz; Leticia Contreras; Rosa Flores; Joaquín Tamariz; Fernando Labarrios; Germán Chamorro; Héber Muñoz |
| 139-146 | β-KETONITROSAMINES AS SYNTHETIC EQUIVALENTS OF α-METHYLENE ALKANOLAMINO ANIONS | Joseph E. Saavedra; David W. Famsworth |
| 147-151 | PREPARATION AND SOME SIMPLE REACTIONS OF 1-SUBSTITUTED IMIDAZOLE-2,4,5-TRIONES | Behzat Altural; Yunus Akcamur; Gert Kollenz |
| 153-156 | ALKYLATION OF PHENYLACETONITRILE USING POTASSIUM CARBONATE AS A BASE | Chengzhi Xu; Xiangjun Mao; Hongbo Shen; Wenquiang Chen |
| 157-162 | A FACILE ONE POT SYNTHESIS OF 3-SUBSTITUTED-1,2,4-TRIAZOLO[4,3-B][4,1,2]BENZOTHIADIAZINE-8-ONES | B. Radha Rani; M. F. Rahman; U. T. Bhalerao |
| 163-172 | AN IMPROVED SYNTHESIS OF NAPHTHO[2,3-d]-1,3-DIOXOLE-5-METHOXY-6-CARBOXYLIC ACID | Jordan Zjawiony; John R. Peterson |
| 173-180 | AN EFFICIENT LARGE SCALE PREPARATION OF (S)-1,1,2-TRIPHENYLETHANEDIOL 2-ACETATE | A. Millar; L. W. Mulder; K. E. Mennen; C. W. Palmer |
| 181-185 | SYNTHESIS OF bis-ISOXAZOLYLNAPHTHOQUINONES | C. S. Ortiz; M. R. Longhi; M. M. De Bertorello; M. C. Briñon |
| 186-188 | SYNTHESIS AND THERMOLYSIS OF CYCLOALKENYL AZIDES. A SIMPLE ROUTE TO POLYCYCLIC ISOXAZOLES | Md. Izhar Sami; Gandhi K. Kar; Jayanta K. Ray |
| 188-190 | AN IMPROVED SYNTHESIS OF 5-METHYLPYRAZINE-2-CARBOXYLIC ACID | I. Iovel; Yu. Goldberg; M. Shymanska |
| 191-192 | OPTIMAL CONDITIONS FOR ACETYLATION OF AROMATIC TERTIARY ALCOHOLS | L. Sipos; M. Zsuga; T. Kelen |
| 193-195 | A CONVENIENT PREPARATION OF trans-3,4-DIPHENYLAND trans, trans-2,3,4-TRIPHENYLVALEROLACTONES | Jean A. Stanley; Susan Dakin; Linda Szabo; Leila Posaw; Christine Lee; Wen Min Hou |
| 196-197 | FACILE SYNTHESIS OF HOMOTRIPTYCENES via ADDITION OF BENZOCYCLOPROPENE AND ANTHRACENES | Katsuhiro Saito; Kazuaki Ito; Kensuke Takahashi; Shinzo Kagabu |
| 198-200 | A NOVEL SYNTHESIS OF SOME ARYLTHIOGLYCOLIC ACIDS | Y. Yildirir; G. Okay |
| 200-203 | AN OPTIMIZED SYNTHESIS OF DIMETHYL 2,2′-DIHYDROXY-1,1′-BINAPHTHALENE-3,3′-DICARBOXYLATE AND OF METHYL 2,2-DIHYDROXY-1,1′-BINAPHTHALENE-3-CARBOXYLATE | Martin Hovorka; Jirí Závada |
| 204-206 | EXPEDITIOUS ROUTES TO SYMMETRICALLY AND ASYMMETRICALLY SUBSTITUTED PYRIDINES FROM CHELIDAMIC ACID | Paolo Scrimin; Paolo Tecilla; Umberto Tonellato |
| C | Editorial Board Page | |
| 547-574 | REARRANGEMENTS OF EPOXY ALCOHOLS AND RELATED COMPOUNDS. A REVIEW | Göran Magnusson |
| 575-578 | DIRECT ALKYLATION OF NITROARENES via VICARIOUS NUCLEOPHLIC SUBSTITUTION OF HYDROGEN | Zbigniew Wrobel; Mieczyslaw Makosza |
| 579-588 | SYNTHESIS OF 2-CHLORO-3-ALKYL- AND ARYLQUINOLINES | Ferenc Korodi; Zoltan Cziaky |
| 589-595 | SYNTHESIS OF α-CHLORO-α,β-UNSATURATED ALDIMINES AND OF α-CHLORO-α,β-UNSATURATED ALDEHYDES | Christian Stevens; Norbert De Kimpe |
| 597-603 | THE PREPARATION OF Nα-t-BOC-2,3-DIAMINOPROPIONIC ACID (DPR) AND OF Nα-t-BOC-2,4-DIAMINOBUTYRIC ACID (DBR) DERIVATIVES SUITABLE FOR SOLID PHASE PEPTIDE SYNTHESIS | C. Freeman Stanfield; Arthur M. Felix; Waleed Danho |
| 605-611 | CONVENIENT C-3 OXIDATION OF DEOXY AND AMINODEOXY SUGARS | Mária Mádi-Puskas; Pál László; István F. Pelyvás; Ferenc Sztaricskai |
| 613-618 | A SIMPLE AND CONVENIENT SYNTHESIS OF 5-SUBSTITUTED BENZOXAZOLES | Kenneth R. Kunz; Ethan Will Taylor; Harold M. Hutton; Barry J. Blackburn |
| 619-622 | CONVENIENT PREPARATION OF METABOLITES OF 6-n-PROPYLTHIOURACIL | F. S. Guziec Jr.; Lynn James Sanfilippo; Loide Mayer Wasmund |
| 623-626 | A FACILE SYNTHESIS OF 5-DEOXY-D-RIBONIC ACID LACTONE AND OF 5-DEOXY-D-RIBOSE | G. M. Escandar; L. F. Sala |
| 627-629 | A SYNTHESIS OF (±)-3-ACETOXY-2,6-DIMETHYL-1,5-HEPTADIENE, THE SEX PHEROMONE OF THE COMSTOCK MEALYBUG | Suk-Ku Kang; Choong-Sil Park |
| 630-632 | IMPROVED METHOD FOR BISALLYLATION OF cis-BICYCLO [3.3.0]OCTANE-3,7-DIONE via THE CLAISEN REARRANGEMENT | K. Sambasivarao; J. M. Cook |
| 632-636 | BIOMIMETIC MODELING OF ASYMMETRIC SYNTHESIS OF ARYLALKYL SULFOXIDES USING β-CYCLODEXTRIN COMPLEXES | K. Rama Rao; H. M. Sumpath Kumar; N. Bhanumathi; P. B. Sattur |
| 636-638 | DIMETHYL 4-NITROPHENYLMALONATE | M. A. E. Bowman; R. E. Bowman |
| 639-641 | AN IMPROVED SYNTHESIS OF 3-NITROFLUORENE | J. R. Moran; G. Emmett |
| 641-643 | AN IMPROVED SYNTHESIS OF 4′,5′-DIAMINOBENZO-15-CROWN-5 | Yasar Gök |
| 643-645 | PREPARATION OF AN o-SUBSTITUTED BENZAMIDINE BY THE PINNER METHOD. A LITERATURE CLARIFICATION | C. C. Cheng |
| 645-648 | AN IMPROVED SYNTHESIS OF 4,8,9,10-TETRAARYL-1,3-DIAZAADAMANTANES | S. Sivasubramanian; M. Sundaravadivelu; N. Arumugam |
| 648-650 | AN IMPROVED OZONOLYTIC APPROACH TO 6-OXOHEPTANAL | M. R. Karim; P. Sampson |
| 651-654 | A CONVENIENT PREPARATION OF (+)-5(S)-METHYL-2(5H)-FURANONE. SYNTHESIS OF (S)-(+)-SULCATOL | Suk-Ku Kang; Dong-Ha Lee; Sung-Gyu Kim |
| C | Editorial Board Page | |
| 399-484 | SYNTHESIS OF α-AMINOALDEHYDES AND α-AMINOKETONES. A REVIEW | Lawrence E. Fisher; Joseph M. Muchowski |
| 485-493 | IMPROVED PROCEDURES FOR THE PREPARATION OF BENZO[c]CINNOLINE, ITS N-OXIDE AND SOME BROMO DERIVATIVES AND SYNTHESIS OF PYRROLIDINO, PIPERIDINO, AND MORPHOLINOBENZO[c]CINNOLINES | Emine Kilic; Celal Tüzün |
| 495-500 | IMPROVED SYNTHESIS OF 1,2-DIMETHOXY-3-ISOPROPYLBENZENE AND GENERAL SYNTHESIS OF 3-SUBSTITUTED-1,2-DIMETHOXYBENZENES | Lorraine M. Deck; Eugenia M. Brazwell; David L. Vander Jagt; Robert E. Royer |
| 501-506 | IMPROVEMENTS IN THE SEMMLER-WOLF REARRANGEMENT OF 19-NORTESTOSTERONE OXIME | William B. Smith; Milind P. Sant |
| 507-511 | A NOVEL METHOD FOR HANDLING ORGANIC REACTIONS IN A BOMB TUBE | G. Csanády; G. Knapp |
| 511-514 | AN IMPROVED SYNTHESIS OF ALKYL 1-ALKYL-3-METHYL-2-PYRAZOLINE-5-ONE-4-DITHIOCARBOXYLATES | Alfonso Oliva; Gerardo Léon; René Maurelia |
| 514-518 | A SIMPLE ROUTE TO SOME SPIROIMIDAZOLONES | C. del Campo; E. F. Llama |
| 519-521 | SYNTHESIS OF 4,4-bis(2-METHOXYETHYL)CYCLOHEXANONE AND OF 4,4-bis(2-METHOXYETHYL)-2-CYCLOHEXEN-1-ONE | Elaine N. Cheeseman |
| 522-525 | EFFECTIVE AND PREFERENTIAL TRANSFORMATION OF COMPOUNDS HAVING 2-HALOETHYL GROUPS ON POSITIVE SULFUR INTO ETHENYL COMPOUNDS UNDER PTC CONDITIONS | Y. Shimizugawa; T. Takahashi; M. Ishii; T. Yamamoto |
| 526-528 | A FACILE SYNTHESIS OF NATURAL MHPG, A METABOLITE OF NOREPINEPHRINE | M. Adamczyk; Y. Y. Chen; J. F. Fishpaugh |
| 528-531 | ULTRASOUND-PROMOTED SODIUM BOROHYDRIDE REDUCTION OF PENTACYCLO[5.4.0.02,6.03.10.05,9]UNDECANE-8,11-DIONE (PCUD-8,11-DIONE) AND OF 4,4-DIMETHOXY-2,3,5,6-TETRACHLORO-PCUD-8,11-DIONE | Alan P. Marchand; G. Madhusudhan Reddy |
| 532-534 | AN IMPROVED SYNTHESIS OF DIMETHYL DIACETOXYFUMARATE AND ITS CONDENSATION WITH HETEROCYCLIC AMINES | M. Tisler; R. Zupet |
| 534-537 | DEOXYGENATION OF EPOXIDES WITH ALUMINUM | Peter W. D. Mitchell |
| 538-540 | ARYL HYDROGEN PHTHALATES | P. C. Crofts; M. Ghahhary; M. Tajbakhsh-Jadidi |
| 540-543 | IMPROVED PREPARATION OF DI-O-ISOPROPYLIDENE-1,2;5,6-D-MANNITOL | C. Morpain; B. Nasser; B. Laude; N. Latruffe |
| 544-546 | PREPARATION OF 4-THIAZOLIDINONE-1-OXIDES | J. B. Lee; S. Y. Yergatian; B. C. Crowther; I. M. Downie |
| C | Editorial Board Page | |
| 131-165 | DIELS-ALDER REACTIONS OF CYCLOALKENONES IN ORGANIC SYNTHESIS | Francesco Fringuelli; Aldo Taticchi; Ernest Wenkert |
| 167-201 | CARBON-CARBON BOND CLEAVAGE BY THE HALLER-BAUER AND RELATED REACTIONS A REVIEW | John P. Gilday; Leo A. Paquette |
| 203-208 | ASYMMETRIC SYNTHESIS OF 2-,3-, AND 4-METHYLOCTANOIC ACIDS | Philip E. Sonnet; Joseph Gazzillo |
| 209-213 | A ONE-POT PROCEDURE FOR THE PREPARATION OF PHOSPHONIC ACIDS FROM ALKYL HALIDES | Alan R. Katritzky; Boguslaw Pilarski; Jack W. Johnson |
| 215-227 | SYNTHESIS AND REACTIONS OF β-SILYLOXYACYLCYCLOPROPANES TRIMETHYLSILYL HALIDE-ZINC HALIDE INDUCED CYCLOPROPYLCARBINYL REARRANGEMENT | A. M. Moiseenkov; B. A. Czeskis; N. M. Ivanova; O. M. Nefedov |
| 229-233 | 2,10-DICHLORO-6-(SUBSTITUTED ARYLOXY)DIBENZO[d,g][1,3,6,2]DIOXATHIA-PHOSPHOCIN 6-OXIDES. SYNTHESIS AND SPECTRAL CHARACTERISTICS | C. Devendranath Reddy; K. Anuradha; K. Darrell Berlin; Prasanna S. Sunthankar; Satish V. Mulekar |
| 235-244 | SYNTHESIS OF SOME 3,4-DIHYDRO-2H-1-BENZOTHIOPYRAN-4-OLS | Vicki L. Pruitt; K. Darrell Berlin; Kenneth S. Hirsch |
| 245-253 | AN EFFICIENT SYNTHESIS OF 2′,3′-DIDEOXYADENOSINE via THE COREY-WINTER REACTION | Russell L. K. Carr; Thomas A. Donovan Jr.; Mahendra N. Sharma; C. Daniel Vizine; Michael J. Wovkulich |
| 255-264 | THE PREPARATION OF AMIDE DERIVATIVES OF 3-AZABICYCLO-[3.3.1]NONANES AS NEW POTENTIAL ANTIARRHYTHMIC AGENTS | Stan A. Zisman; K. Darrell Berlin; B. J. Scherlag |
| 265-268 | SYNTHESIS OF 2′,3′-DIDEOXY-5-METHYLCYTIDIN-2-ENE, A CYTIDINE ANALOG OF 3′-DEOXYTHYMIDIN-2′-ENE (d4T) | Tai-Shun Lin; Jing-Hua Yang |
| C | Editorial Board Page | |
| 1-36 | RECENT ADVANCES IN THE USE OF ACYLIUM SALTS IN ORGANIC SYNTHESIS. A BRIEF REVIEW | Mahmoud Al-Talib; Hasan Tashtoush |
| 37-45 | SYNTHESIS OF 1,4-DIMETHOXYBENZ[a]ANTHRACENES AND OF 7,10-DIMETHOXYCHOLANTHRENES | Melvin S. Newman; A. R. Choudhary; A. Kumar |
| 47-55 | SYNTHESIS OF MANNICH COMPOUNDS FROM FLAVANONES | György Litkei; Tamás Patonay; Jenó Kardos |
| 57-61 | REGIOSPECIFIC 5′-SILYLATION OF NUCLEOSIDES | Vasu Nair; Greg S. Buenger |
| 63-70 | AN INEXPENSIVE AND CONVENIENT PREPARATION OF METHOXYMETHYL AND PHENYLTHIOMETHYL ETHERS | R. Karl Dieter; Ravindra Datar |
| 71-76 | A CONVENIENT SYNTHESIS OF N-[2-[[[5-[(DIMETHYLAMINO)METHYL]-2-FURANYLMETHYL]THIO]ETHYL]THIENO-[3,4-d]ISOTHIAZOL-3-AMINE-1,1-DIOXIDE HYDROCHLORIDE, A POTENT GASTRIC ACID ANTISECRETORY AGENT | Arthur A. Santilli; Robert L. Morris; Anthony C. Scotese; Donald P. Strike |
| 77-84 | COMPETITIVE BIMOLECULAR REDUCTION IN THE SYNTHESIS OF KETONES MICHAEL ADDITION OF GRIGNARD REAGENTS TO α-ENONES | C. Alvarez-Ibarra; M. S. Arias-Pérez; E. Moya; M. A. Rodríguez-Barranco |
| 85-87 | A NEW ROUTE TO NITRO-AND BENZOYLPHTHALIDES | Wenjeng Guo; Y. F. Duann |
| 87-94 | SYNTHESIS OF 3-QUINUCLIDINYL BENZILATE DERIVATIVES | G. W. Kabalka; S. B. Mathur; Y. -Z. Gai |
| 94-97 | AN EFFICIENT SYNTHESIS OF α,β-UNSATURATED CARBOXYLIC ACIDS AND NITRILES | Chang Kiu Lee; Jeung Yeop Shim |
| 97-99 | SYNTHESIS OF N-DESMETHYL MESORIDAZINE | T. Mohammad; E. M. Hawes; K. K. Midha |
| 99-102 | MONOMETHYLATION OF 3,4-DIHYDROXYBENZALDEHYDE AS AN ALTERNATE ROUTE TO ISOVANILLIN | Andre Loupy; Mustapha Majdoub |
| 102-104 | A CONVENIENT SYNTHESIS OF 2,3-DIBROMOANTHRACENE | Murthy R. Akula |
| 104-105 | THE PREPARATION OF 5-CHLORO-2-INDOLINONE BY DIRECT CHLORINATION OF 2-INDOLINONE | Paul Pranc |
| 106-108 | BENZIMIDAZOLE ANTIVIRALS. REGIOSPECIFIC SYNTHESIS OF ARYL BENZIMIDAZOYL KETONES BY SULFONAMIDE ANION DISPLACEMENT OF AROMATIC FLUORIDE | Samuel J. Dominianni |
| 109-111 | 2,2-DIMETHYL-6-[(TRIPHENYLPHOSPHORANYLIDENE)METHYL]-4H-1,3-DIOXIN-4-ONE. A FOUR-CARBON HOMOLOGATING AGENT REQUIRING NO ACTIVATION | Christina Bodurow; Michael A. Carr; Larry L. Moore |
| 112-113 | A CONVENIENT ONE-POT SYNTHESIS OF 2-METHYL-2-BENZYLTHIOPROPANAL | Gerald S. Jones Jr.; David R. Elmaleh |
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| 521-618 | SYNTHESIS OF QUASSINOIDS. A REVIEW | Kenji Kawada; Moonsun Kim; David S. Watt |
| 619-627 | SYNTHESIS OF CHROMOPHORIC ANALOGS OF ACETYLCHOLINE HALIDES | Leroy H. Klemm; Warner L. Peticolas; Kori L. Clement; K. Jeffry Wilson |
| 629-632 | A FACILE PREPARATION OF 2(Z), 5(Z), 8(Z)-TETRADECATRIEN-1-OL, A KEY INTERMEDIATE FOR EICOSANOID SYNTHESIS | Domenico Badone; Roberto Pagliarin; Massimo Sisti; Paolo Tavecchia |
| 633-641 | PREPARATION OF AZULENE DERIVATIVES: AN AMINOACID, DICARBOXYLATES, AN ISOTHIOCYANATE, AND RELATED COMPOUNDS | LeRoy H. Klem; Bruce S. Hudson; Jennifer J. Lu |
| 643-645 | AN IMPROVED SYNTHESIS OF 1-(4-NITROBENZYL)-1.2-ETHYLENEDIAMINE, PRECURSOR OF THE CORRESPONDING ETHYLENEDIAMINETETRAACETIC ACID | Rene C. Gaudreault; Antoine A. Noujaim |
| 645-648 | SYNTHESIS OF 2-HEXYLNAPHTHALENE | B. Dewprashad; E. J. Eisenbraun |
| 649-652 | THE 2- AND 4-NITRO AND 2- AND 4-ACETAMIDO 5,6,7,8,9,10-HEXAHYDRO DERIVATIVES OF CYCLOHEPTA[b]INDOLE | Arthur G. Anderson Jr.; Harry F. Richards; Ralph D. Haddock |
| 653-655 | 2,3,4,5,6,7-HEXAHYDROCYCLOPENTA-1,4-THIAZINE AND THE 8,9-DIHYDRO-, 4-ACETYL AND l-OXO - 4-ACETYL DERIVATIVES | Arthur G. Anderson Jr.; Russell A. Labar; Ralph D. Haddock |
| 655-656 | A FACILE REDUCTION OF 1,8-NAPHTHALIMIDE TO 1,2,3,4-TETRAHYDRO-1,8-NAPHTHALIMIDE | Michael D. Crenshaw; C. C. Cheng |
| 657 | CORRIGENDUM | |
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| 257-296 | USE OF SUBSTITUTED 3-SULFOLENES AS PRECURSORS FOR 1,3-BUTADIENES | Ta-Shue Chou; Hsi-Hwa Tso |
| 297-301 | CYCLZATION OF ω-HALONITRILES WITH ORGANOLITHIUMS | Vincent Gallulo; Liberty Dimas; Charles A. Zezza; Michael B. Smith |
| 303-308 | SYNTHESIS OF TWO PHOTOLABILE BENZYL MANGANESE DERIVATIVES INCORPORATING A GEOMETRICALLY INACCESSIBLE RADICAL TRAP | John F. W. Keana; Sovitj Pou |
| 309-314 | SYNTHESIS OF (±)-NOROORALYDINE AND (±)-TETRAHYDROPALMATINE | Kazuhiko Orito; Tsutomu Matsuzaki; Hiroshi Suginome |
| 315-319 | A SIMPLIFIED PROCEDURE FOR PREPARING THE CHOLINERGIC NEUROTOXIN 1-ETHYL-1-(2-EYDROXYETHYL)AZIRIDINIUM ION (AF64A) | Walter H. Moos; Robert E. Davis; Roy D. Schwarz |
| 321-326 | ACYLATION OF 1,2,4,5-TETRAHYDRO-3-MEIHYL-3H-3-BENZAZEPIN-2-ONE IN THE PRESENCE OF SODIUM HYDRIDE | Kazuhiko Orito; Harumi Kaga; Hiroshi Suginome |
| 327-335 | SYNTHESIS OF 2,6-DIARYLTETRAHYDROPYRAN-4-ONES | Timothy M. Fakler; K. Darrell Berlin |
| 337-339 | SYNTHESIS OF 1,3-bis(2-BROMOPHENYL)PROPANE | Richard A. Bunce; Vicki L. Taylor; Henry D. Reeves |
| 340-341 | A PRACTICAL SYNTHETIC METHOD FOR N-METHYL-o-TOLUIDINE | Alan R. Katritzky; Kunihiko Akutagawa |
| 341-343 | 4-(2-ARYLALKENYL)-3-CYANO-2H-1-BENZOPYRAN-2-ONES | Y. Anghelova; E. Dimitrova |
| 344-346 | AN IMPROVED SYNTHESIS OF 5-HYDROXYPENTANAL | Peter Vinczer; Zoltan Juvancz; Lajos Novak; Csaba Szantay |
| 346-348 | A SIMPLE SYNTHESIS OF (+)-trans-VERBENYL PROPIONATE, A PHEROMONE ANALOG OF AMERICAN COCKROACH USING LEAD(IV) PROPIONATE | Peter Vinczer; Maria Kajtar-Peredy; Zoltan Juvancz; Lajos Novak; Csaba Szantay |
| 348-351 | SYNTHESIS OF (2-BUTYL-3-BENZOFURANYL)[4-[2-(DIETHYLAMINO)ETHOXY]-3,5-DIIODOPHENYL)METHANE DERIVATIVES | George W. Kabalka; Thomas P. Kennedy; Naganna M. Goudgaod; Rajender S. Varma |
| 351-353 | L-DOPA-3-0-SULFATE BY THE PERSULFATE OXIDATION OF L-TYROSINE | E. J. Behrman; J. M. Bidinger |
| 354-355 | A FACILE SYNTHESIS OF DIARYLACETONITRILE FROM DIARYKETONES AND TRIMETHYLSILYL CYANIDE | Katsuhiro Saito; Shinzo Kagabu; Yoichi Horie; Kensuke Takahashi |
| 355-358 | AN IMPROVED PROCEDURE FOR THE DICHLOROACETYLATION OF PRIMARY AND SECONDARY AMINES | Braja G. Hazra; V. S. Pore; S. P. Maybhate |
| 359-360 | THE LITHIATION OF 1,4-DIMETHOXYNAPHTHALENE AND CARBOXYLATION OF THE PRODUCTS | Melvin S. Newman; Anil R. Choudhary |
| 360-363 | AN EFFICIENT PREPARATION OF 1,2-DIHYDROCYCLOBUTA[a]NAPHTHALENE | David A. Hunt |
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| 129-133 | SYNTHESIS OF BRANCHED LONG CHAIN ALIPHATIC PRIMARY ALKYL BROMIDES | Alan R. Katritzky; Adam Bieniek; Long Chiang |
| 135-139 | THE PREPARATION OF 1-(α-AMINOALKYL) - BENZOTRIAZOLES IN AQUEOUS SOLUTION | Alan R. Katritzky; Boguslaw Pilarski; Laszlo Urogdi |
| 141-146 | A SIMPLE PREPARATION OF 2-UNSUBSTITUTED 4-AMINOOXAZOLES | Ram Lakhan; Ram Lakhan Singh |
| 147-156 | REGIOSELECTTVE SYNIHESIS OF CHOLESTANE-3β,5α,6α-TRIOL-7-ONE 3-ACETATE AND EIGHT STEREOISOMERIC CHOLESTANE-3β,4,5α,6 AND OF 3β,5α,6,7-TETROL TRIACETATES | James Warren; Stephen O'brien; Harold R. Nace |
| 157-162 | CONVENIENT LARGE SCALE PREPARATION OF 5-METHYL- AND 4-NITRO- 2-IODOSOBENZOIC AND OF 4-NITRO-2-IODOXYBENZOIC ACIDS | Alan R. Katritzky; G. Paul Savage; John K. Gallos; H. Dupont Durst |
| 163-171 | SYNTHESIS OF NOVEL 1,2,4-TRIAZOLOQUINAZOLINE RING SYSTEMS | József Reiter; László Pongo |
| 173-178 | SYNTHESIS OF ANALOGS OF PROPRANOLOL HYDROCHLORIDE | James S. Farina; Steven A. Jackson; Corbin L. Cummings |
| 179-217 | RECENT PROGRESS IN TEE CONTROL OF CARBON VERSUS OXYGEN ACYLATION OF ENOLATE ANIONS | T. Howard Black |
| 219-221 | A SHORT SYNTHESIS OF cis-1,7,7-TRIMETHYLBICYCLO[4.4.0]DEC-3-ENE | William A. Donaldson; Joseph W. Strohbach |
| 221-223 | A FACILE SYNTHESIS OF 3,4-DIHYDRO-1,5-BENZODIOXEPIN-2-ONES | M. S. Reddy; G. L. D. Krupadanam; G. Srimannarayana |
| 223-225 | A SIMPLE PREPARATION OF 1-HYDROXYPYRENE | Raj K. Sehgal; Subodh Kumar |
| 225-228 | AN IMPROVED SYNTHESIS OF (1R, 2R)-(-)-a-(1-ISOPROPYLAMINOETHYL)BENZYL ALCOHOL | Duy H. Hua; Roch Chan-yu-King; Robert A. Ostrander; Jeffrey A. McKie |
| 228-230 | A FACILE SYNTHESIS OF BENZYL ISOTHIOCYANATES BY USE OF 18-CROWN-6 ETHER | S. Muthusamy; V. T. Ramakrishnan |
| 230-232 | A NEW METHOD FOR THE CONVERSION OF ALDOXIMES INTO NITRILES WITH ZEOLITES | M. Narayana Rao; Pradeep Kumar; Kamini Garyali |
| 232-237 | SIMPLE SYNTHESIS OF ALKYNES FROM 1,2-DIBROMOALKANES USING PTC CONDITIONS | Peter Vinczer; Terez Kovacd; Lajos Novak; Csaba Szantay |
| 237-240 | REDUCTION OF 1,3,5-TRISUBSTITUTED 2-ALKYLPYRAZOLIUM SALTS WITH COMPLEX METAL HYDRIDES. SYNTHESIS OF 3-PYRAZOLINES | Angel Alberola; Luis A. Banuelos; Purification Cuadrado; Ana Ma Gonzalez; Fco. Jose Pulido |
| 241-242 | A SIMPLE ONE-STEP SYNTHESIS OF 5-ACETOXY-6-CHLORO-2-HEXANONE | Naresh K. Sangwan; Kuldip Singh Dhindsa |
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| 199-204 | A SHORT SYNTHESIS OF (±)-α-CHAMIGRENE | Emil R. Koft; Thomas A. Broadbent |
| 205-211 | PREPARATION OF STYRYL BENZYLSULFONES AND 1, 2-BIS (STYRYLSULFONYLMETHYL)-4, 5-DIMETHYLBENZENES | D. Bhaskar Reddy; N. S. Reddy; S. Reddy; H. V. R. Reddy; S. Balasubramanyan |
| 213-222 | SYNTHESIS OF ACENAPHTHO[1, 2-b]BENZO[d]THIOPHENE | Gandhi K. Kar; Basanta G. Chatterjee; Jayanta K. Ray |
| 223-230 | THE SYNTHESIS OF PEROPYRENE-TYPE POLYCYCLIC AROMATIC HYDROCARBONS | J. C. Fetzer; W. R. Biggs |
| 231-236 | 4-PHENYL-Δ3-DIHYDROPYRANS BY REDUCTION OF PYRILIUM SALTS WITH SODIUM BOROHYDRIDE IN ACETIC ACID | Teodor-Silviu Balaban; Alexandru T. Balaban |
| 237-243 | SYNTHESIS OF ALKYL INDOLIZINES FROM PYRYLIUM SALTS | Antonie Dinculescu; Teodor-Silviu Balaban; Alexandru T. Balaban |
| 245-252 | SYNTHESIS OF 4-HYDROXY-4-(2-THIENYL)PENTAMIDE | R. Cruz-Almanza; F. García; B. Ramírez; M. Ordoñez |
| 253-260 | SYNTHESIS OF THE ANTIHYPERTENSIVE AGENT 1-(1-METHYLETHYL)-2-(2-[4-(3-TRIFLUOROMETHYLPHENYL)-1-PIPERAZINYL]ETHYL)-1H-NAPHTH[1, 2-d] IMIDAZOLE CITRATE | E. Toja; A. Trani |
| 261-269 | APPROACH TO THE SYNTHESIS OF AN OPTICALLY ACTIVE POLYNUCLEOTIDE ANALOG | Ming-Jye Lan; C. G. Overberger |
| 271-274 | S, S-DIARYL- AND S-(2-SUBSTITUTED ETHYL)-S-PHENYL-N-TOSYLSULFILIMINES FROM CHLORAMINE T UNDER PTC CONDITIONS | Tamotsu Yamamoto; Daisaburo Yoshida |
| 275-279 | A SIMPLE PREPARATION OF 1-ALKOXY-1-ALKYN-3-OLS | Wayne M. Stalick |
| 279-284 | “ONE POT” FISCHER SYNTHESIS OF (2, 3, 3-TRIMETHYL-3-H-INDOL-5-YL)-ACETIC ACID. DERIVATIVES AS INTERMEDIATES FOR FLUORESCENT BIOLABELS | Philip L. Southwick; Jennifer G. Cairns; Lauren A. Ernst; Alan S. Waggoner |
| 285-289 | SYNTHESIS OF 3- AND 4-CHLORO-1H-PYRROLO[3, 2-c]PYRIDIN-4(5H)-ONE | G. Cristalli; P. Franchetti; M. Grifantini; E. Nasini; S. Vittori |
| 289-292 | PREPARATION OF 2, 6-DIMETHYL-4-PHENYLPYRYLIUM SULFOACETATE | T. S. Balaban; A. Dinculescu; A. T. Balaban |
| 293-295 | LARGE SCALE PREPARATION OF 1, 3-DIMETHYLADAMANTANE | Thomas J. Dooley; William Rowe |
| 295-298 | A CONVENIENT SYNTHESIS OF 10, 10′-DIMETHYL-9, 9′-BIACRIDYLIDENE | Marion R. Surgi; Julian Tirado-Rives |
| 299-302 | AN IMPROVED SYNTHESIS OF ETHYL 4-HYDROXY-3-METHYLBENZOFURAN-2-CARBOXYLATE | P. C. Bélanger; C. Dufresne; C. K. Lau; J. Scheigetz |
| 302-305 | IODIDE SALTS OF NITROGEN HETEROCYCLES BY BROMIDE-IODIDE EXCHANGE | In-Sook Han Lee; Chang Kiu Lee; In Sup Han |
| 305-311 | SYNTHESIS OF 3-METHYL- AND 3-tert-BUTYLPHENANTHRENE | R. C. Bansal; S. A. Samad; J. S. Thomson; E. J. Eisenbraun |
| 311-316 | SYNTHESIS OF 2-[4-METHOXY-2-[2-(METHYLSULFINYL)ETHOXY]PHENYL]-1H-IMIDAZO[4, 5-b]PYRIDINE, A POTENT NONGLYCOSIDE INHIBITOR OF Na+, K+-ATPASE | David W. Robertson; Joseph H. Krushinski |
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| 83-159 | RECENT SYNTHETIC APPLICATIONS OF N-NITROSAMINES AND RELATED COMPOUNDS | Joseph E. Saavedra |
| 161-166 | FORMATE ESTERS BY CANNIZZARO-TISHCHENKO REACTION OF GRIGNARD AND SODIUM ALKOXIDES WITH FORMALDEHYDE | Richard A. Bunce; A. Joe Shellhammer Jr. |
| 167-172 | A NEW AND CONVENIENT SYNTHESIS OF 4-AMINO-3-NITROBENZOPHENONE AND 2-AMINO-5-NITROBENZOPHENONE AND THEIR N-ALKYL DERIVATIVES | N. R. Ayyangar; R. J. Lahoti; K. V. Srinivasan; Thomas Daniel |
| 173-180 | REGIOSELECTIVE DEOXYGENATION OF CHLORAMPHENICOL AND OF (1R,2R)-(+)-2-AMINO-1-PHENYL-1,3-PROPANEDIOL | P. Ramaiah; A. S. Rao |
| 181-186 | SYNTHESIS OF DIIMINES FROM 1,2-DICARBONYL COMPOUNDS BY DIRECT CATALYZED CONDENSATION | D. Armesto; P. Bosch; M. G. Gallego; J. F. Martin; M. J. Ortiz; R. Perez-Ossorio; A. Ramos |
| 187-195 | PREPARATION OF THE 9-cis, 13-cos-. AND ALL trans-ISOMERS OF α- AND β2-RETINAL | Michael F. Vaezi; Cynthia Y. Robinson; Kenneth D. Hope; Wayne J. Brouillette; Donald D. Muccio |
| 197-208 | SYNTHESIS OF BIOLOGICAL MARKERS IN FOSSIL FUELS 5. A SYNTHESIS OF 5α-CHOLAN-24-OIC ACID | Ayhan S. Demir; Mark R. Sabol; Alwarsamy Jeganathan; Eric Kurt Dolence; David S. Watt; J. Michael Moldowan |
| 209-214 | A CONVENIENT SYNTHESIS OF (dl)-1-AMINO-4-CARBOXYCYCLOHEXANE-1-13C-CARBOXYLIC ACID | N. Dale Ledford; Cathy R. Cutcliff; H. Blair Wood Jr.; Michael Barfield |
| 215-248 | RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF TETRAZINES. A BRIEF REVIEW | Michael J. Hearn; Fiona Levy |
| 249-250 | A SIMPLE PREPARATION OF 6-CHLORO-5, 8-QUINOLINEDIONE | Arthur Haber |
| 251-252 | ONE-STEP PREPARATION OF 4-BROMOMETHYL-2,3,5,6-TETRABROMOPHENOL | Wenjeng Guo; George Wu |
| 252-255 | [2-CARBOXY-2′-CHLORO-4,4′, 5.5′-TETRA(BENZYLOXY)] AZOBENZENE FROM THE BENZYNE DECOMPOSITION OF 2-CARBOXY-4, 5-DIBENZYLOXYBENZENEDIAZONIUM CHLORIDE | Frank W. Muellner; Ashraf N. Abdel-Sayed; Ludwig Bauer; James N. Shoolery |
| 255-257 | THREE NEW PRODUCTS FROM METHYL 3,4-DIPHENYL-5-NITRO-2-FUROATE BY CATALYTIC REDDCTION | K. Yamamoto; A. Tanaka; M. Ichikawa; S. Swaminathan; G. T. Bryan |
| 258-260 | THE IODINATION OF FLUORENE TO 2,7-DIIODOFLUORENE | R. C. Bansal; E. J. Eisenbraun; R. J. Ryba |
| 261 | OPPI-CORRIGENDUM | |
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| 219-226 | α,β-UNSATURATED ALDEHYDES BY ONE-STEP VINYLOGATION OF CARBONYL COMPOUNDS | Lucette Duhamel; Gérard Plé; Béatriz Contréras |
| 227-236 | SYNTHESIS OF OXYGEN HETEROCYCLES FROM 2-ARYLIDENE-1,3-D1 KETONES | J. A. Ciller; N. Martín; M. Quinteiro; C. Seoane; J. L. Soto |
| 237-244 | SYNTHESIS AND OPTICAL RESOLUTION OF 1-(1-NAPHTHYL)-2-DIMETHYLAMINOETHANOL | Leroy H. Klemm; Jennifer J. Lu |
| 245-252 | REACTION OF 2,7-DI-t-BUTYL-2,4,5,7,9,10-HEXACHLORO-trans-10b,10c-DIMETHYL-2,7,10b,10c-TETRAHYDROPYRENE WITH ALCOHOLS AND WATER AND THE CHEMISTRY OF THE PRODUCTS OBTAINED | Takehiko Yamato; Kazumasa Kobayashi; Masashi Tashiro |
| 253-262 | SYNTHESIS OF ANTIFUNGAL ISOCOUMARINS | H. Kaji; M. Yamada; K. Nozawa; K. Kawai; S. Nakajima |
| 263-268 | A CONVENIENT SYNTHESIS OF (d1)-o-CARBOXY13C-PHENYLALANINE | N. Dale Ledford; Pamala C. Gibbs; H. Blair Wood Jr.; Michael Barfield |
| 269-272 | A FACILE SYNTHESIS OF N-CHLORO FATTY AMIDES | W. A. Henderson Jr.; L. W. Chang |
| 272-275 | SYNTHESIS OF 1,3,4-THIADIAZOLYL UREAS | E. V. P. Tao; Stanislaw Rolski |
| 275-278 | 1-METHYL-4-NITRO-5-IMIDAZOLYL SULFONES | Ned D. Heindel; C. Jeffrey Lacey; Belle A. Mease; David V. Woo |
| 278-281 | A CONVENIENT SYNTHESIS OF PYRROLE-3-CARBOXALDEHYDE | Vassilis J. Demopoulos |
| 281-283 | DIRECT PREPARATION OF 1,3,5-TRIAZA-1,3,5-TRINITROCYCLOHEXANE FROM HEXAMETHYLENETETRAMINE | John W. Fischer; Ronald L. Atkins |
| 283-285 | A FACILE AND EFFICIENT SYNTHESIS OF PYRROLE-3-CARBOXYLIC ACID FROM PYRROLE | Carlos Cativiela; Jose I. Garcia |
| 286-289 | SYNTHESIS OF 3-CARBOXYTHIOPHENE-2-ACETIC ACID AND ITS DERIVATIVES | Reinhold Bender; Dimitri Sarantakis |
| 290-295 | AN IMPROVED SYNTHESIS OF TRIBENZO[a,cd,1m]PERYLENE | J. C. Fetzer; W. R. Biggs |
| 295-297 | 3-METHYLSUCCINIMIDE AND 3-METHYLPYRROLIDINE | R. S. Budhram; N. Pourahmady; A. -S. Syed; E. J. Eisenbraun |
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| 155-162 | REDUCTIVE CLEAVAGE OF N-NITROSOOXAZOLIDINES TO AMINES WITH Al-Ni ALLOY. REDUCTION TO SECONDARY N-ALKYLALKANOLAMINES | Joseph E. Saavedra |
| 163-167 | SYNTHESIS OF 3-MERCAPTOTHIOPHENE-2-AND 4-CARBOXYLIC ACIDS | C. Corral; J. Lissavetzky; A. S. Alvarez-Insúa; A. M. Valdeolmillos |
| 169-173 | AN IMPROVED SYNTHESIS OF 5,5,9,9-TETRAMETHYL-5H, 9H-QUINO[3,2,1-DE]ACRIDINE | John L. Fox; Chin H. Chen; John F. Stenberg |
| 175-181 | AN EFFICIENT SYNTHESIS OF D,L-CARNITINE HYDROCHLORIDE via THE ACYLATION OF AN α-AMINOKETONE | Robert N. Comber; Wayne J. Brouillette |
| 183-186 | A MODIFIED STRECKER SYNTHESIS | Khuong Mai; Ghanshyam Patil |
| 187-190 | A FACILE SYNTHESIS OF 6,7-DIHYDRO-5H-DIBENZO[a,c]CYCLOHEPTENE | G. William Griffin; Keith A. Horn |
| 190-192 | ORGANIC SONOCHEMISTRY. A FACILE SYNTHESIS OF 1-METHYLISOQUINOLINE | J. Ezquerra; J. Alvarez-Builla |
| 192-194 | STEROIDAL ALLYLIC OXIDATION WITH CHROMIUM TRIOXIDE IN THE PRESENCE OF PYRAZOLE | Edward J. Parish; Sarawanee Chitrakorn; Kenneth L. Todd III |
| 195-198 | A NEW SYNTHESIS OF 2-BROMO-1-(9-PHENANTHRYL)ETHANE | Magid Abou-Gharbia; Bruce R. Hoffman |
| 198-203 | SYNTHESIS OF SOME 2-PYRAZOLIN-5-ONE DERIVATIVES STRUCTURALLY RELATED TO CERTAIN ANALGESIS AND ANTIPYRETIC DRUGS | M. A. Metwally; A. A. Fadda; H. M. Hassan; E. Afsah |
| 203-205 | OXIDATION OF FURFURALDEHYDES WITH SODIUM CHLORITE | J. A. Moore; Emmett M. Partain III |
| 206-210 | SYNTHESIS OF THIADIAZINE AND ARYLMETHINEAZOTHIAZOLONE DERIVATIVES OF COUMARIN | R. Djudjic; M. Trkovnik; D. Kitan |
| 210-212 | AN EFFICIENT SYNTHESIS OF N-(2,4-DIFLUOROPHENYL)-N-METHYL-2,4-DINITRO-6-(TRIFLUOROMETHYL)ANILINE | E. V. P. Tao; H. A. Corbitt |
| 212-214 | A CONVENIENT, TWO-STEP SYNTHESIS OF BICYCLO[3,3,0]OCT-1(5)-ENE | Paul J. Okarma; Joseph J. Caringi |
| 215-218 | AN IMPROVED SYNTHESIS OF METHYL [5-BENZOYL- AND 5-p-FLUOROBENZOYLBENZIMIDAZOL-2-YL]CARBAMATES | Siya Ram; Dean S. Wise; Leroy B. Townsend |
| 219-223 | REACTIVE ALUMINUM POWDERS FOR THE REDUCTION OF HALOARENES. APPLICATION OF THE “PLANNING OF EXPERIMENTS” METHOD FOR THE OPTIMISATION OF OBTAINING REACTIVE METAL POWDER | A. Akagah; J. -C. Poite; M. Chanon |
| 223-227 | A CONVENIENT PREPARATION OF 9-DIMETHYLAMINO-10-CARBOMETHOXYANTHRACENE | Andrew T. Brown; Geoffrey Hallas |
| 227-230 | MILD SELECTIVE OXIDATION OF SULFIDES TO SULFONES | Suzanne T. Purrington; Anne G. Glenn |
| 230-235 | INDIRECT IODINATION WITH 2-(3,5-DIIODO-4-METHOXYPHENYL)-1,3,4-OXADIAZOLE AS A PRECURSOR OF AN AROYL HYDRAZINE | Ned D. Heindel; Marcian Van Dort |
| 235-238 | A CONVENIENT SYNTHESIS OF N-5-(1,1-DIMETHYLETHYL)-3-ISOXAZOLYL-N,N-DIMETHYLUREA | E. V. P. Tao; G. S. Staten |
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| 83-89 | SYNTHESIS OF N-(p-CARBOBENZOXYAMINOBENZOYL)-L-GLUTAMIC ACID α-BENZYL ESTER | Leszek Krzyzanowski; Barbara Rzeszotarska |
| 91-97 | AN IMPROVED PREPARATION OF (±) 3-HYDROXY-2-PYRROLIDINONE | O. P. Goel; U. Krolls; E. P. Lewis |
| 99-105 | PREPARATION OF β-BROMOTRIMETHYLSILOXYENOLETHERS FROM α-BROMOCARBONYL COMPOUNDS | Lucette Duhamel; Francis Tombret; Jean-Marie Poirier |
| 107-114 | ACTIVATED NITRILES IN HETEROCYCLIC SYNTHESIS. NOVEL SYNTHESES OF PYRIMIDINES AND PYRIDINES | N. M. Abed; N. S. Ibrahim; S. M. Fahmy; M. H. Elnagdi |
| 115-120 | PREPARATION OF 6-SUBSTITUTED-6H-7-AZA-INDENO[1,2-c] ISOQUINOLINE-5, 11-DIONES | S. Wawzonek; M. C. Chen |
| 121-131 | PREPARATION OF n-MONOALKYL MALEATES AND n-MONO- AND DIALKYL FUMARATES | Michael Dymicky; Robert L. Buchanan |
| 133-137 | CHEMISTRY OF COUMARINS. ANNELATION OP COUMARIN SING via REACTIONS OF 3-AMINO-4-HYDROXYCOUMARIN | I. Tabakovic; K. Tabakovic; M. Trkovnik; Z. Stunic |
| 138-140 | 1,2,3,4-TETRAHYDRO-1,4,d2-NAPHTHALENE-1,4.5,6,7.8.-d6 | Mark H. Gaston; Duane R. Skidmore |
| 140-142 | ONE-POT SYNTHESIS OF NITROSTYRENE OXIDES | Karim Rafizadeh; Keith Yates |
| 143-146 | LOW TEMPERATURE OZONOLYSIS OF METHYL O-METHYL PODOCARPATE | Edward J. Parish; Garvis G. McKeen; D. Howard Miles |
| 146-151 | SYNTHESIS AND ELECTROPHILIC SUBSTITUTION REACTIONS OF FLUORINE CONTAINING ARYLGLYOXAL 2-ARYLHYDRAZONES | Krishna C. Joshi; Vijai N. Pathak; Sharda Sharma |
| 152-154 | 3-ARYL-1,2,5-THIADIAZOLES FROM THE REACTION OF TETRASULFUR TETRANITRIDE WITH ARYL METHYL KETONES | Shuntaro Mataka; Kazufumi Takahashi; Masashi Tashiro |
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| 299-307 | IMPROVED SYNTHESIS OF POLYAZOLYLMETHANES UNDER SOLID-LIQUID PHASE-TRANSFER CATALYSIS | Sebastián Juliá; José Ma del Mazo; Luis Avila; José Elguero |
| 309-314 | STUDIES IN THE SYNTHESIS OF HALOGENATED ANTHRAQUINONES. II. A FACILE PREPARATION, OF 1,4-DICHLORO-5,6,8-TRIHYDROXY-9,10-ANTHRACENEDIONE (5,8-DICHLOROPURPURIN) | H. D. Hollls Showalter; Jeanne M. Hoftiezer |
| 315-319 | A SIMPLE PROCEDURE FOR THE CYCLIZATION OF 2′-HYDROXYCHALCONES INTO FLAVANONES | Tamas Patonay; György Litkei; Miklós Zsuga; Anikó Kiss |
| 321-328 | A CONVENIENT SYNTHESIS OF ISOMERICALLY PURE 1-METHYL-2-VINYLCYCLOHEXENE AND 1-VINYLCYCLOHEXENE | George W. Kabalka; Mohammad Mohammadi; Mark Hylarides; Ronald D. Finn |
| 329-333 | IMPROVED PREPARATION OF 2-CHLORO-6-METHYLANTHRAQUINONE, A PRECURSOR FOR THE CORRESPONDING 6-CARBOXYLIC ACID ESTERS AND 2-CHLORO-6,9,10-TRIMETHYLANTHRACENE | V. S. Prabhu; John F. W. Keana |
| 335-372 | AMINE BORANES AS SELECTIVE REDUCING AND HYDROBORATING AGENTS. A REVIEW | Robert O. Hutchins; Keith Learn; Behrooz Nazer; David Pytlewski; Andrew Pelter |
| 373-376 | METHYL 2-(5-ISOPROPYL-3-ISOXAZOLYL) BENZOATE | Robert K. Howe; Becky R. Shelton |
| 376-379 | CHLORINATION OF 5,13-DI-t-BUTYL-8,16-DIMETHYL[2.2]METACYCLOPHANE | Masashi Tashiro; Takehiko Yamato |
| 379-383 | PREPARATION OF HROMOBENZOIC ACIDS FROM THE CORRESPONDING BROMOTOLUENES VIA THE KROHNKE METHOD | Masashi Tashiro; Kouji Nakayama |
| 384-387 | AN IMPROVED SYNTHESIS OF METHIL- AND BENZYL-ESTERS AS WELL AS HYDRAZIDE OF L-PYOGLUTAMYL-L-HISTIDYL-L-TRYPTOPHAN | B. Rzeszotarska; E. Masiukiewicz |
| 388-391 | PARTIAL DEPROTECTION OF 1.2.5.6-DI-O-ISOPROPYLIDENE-D-GLUCOFURANOSES | Ratnasamy Somanathan; Lars H. Hellberg |
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| 79-83 | THIOCARBONYL-ACTIVATED TRANSAMINATION. A FACILE SYNTHESIS OF N4-MONO AND N4,N4-DISUBSTITUTED THIOSEMICARBAZONES | Daniel L. Klayman; Ai J. Lin |
| 85-89 | STUDIES IN THE SYNTHESIS OF HALOGENATED ANTHRAQUINONES. I. A CONVENIENT PREPARATION OF 1,4-DICHLORO-5-HYDROXY-9,10-ANTHRACENEDIONE | Judith L. Johnson; H. D. Hollis Showalter |
| 91-96 | A RAPID AND EFFICIENT SYNTHESIS OF 2H-1,4-BENZOXAZINE-3(4H)-THIONES AND 2H-1,4-BENZOTHIAZINE-3(4H)-THIONES | D. R. Shridhar; M. Jogibhukta; V. S. H. Krishnan |
| 97-114 | THE REACTION OF AMINES WITH METHYLENE CHLORIDE. A BRIEF REVIEW | John E. Mills; Cynthia A. Maryanoff; Robin M. Cosgrove; Lorraine Scott; David F. McComsey |
| 115-119 | PHASE-TRANSFER CATALYZED DOUBLE MICHAEL CONDENSATION. PREPARATION OF 7,11-BISARYLSPIRO[5,5]UNDECANE-1,9-DIONES | D. Loganathan; T. Varghese; G. K. Trivedi |
| 119-125 | A SYNTHESIS OF THE SIDEROPHORE 1,3,5-TRIS(N,N′,N-2,3-DIHYDROXYBENZOYL)AMINOMETHYLBENZENE | Paul F. Schuda; Catherine M. Botti; Michael C. Venuti |
| 126-130 | SELECTIVE PREPARATION. 41. CONVERSION OF 2,2′-DIHYDROXY-3,3′-DI-t-BUTYL-5,5′-DIMETHYLBIPHENYL TO SOME NOVEL DIBENZOFURAN | Masashi Tashiro; Haruo Yoshiya |
| 130-136 | SYNTHESIS OF N-ARYL ENAMINOSULFONES AND IMPROVED PREPARATION OF N-SUBSTITUTED ENAMINONITRILES | Tatsuo Yamamoto; Motowu Muraoka |
| 136-139 | SYNTHESIS OF t-BUTOXYCARBONYL AND BENZYLOXYCARBONYL AMINO ACID AMIDES | B. Rzeszotarska; M. Makowski; Z. Kubica |
| 140-143 | SYNTHESIS OF A NEW POLYMER POLY(4′-VINYLDIBENZO-14-CROWN-4) | T. C. Kuan; S. J. Wang |
| 144-148 | THE FRIEDEL-CRAFTS ACYLATION AND BENZOYLATION OF PYRENE | Ronald G. Harvey; John Pataki; Hongmee Lee |
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| 297-302 | THE VON BRAUN REACTION BETWEEN N-t-BUTYLAMIDES AND PHOSPHORUS OXYCHLORIDE. A CONVENIENT NITRILE SYNTHESIS | Robert B. Perni; Gordon W. Gribble |
| 303-313 | SYNTHESIS OF URACIL, 6-METHYLURACIL AND SOME DIHYDROURACILS | K. S. Bhat; A. S. Rao |
| 315-319 | AN IMPROVED METHOD FOR THE PREPARATION OF 2-SUBSTITUTED 1,2-BENZISOTHIAZOL-3 (2H)-ONES. NOVEL CYCLIZATION OF N-SUBSTITUTED 2-CARBAMOYLBENZENESULFENYL BROMIDES ON ACTIVATED BASIC ALUMINA | Nobumasa Kamigata; Satoshi Hashimoto; Michio Kobayashi |
| 321-327 | SYNTHESIS OF SOME BICOUMARYL SULPHIDES AND SULPHONES | J. R. Merchant; N. M. Koshti |
| 329-333 | SUGAR 1,3,4-OXADIAZOLES VII. CYCLIZATION OF ACETATES OF SUGAR AROYLHYDRAZONES USING LEAD TETRAACETATE | Mahmoud A. M. Nassr |
| 335-340 | SYNTHESIS OF 3-HYDROXYDIBENZ [a,c] ANTHRACENE | Ronald G. Harvey; Jayanta K. Ray; Kutikat B. Sukumaran |
| 341-348 | SYNTHESIS OF 6-BROMO-, 8-BROMO- AND 6, 8-DIBROMOCATECHIN | Eberhard Kiehlmann; Pieter J. Van der Merwe; Hans K. L. Hundt |
| 349-359 | PREPARATION OF 11-HYDROXYMETHYL-2, 3-NAPHTHO-18-CROWN-6 AND ITS CONVERSION INTO A HIGHLY LIPOPHILIC CROWN CARBOXYLIC ACID | Bronislaw Czech; Anna Czech; Richard A. Bartsch |
| 361-364 | THE SYNTHESIS OF HIGH PURITY Nα-BENZYLOXYCARBONYL Nε-t-BUTYLOXYCARBONYL-L-LYSINE | S. T. Chen; K. T. Wang |
| 365-367 | A SIMPLIFIED, ONE STEP SYNTHESIS OF CHOLEST-5-EN-3-ONE | Edward J. Parish; Sarawanee Chitrokorn |
| 368-369 | A FACILE SYNTHESIS OF 2, 2′-BIPYRIDYL-3, 3′-DICARBOXYLIC ACID | Franz L. Wimmer; Smita Wimmer |
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| 309-317 | THE SYNTHESIS OF PHENOLIC ANTIOXIDANTS. 3,5-BIS(3,5-DI-TERT-BUTYL-4-HYDROXYBENZYL)-2,3,6-TRIMETHYLBENZYL DERIVATIVES | Luke K. T. Lam; Alex Chung; Alan V. Fladmoe; Lee W. Wattenberg |
| 319-326 | SYNTHESIS OF 2-AROYL-4-CYANO-4-CARBETHOXY-1,3,5-TRIARYLCYCLOHEXANOLS | J. L. Soto; C. Seoane; A. M. Mansilla; M. Quinteiro |
| 327-331 | A CONVENIENT SYNTHESIS OF ETHYL α-CARBETHOXY-β-(ARYLAMINO) ACRYLATES AND RELATED COMPOUNDS | Nagaraj R. Ayyangar; Rajgopal J. Lahoti; Thomas Daniel |
| 333-336 | AN IMPROVED PREPARATION OF 2,3,4-TRIMETHOXYBENZSUBER-6-ONE | Joseph G. Cannon; Basil J. Demopoulos |
| 337-342 | 7-ETHOXY-6-METHOXY-2,2-DIMETHYL-2H-1-BENZOPYRAN | E. Kiehlmann; J. E. Conn; J. H. Borden |
| 343-346 | A CONVENIENT SYNTHESIS OF 1-BENZYLINDOLES | Robert B. Perni; Gordon W. Gribble |
| 347-349 | SYNTHESIS OF (2R,3R) 0,0-DIPIVALOYLTARTARIC ACID (DPTA) AND OF (2R,3R) 0,0-DI(ADAMANTANE-1 CARBONYL) TARTARIC ACID (DATA), USEFUL CHIRAL REAGENTS FOR ASYMMETRIC PROTONATIONS | L. Duhamel; J. C. Plaquevent |
| 350-353 | SYNTHESIS OF 4'-ALKYLDIBENZO CROWN ETHERS | C. S. Chen; S. J. Wang; S. C. Wu |
| 354-356 | A SIMPLIFIED APPARATUS FOR GENERATION OF DIAZOMETHANE | Milos Hudlicky |
| 357-359 | NITROSYLSULFURIC ACID HYDROLYSIS OF PRIMARY AMIDES | L. G. Wade Jr.; William B. Silvey |
| 359-362 | SYNTHESIS OF ARYL HALIDES via ORGANOBORANE CHEMISTRY | George W. Kabalka; Kunda A. R. Sastry; Usha Sastry; Vishwanatha Somayaji |
| 362-365 | FACILE OXIDATIVE CLEAVAGE OF CARBON-CARBON MULTIPLE BONDS WITH CHROMIUM(V) REAGENT [(BiPy)H2CrOCl5] | T. K. Chakraborty; S. Chandrasekaran |
| 365-369 | O-CYANOMETHYLOXIME OF NITROGLYOXYLONITRILE | T. Perumal Pillai; Joseph H. Boyer |
| 369-372 | A SIMPLE, INEXPENSIVE SYSTEM FOR PERFORMING HIGH PRESSURE REACTIONS | Philip Deshong; C. Michael Dicken; Joseph J. Perez; Robert M. Shoff |
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| 157-162 | SYNTHESIS OF γ-L-GLUTAMYL-TAURINE (GLUTAURINE) | Arthur M. Felix |
| 163-168 | SYNTHESIS OF 6-SUBSTITUTED-6H-INDENO[1,2-c]ISOQUINOLINE-5,11-DIONES | Stanley Wawzonek |
| 169-175 | A MODIFIED APPROACH IN THE SYNTHESIS OF 5- AND 6-METHYLBENZ[a]ANTHRACENES | Peter P. Fu; Frederick E. Evans; Dwight W. Miller; J. P. Freeman; Shen K. Yang |
| 177-181 | A GENERAL METHOD FOR THE PREPARATION OF FORMATES | M. Dymicky |
| 183-187 | A CONVENIENT METHOD FOR THE SYNTHESIS OF KAEMPFEROL | Masataka Ichikawa; A. Mahir Pamukcu; George T. Bryan |
| 189-194 | ALKOXYETHYNYL KETONES | G. Himbert; L. Henn |
| 195-197 | A GENERAL AND CONVENIENT SYNTHESIS OF 2H-1,4-BENZOXAZIN-3(4H)-ONES | D. R. Shridhar; M. Jogibhukta; V. S. H. Krishnan |
| 197-198 | AN UNUSUAL SYNTHESIS OF 2,6-Di-t-BUTYL-4-ISOPROPENYLPHENOL | Lajos Avar |
| 199-200 | PREPARATION OF ISATOIC ANHYDRIDE FROM PHTHALIMIDE | Y. R. Rao; M. Bapuji; S. N. Mahapatra |
| 200-202 | HIGH-YIELD, ONE STEP PHOTOCHEMICAL SYNTHESIS OF 3- AND 4-BROMOMETHYLBENZOIC ACIDS | Ravi Subramanyam; A. G. Pinkus |
| 202-203 | SYNTHESIS OF BENZ(a)ANTHRACENE-5,6-DIONE | Dominic T. C. Yang; W. M. Trie |
| 204-205 | SYNTHESIS OF 2-CHLORO-4-FLUORANILINE | Jeffery B. Press; Corris M. Hoffman |
| 206-208 | 2,4-BIS(BROMOMETHYL)-5-METHYL-N-ACETYL BENZYLAMINE AND 2,4-BIS(CYANOMETHYL)-5-METHYL-N-ACETYLBENZYLAMINE | Nitya G. Kundu; James Peck; Dennis W. Evangelatos |
| 208-213 | PHOTOCHEMICAL SYNTHESIS OF BULLVALENEDIONE | T. Miyashi; Y. Takahashi; K. Okada; T. Mukai |
| 213-215 | AN IMPROVED SYNTHESIS OF TRIALKYLKETENIMINES | N. De Kimpe; R. Verhé; L. De Buyck; N. Schamp |
| 216-219 | METACYCLOPHANES AND RELATED COMPOUNDS. 2.† NITRATION AND ACETYLATION OF 2,7-DI(t-BUTYL)-trans-10b,10c-DIMETHYL-10b,10c-DIHYDROPYRENE | Masashi Tashiro; Takehiko Yamato |
| 220-224 | SYNTHESIS OF α-AMINOKETONES BY CATALYTIC HYDROGENATION OF BENZILMONOIMINES | Benito Alcaide; Gerardo Escobar; Rafael Pérez-Ossorio; Joaquin Plumet |
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| 71-79 | MICHAEL ADDITION OF DITHIOBENZOIC ACID TO α,β-UNSATURATED KETONES. A NEW SERIES OF DITHIOESTERS | Jayalakshmi Ramachandran; S. R. Ramadas; C. N. Pillai |
| 81-86 | SYNTHESIS OF 4-ARYL-5,6-BIS (CARBOMETHOXY)-2H-THIOPYRAN-2-THIONES. A NEW SERIES OF CYCLIC DITHIOESTERS OR α-DITHIOPYRONES | Jayalakshmi Ramachandran; S. R. Ramadas; C. N. Pillai |
| 87-92 | POLYETHERS. 2. PREPARATION OF ω,ω′-DISUBSTITUTED POLYARYLETHERS | Masashi Tashiro; Haruo Yoshiya; Gouki Fukata |
| 93-96 | STUDIES ON FRIEDEL-CRAFTS CHEMISTRY. 5. THE AlCl3-CH3NO2-CATALYZED FRIEDEL-CRAFTS REACTIONS OF BIS (BROMOMETHYL) BENZENES WITH BENZENE | Shuntaro Mataka; Yuhsuke Tsuda; Kazufumi Takahashi; Masashi Tashiro |
| 97-101 | MILD PREPARATION OF PYRROLE-2-CARBOXALDEHYDES | J. A. de Groot; G. M. Gorter-La Roy; J. A. van Koeveringe; J. Lugtenburg |
| 103-108 | ISOMER-SELECTIVE SYNTHESES OF 2,6-DICHLORO-4-NITROTOLUENE AND 2,4-DIFLUOROANILINE | Leonard M. Weinstock; Anthony M. Demarco; Roger J. Tull; Ichiro Shinkai |
| 109-112 | A GENERAL SYNTHESIS OF UNSUBSTITUTED POLYCYCLIC ARENE IMINES. 3-METHYLCHOLANTHRENE 11,12-IMINE | Irene Yona; Jochanan Blum |
| 112-115 | PREPARATION OF p-TOLUENESULFONYL AZIDE. A CAUTIONARY NOTE | Thomas J. Curphey |
| 116-118 | 3-CHLOROMETHYL-2,4,6-TRIMETHYLBENZOIC ACID | F. H. C. Stewart |
| 118-123 | SYNTHESIS OF p-BIS (DIMETHYLHYDROXYSILYL) BENZENE | H. Matsumoto; K. Shono; Y. Nagai |
| 123-126 | THE SYNTHESIS OF 3-R-7-CARBOMETHOXYMETHYLENE-7H-1,2,4-TRIAZOLO[3,4-b]-1,3,4-THIADIAZIN-6-ONES | Ned D. Heindel; Jack R. Reid |
| 126-129 | REDUCTION OF 5-HYDROXYMETHYL-1-AZA-3,7-DIOXABICYCLO[3.3.0]OCTANE AND OF 2-PHENYL-4,4-DIMETHYLOXAZOLIDINE WITH FORMIC ACID | S. Wawzonek |
| 129-134 | REACTION OF DIAZOMETHANE WITH N-NITROSO-4-PIPERIDINONES | Joseph E. Saavedra |
| 134-136 | LEWIS ACID CATALYZED PREPARATION OF TETRAMETHYLHEXATHIOADAMANTANE | C. S. Giam; R. L. Tabor; T. E. Goodwin |
| 137-140 | A CONVENIENT PREPARATION OF ALKYL- AND ARYLSULFONYLPYRIDINES | C. S. Giam; K. Kikukawa; D. A. Trujillo |
| 140-144 | A CONVENIENT PREPARATION OF cis-DIHYDROIONONE | Crist N. Filer; James C. Pugliese; John C. Morrison; David G. Ahern |
| 144-149 | A CONVENIENT PREPARATION OF α,α-DIPHENYLACETOPHENONE | N. Sbarbati Nudelman; A. A. Vitale |
| 149-151 | AN IMPROVED PREPARATION OF CORONENE | A. G. Holba; E. J. Eisenbraun |
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| 181-184 | THIOL ESTERS OF Nα-TOSYL-L-ARGININE | T. R. Herrin; J. J. Plattner; J. W. Cole; M. R. Shaffar |
| 185-189 | S-CARBOXYMETHYL DERIVATIVES OF L-CYSTEINYLGLYCINE AND GLYCYL-L-CYSTEINE | Marvin D. Armstrong |
| 191-195 | A PREPARATIVE SCALE SYNTHESIS AND CHROMATOGRAPHIC SEPARATION OF METHOTREXATE-α AND γ-MONOBUTYL ESTERS | J. D. Warren; R. B. Angier; George Morton; Andre Rosowsky |
| 197-200 | DINITRONATE SALTS OF SUCCINONITRILE | Edward F. Witucki; Walter Maya; Milton B. Frankel |
| 201-202 | A CONVENIENT SYNTHESIS OF p-HYDROXYBENZAL DEHYDES | C. W. Bird; Y. -P. S. Chauhan |
| 203-206 | AN IMPROVED PROCEDURE FOR THE CONVERSION OF 2H-(1, 4)-BENZO-THIAZIN- AND 2H-(1, 4)-BENZOXAZIN-3(4H)-ONES INTO 3(4H)-THIONES | D. R. Shridhar; C. V. Reddy Sastry; L. C. Vishwakarma; G. K. A. S. S. Narayan |
| 207-212 | A GENERAL, HIGHLY EFFICIENT SYNTHESIS OF ACETYL AMINO ACID ETHYL ESTERS | M. Dymicky |
| 213-218 | SYNTHESIS OF α,α′-DIFUNCTIONAL CONJUGATED ENYNES | Jean-Paul Charpentier; Danielle Mesnard; Léone Miginiac |
| 219-223 | A FACILE BASE CATALYZED CONDENSATION FOR THE SYNTHESIS OF FUSED PYRIMIDINE-2-CARBOXYLIC ACID ESTERS | Susumu Nakanishi; Stephen S. Massett |
| 225-228 | A NEW RAPID ESTERIFICATION PROCEDURE UTILIZING EXCEPTIONALLY MILD REACTION CONDITIONS | C. Gundu Rao |
| 229-230 | AN IMPROVED METHOD FOR THE SYNTHESIS OF DISULFONYLMETHYL THIOLSULFONATES | Nils Henning Nilsson; Alexander Senning |
| 230-232 | SYNTHESIS OF dl-2-METHYL-2-(4-METHYL-3-PENTENYL) 5-OXYMETHYLENEMETHOXY-2H-BENZOPYRAN. A CANNABICHROMENE HOMOLOGUE | F. Garcia; R. Laureles; R. Cruz |
| 233-234 | 3-ARYL-5-CARBOMETHOXY-5-CARBOMETHOXYMETHYL-1,4,2-OXATHIAZOLES | Ned D. Heindel; Gail K. Friedrich; Maria C. Tsai |
| 234-237 | IMPROVED PREPARATION OF PYRIDO[3′,4′(4′,3′):4,5]IMIDAZO [1,2-c] [1,2,3]BENZOTRIAZINES | Jessie Lee; Anne Guthrie; Madeleine M. Joullié |
| 238-242 | IMPROVED SYNTHESES OF 9-HYDROXY- AND 9-BUTOXY-1-PHENALENONE | K. D. Franz; R. C. Haddon |
| 242-243 | t-BUTYL PHENYL CARBONATE | John W. Scott; David Parker |
| 243-244 | AN IMPROVED SYNTHESIS OF 2,2′-DIPYRIDYL-1-OXIDE | Willem Sont; Howard Alper |
| 244-246 | 13C-LABELLED ALIPHATIC NITRILES AND KETONES | Gert Kollenz; Hans Waldenberger |
| C | Editorial Board Page | |
| 257-262 | CONVENIENT ONE-STEP CONVERSIONS OF ALCOHOLS OR PHENOLS TO N,N-DIPROPYL ALKOXYACETAMIDES | Irving J. Borowitz; Ven-Shun Li; Irwin Gross |
| 263-266 | DEOXYGENATION OF QUINOXALINE 1,4-DIOXIDES WITH TITANIUM TRICHLORIDE | Berkeley W. Cue Jr.; John P. Dirlam; Edward A. Glaser |
| 267-270 | SUGAR 1,3,4-OXADIAZOLES. IV: THE SYNTHESIS OF SUGAR 1,3,4-OXADIAZOLINE DERIVATIVES | M. A. E. Shaban; M. A. M. Nassr; E. H. El. Ashry; V. N. Reinhold |
| 271-276 | A CONVENIENT N-ACETYLATION OF INDOLES | Gordon W. Gribble; Laurence W. Reilly Jr.; Jerry L. Johnson |
| 277-280 | AN IMPROVED SYNTHESIS OF 1-BENZOYL-4-KETO-1,2,2A,3,4,5-HEXAHYDROBENZ [cd]INDOLE | David E. Nichols; J. Michael Robinson; George S. Li; John M. Cassady; Heinz G. Floss |
| 281-284 | PREPARATION OF 2-PHENYLPERHYDROAZEPINE | S. Wawzonek; J. M. Shradel |
| 285-288 | A SIMPLE SYNTHESIS OF 4-CYCLOHEXENE-1,2-cis-DIOL AND ITS USE AS THE PRECURSOR OF A FUNCTIONALIZED CYCLOHEXENONE SYNTHON | Grant R. Krow; Richard Carmosin; Anthony Mancuso |
| 289-296 | SYNTHESIS OF NITROXYL DERIVATIVES OF BENZO[a]PYRENE | H. Schlude |
| 297-299 | REDUCTIVE ALKYLATION OF ANILINE WITH 2-INDANONE AND 2-TETRALONE | Jack B. Campbell; E. R. Lavagnino |
| 299-303 | SULTAMO-STEROIDS II | S. H. Doss; S. S. A. Dimitry |
| 303-307 | ETHYL 2-(4-AMINOPHENYL) PROPIONATE | M. Perchinunno; A. Guerrato; F. Pregnolato |
| 309 | OPPI-CORRIGENDUM | |
| 311-318 | INDEXES | |
| C | Editorial Board Page | |
| 49-52 | SYNTHESIS OF THE SELECTIVE BLADDER CARCINOGEN, N-(n-BUTYL)-N-(3-CARBOXYPROPYL)NITROSAMINE (BCPN) | William Gaffield; Larry K. Keefer; Peter P. Roller |
| 53-56 | USE OF SODIUM CYANOBOROHYDRIDE IN THE SYNTHESIS OF BIRADICAL NITROXIDES | Elmer J. Rauckman; Gerald M. Rosen; W. Winn Hord |
| 57-62 | COMPARISON OF SYNTHETIC ROUTES TO DL-CANALINE | Timo Korpela; Juhani Lundell; Paavo Pasanen |
| 63-83 | DEXYGENATION OF SULFOXIDES. A REVIEW | Jozef Drabowicz; Tatsuo Numata; Shigeru Oae |
| 85-87 | AN IMPROVED SYNTHESIS OF 5β-CHOLEST-3-ENE | D. T. C. Yang; G. W. Kabalka |
| 87-89 | IMPROVED PROCEDURE FOR THE PREPARATION OF “OXAURACIL”, 2H-1,3(3H)-OXAZINE-2,6-DIONE | John H. Macmillan |
| 89-91 | NOVEL ACID HYDROLYSIS OF 2,3,5,6-DIEPOXY-2,5-DIMETHYL-1,4-BENZOQUINONE | Aspi B. Daruwala |
| 91-94 | A RAPID AND MILD PROCESS FOR THE OXIDATION OF 2,3-DICHLORO-5,6-DICYANOBENZOQUINONE (DDQ) FROM 2,3-DICHLORO-5,6-DICYANOHYDROQUINONE (DDHQ) | John W. Scott; David R. Parrish; Fred T. Bizzarro |
| 94-96 | A BRIEF PREPARATION OF THIAN-4-CARBOXYLIC ACID 1,1-DIOXIDE | E. Carlon; R. W. Draper; R. Friary |
| 96-98 | AN EFFICIENT SYNTHESIS OF 4-HYDROXYBENZOTRIFLUORIDE | E. R. Lavagnino; B. B. Molloy; J. W. Paschal |
| 99-101 | SYNTHESIS OF NOPALINE AND ISO-NOPALINE | D. Cooper; J. L. Firmin |
| C | Editorial Board Page | |
| 103-106 | THE N-DEMETHYLATION OF MORPHINE AND CODEINE USING METHYL CHLOROFORMATE | George A. Brine; Karl G. Boldt; Carolyn King Hart; Frank I. Carroll |
| 107-112 | SACCHARIDE 1,3,4-OXADIAZOLES | M. Shaban; M. Nassr |
| 113-118 | SUGAR 1,3,4-OXADIAZOLES. III. THE SYNTHESIS OF 1,2,3,4-TETRA-O-ACETYL-1,4-BIS(5-ARYL-1,3,4-OXADIAZOL-2-YL)-GALACTO-TETRITOLS | M. Shaban; M. Nassr |
| 119-124 | REDUCTION OF SULFOXIDES WITH METHANE- AND p-NITROBENZENESULFINYL CHLORIDE BY OXYGEN TRANSFER REACTION | Tatsuo Numata; Katsuyata Ikura; Yasutaka Shimano; Shigeru Oae |
| 125-132 | SYNTHESIS OF 2-(1-NAPHTHYLMETHYL)-3,4-DIHYDRONAPHTHALENE, 2-(1-NAPHTHYLMETHYL)-1,2,3,4-TETRAHYDRONAPHTHALENE, 7a, 8, 9, 13b-TETRAHYDRO-7H-DIBENZ [a, k L] ANTHRACENE, AND 5,6-DIHYDRO-4H-DIBENZ[a, k L]ANTHRACENE | L. L. Ansell; T. E. Webb; J. W. Burnham; E. J. Eisenbraun; M. C. Hamming; G. W. Keen |
| 133-140 | THE SYNTHESIS OF 1,2,3,7,8,9-HEXAHYDRODIBENZO[def, mno]CHRYSENE AND THE USE OF HYDRIODIC ACID-RED PHOSPHORUS IN THE DEOXYGENATION OF KETONES | L. L. Ansell; T. Rangarajan; W. M. Burgess; E. J. Eisenbraun; G. W. Keen; M. C. Hamming |
| 141-143 | A RAPID, CONVENIENT, HIGH YIELD PROCEDURE FOR THE REGENERATION OF 2,3-DICHLORO-5,6-DICYANOBENZOQUINONE (DDQ) FROM THE CORRESPONDING HYDROQUINONE (DDHQ) | Ki Hwan Kim; Gary L. Grunewald |
| 143-146 | A SIMPLIFIED PROCEDURE FOR THE SYNTHESIS OF THE 6,7-BENZOMORPHAN NUCLEUS | E. Bellora; E. Cereda; A. Donetti |
| 146-148 | SYNTHESIS OF NEW PHENYLQUINOXALINES | J. A. Harvey; M. A. Ogliaruso |
| 148 | DIETHYL 2,5-DI [BENZYLOXY] TEREPHTHALATE | S. Wawzonek; J. E. Durham |
| C | Editorial Board Page | |
| i | NOTICE | |
| ii | PREFACE | J. P. Anselme |
| 1-5 | 1-ACYL-4-SUBSTITUTED PIPERAZINES | James A. Moore; E. A. Steck |
| 6-11 | SOME BENZIMIDAZOLE DERIVATIVES | Edgar A. Steck; R. Pauline Brundage |
| 11-14 | SYNTHESIS OF METHYL 2,3,4-TRI-0-ACETYL-6-DEOXY-6-IODO-α-D-GLUCOPYRANOSIDE | Tai-Shun Lin; Robert E. Harmon |
| 14-16 | AN IMPROVED SYNTHESIS OF 2-ETHYL-2-PHENYL-GLUTACONIMIDE | Hassan Y. Aboul-Enein |
| 16-21 | THE SYNTHESIS OF STEROLS WITH MODIFIED SIDE CHAINS BY THE WITTIG REACTION | J. E. Herz; S. M. Cruz |
| 21-22 | THE SPECTRAL CHARACTERIZATION OF endo-4-OXATRICYCL[5,2,1,02,6]DEC-2-ENE | Bradford P. Mundy |
| 23-26 | NEW MIXED KETENE DIALKYL ACETALS | G. R. Cliff; D. J. Dunn |
| 26-30 | 4H-BENZPYRANO [3,4-d]OXAZOL-4-ONES AND 3-[N,N-BIS(CARBOXYMETHYL)AMINO]-4-HYDROXYCOUMARIN DERIVATIVES | M. Trkovnik; M. Kules; K. Krunic |
| 31-34 | HYDROGENOLYSIS OF ARYL HALIDES IN THE PRESENCE OF RANEY NICKEL IN ALKALINE MEDIUM | A. J. De Koning |
| 35-37 | SYNTHESIS OF DIMETHYL 1,2-DIHYDROPYRIDAZINE-1,2-DICARBOXYLATE | L. J. Altman; M. F. Semmelhack; R. B. Hornby; J. C. Vederas |
| 39-42 | A NEW PORPHINOGEN TYPE COMPOUND | O. Tsuge; M. Tashiro; Y. Kiryu |
| 43-46 | STUDIES ON POSITIONAL PROTECTIVE GROUPS III. A NEW PREPARATIVE METHOD FOR CHLOROPHENOLS WITH THE BROMO GROUP AS A PROTECTIVE GROUP | M. Tashiro; H. Watanabe; O. Tsuge |
| 47-50 | ELECTROCHEMICAL SYNTHESIS OF 3-AMINO-4-HYDROXYCOUMARIN | M. Trkovnik; M. Laćan; Z. Stunić; D. Nahmijaz |
| 51-54 | ROBINSON ANNELATION WITH A β-HYDROXYKETAL IN THE PRESENCE OF AN ACID | P. A. Zoretic; B. Branchaud; T. Maestrone |
| C | Editorial Board Page | |
| 259-263 | A SIMPLE, TWO STEP SYNTHESIS OF 1-(2-CHLOROETHYL)-1-NITROSO-3-(D-GLUCOS-2-YL) UREA | H. Donald Burns; Ned D. Heindel |
| 265-267 | PREPARATION OF 3, 6-EXO-OXO-HEXAHYDROPHTHALIDE | Humberto Cervantes Cuevas; Federico García Jiménez |
| 269-273 | cis-OLEFINS FROM THE WITTIG REACTION | P. E. Sonnet |
| 275-280 | A CONVENIENT PREPARATION OF HOMOGENEOUS 2,3,6-TRICHLOROBENZOIC ACID AND ITS CONVERSION TO 2,2′,3,3′,6,6′-HEXACHLOROBIPHENYL | Louis A. Levy |
| 281-285 | N-BENZOYLBENZILIMINE | Peter Yates; E. M. Levi |
| 287-293 | SYNTHESIS OF 2-METHOXYDIBENZO [b,f] (1,4)-THIAZEPIN-11(10H)-ONE-5,5-DIOXIDE | O. Francis Bennett; James Johnson; John Tramondozzi |
| 295-298 | PREPARATION OF 1,2,3-TRIAZOLO[4,5-f]QUINOLINE N-OXIDES FROM 6-NITRO-5,8-DIMETHOXYQUINALDINE | Paul C. Unangst; Ned D. Heindel |
| 299-303 | REDUCTIVE ALKYLATION OF ACRYLONITRILES AND ACRYLATES | T. Caronna; A. Citterio; A. Clerici; R. Galli |
| 305-311 | HYDROXYL GROUP ELIMINATION IN THE MORPHINE SERIES | R. Bognár; Gy. Gaál; P. Kerekes; G. Horváth; M. T. Kovács |
| 313-324 | INDEXES | |
| C | Editorial Board Page | |
| 103-106 | CATALYTIC REDUCTION OF 1,1,1-TRIS(AZIDOMETHYL)ETHANE TO 1,1,1-TRIS(AMINOMETHYL)ETHANE | L. J. Zompa; J. P. Anselme |
| 107-115 | STUDIES ON POSITIONAL PROTECTIVE GROUPS ON AROMATIC RINGS I. A NEW PREPARATIVE METHOD FOR HALOPHENOLS WITH THE t-BUTYL OR BENZYL GROUP AS A PROTECTIVE GROUP | M. Tashiro; H. Watanabe; O. Tsuge |
| 117-122 | STUDIES ON POSITIONAL PROTECTIVE GROUPS ON AROMATIC RINGS II. A NEW PREPARATIVE METHOD FOR DIHYDROXYDI-PHENYLS WITH t-BUTYL GROUP AS A PROTECTIVE GROUP | M. Tashiro; H. Watanabe; O. Tsuge |
| 123-130 | THE PREPARATION OF DIHYDROXYDIPHENYLMETHANE DERIVATIVES CONTAINING NITRO GROUPS. I. SYMMETRICALLY SUBSTITUTED COMPOUNDS | W. Lotz; V. Böhmer |
| 131-134 | 4-METHYLPENT-4-EN-2-ONE (iso-MESITYL OXIDE) | R. D. Gillard; B. T. Heaton; M. P. Pilbrow |
| 135-139 | 1,5-DIMETHYLTETRAZOLE | F. E. Condon; Robert Waldman; Nitya Kundu; J. P. Trivedi |
| 141-144 | THE STUDIES ON DIHYDROISOCOUMARIN (III). THE SYNTHESIS OF 3-(3′-HYDROXY-4′-METHOXYPHENYL)-3,4-DIHYDROIROCOUMARIN | Y. Naoi; K. Sakai; T. Nakano; H. Ito; S. Higuchi; T. Matsui; Y. Takahashi; S. Wagatsuma; A. Nishi; S. Sano |
| 145-147 | NEW 2,4- AND 4,5-DIALKYLOXAZOLES | James A. Moore; P. B. Terentiev; A. N. Kost; N. P. Lomakina; V. G. Kartev |
| 148-149 | 4-(α,β-DIBROMOETHYL)PHENYLPHOSPHONIC ACID | M. A. Rea; T. L. Slapar; W. A. Trinler |
| 149-153 | 3,4-DIALKYLQUINOLINES BY AN EXTENSION OF THE BEYER SYNTHESIS | Paul A. Claret; A. G. Osborne |
| 153-156 | 2-CYCLOHEXYLIDENECYCLOPENTANONE | Richard D. Sands |
| 156-157 | 4-AMINO-3-HYDRAZINO-5-MERCAPTO-1,2,4-TRIAZOLE | R. G. Dickinson; N. W. Jacobsen |
| 159 | CORRIGENDA | |
| C | Editorial Board Page | |
| 255-260 | FERROCENES FROM CYCLOPENTADIENES. 1,1′-DIMETHYLFERROCENE | Ilgvars J. Spilners; Robert J. Hartle |
| 261-264 | SYNTHESIS OF 5-BENZOYL-6-PHENYL-1,3-0XAZINONES+ (SYNTHESES OF HETEROCYCLES, 179.) | G. Kollenz; E. Ziegler; W. Ott |
| 265-269 | SYNTHESIS OF α-AMINO-β-(p-HYDR0XYPHENOXY) PROPIONAMIDE HYDROCHLORIDE | S. Wawzonek; W. P. Gaffield Jr. |
| 271-273 | 2,4,6-TRINITRORESORCINOL | B. A. Bydal |
| 275-279 | AN IMPROVED STEREOSELECTIVE REDUCTION FOR THE PREPARATION OF endo-7-PHENYLNORCARANE | Paul R. Morris; James D. Woodyard |
| 281-284 | METHYLAMINOACETONE ETHYLENE KETAL HYDROCHLORIDE | F. Benington; R. D. Morin |
| 285-290 | THE SYNTHESIS OF 5-TERT-BUTYL-1,2,3,4-TETRAHYDRONAPHTHALENE | J. W. Burnham; W. P. Duncan; E. J. Eisenbraun; G. W. Keen; M. C. Hamming |
| 291-298 | SYNTHESIS OF POLYMETHOXY-1-TETRALOUES | Theodore E. Snider; Mohamed M. Hashem; K. D. Berlin; R. W. Chesnut; N. N. Durham |
| 299-301 | AN IMPROVED SYNTHESIS OF 1,4-DIHYDRO-3-[2H]-ISOQUINOLONE | R. E. Lyle; D. A. Walsh |
| 303-304 | exo-TRICYCLO[4.2.1.02,5] NON-7-EN-3-ONE | Roy C. De Selms |
| 305-306 | AN IMPROVED SYNTHESIS OF 2-IODO-5-NITROPYRIDINE | Frank L. Setliff |
| 307-318 | INDEXES | |
| C | Editorial Board Page | |
| 1-3 | 2,2-′AZOBIS(2-CYANO-n-PROPANOL). A NEW FREE RADICAL INITIATOR | P. O. McCoy |
| 5-8 | A SYNTHESIS OF 2,3-DIMETHOXY-6-(3,4-DIMETHOXYPHENYLACETYL)TOLUENE | J. A. Bakker; H. C. Beyerman; L. Maat |
| 9-11 | 4-NITROISOQUINOLINE | John W. Bunting; William G. Meathrel |
| 13-18 | PREPARATION OF HOMOMIRISTICINIC ACID | G. Y. Moltrasio; D. Giacopello; M. J. Vernengo |
| 19-21 | INEXPENSIVE STEEL REACTION VESSELS AND ACCESSORIES FOR ORGANIC REACTIONS | E. J. Eisenbraun; H. Hall |
| 23-26 | HYDROLYSIS OF 2-OXOCYCLOPENTYL PHENYL KETIMINE | Stuart S. Kulp; Bartholomew Palenchar; Robert K. Sharer |
| 27-30 | 3-METHYL-3-BUTEN-1-OL AND 3-BUTEN-1-OL | R. B. Kinnel; B. B. Molloy; D. W. Graham; K. E. Harding |
| 31-34 | AN IMPROVED PREPARATION OF DIETHYL 1,4-DIHYDROXY-CYCLOHEXA-1,4-DIENE-2,5-DICARBOXYLATE | J. A. Moore |
| 35-42 | THE SYNTHESIS OF 1H, 3H-NAPHTHO[1,8-cd]PYRAN-1-ONE, 1,8-DIMETHYL-1, 2,3,4TETRAHYDRONAPHTHALENE, 1,3,3a,4,5,6-HEXAHYDRONAPHTHO[1,8-cd] PYRAN, AND 1,2,3,4-TETRAHYDRO-8-METHYL-1-NAPHTHALENEMETHANOL | J. W. Burnham; E. J. Eisenbraun; M. C. Hamming; G. W. Keen |
| 43-47 | 4-(7-BENZ[a]ANTHRACENYL)-N-(2-SUBSTITUTED ETHYL)BENZAMIDES | F. A. Vingiello; M. P. Rorer; M. A. Ogliaruso |
| 49 | 2,4-DINITROPHENYLHYDRAZONES | D. E. Pearson |
| C | Editorial Board Page | |
| 213-215 | 3-(2-HYDROXYETHYL) TETRAHYDROFURAN. CYCUZATIONS IN LITHIUM ALUMINUM HYDRIDE REDUCTIONS | Leonard O. Moore |
| 217-222 | THE SYNTHESIS OF TWO NEW 2,3-DIHALO-5-METHYLPYRIDINES | Prank L. Setliff |
| 223-226 | DDQ DEHYDROGENATION OF DIHYDRODICTAMNINE | F. Piozzi; P. Venturella; A. Bellino |
| 227-230 | DIAZOACETALDEHYDE | John Hooz; Geoffrey F. Morrison |
| 231-233 | SYNTHESES WITH AMMONIUM PEROXYDISULPHATE. α,β-DIAZIDOETHYLBENZENE AND α-CHLORO-β-AZIDOETHYLBENZENE | R. Galli; V. Malatesta |
| 235-238 | 3- AND 4-(BENZ[a]ANTHRACENYL)PHENYL-2-THIAZ0LINES AND 3- AND 4-(9-ANTHRACENYL)PHENYL-2-THIAZ0LINES. A NEW METHOD OF PREPARATION OF THIAZOLINES | F. A. Vingiello; M. P. Rorer; M. A. Ogliaruso |
| 239-242 | AN IMPROVED SULFONIC ACID-RESIN CATALYZED CYCLIDEHYDRATION OF 2-METHYL-4-PHENYL-2-BUTANOL TO 1,1-DIMETHYLINDAN | W. M. Harms; E. J. Eisenbraun |
| 243-248 | PREPARATION OF 4H-PYRAN-2,6-DICARBOXYLIC ACID AND 4-METHYL-4H-PYRAN-2,6-DICARBOXYLIC ACID | J. C. Lewis; R. M. Seifert |
| 249-254 | AN EFFICIENT TECHNIQUE FOR THE CLEAVAGE OF HYDROCARBON PICRATES. THE PURIFICATION OF 1,8-, 2,6-, and 2,7-DIMETHYLNAPHTHALENE | E. J. Eisenbraun; T. E. Webb; J. W. Burnham; L. E. Harrisld |
| 255-260 | DI-2-PYRIDYLMETHANOL AND 1,1-DI-2-PYRIDYLETHANOL | Joe Murphy; John W. Bunting |
| 261-267 | 1-ETHYL-4-CARBOMETHOXYPYRIDINYL (Pyridinyl, 1-ethyl-4-carbomethoxy) | E. M. Kosower; Harold P. Waits |
| 269 | STYRYL CARBONATES FROM ARYLACETONES. A CORRECTION | John L. Wong; Calvin H. Savells Jr. |
| C | Editorial Board Page | |
| 109-112 | SYNTHESIS OF 4-ETHYL-2,6-DINITRO-N,N-DIPROPYLANILINE-A NEW PLANT-GROWTH REGULATOR AND SELECTIVE HERBICIDE | C. S. Giam; R. C. Hall |
| 113-116 | A NEW SYNTHESIS OF 10, 11 -DIHYDRO-5H-DIBENZO (a, d)CYCLOHEPTEN-5-ONE | Jasjit S. Bindra; Shiv N. Rastogi; Randhir S. Kapil; Nitya Anand |
| 117-120 | OXIDATIVE PHOSPHORYIATION OF PHENOLS AND RELATED COMPOUNDS | Roger P. Napier; S. T. D. Gough |
| 121-124 | 4-PYRIDYLETHYLENE OXIDE | F. I. Carroll |
| 125-126 | 1-BROMOPHENANTHRIDINE | J. P. Casey; A. Catala Casey; F. D. Popp |
| 127-130 | 2,6-DIMETHYL-4-(MONO- AND DI-p-NITROBENZENESULFENYLMETHYLENE)-4H-PYRAN | R. A. Abramovitch; E. P. Kyba |
| 131-133 | 3,5-PYRIDINEDICARBOXYLIC ACID (Dinicotinic acid) | Bruce E. Maryanoff; Robert O. Hutchins |
| 135-138 | SYNTHESIS OF THIOKETONES AND OF TETRAARYLETHYLENES | Riaz Ahmed; Walter Lwowski |
| 139-142 | PREPARATION OF MONO, BIS, TRIS AND TETRAKIS(CHLOROMETHYL) DERIVATIVES BY PHOTOCHLORINATION OF HEXAMETHYLBENZENE | E. Henzelmann; J. Schwarcz; A. R. Frasca |
| 143-148 | SYNTHESES WITH BENZENEDIAZONIUM SALTS. DIPHENYLOCTADIENES AND TETBBPHENYLBUTANFS | R. Galli; M. Perchinunno; A. Arnone |
| 149-154 | DIRECT CHLORINATION OF SATURATED CYCLIC ETHERS USING TRICHLOROISOCYANURIC ACID | W. P. Duncan; G. D. Strate; B. G. Adcock |
| 155-157 | A FACILE SYNTHESIS OF 4-ALKYL-2,6-DINITROCHLOROBENZENES | C. S. Giam; R. C. Hall |
| 159-162 | THE PREPARATION OF 1,3-DIBROMOADAMANTANE | T. M. Gorrie; P. v. R. Schleyer |
| C | Editorial Board Page | |
| i | PREFACE | |
| 51-53 | AZIDOMETHYLDIPHENYLPHOSPHINE OXIDE | Dietmar Seyferth; Peter Hilbert |
| 55-59 | POLYARYLPYRYLIUM HEXA CHLOROANTIM ONATES | D. Frcaŝiu; Irina Elian |
| 61-70 | A VARIABLE TEMPERATURE PREPARATIVE SCALE PHOTOCHEMICAL REACTOR. CIS-DIMETHYL BICYCLO[3.2.0]HEPTANE-1,5-DICARBOXYLATE | Dennis C. Owsley; Jordan J. Bloomfield |
| 71-76 | OPTICAL RESOLUTION OF 4,6,4′,6′-TETRACHLORODIPHENIC ACID | Edward R. Atkinson |
| 77-81 | REACTION OF ENAMINES OF SOME BICYCLIC AND MONOCYCLIC KETONES WITH 2,4-DINITROCHLOROBENZENE AND 2-CHLORO-3,5-DINITROTHIOPHENE | Lars H. Hellberg; Charles C. Adams; Robert J. Milligan; Robert N. Wilke |
| 83-86 | 1,1,2,2-TETRAMETHYLCYCLOHEXANE | A. J. M. Reuvers; J. A. Jongejan; J. Klomp; H. van Bekkum |
| 87-91 | A SIMPLE PREPARATION OF 4-AMINO-2,3,5-TRICHLOROPYRIDINE | C. S. Giam; S. D. Abbott; R. C. Hall |
| 93-95 | 6,7-DIMETHOXYCARBOSTYRIL | George R. Pettit; Benjamin Stevenson; Gabriel Gever |
| 97-98 | CATALYTIC SYNTHESIS OF METAL-FREE PHTHALOCYANINE | M. V. Twigg |
| 99-102 | USE OF DIETHYL PHENYLMALONATE AS A NUCLEOPHILIC DONOR IN THE MICHAEL REACTION | Wayland E. Noland; Richard B. Hart |
| 103-107 | 3- AND 4-(7-BENZ[a]ANTHRACENYL)PHENYL-2-OXAZOLINES AND 3- AND 4-(9-ANTHRACENYL)PHENYL-2-OXAZOLINES AND THEIR HYDROCHLORIDE SALTS | F. A. Vingiello; M. P. Rorer; M. A. Ogliaruso |
| C | Editorial Board Page | |
| 1-4 | NOVEL METHODS OF PREPARATION OF 2-OXAZOLIDONES | Z. Lukasiewicz; T. Urbanski |
| 5-8 | 2-OXO-3-OXA-5-anti-6-syn-DIPHENYLBICYCLO[2.1.1]HEXANE. A gamma LACTONE FROM LEAD TETRAACETATE OXIDATION OF alpha-TRUXILLIC ACID | Donald G. Farnum; Abdol J. Mostashari |
| 9-15 | 3- AND 4-(7-BENZ[a]ANTHRACENYL)-N-BENZOYLAZIRIDINES AND 3- AND 4-(9-ANTHRACENYL)-N-BENZOYLAZIRIDINES | F. A. Vingiello; M. P. Rorer; M. A. Ogliaruso |
| 17-20 | PREPARATION AND PROPERTIES OF N-α-CARBOBENZOXY-N-IMIDAZOLE ADAMANTYLOXYCARBONYL-L-HISTIDINE | Manohar A. Tilak; Ralph Russell; Mary L. Hendricks |
| 21-25 | 1,3-DIALKYL-5,5-DIMETHYLHEXAHYDROPYRIMIDINES | H. Piotrowska; T. Urbanski; W. Bednarska |
| 27-32 | 1-THIA-3-AZACYCLOHEPTANE DERIVATIVES | Z. Olszenko-Piontkowa; T. Urbanski |
| 33-36 | AN IMPROVED SYNTHESIS OF 3,4-DIHYDRO-1H-2,1-BENZOTHIAZIN-4-ONE 2,2-DIOXIDE | J. G. Lombardino; N. W. Treadway Jr. |
| 37-38 | HEXALOCYCLOPENTANTADIENES IV. SYNTHESIS AND PYROLYSIS OF OCTABROMO-3a,4,7,7a-TETRAHYDROMETHANOINDENE-1,8-DIONE | R. G. Pews |
| 39-44 | THE (±)-p-MENTHANE-2,5-DIONES AND THE (±)-2-t-BUTYL-5-METHYL-1,4-CYCLOHEXANEDIONES | Robert D. Stolow; Robert R. Krikorian |
| 45-46 | 2-BENZYLQUINOXALINE | K. C. Bass; P. Nababsing |
| 47-50 | VINYLDIAZOMETHANE | John Hooz; Hiromichi Kono |
| C | Editorial Board Page | |
| 245-248 | IMPROVED PREPARATIONS OF CYCLONONEN-3-OL, CYCLONONEN-3-ONE, CYCLONONANONE AND CYCLONONANOL | Goverdhan Mehta |
| 249-252 | ARYLGLYOXYLIC ESTERS, FRIEDEL-CRAFTS REACTION | R. G. Micetich |
| 253-254 | NOTICE TO AUTHORS | |
| 255-258 | AN IMPROVED SYNTHESIS OF L-HISTIDINE BENZYL ESTER | A. M. Felix; D. P. Winter |
| 259-263 | THE REACTION OF 2,3-DICHLORO-1,4-NAPHTHOQUINONE WITH p-NITROBENZHYDRAZIDE1 | F. I. Carroll; H. Wayne Miller |
| 265-269 | 4-(ISOPROPYLIDENE)-2-(2′-PHENYLETHYL)-5-OXAZOLONE | D. N. Reinhoudt; P. R. M. van der Kamp |
| 271-273 | 2,3-DIAZABICYCLO[2.2.1]-2-HEPTENE M-OXIDE | Robert C. Kerber; Thomas J. Ryan |
| 275-279 | 1-ACYL- AND 1,1-DIACYL-2,2-DIMETHYLHYDRAZINES | E. A. Sedor; R. E. Freis; H. J. Richards |
| 281-283 | CORYPALLINE | A. Brossi; J. O'brien; S. Teitel |
| 285-289 | SYNTHESIS OF METHOXYPYRIDYL PHENYL KETONES VIA PYRIDYLLITHIUM COMPOUNDS | Ellis V. Brown; M. B. Shambhu |
| 291-294 | 1-TERT-BUTYL-1,3-PROPANEDIOL | R. O. Hutchins; Frank J. Dux |
| 295-296 | METHYL γ-RESORCYLATE | Arthur Mendel |
| 297-303 | AN IMPROVED SYNTHESIS OF INDOLE-3-CARBOXYLIC ACIDS | A. S. Katner |
| 305-308 | 2,4-DIETHYLQUINOLINE - AN EXTENSION OF THE COMBES SYNTHESIS | P. A. Claret; A. G. Osborne |
| 309-310 | CONVENIENT SYNTHESIS OF 4-NITROBENZOYL CHLORIDE | Pankaja K. Kadaba |
| 313-315 | MICRO-DISTILLATION OF ORGANIC LIQUIDS | Kenn E. Harding; Robin B. Kinnel |
| 317-319 | A SOLVENT PAIR RECRYSTALLIZATION APPARATUS FOR GROWING SINGLE CRYSTALS | J. N. Brown; L. M. Trefonas |
| 321-325 | ANHYDRIDE FORMATION WITH THIONYL CHLORIDE | Jerry M. Adduci; Rene S. Ramirez |
| 325-329 | MONO- AND DIKETONES FROM ALKYLTIN CARBOXYLATES | Bernard R. Laliberte; Helmut F. Reiff; Wenzel E. Davidsohn |
| C | Editorial Board Page | |
| 79-81 | THE NITRATION OF DIPHENYLCYCLOPROPENONE | C. W. Bird; A. F. Harmer |
| 83-87 | THE PREPARATION OF 1,2:5,6-Di-O-Cyclohexylidene-α-D-Gulofuranose | Susanne L. von Schuching; Glenn H. Frye |
| 89-92 | REDUCTION OF 1,1-DICHLOROBENZOCYCLOBUTENES | David J. Hart; Harold Hart |
| 93-100 | THE RESOLUTION OF (±)-3-METHYLCYCLOHEXANONE AND (±)-3-tert-BUTYLCYCLOHEXANONE | G. Adolphen; E. J. Eisenbraun; G. W. Keen; P. W. K. Flanagan |
| 101-115 | N,N′-DIALKYLATION OF SULFONYLAMIDES OF p-PHENYLENEDIAMINES | T. Doornbos; J. Strating |
| 117-119 | SOME NITRO-1,2,3-TRIAZOLES | T. E. Eagles; M. A. Khan; B. M. Lynch |
| 121-124 | ARYL N, N-DIFLUOROSULFONAMIDES1 | Travis E. Stevens; Royland D. Shoults |
| 125-128 | 1,1-DIARYLHYDRAZINES | J. -P. Anselme; N. Koga |
| 129-135 | cis- AND trans-N,N′-DIMETHYL-1,4-CYCLOHEXANEBIS (METHYLAMINE) BY METHYLATION OF THE BENZALDEHYDE IMINES | J. Richard Hall; Thomas A. Hollingworth Jr. |
| 137-139 | ALKYLATION AND OXIDATION OF DIARYLACETONITRILES | Stuart S. Kulp |
| 141-144 | KETALIZATION OF 5-KETO STEROID ESTERS1 | David M. Piatak; Eliahu Caspi |
| 145-147 | PREPARATION OF N-BENZOYL-N-METHYLPHENYLGLYCINE | Donald F. McLaen |
| 149-156 | AN IMPROVED SYNTHESIS OF KETIMINES | E. P. Kyba |
| C | Editorial Board Page | |
| 1-4 | UNSYMMETRICALLY ALKOXYLATED DISILAZANES | R. E. Goldsberry; W. E. Weibrecht |
| 5-10 | PREPARATION OF PHOSPHANILIC ACID (p-AMINOBENZENEPHOSPHONIC ACID) | O. Grummitt; N. Vourlogianes; J. Mehaffey; R. Tebbe |
| 11-17 | SOME DERIVATIVES OF 3-CARBOXYMETHYLSYDNONE | F. H. C. Stewart |
| 19-23 | THE SYNTHESIS OF TRICHLOROTRIS (4-BIPHENYLYL-1-NAPHTHYLPHENYL PHOSPHINE) RHODIUM(III). A NEW OCTAHEDRAL COMPLEX | Robert E. Harmon; Jack L. Parsons; S. K. Gupta |
| 25-27 | PROCEDURE FOR THE HOMOGENEOUS CATALYTIC HYDROGENATION OF α, β-UNSATURATED NITRO COMPOUNDS USING TRIARYLPHOSPHINE-RHODIUM COMPLEXES | Robert E. Harmon; Jack L. Parsons; S. K. Gupta |
| 29-31 | DIAZEPINES. VIII. 3,8-DINITRO-11H-DIBENZO[c, f] [1, 2]-DIAZEPINE-5-OXIDE | A. Catala Casey; F. D. Popp |
| 33-36 | THE PREPARATION OF A FORMALDEHYDE ADDUCT OF 3-DIMETHYLAMINO-2,2-DIMETHYLPROPIONALDEHYDE | Lloyd D. Taylor; Paul McLaughlin; Martin Mach |
| 37-43 | A CONVENIENT SYNTHESIS OF 2-BENZYLNAPHTHALENE AND 2-BENZYL-1,2,3,4-TETRAHYDRONAPHTHALENE | R. G. Melton; E. J. Eisenbraun; P. W. K. Flanagan; M. C. Hamming |
| 45-50 | GRADIENT ELUTION CHROMATOGRAPHY OF S-PALMITYL COENZYME A* | Steven S. Kuwahara |
| 51-52 | DL-4-ACETAMIDO-4-HYDROXY-2-BUTENOIC ACID γ-LACTONE | Joan A. Gratz; C. E. Cook; Monroe E. Wall |
| 53-58 | PREPARATION OF 4,4-BIS(DIFLUORAMINO)CYCLOHEXANONE AND 5,5-BIS(DIFLUORAMINO)-2-AZACYCLOHEPTANONE | Travis E. Stevens |
| 59-63 | ALKYLATION OF 2,6-DI-TERT-BUTYLPHENOL IN DIMETHYL SULFOXIDE | Eugene R. Wagner |
| 65-67 | 2,5-BIS-(2-PYRROLYL)-1-PYRROLINES | V. Bocchi; G. P. Gardini |
| 69-70 | SYNTHESIS OF 4,4′-DIHYDROXY-3,3′,5,5′-TETRA-t-BUTYLBENZOPHENONE | Mary K. Conner; E. Legoff |
| 71-74 | 5,6-DIHYDRO-4H-1,3-OXAZINES BY A MODIFICATION OF THE TILLMANNS-RITTER PROCEDURE | Samuel P. McManus; John T. Carroll |
| 75-78 | 3-NITRO-1,3,5-HEXATRIENE | Charles W. Spangler; Ronald P. Hennis |
| C | Editorial Board Page | |
| 221-224 | SANDMEYER TYPE REACTION IN DIMETHYL SULFOXIDE | Michio Kobayashi; Eiichi Yamada; Mikio Matsui; Nobumasa Kobori |
| 225-228 | PREPARATION OF TOSYLATES OF PHENOLS AND ACIDIC ALCOHOLS | Stanley E. Wentworth; Patrick L. Sciaraffa |
| 229-233 | 2-METHOXY-1,3-BUTADIENE | L. J. Dolby; K. S. Marshall |
| 235-238 | 2,5,5-TRIMETHYL-2-OXAZOLINE | S. P. McManus; J. T. Carroll; P. M. Grohse; C. U. Pittman Jr. |
| 239-241 | ACRYLYLOXYMETHYL METHYL SULFIDES | R. L. Harville; Samuel F. Reed Jr. |
| 243-248 | PREPARATION OF 3-PHENYL-1,2-CYCLOPROPANEDICARBOXYLIC ACIDS | S. Wawzonek; A. R. Zigman |
| 249-251 | α-ACETAMIDO-β-(1-AZULYL) PROPIONIC ACID | Arthur G. Anderson Jr.; Robert C. Rhodes |
| 253-254 | N-METHYL OCTAHYDROCARBAZOLE | E. Schmitz; H. Fechner |
| 255-258 | 1,2,5-THIADIAZOLID-3,4-DIONE-1-OXIDE | Marvin Carmack; Ian W. Stapleton; Richard Y. Wen |
| 259-261 | cis-1,2-VINYLENEBIS (DIPHENYLPHOSPHINE) | J. P. Mitchener; A. M. Aguiar |
| 263-266 | PREPARATION OF 2-BENZYLPHTHALIMIDINE VIA INTRAMOLECULAR FRIEDEL-CRAFTS RING CLOSURE OF N,N-DIBENZYLCARBAMOYL CHLORIDE | D. E. Rivett; J. F. K. Wilshire |
| 267-269 | β- AND δ-TRUXINIC ACIDS | M. Freedman; Y. Mohadger; J. Rennert; S. Soloway; I. Waltcher |
| 271-277 | γ-ARYL-γ-AMINO ACIDS | V. Bocchi; G. P. Gardini |
| 279-281 | 3-NITRO-7-CHLOROQUINOLINE | Ned D. Heindel; Stephen A. Fine |
| 283-285 | AN IMPROVED SYNTHESIS OF METHYLENECYCLOPROPANE | I. S. Krull; D. R. Arnold |
| 287-303 | THE COMPLETE N-ALKYLATION OF 1,4-DIAMINO-2,5-DIBROMOBENZENE AND OF 1,4-DIAMINO-2,5-DIMETHOXYBENZENE | T. Doornbos; J. Strating |