Organic Preparations and Procedures International (1969-2010)

Volume 42, Issue 6 (2010)

503-555Recent Progress in the Use of Vilsmeier-Type ReagentsWeike Su; Yiyi Weng; Ling Jiang; Yanyan Yang; Linyao Zhao; Zhiwei Chen; Zhenhua Li; Jianjun Li
557-5634(1H)-Quinolinones by a Tandem Reduction-Addition-Elimination ReactionRichard A. Bunce; Baskar Nammalwar

Volume 42, Issue 5 (2010)

387-4311,3-Dipolar Cycloadditions of Nitrones to Heterosubstituted Alkenes. Part 1: Oxa and Aza-substituted AlkenesThanh Binh Nguyen; Arnaud Martel; Catherine Gaulon; Robert Dhal; Gilles Dujardin
433-465Recent Synthetic Approaches to 1H- and 2H-Indazoles. A ReviewNaděžda Cankařová; Jan Hlaváč; Viktor Krchňák
467-477Chemistry of 3-Alkynals. A ReviewRonald Blankespoor
479-484A Practical and Efficient Vilsmeier Synthesis of 3-Chloroindole-2-carboxaldehydesZ. H. Li; Z. R. Hu; R. E. Chen; W. K. Su
485-489Preparation of 4,6-Diarylindazole Derivatives in Ionic Liquid under Solvent-free ConditionsJavad Safaei-Ghomi; Mahdi Taheri; Mohammad Ali Ghasemzadeh
490-4938-Chloro- and 5,8-Dichloro-1-naphthoic AcidsJianhong Chen; Valerie J. Smith; John W. Huffman
494-498Facile One-Pot Synthesis of Tetrahydrobenzo[a]xanthene-11-one and Aryl-14H-dibenzo[a.j]xantheneRamin Ghorbani-Vaghei; Seyedeh Mina Malaekehpoor
499-502A Simple Synthesis of 8-Methoxy-1-tetraloneElvia V. Cabrera; Ajoy K. Banerjee

Volume 42, Issue 4 (2010)

285-362Acidic Bronsted Ionic LiquidsAbdol R. Hajipour; Fatemeh Rafiee
363-371Bismuth(III) Triflate Catalyzed Allylation of Cyclic Acetals and Dithianes Followed by in situ Derivatization to Generate Highly Functionalized EstersScott W. Krabbe; Matthew J. Spafford; Ram S. Mohan
373-378A Practical Route for the Preparation of Aromatic trans-β-NitroolefinsG. Groszek
379-385Aromatization of 1,3-Cyclohexanediones Mediated by bis-(Trichloromethyl) Carbonate/DMF SystemX. R. Liang; F. Shi; R. E. Chen; W. K. Su

Volume 42, Issue 3 (2010)

191-283Synthesis of 2′-C-Branched NucleosidesNan-Sheng Li; Jun Lu; Joseph A. Piccirilli

Volume 42, Issue 2 (2010)

111-132Progress towards the Synthesis of Sordarin and its AnalogsHuan Liang; Marco Ciufolini
133-141Regioselective Nucleophilic Aromatic Substitution of Benzo[c][2,7]naphthyridinesCharles F. Nutaitis; Katrin Przyuski; Vincent Ross
143-150Synthesis of Various 2,8-Cyclooctadiene-1,2-dicarboxylatesAyse Uzgoren-Baran; Nazan Tunoglu; Gurol Okay
151-160An Improved Non-chromatographic Scale-up Synthesis of a New 1,6,7,8-Substituted-4-oxo-1,4-dihydroquinoline-3-carboxylic Acid as a Potent Bacterial Topoisomerase InhibitorXun Li; Scott Youells; Ronald K. Russell; Armin Roessler; Tobias Schmid; Roger Faessler; Michele A. Weidner-Wells; Eugene B. Grant; Mark J. Macielag
161-167Practical and Efficient Synthesis of 4,4′-Dihydroxy-3,3′-dinitrodiphenyl Ether and 1,3-bis(4-Hydroxy-3-nitrophenoxy)benzene in Aqueous Alkaline MediumMitsutaka Imoto; Motonori Takeda; Akihiro Tamaki; Hisaji Taniguchi; Kazuhiko Mizuno
169-173Efficient Iodine-catalyzed Synthesis of 3-Aryl 4(3H)-quinazolinonesMin Wang; Zhi-Guo Song; Ting-Ting Zhang
175-182Facile and Mild Synthesis of bis(3-Indolyl)methanesR. Ghorbani-Vaghei; S. M. Malaekehpoor
183-185A New Route for the Synthesis of Ozagrel HydrochlorideChenglong Yu; Baohai Zhao; Yihong Zhao; Jimao Lin
187-190Expedient Preparation of 4,6-Dihalo-3-arylisobenzofuran-1(3H)-ones from 3,5-Dihalo-N-ethylbenzamidesLynn M. Bradley; Carleton G. Collins; Erica R. Tabakin; David A. Hunt

Volume 42, Issue 1 (2010)

1-69Arylcyclopropanes: Properties, Synthesis and Use in Medicinal ChemistryAlexandre Gagnon; Martin Duplessis; Lee Fader
71-826-Nitro-1,2,3,4-tetrahydroquinoline-4-carboxylic Esters and 7-Nitro-3,4-dihydroquinoxaline- 1(2H)-carboxylic Esters by a Tandem Reductive Amination-SNAr ReactionRichard A. Bunce; James E. Schammerhorn
83-93Tetrahydronaphthalene Derivatives by Amberlyst® 15-Promoted Friedel-Crafts CyclizationsRichard A. Bunce; Andrew N. Cox
95-102Ionic Liquid 3-Methyl-1-sulfonic Acid Imidazolium Chloride as a Novel and Highly Efficient Catalyst for the Very Rapid Synthesis of bis(Indolyl)methanes under Solvent-free ConditionsMohammad Ali Zolfigol; Ardeshir Khazaei; Ahmad Reza Moosavi-Zare; Abdolkarim Zare
103-106An Efficient Methodology for the Synthesis of 1-(Trimethylammoniummethyl)cyclohexaneacetic Acid Iodide: A Trimethylammonium Iodide Salt of GabapentinMorshed A. Chowdhury; Peter A. Smith; Edward E. Knaus
107-109A Practical Synthesis of 2-Bromo-6-methoxynaphthaleneWei-Ming Xu; Hong-Qiang He

Volume 41, Issue 6 (2009)

429-478Recent Advances in Stereoselective Synthesis and Application of β-Amino AcidsBrad E. Sleebs; T. T. Van Nguyen; Andrew B. Hughes
479-514Advances in the Synthesis of 5- and 6-Substituted Uracil DerivativesJavier I. Bardagí; Roberto A. Rossi
515-532Synthesis of Cytosine Derivatives and Study of their Alkylation under Mild ConditionsDilip R. Birari; Maruti G. Ghagare; Muddassar A. Kazi; Sandeep M. Bagul; Bhausaheb K. Ghotekar; Raghunath B. Toche; Madhukar N. Jachak
533-538A Convenient Method for the Synthesis of 3,5,6-Trisubstituted-2-chloropyridines with bis-(Trichloromethyl) CarbonateZ. H. Li; B. Hong; W. K. Su
539-541A Practical Synthesis of 2-Fluoro-4-bromobiphenylYa-Yu Qiu; Haining Gu; Peng-Fei Zhang; Wei-Ming Xu
543-548An Efficient Procedure for the Synthesis of Some New 9-Hydroxy-6-methyl-7H-benzo[c] chromene-7-one DerivativesA. Zonouzi; Z. Izakian; M. Biniaz

Volume 41, Issue 5 (2009)

331-358Synthesis of TerphenylsLuis A. Adrio; José M. Antelo Míguez; King Kuok Hii
359-383Syntheses of the Crocacins. A ReviewRodrigo B. Andrade
385-418Recent Progress in the Synthesis of 2,3-DihydrobenzofuransFerruccio Bertolini; Mauro Pineschi
419-421A Practical Synthesis of 2′-Fluoro- 4′-hydroxyacetophenoneXiao-Bo Zhang; Qun Lu; Wei-Ming Xu
423-427A Novel and Practical Synthesis of 2-Amino-5-hydroxypropiophenoneXiao-Dong Xiong; Wen-Xue Chen; Yun-Yan Kuang; Fen-Er Chen

Volume 41, Issue 4 (2009)

253-290Recent Advances in the Synthesis of Pyrazoles. A ReviewSantos Fustero; Antonio Simón-Fuentes; Juan F. Sanz-Cervera
291-299Potassium Fluoride as an Efficient and Reusable Reagent for the Synthesis of N,N-Dialkylsulfonamides via Aza-Conjugate Addition Reaction Under Microwave IrradiationAlireza Hasaninejad; Abdolkarim Zare; Abolfath Parhami; Ahmad Reza Moosavi-Zare; Raheleh Bargebid; Mohammad Hassan Beyzavi; Ali Khalafi-Nezhad; Azam Arghoon; Maria Merajoddin; Sayyed Ali Moosavi; Abdoreza Dara; Mohsen Shekouhy
301-307Preparation of Mono Boc-Protected Unsymmetrical DiaminesHongbo Li; Meng-an Hao; Liping Wang; Wu Liang; Kai Chen
309-314An Efficient Synthesis of 1,2,6,7-Tetrahydro-8H-indeno[5,4-b]furan-8-oneBo Wang; Lijuan Zhang; Kaiyong Fu; Yu Luo; Wei Lu; Jie Tang
315-321Three-Component Mannich Reaction of Aromatic Ketones, Aldehydes and Amines Catalyzed by Reusable Aluminium MethanesulfonateMin Wang; Zhi-Guo Song; Heng Jiang
323-326New Synthetic Routes for the Preparation of 2-Amino-3-hydroxy-1,4-naphthoquinoneAcácio I. Francisco; Annelise Casellato; Maria D. Vargas
327-330Convenient Synthesis of Wogonin, A Flavonoid Natural Product with Extensive Pharmacological ActivityZhi-Yu Li; Xin Cao; Xin Wang; Qing-Long Guo; Qi-Dong You

Volume 41, Issue 3 (2009)

173-210Properties, Preparation and Synthetic Uses of Amine N-Oxides. An UpdateDavid Bernier; Ulrike K. Wefelscheid; Simon Woodward
211-215An Improved One-pot Procedure for the Preparation of β-Lapachone and nor-β-Lapachone, Two Potent Drug PrototypesSabrina Baptista Ferreira; Carlos Roland Kaiser; Vitor Francisco Ferreira
217-227Synthesis and Structure of Tetratosyl Bora Derivatives of Resorcinarenes From l-Proline and l-ProlinolBarbara Gawdzik; Alicja Wzorek; Jochen Mattay; Waldemar Iwanek
229-236Fries Rearrangement of Anilides in the Presence of Phosphorus Pentoxide in Methanesulfonic AcidBabak Kaboudin; Yaghoub Abedi
237-242Oxidative Aromatization of 1,3,5-Trisubstituted Pyrazolines Using Hydrogen Tetrachloroaurate as Catalyst Under an Oxygen AtmosphereYunkui Liu; Dajie Mao; Shaojie Lou; Jianqing Qian; Zhen-Yuan Xu
243-247New and Convenient Syntheses of 1-Amino-1-phenylbutane from n-ButylbenzeneLingaiah Nagarapu; Satyender Apuri; Chandana Gaddam; Rajashakar Bantu
249-252A Novel Synthesis of PendimethalinXiao-Hua Du; Da-Wei Luo; Zhen-Yuan Xu

Volume 41, Issue 2 (2009)

93-141Recent Developments in the Use of bis-(Trichloromethyl) Carbonate in SynthesisWeike Su; Yiyi Weng; Cun Zheng; Ying Zhang; Fei Shi; Bin Hong; Zhiwei Chen; Jianjun Li; Zhenhua Li
143-147Unexpected Incorporation of Bromine at a Non-anomeric Position during the Synthesis of an O2-Glycosylated DiazeniumdiolateJoseph E. Saavedra; Keith M. Davies; Joseph J. Barchi Jr.; Larry K. Keefer
147-152Syntheses of C-1 Axial Derivatives of l-MentholDebra K. Dillner
152-155A Practical Synthesis of α-Asarone via Iodine-catalyzed Isomerization of α/β-AsaroneGuangyu Xu; Chang Liu; Wei Zhang; Gaolei Zuo
156-161Intramolecular Cyclization of 2′-Aminochalcones by Halomethyleniminium Salts Derived from BTC/DMFZhen-Hua Li; Cun Zheng; Ren-Er Chen; Weike Su
162-164A Practical Synthesis of 5,5′-Methylene-bis(benzotriazole)Haining Gu; Biao Yu; Peng-Fei Zhang; Wei-Ming Xu
164-168A Practical Synthesis of (7-Methoxynaphth-1-yl)acetic AcidJia-Deng Tang; Jun-Da Cen
168-171A Simple and Convenient Synthesis of TriprolidineG. Venkateswara Rao; B. Narayana Swamy; P. Hareesh Kumar; G. Chandrasekara Reddy

Volume 41, Issue 1 (2009)

1-68Recent Progress in Three-Component Reactions. An UpdateM. Syamala
69-75First Vilsmeier-Haack Synthesis of Flavones using bis-(Trichloromethyl) Carbonate/DimethylformamideW. K. Su; X. Y. Zhu; Z. H. Li
77-82One-Pot Synthesis of Tetrahydrobenzo[b]pyran Derivatives Catalyzed by Amines in Aqueous MediaLi-Qin Yu; Fei Liu; Qi-Dong You
83-87Thermal and Photochemical Approaches to the Synthesis of vic-Tricarbonyl Compounds from 4-Hydroxyquinolin-2(1H)-onesJia-Hai Ye; Zhichun Qin; Bin Zhou; Wenchao Zhang; Guirong Tian; Lei Yuan; Jian-Hua Xu
87-91Iodination of Alcohols using Triphenylphosphine/Iodine in Ionic Liquid under Solvent-Free ConditionsAbdol Reza Hajipour; Majid Mostafavi; Arnold E. Ruoho

Volume 40, Issue 6 (2008)

CEditorial Board Page
505-542α-, β-,γ- AND ω-CYCLOPROPYLPHOSPHONATES. PREPARATION AND BIOLOGICAL ACTIVITYAbed Al Aziz Al Quntar; Valery M. Dembitsky; Morris Srebnik
543-550A SIMPLE AND EFFICIENT PROCEDURE FOR THE BECKMANN REARRANGEMENT OF OXIME USING bis-(TRICHLOROMETHYL) CARBONATE/DMFW. K. Su; Y. Zhang; J. J. Li; P. Li
551-556SYNTHESIS OF 4-CYANO- AND 5-AMINOPYRAZOLES AND DEAMINATION OF 5-AMINOPYRAZOLESR. B. Toche; M. A. Kazi; M. N. Jachak
557-5614-IODO-6-METHOXYQUINOLINEAlex C. Bissember; Martin G. Banwell
561-566A SHORT SYNTHESIS OF THE NATURALLY OCCURRING 2,3,3′,4,4′,5,5′-HEPTACHLORO- (“Q1”) AND HEPTABROMO-1′-METHYL-1,2′-BIPYRROLESLiangfeng Fu; Gordon W. Gribble
566-571SYNTHESIS OF SUBSTANCES RELATED TO FLUTICASONE PROPIONATEJin Zheng; Qinglin Lai; Yiru Dai; Qingjie Zhao; Jingshan Shen
572-574AN EFFICIENT ONE-STEP METHOD FOR THE LARGE-SCALE SYNTHESIS OF 2,4-THIAZOLIDINEDIONEGe Meng; Zhen-Yu Li; Mei-Lin Zheng
574-579AN IMPROVED APPROACH TO N-SUBSTITUTED MALEIMIDES AND PHTHALIMIDES BY MICROWAVE-PROMOTED MITSUNOBU REACTIONChristoph D. Mayer; Marcus Kehrel; Franz Bracher
579-585A NOVEL ACCESS TO SOME 1,4-DICHLOROISOQUINOLINES FROM PHENACYL AZIDESR. E. Chen; X. H. Zhou; W. H. Zhong; W. K. Su
586-589SYNTHESIS OF ARYL 14H-DIBENZO[A,J]XANTHENES USING ZIRCONIUM(IV) OXIDE CHLORIDE AS A CATALYSTElaheh Mosaddegh; Mohammad Reza Islami
591-596INDEXES

Volume 40, Issue 5 (2008)

CEditorial Board Page
411-445TURNING THE CORNER: RECENT ADVANCES IN THE SYNTHESIS OF THE WELWITINDOLINONESLauren E. Brown; Joseph P. Konopelski
447-455IMPROVED THREE-COMPONENT LEWIS ACID-FREE APPROACH FOR THE SYNTHESIS OF PROTECTED RACEMIC CYANOHYDRINSG. Kumaraswamy; K. Ankamma
457-463A GREEN SOLVENTLESS PROTOCOL FOR THE SYNTHESIS OF N-SULFONYLIMINES IN THE PRESENCE OF SILICA SULFURIC ACID AS AN EFFICIENT, HETEROGENEOUS AND REUSABLE CATALYSTAbdolkarim Zare; Alireza Hasaninejad; Mohsen Shekouhy; Ahmad Reza Moosavi Zare
465-467A PRACTICAL SYNTHESIS OF 4-HYDROXYETHYL-2,3-DIHYDROBENZOFURANHaining Gu; Wei Ming Xu
467-470AN IMPROVED SYNTHETIC PROCESS FOR YF-6, A PROMISING ANTI-HBV DRUG CANDIDATESai Hong Jiang; Peng Lu; Xiao Zhong Fu; Yu She Yang; Ru Yun Ji
471-477SIMPLE AND RAPID PROCEDURE FOR THE SYNTHESIS OF SOME NEW 2H-CHROMENESA. Zonouzi; M. Sadeghi Googheri; P. S. Miralinaghi
477-481AN EFFICIENT, ONE-POT SYNTHESIS OF ALKYL ARYLSELENOFORMATES USING THE ZINC-RUTHENIUM CHLORIDE SYSTEM IN AQUEOUS MEDIABarahman Movassagh; Ameneh Tatar
481-487SYNTHESIS OF SUBSTITUTED AROMATIC COMPOUNDS USING BTC/DMF AS VILSMEIER REAGENTW. K. Su; Z. C. Lu; X. X. Zhang
487-489AN EFFICIENT SYNTHESIS OF 3, 5-bis(2-CYANOISOPROPYL)TOLUENEYu-Hua Mei; Yu Luo; Wei Lu
490-493A PRACTICAL SYNTHESIS OF 4-ACETYL-2,3,4,5-TETRAHYDRO-1H-1,4-BENZODIAZEPINEQingjie Zhao; Haihong Li; Fuqiang Zhu; Hongli Guo; Jingshan Shen
493-498SYNTHESIS OF 3-(2-ARYL-1H-INDOL-3-YL)-4-AROYL-5-ARYLISOXAZOLINESVijai N. Pathak; Meenakshi Jain; Anjali Tiwari
499-504SYNTHESIS OF BIVALENT ORGANOPHOSPHORUS COMPOUNDS AS ACETYLCHOLINESTERASE INHIBITORSGuoquan Yang; Qianfei Zhao; Yonghong Li; Huizhu Yuan; Xiangdong Mei; Jun Ning

Volume 40, Issue 4 (2008)

CEditorial Board Page
317-363RECENT PROGRESS IN THE SYNTHESIS OF LABDANE DITERPENOIDS. A REVIEWBahlul Z. S. Awen; Masato Nozawa; Hisahiro Hagiwara
365-3785-CARBETHOXY- AND 5-ACETYLPYRAZOLES AS PRECURSORS FOR THE SYNTHESIS OF SOME NOVEL 1-p-CHLOROPHENYLPYRAZOLE-3-CARBONITRILESHatem M. Gaber
379-384SYNTHESIS OF (+)-9-O-DESMETHYL-α-DIHYDROTETRABENAZINE, PRECURSOR FOR THE HIGH AFFINITY VMAT2 IMAGING PET RADIOLIGAND [11C]-(+)-α-DIHYDROTETRABENAZINEKarl G. Boldt; George A. Brine; Ken Rehder
385-391AN EFFICIENT AND CHEMOSELECTIVE SYNTHESIS OF ALDEHYDE 1,1-DIACETATES USING MORPHOLINIUM BISULFATE AS A BRÖNSTED ACIDIC IONIC LIQUID UNDER SOLVENT-FREE CONDITIONSAbdol Reza Hajipour; Zahra Nasreesfahani; Arnold E. Ruoho
391-394FACILE SYNTHESIS OF ANXIOLYTIC BUSPIRONEJie Mou; Zhi-Min Zong; Xian-Yong Wei
395-398HIGH-YIELD SYNTHESIS OF ANDROST-4-ENE-3,6,17-TRIONE AND ANDROST-4-ENE-3B,6B,17B- TRIOLHuyue Zhang; Guanghui Deng; Zhuibai Qiu
399-404A SIMPLE AND CONVENIENT METHOD FOR THE SYNTHESIS OF PHOSPHOROAMIDATES AND PHOSPHOROAMIDOTHIOATES UNDER SOLVENT-FREE CONDITIONBabak Kaboudin; Mansoureh Karimi; Hazegh Zahedi
405-410FACILE AND EFFICIENT SYNTHESIS OF ISOLONGIFOLENONEShifa Wang; Aijun Zhang

Volume 40, Issue 3 (2008)

CEditorial Board Page
215-291RECENT APPLICATIONS OF ARYNE CHEMISTRY TO ORGANIC SYNTHESIS. A REVIEWRoberto Sanz
293-301AN IMPROVED COPPER-CATALYZED CROSS-COUPLING REACTION OF ALKYL TRIFLATES WITH PRIMARY ALKYL GRIGNARD REAGENTSShifa Wang; Aijun Zhang
303-306CONVENIENT TREMETHYLSILYLATION OF HYDROXY GROUPS WITH HEXAMETHYLDISILAZANE UNDER SOLVENT-FREE CONDITIONSAmin Rostami; Ardeshir Khazaei; Marjan Mahboubifar; Sadegh Rahmati
307-310IMPROVED PROCEDURE FOR THE PREPARATION OF 1-(2-PHENETHYL)-4-PIPERIDONEH. Fakhraian; M. Babaei Panbeh Riseh
311-315CONVENIENT SYNTHESIS OF 1-ACETYL-2,2-DIMETHYL-3-ARYLCYCLOPROPANESLakshmi Muthusubramanian; Rajat B. Mitra

Volume 40, Issue 2 (2008)

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107-161TOTAL SYNTHESES OF PANCRATISTATIN. A REVIEWMadhuri Manpadi; Alexander Kornienko
163-200TARTARIC ACID AND ITS O-ACYL DERIVATIVES. PART 2. APPLICATION OF TARTARIC ACID AND OF O-ACYL TARTARIC ACIDS AND ANHYDRIDES. RESOLUTION OF RACEMATESLudwik Synoradzki; Urszula Bernaś; Pawel Ruśkowski
201-204IMPROVED SYNTHESIS OF 11-ACETOXY-8α-DRIMANOLSudhakarrao Vadapalli; Charles T. Kane Jr.
204-208AN IMPROVED SYNTHESIS OF ETHYL 5-CHLORO-4-FLUORO-1H-INDOLE-2-CARBOXYLATEFrancesco Piscitelli; Giuseppe La Regina; Romano Silvestri
209-213IMPROVED PROCEDURE FOR THE SYNTHESIS OF (2R)-N-PROPENOYLBORNANE-2,10-SULTAMJoydev K. Laha

Volume 40, Issue 1 (2008)

CEditorial Board Page
1-65APPLICATION OF CLAY CATALYSTS IN ORGANIC SYNTHESIS. A REVIEWSujaya Dasgupta; Béla Török
67-91SYNTHESIS OF CONAGENIN AND α-METHYLSERINE. A REVIEWKeiji Nakano; Hiyoshizo Kotsuki; Yoshiyasu Ichikawa
93-96REGIOSELECTIVE TRANSFER OF THE PRENYL ANION IN THE TOTAL SYNTHESIS OF (±)-SHIKONINDe-Feng Xu; Li-Ming Zhao; Zhi-Qiang Mao; Shao-Shun Li
97-101MICROWAVE-ASSISTED SYNTHESIS OF ERYTHROMYCIN DERIVATIVES ON SODIUM ACETATE-DOPED CALCIUM CHLORIDEKai Bao; Wei-Ge Zhang; Ying-Wei Qu; Chuan-Liang Zhang; Liang Tian; Mao-Sheng Cheng
101-105IODINE AS AN EFFICIENT CATALYST FOR THE SYNTHESIS OF BENZIMIDAZOLES AND IMIDAZOLINES FROM PRIMARY ALCOHOLS AND DIAMINESYi-Ming Ren; Chun Cai

Volume 39, Issue 6 (2007)

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523-559TRANSITION METAL-CATALYZED HYDROSILYLATION OF CARBONYL COMPOUNDS AND IMINES. A REVIEWSilvia Díez-González; Steven P. Nolan
561-590PREPARATION AND APPLICATION OF CYCLOPROPYLIMINES IN ORGANIC SYNTHESIS. A REVIEWAlberto Soldevilla; Diego Sampedro
591-602SOLID-PHASE SYNTHESIS OF DIFLUOROBENZIMIDAZOLES AND DIFLUORO-2-QUINOXALINOLSYafei Ji; Xianyong Wei
603-608IMPROVED SYNTHESIS OF 2-CHLORO- AND 2, 9-DICHLORO-1, 10-PHENANTHROLINESA. Paul Krapcho; Jennifer Brett Lanza
608-611FERRIC CHLORIDE-CATALYZED REDUCTIVE HALOGENATION OF CARBONYL COMPOUNDS TO BROMIDES AND IODIDESZhifang Li; Chunqi Sheng; Chengjun Yang; Huayu Qiu
611-615PREPARATION OF NOVEL QUINO[3, 4-C]-, QUENO[4, 3-C], QUINO[5, 6-C]-, QUINO[6, 5-C]-, AND QUINO[7, 8-C][2, 7]NAPHTHYRIDINECharles F. Nutaitis; Kimberly Smith
616-6203-CARBOXYPYRIDINIUM TRIFLUOROACETATOCHROMATE AND 3-CARBOXYPYRIDINIUM TRICHLOROACETATOCHROMATE, TWO NEW AND EFFICIENT REAGENTS FOR THE OXIDATION OF ALCOHOLS, BENZYLIC HYDROCARBONS AND POLYCYCLIC AROMATIC COMPOUNDSFatma Aydin; Recep Ozen

Volume 39, Issue 5 (2007)

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417-446o-AMINOMETHYL DERIVATIVES OF PHENOLS. PART 2. BENZOXAZINES AND DIBENZYL AMINES: PROPERTIES, STRUCTURE, SYNTHESIS AND PURIFICATIONKrzysztof Bujnowski; Agnieszka Adamczyk; Ludwik Synoradzki
447-494SULFANYLATION REACTIONS OF CARBONYL COMPOUNDS AND CARBOXYLIC ACID DERIVATIVES EMPLOYING SULFUR ELECTROPfflLES. A REVIEWBlanka Wladislaw; Liliana Marzorati; Claudio Di Vitta
495-502ONE-POT SYNTHESIS OF 3-FORMYLCHROMONES FROM bis-(TRICHLOROMETHYL) CARBONATE/DMFW. K. Su; Z. H. Li; L. Y. Zhao
503-508A PRACTICAL ONE-POT SYNTHESIS OF WEINREB-LIKE AMIDES OF (S)- AND (R)-N-BOC-PIPECOLIC ACIDS FROM (+)-PIPERIDINE-2-CARBOXYLIC ACIDIstván Moldvai; Gábor Dömyei; Eszter Temesvári-Major; Csaba Szántay
509-513AN EFFICIENT SYNTHESIS OF (R)-GABOB AND OF (+)-GABOBEngin Sahin; Nurhan Kishali; Latif Kelebekli; Ebru Mete; Hasan Secen; Ramazan Altundas; Yunus Kara
514-517AN IMPROVED PROCEDURE FOR SYNTHESIS OF α-ASARONEGuangyu Xu; Yi Zhouf; Gaolei Zuo; Yongjun Jiang
517-522SYNTHESIS OF INDAZOLE DERIVATIVES FROM 3, 5-DIARYL-6-ETHOXYCARBONYL-2-CYCLOHEXEN-1-ONESJavad Safaei-ghomi; Zohreh Alishahi

Volume 39, Issue 4 (2007)

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311-353THE CONQUEST OF VINIGROL. CREATIVITY, FRUSTRATIONS, AND HOPEGuillaume Tessier; Louis Barriault
355-383UNSYMMETRICAL UREAS. SYNTHETIC METHODOLOGIES AND APPLICATION IN DRUG DESIGNIsabelle Gallou
385-393MICROWAVE-ASSISTED REACTION OF HYDRAZONOYL HALIDES WITH CARBODITHIOIC ACID HYDRAZONESSayed M. Riyadh; Hamad M. Al-matar
395-398OPPI BRIEFS NEW SYNTHESIS OF HYDRANGETIN AND COLLBSINDominick Maes; Stijn Vervisch; Norbert De Kimpe
399-402IMPROVED SYNTHESIS OF MIRTAZAPINED. V. N. Srinivasa Rao; R. Dandala; V. K. Handa; M. Sivakumaran; A. V. Raghava Reddy; A. Naidu
403-412AN EFFICIENT METHOD FOR THE THIOACETALIZATION OF CARBONYL COMPOUNDS IN THE PRESENCE OF CATALYTIC AMOUNTS OF BENZYLTRIPHENYLPHOSPHONIUM TRIBROMIDEA. R. Hajipour; S. A. Pourmousavi; A. E. Ruoho
412-415FERRIC CHLORIDE-CATALYZED DEOXYGENATIVE CHLORINATION OF CARBONYL COMPOUNDS TO HALIDESZ. Li; C. Sheng; H. Qiu; Y. Zhang

Volume 39, Issue 3 (2007)

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203-296SYNTHESIS AND CLEAVAGE OF LACTONES AND THIOLACTONES. APPLICATIONS IN ORGANIC SYNTHESIS. A REVIEWZdzislaw Paryzek; Iwona Skiera
297-305AN EFFICIENT SYNTHESIS OF THE POTENTIAL MARINE TOXIN PTYCHODISCUS BREVIS [PB-1] AND ITS ANALOGUESArvind K. Gupta; D. K. Dubey; Mamta Sharma; M. P. Kaushik
305-3092, 6-DIISOPROPYL-4-METHYLPYRYLIUM HEXAFLUOROPHOSPHATET. S. Balaban; V. L. Horhoiu; A. T. Balaban

Volume 39, Issue 2 (2007)

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107-133SYNTHESIS OF FUROPYRANYL PYRIMIDINE NATURAL PRODUCTS. A REVIEWJesse D. More
135-152SYNTHESIS OF ANTIMYCINS. A REVIEWYong-Qing Yang; Yikang Wu
153-184o-AMINOMETHYL DERIVATIVES OF PHENOLS. PART 1. BENZYLAMINES: PROPERTIES, STRUCTURE, SYNTHESIS AND PURIFICATIONKrzysztof Bujnowski; Agnieszka Adamczyk; Ludwik Synoradzki
185-189OXIDATIVE CLEAVAGE OF 1, 2-DIOLS, α-KETOLS AND 1, 2-DIKETONES WITH AQUEOUS SODIUM HYPOCHLORITEJ. M. Khurana; P. Sharma; A. Gogia; B. M. Kandpal
190-195AN EFFICIENT AND STEREOSELECTIVE SYNTHESIS OF (Z)-ALLYL CHLORIDES FROM BAYLIS-HILLMAN ADDUCTS USING VILSMEIER-HAACK REAGENTY. Liu; H. Zheng; D. Xu; Z. Xu; Y. Zhang
195-199A CONVENIENT SYNTHESIS OF β-CHLOROVINYLALDEHYDES WITH bis-(TRICHLOROMETHYL) CARBONATEW. K. Su; Y. G. Zhuang; D. Z. Wu; W. H. Zhong
199-202A RELIABLE, HIGH-YIELDING PREPARATION OF 2, 6-DIMETHYL-4-HYDROXYBENZALDEHYDEGary M. Coppola; Yongjin Gong

Volume 39, Issue 1 (2007)

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1-70THE SYNTHESIS OF FLUORINATED HETEROAROMATIC COMPOUNDS. PART 2. FIVE-MEMBERED RINGS WITH TWO HETEROATOMS. A REVIEWAndrea Pace; Silvestre Buscemi; Nicolò Vivona
71-75YTTERBIUM PERFLUOROOCTANESULFONATE-CATALYZED KNOEVENAGEL CONDENSATION IN A FLUOROTJS BIPHASIC SYSTEMWen-Bin Yi; Ya-Qing Yin; Chun Cai
76-80SYNTHESIS AND ESI-MS STUDY OF NEW N-FUNCTIONALIZED MACROCYCLIC POLYAMINE AND AZACROWN ETHER DERIVATIVESBlazej Gierczyk; Joanna Wyrwal; Grzegorz Schroeder
81-85SIMPLE AND RAPID SYNTHESIS OF BIOLOGICALLY ACTIVE PHTHALEMIDE AND N-HYDROXYPHTHALIMIDE DIMERS USING POLYMER-SUPPORTED ANIONSD. S. Dalal; N. S. Pawar; P. P. Mahulikar
86-90IMPROVED SYNTHESIS OF 8-METHYL-3, 8-DIAZABICYCLO [3.2.1] OCTANEOsvaldas Paliulis; Dan Peters; Linas Miknius; Algirdas Šačkus
90-93AN IMPROVED IODBMATION OF 2-AMINO-5-NITROBENZONITRILEYe Zhang; Tianrui Ren; Weiwen Zhu; Yanhong Xie
93-96AN IMPROVED METHOD FOR THE PREPARATION OF 2-(2′-AMINOARYL) OXAZOLINES FROM SUBSTITUTED ISATOIC ANHYDRIDES AND 2-CHLOROETHYLAMINE HYDROCHLORIDEDavid A. Hunt
96-101AN IMPROVED PREPARATION OF 2, 2, 4, 4-TETRAMETHYL-6-AMINOTHIOCHROMAN, A KEY INTERMEDIATE TO UREA AND THIOUREA HETEROAROTINOIDS FOR ANTICANCER STUDIESC. R. Tallent; C. E. Twine Jr.; P. Risbood; H. H. Seltzman
101-106SYNTHESIS OF NOVEL 5-SUBSTITUTED-6-METHYL-4-[5-CHLORO-3-METHYL-1-PHENYL-1H-PYRAZOL-4-YL]-3, 4-DIHYDROPYRIMIDIN-2(1H)-ONESRakesh Kumar; Sakshi Malik; Ramesh Chandra

Volume 38, Issue 6 (2006)

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505-591THE PICTET-SPENGLER REACTION: EFFICIENT CARBON-CARBON BOND FORMING REACTION IN HETEROCYCLIC SYNTHESISSo Won Youn
593-599A SHORT SYNTHESIS OF THE CARBAZOLE ALKALOID CLAUSINE EJan Bergman; Ann-Louise Johnson
601-604FACILE PREPARATION OF TERMINALLY FUNCTIONALIZED THIOLS FROM 6-BROMOHEXANENITRILEJ. H. Wynne; C. T. Lloyd
604-608A PRACTICAL METHOD FOR PHOSPHORYLATION OF COMBRETASTATIN A-4 WITH PHOSPHORUS OXYCHLORIDEGurmit S. Gill; Damian Grobelny; Bernard Flynn
609-614INDEXES

Volume 38, Issue 5 (2006)

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427-465AZETIDINE-2-CARBOXYLIC ACID. FROM LILY OF THE VALLEY TO KEY PHARMACEUTICALS. A JUBILEE REVIEWFrançis Couty; Gwilherm Evano
467-469A PRACTICAL SYNTHESIS OF 3-BUTYN-1-OLXiao-Chun Yu; Haining Gu; Wei-Ming Xu
469-473SYNTHESIS OF INDOLOSULFONYLUREAS, POTENT ACETOLACTATE SYNTHASE INHIBITORSYe Zhang; Tianrui Ren
473-476DIRECT α-HYDROXYLATION OF ARYL KETONES USING A HYPERVALENT IODINE(III) SULFONATEH. -Y. Huang; R. -S. Hou; H. -M. Wang; L. -C. Chen
476-480IMPROVED METHOD FOR THE CYCLIZATION OF ortho-ALKYNYLBENZENEDIAZONIUM SALTSNataliya A. Zolnikova; Lidiya G. Fedenok; Nikolay E. Polyakov
480-483IMPROVED SYNTHESIS AND PURIFICATION OF CAVITANDSJorden P. Kass; Leslie A. Slasor; Cesar H. Zambrano; Eric E. Dueno
484-4901,3-DIBROMO-5,5-DIMETHYLHYDANTOIN AS AN EFFICIENT AND CHEMOSELECTIVE AGENT FOR THE REGENERATION OF CARBONYL COMPOUNDS FROM SEMICARBAZONES AND OXIMESArdeshir Khazaei; Amin Rostami
490-494CONVENIENT AND RAPID PREPARATION OF INDENE DIMERS FROM INDENES OR INDANOLSFei Liu; Qi-Dong You; Min-Yong Li; Wen-Bin Shen; Lin Xia
495-500AN EFFICIENT AND RAPID SYNTHESIS OF N-SUBSTITUTED PYRROLES BY MICROWAVE ASSISTED SOLID ACID CATALYSISMohammed Abid; Shainaz M. Landge; Béla Török
500-504NEW AND SIMPLE SYNTHESIS OF THE PHEROMONE COMPONENT OF MALE MELON FLYYao-Pin Yen; Jay-Hung Chen

Volume 38, Issue 4 (2006)

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347-399DIPYRRINONES-CONSTITUENTS OF THE PIGMENTS OF LIFE. A REVIEWStefan E. Boiadjiev; David A. Lightner
401-404AN EFFICIENT SYNTHESIS OF 4,4′-DIAMINODIPHENIC ACIDArkadiy Rubezhov
404-410A CONVENIENT, ONE-POT SYNTHESIS OF THIOCARBAMATES USING BIS(TRICHLOROMETHYL) CARBONATEW. K. Su; J. P. Zhang; X. R. Liang
410-412AN IMPROVED SYNTHESIS OF 2-n-(PROPYL)-1H-IMIDAZOLE-4,5-DICARBOXYLIC ACID DIETHYL ESTERXinmin Wen; Xinhong Yu; Jan Tang
412-417A NEW, EFFICIENT AND SIMPLE METHOD FOR THE SYNTHESIS OF THIOAMIDES FROM NITRILESBabak Kaboudin; Dawood Elhamifar; Fatemeh Farjadian
417-422AN IMPROVED PROCEDURE FOR THE ROBINSON ANNULATION REACTION OF SOME CHALCONES CATALYZED BY K2CO3 UNDER ULTRASOUNDJavad Safaei-Ghomi; Zohreh Alishahi
423-426AN IMPROVED RESOLUTION PROCESS FOR THE PREPARATION OF ANTIDE-PRESSANT DRUG: ESCITALOPRAMAlka Mital; Rakesh Kumar; Uma Ramachandran

Volume 38, Issue 3 (2006)

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217-305SYNTHESIS OF MODIFIED STEROIDS IN THE ANDROSTANE AND ANDROSTENE SERIESElie Stéphan
307-312AN EFFICIENT ONE-POT SYNTHESIS OF 2-AMINO-4H-PYRANSA. Zonouzi; D. Kazemi; M. Nezamabadi
313-324SYNTHESIS OF NOVEL BENZOCHROMENE, BENZOQUINOLINE, BENZOCHROMENOPYRIMIDINE AND PYRIMIDOBENZOQUINOLINE DERIVATIVESM. N. Jachak; D. B. Kendre; A. B. Avhale; R. B. Toche; V. J. Medhane
325-331SYNTHESIS OF 3,6-DIHALOPHENANTHRENE DERIVATIVESDane W. Scott; Richard A. Bunce; Nicholas F. Materer
331-336THE SELECTIVE SOLID-PHASE OXIDATION OF ALCOHOLS AND OTHER ORGANIC SUBSTRATES BY 3,5-DIMETHYLPYRAZOLIUM FLUOROCHROMATEM. K. Chaudhuri; S. K. Dehury; S. Hussain; A. Duarah; N. Gogoi
337-340DIMERIZATION OF LITHOCHOLATE UNSATURATED ESTERS USING THE ‘SECOND GENERATION’ GRUBBS' REAGENTChristopher Dallstream; Jerry Ray Dias
341-344SYNTHESIS OF NOVEL 4,4′-BENZIDINE DERIVATIVES WITH SULFONIC ACID GROUPSM. Nanasawan; S. Yamashita; M. Hirai; K. Miyatake; M. Watanabe
344-346TEMPERATURE DEPENDENT MIGRATION OF THE NITRO GROUP OF POTASSIUM 4-AMINO-3,5-DINITROBENZENESULFONATE VS DESULFONATIONViktor Milata; Maroš Bella

Volume 38, Issue 2 (2006)

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101-176SYNTHESIS AND PROPERTIES OF PSICO-NUCLEOSIDESStewart K. Richardson; Amy R. Howell; Rosa Taboada
177-216USES OF SODIUM CHLORITE AND SODIUM BROMATE IN ORGANIC SYNTHESIS. A REVIEWA. Paul Krapcho

Volume 38, Issue 1 (2006)

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1-80RECENT PROGRESS IN THE SYNTHESIS OF ARTEMISININ AND ITS DERIVATIVESByung Ju Kim; Tomikazu Sasaki
81-85A CONVENIENT SYNTHESIS OF 5-ARYLIDENETHIAZOLIDINE-2,4-DIONES ON POTASSIUM FLUORIDE-ALUMINIUM OXIDEDe-Hong Yang; Ben-Yong Yang; Zhen-Chu Chen; Song-Ying Chen
87-88A SIMPLE PROCEDURE FOR THE PREPARATION OF 6-CHLORO-3-ACETOXY-1-ACETYLINDOLEAlexander Balbuzano-Deus; Juan C. Rodríguez-Domínguez; Anaís Fernández-Villalobo; Miguel López-López; Gilbert Kirsch
89-94A CONVENIENT SYNTHESIS OF 2-METHYL-3-SUBSTITUTED-4(3H)-QUINAZOLINONES USING BIS(TRICHLOROMETHYL) CARBONATE AS CONDENSING AGENTW. K. Su; D. Z. Wu; Y. Y. Xie; J. J. Li
94-99SYNTHESIS OF OCTANDRENOLONE, FLEMICULOSIN, (±)-3-DEOXY-MS-II AND LAXICHALCONEMandar Deodhar; David StC Black; Naresh Kumar

Volume 37, Issue 6 (2005)

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513-538THE ASYMMETRIC AZA-MICHAEL REACTION. A REVIEWJose L. Vicario; Dolores Badía; Luisa Carrillo; Juan Etxebarria; Efraim Reyes; Nerea Ruiz
539-546SYNTHESIS OF 2-MERCAPTOBENZOTHIAZOLE AND OF 2-MERCAPTO-BENZIMIDAZOLE DERIVATIVES USING POLYMER-SUPPORTED ANIONSD. S. Dalal; N. S. Pawar; P. P. Mahulikar
546-550AN EFFICIENT SYNTHESIS OF TRICYCLIC COMPOUNDS, (±)-(4aβ,8aβ,10aα)-1,2,3,4,4a,6,7,8,8a,9,10,10a-DODECAHYDRO-1,1,4a-TRIMETHYL-2-OXOPHENANTHRENE-8a-CARBOXYLIC ACID, ITS METHYL ESTER, AND (±)-(4aβ,8aβ,10aα)-3,4,4a,6,7,8,8a,9,10,10a-DECAHYDRO-8a-HYDROXYMETHYL-1,1,4a-TRIMETHYLPHENANTHREN-2(1H)-ONETadashi Honda; Yukiko Honda; Hidenori Yoshizawa; Gordon W. Gribble
550-555A SYNTHESIS OF SELECTED o,o'-DISUBSTITUTED DIARYLACETIC ESTERS AND DIARYLMETHANESRichard A. Bunce; James E. Schammerhorn
555-559A CONVENIENT SYNTHESIS OF 3-ETHOXYCARBONYLAMINO-2-HYDROXY-4-PHENYLBUTYRIC ACIDLi Jun Lei; Xu Chang He
560-565SYNTHESIS OF 2,4(1H,3H)-QUINAZOLINEDIONE AND 3-SUBSTITUTED 2,4(1H,3H)-QUINAZOLINEDIONESJ. S. Petrov; G. N. Andreev
566-569A NOVEL SYNTHESIS OF 2-CHLORO-4-FLUORO-5-NITROBENZENESULFONYL CHLORIDEXiao-Hua Du; Sheng Chen; Mei Zheng; Zhen-Yuan Xu
569-574EFFICIENT AND COST-EFFECTIVE SYNTHESIS OF DIALKYL CHLOROPHOSPHATESP. D. Shakya; D. K. Dubey; Deepak Pardasani; Meehir Palit; A. K. Gupta
575-579REGIOSELECTIVE SYNTHESIS OF E-OXIMES CATALYZED BY FERRIC CHLORIDE UNDER SOLVENT-FREE CONDITIONSHossein Eshghi; Asadollah Hassankhani
579-584TWO-STEP PROTIC SOLVENT-CATALYZED REACTION OF PHENYLETHYLAMINE WITH METHYL ACRYLATEH. Fakhraian; M. Babaie Panbeh Riseh
585-589NITRIC ACID AND PHOSPHORUS PENTOXIDE SUPPORTED ON SILICA GEL AS A MILD AND EFFICIENT SYSTEM FOR THE OXIDATION OF BENZYLIC ALCOHOLS UNDER SOLVENT-FREE CONDITIONSAbdol R. Hajipour; Behzad Kooshki; Arnold E. Ruoho
589-594ALTERNATE SYNTHESES OF PRODAN AND ACRYLODANSteven S. Silvonek; Carl B. Giller; Christopher J. Abelt
595-602INDEXES

Volume 37, Issue 5 (2005)

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411-445APPROACHES TO THE SYNTHESIS OF THE LAMELLARINS AND RELATED NATURAL PRODUCTS. A REVIEWScott T. Handy; Yanan Zhang
447-506THE SYNTHESIS OF FLUORINATED HETEROAROMATIC COMPOUNDS. PART 1. FIVE-MEMBERED RINGS WITH MORE THAN TWO HETEROATOMS. A REVIEWAndrea Pace; Silvestre Buscemi; Nicolò Vivona
507-511REDUCTION OF π-DEFICIENT HETEROCYCLIC SECONDARY CARBINOLS WITH SODIUM BOROHYDRIDE/TRIFLUOROACETIC ACIDCharles F. Nutaitis; Brett D. Swartz

Volume 37, Issue 4 (2005)

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307-336SMALL PEPTIDES WITH A β-HAIRPIN STRUCTURES. Miltschitzky; B. Koenig
337-375SYNTHETIC GLYCODIVERSIFICATION. FROM AMINOSUGARS TO AMINOGLYCOSIDE ANTIBIOTICS. A REVIEWRavi Rai; Ian McAlexander; Cheng-Wei Tom Chang
377-385REEXAMINATION OF THE FRIEDEL-CRAFTS REACTION OF METHYL CHLORIDE WITH PHOSPHORUS TRICHLORIDE FOR THE PREPARATION OF METHYL PHOSPHONIC DICHLORIDEH. Fakhraian; M. Zarinehzad; H. Ghadiri
387-396NITRATION OF PHENOL, CRESOL, AND ANISOLE USING CERIC AMMONIUM NITRATE SUPPORTED ON A CLAY AND ON A PILLARED CLAYCuauhtemoc Pérez; Salud Pérez-Gutiérrez; Sergio A. Gómez; Gustavo A. Fuentes; Miguel A. Zavala
397-402REINVESTIGATION OF THE SYNTHESIS OF 2-BENZYL-3-ARYL-QUINAZOLIN-4-[3H]-ONES. AN IMPROVED MULTI-COMPONENT PROCEDURE USING MICROWAVESAnshu Dandia; Ruby Singh; Pritima Sarawgi
403-405AN IMPROVED SYNTHESIS OF 1-METHYL-2-TRICHLOROACETYLIMIDAZOLEElżb�eta Masiukiewicz; Damian Mrugala; Barbara Rzeszotarska
405-408FORMATION OF OXIRANES DURING THE PREPARATION OF AROYLACETONITRILESR. B. Toche; M. N. Jachak; N. S. Badgujar; A. B. Avhale; D. B. Kendre
409CORRIGENDUM

Volume 37, Issue 3 (2005)

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205-212RAPID FUNCTIONALIZATION AND LOADING OF SOLID SUPPORTSRadhakrishnan P. Iyer; John E. Coughlin; Seetharamaiyer Padmanabhan
213-222SYNTHESIS OF SUBSTITUTED 1,3,4-THIADIAZOLES USING LAWESSON'S REAGENTB. Gierczyk; M. Zalas
223-230ENAMINONES IN THE SYNTHESIS OF HETEROCYCLES BY MICROWAVE IRRADIATIONMariam A. Al-Shiekh
231-237IMPROVED PROCEDURES FOR THE BAYLIS-HILLMAN REACTIONSan-Hu Zhao; Hong-Yan Bie; Zhao-Bin Chen
239-246DIASTEREOSPECIFIC SYNTHESIS OF trans-2,3-DIARYL-1-AMINOCYCLOPROPANECARBOXYLIC ACIDSChengxue Pan; Guifa Su; Jiangke Qin
247-256SYNTHESIS OF ISOMERIC PYRIDOOXAZINONES, PYRIDOPYRIDAZINES AND TRIAZOLOPYRIDOPYRIDAZINES FROM o-AROYLPYRIDINECARBOXYLIC ACIDSMohamed Salah K. Youssef; Amin F. Fahmy; Mohamed S. Abdel Halim; Mamdouh A. Hassan; Jürgen Sauer
257-263FLUOROUS SILYL PROTECTING GROUP FOR 5'-HYDROXYL PROTECTION OF OLIGONUCLEOSIDESSnehlata Tripathi; Krishna Misra; Yogesh S. Sanghvi
265-2675-CHLORO- AND 5,7-DICHLOROISATIN BY CHLORINATION OF ISATIN WITH TRICHLOROISOCYANURIC ACIDN. M. Ribeiro; B. V. Da Silva; F. de Almeida Violante; C. M. Rezende; A. C. Pinto
268-272FACILE ONE-STEP SYNTHESIS OF DITHIAALKANEDIOLSMahabir P. Kaushik; Hemlata Rana
272-275A NOVEL AND CONVENIENT METHOD FOR THE SYNTHESIS OF PHENSTATINMaojiang Wu; Qinggang Ji; Chunhao Yang; Yuyuan Xie
275-279EXPLOITATION OF CO-OPERATIVE DIRECTED ortho-METALLATION (DoM) BY 1,3-RELATED -OMOM GROUPS IN THE DEVELOPMENT OF A FULLY REGIO-CONTROLLED SYNTHESIS OF ATRANOL FROM ORCINOLMartin G. Banwell; Satish Chand
279-283METHYLTRIPHENYLPHOSPHONIUM PEROXYDISULFATE AND IODINE AS MILD REAGENTS FOR THE IODINATION OF ACTIVATED AROMATIC COMPOUNDSAbdol R. Hajipour; A. E. Ruoho
283-285A PRACTICAL LARGE-SCALE PREPARATION OF 5'-BROMOSPIRO(CYCLOHEXANE-1,3-[3H]INDOL)-2'(1'H)-ONEBogdan K. Wilk; Arkadiy Rubezhov; Jean L. Helorn; Lisa R. Routel; John R. Potoski
286-290CONVENIENT MICROWAVE ASSISTED SYNTHESIS OF NATURALLY OCCURRING METHYL (E)-CINNAMATESRajesh P. Mahajan; Shamkant L. Patil; Raghao S. Mali
290-293SYNTHESIS OF FUSED BICYCLO[3.2.2]NONENONESXinglong Jiang; Kapa Prasad; Oljan Repič
294-298A SIMPLE AND EFFICIENT METHOD FOR THE SYNTHESIS OF gem-CHLORONITROSO COMPOUNDSA. K. Gupta; D. K. Dubey; Mahabir P. Kaushik
298-303SOLID STATE DEPROTECTION OF THIOACETALS AND THIOKETALS USING 1-BENZYL-4-AZA-1-AZONIABICYCLO[2.2.2]OCTANE PERIODATE AND ALUMINUM CHLORIDEAbdol Reza Hajipour; Arnold E. Ruoho
305CORRIGENDUM

Volume 37, Issue 2 (2005)

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103-171A DECADE OF ADVANCES IN THREE-COMPONENT REACTIONSM. Syamala
173-177AN IMPROVED AND FACILE SYNTHESIS OF SCHIFF BASES IN AQUEOUS MEDIUMM. S. Singh; A. K. Singh; Pratibha Singh; Ruchi Jain
178-183REGIOSELECTIVITY OF THE METHYL-TOSMIC REACTION WITH SUBSTITUTED ETHYL CINNAMATESRoberto Di Santo; Roberta Costi; Carlo Galeffi; Michela Forte
184-188A CONVENIENT AND EFFICIENT ASYMMETRIC SYNTHESIS OF (S)-α-ARYLTHIOMETHYL-α-HYDROXYBUTYRIC ACID ESTERSYun-Yan Kuang; Fen-Er Chen
189-194REDUCTION AND OXIDATION OF 1-METHYLCYCLOHEXA-2,5-DIENE-1-CARBOXYLIC ACIDSLiliana E. Luna; Raquel M. Cravero
194-197REDUCTIVE THIOLATION APPROACH TO PURE CYCLOBUTYL PHENYL SULFIDEMatthew C. T. Fyfe; Chrystelle M. Rasamison
198-203A SIMPLE PROCEDURE FOR THE CONVERSION OF CARBOXYLIC ACIDS TO THE CORRESPONDING AMIDESKi-Jong Han; Beom Seok Tae; Misoo Kim

Volume 37, Issue 1 (2005)

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1-35SYNTHESIS OF THE HAMIGERANS. A REVIEWDerrick L. J. Clive; Jian Wang
37-63TARTARIC ACID AND ITS O-ACYL DERIVATIVES. PART 1. SYNTHESIS OF TARTARIC ACID AND O-ACYL TARTARIC ACIDS AND ANHYDRIDESLudwik Synoradzki; Pawel Ruśkowski; Urszula Bernaś
65-73STEREOSELECTIVE SYNTHESIS OF α-AMINO ACIDS FROM O-PIVALOYL-D-GLUCOPYRANOSYLALDIMINEGuobin Zhou; Pengfei Zhang; Yuanjiang Pan; Junli Guo
75-79α,α-bis(BENZYLIDENE)CYCLOALKANONES BY CONDENSATION IN WATER UNDER PTC CATALYSIS AND MICROWAVE IRRADIATIONJianfeng Zhou
80-83DIATOMITE-SUPPORTED PERACETIC ACID OXIDATION OF 1,4-DIHYDROPYRIDINESBu-Lan Wu; Zhao-Bin Chen
83-86OXIDATION OF TOLUENES TO AROMATIC ALDEHYDES WITH MOLECULAR OXYGEN IN SUBCRITICAL WATERBerkant Kayan; Recep Özen; Ahmet M. Gizir; N. Simsek Kus
87-92EFFICIENT ESTERIFICATION OF ALIPHATIC CARBOXYLIC ACIDS CATALYZED BY COPPER METHANESULFONATEJie Ma; Heng Jiang; Hong Gong
93-98THE SYNTHESIS OF E-2-(BROMOMETHYLENE)CYCLOHEXANONE AND E-2-(BROMOMETHYLENE)CYCLOHEPTANONEMartin G. Banwell; Xinghua Ma; Anthony C. Willis
99-102IMPROVED SYNTHESIS OF TADALAFILYunlong Zhang; Qian He; Huasheng Ding; Xihan Wu; Yuyuan Xie

Volume 36, Issue 6 (2004)

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499-547RECENT ADVANCES IN THE CHEMISTRY OF TRICHLOROMETHYL CHLOROFORMATE AND bis-(TRICHLOROMETHYL) CARBONATEWeike Su; Weihui Zhong; Gaofeng Bian; Xiangjun Shi; Jianping Zhang
549-572A CRITICAL EXAMINATION OF THE PREPARATION OF POLYCHLORINATED ACETONESBaldur Föhlisch; Hartmut Zinser
573-579PRACTICAL PROCEDURE FOR THE PREPARATION OF FUNCTIONALIZED (E)-1-ALKENYLBORONIC ACIDS INCLUDING THE UNPRECEDENTED 1-ALKOXYCARBONYL DERIVATIVESMichel Gravel; Barry B. Touré; Dennis G. Hall
581-586ZEOLITE-MEDIATED CONVERSION OF ALCOHOLS TO p-METHOXYBENZYL ETHERSG. V. M. Sharma; Sreenivas Punna; A. Ratnamala; V. Durga Kumari; M. Subrahmanyam
587-596KILOGRAM-SCALE SYNTHESIS OF bis(6-HYDROXY-5,5-DIMETHYLHEXYL)ETHER (ESP24232), A NOVEL LIPID LOWERING AGENTJing Yang; Ralf Mueller; Emil Pop; Jean-Louis H. Dasseux; Daniela C. Oniciu
597-600IMPROVED SYNTHESIS OF NTTRILES OF QUINOLONE ANTIBIOTICSKeith A. Korthals; Thomas J. Delia
600-604REACTION OF 5-CHLORO-2-HYDROXYBENZOPHENONE WITH PHOSPHORUS OXYCHLORIDE AND RELATED REACTIONSA. G. Pinkus; Tsung C. Chang; Lily Y. C. Meng
605-614INDEXES

Volume 36, Issue 5 (2004)

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391-443RECENT DEVELOPMENTS IN HYDANTOIN CHEMISTRY. A REVIEWManuela Meusel; Michael Gütschow
445-452SYNTHESIS OF UNSYMMETRICAL DIALKOXY QUINAZOLINESMatthieu Desroses; Guillaume Laconde; Patrick Depreux; Jean-Pierre Hénichart
453-457SYNTHESIS OF RING-A HYDROXYLATED FLAVONES BY SODIUM HYDROXIDE-CATALYZED CYCLIZATION OF 1,3-DIKETONES IN WATERLijun Tang; Shufen Zhang; Jinzong Yang; Wentao Gao; Jian Cui
459-467AN EFFICIENT LARGE SCALE SYNTHESIS OF NATEGLINIDEBatchu Chandrasekhar; Mangesh S. Sawanth; Sameer J. Naik; Nandakumar B. Gaikwad; Pramila V. Kulkarni; Shekar B. Bhirud
469-472A RELIABLE MULTI-KILOGRAM PREPARATION OF 4-PHENYLURAZOLEB. Chandrasekhar; G. B. Kumar; S. Mallela; S. B. Bhirud
472-475A CONVENIENT METHOD FOR PREPARATION OF TRIAZOLINEDIONESAbdol Reza Hajipour; Morteza Malakoutikhah
476-479A PRACTICAL PROCEDURE FOR THE SYNTHESIS OF 3-((E)-5-(2,3,4,5-TETRAMETHOXY-6-METHYLPHENYL)-3METHYLPENT-3-ENYL)-2,2-DIMETHYLOXIRANEYong Chu; Yunyan Kuang; Huifang Dai; Liang Lu; Fener Chen
479-481A PRACTICAL PREPARATION OF N,N,-PHTHALYL-L-GLUTAMIC 1,5-ANHYDRIDEHaining Gu; Yongxiang Jiang
482-487N-(NITROPHENYL) BENZAMIDE AND BENZENESULFONAMIDE DERIVATIVES BY NUCLEOPHILIC AROMATIC SUBSTITUTIONRichard A. Bunce; Christopher L. Smith; Christopher L. Knight
487-490A NOVEL AND CONVENIENT SYNTHESIS OF 4-HALOBUTYRALDEHYDE ACETALSJohn A. Hyatt
491-494EFFICIENT SYNTHESIS OF IMIDAZO[2,1-α]ISOQUINOLINES USING A HYPERVALENT IODINE(III) SULFONATER. -S. Hou; H. -M. Wang; H. -Y. Huang; L. -C. Chen
494-498A CLEAN AND RAPID SYNTHESIS OF 5-AMINO AND 5-ALKOXYCARBONYLPYRAZOLES USING MONTOMORILLONITE UNDER ACID FREE CONDITIONSG. Jagath Reddy; D. Latha; K. Srinivasa Rao

Volume 36, Issue 4 (2004)

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297-330DIBENZO[bf]OXEPINES: SYNTHESES AND APPLICATIONS. A REVIEWRoberto Olivera; Raul Sanmartin; Fátima Churruca; Esther Domínguez
331-335PRACTICAL ROUTE TO A β-KETOPHOSPHONATE, A KEY INTERMEDIATE FOR THE TOTAL SYNTHESIS OF 20(S)-CPT AND RELATED ANALOGUESMing Huo; Yun-Yan Kuang; Fen-Er Chen
337-340VILSMEIER-HAACK SYNTHESIS OF AROMATIC ALDEHYDES USING bis-(TRICHLOROMETHYL) CARBONATE AND DIMETHYLFORMAMIDEW. G. Shan; X. J. Shi; W. K. Su
341-345AN EXPEDITIOUS, PRACTICAL LARGE SCALE SYNTHESIS OF 4-AMINO-2-CHLORO-6,7-DIMETHOXYQUINAZOLINAZOLINEG. Kumaraswamy; Nivedita Jena; M. N. V. Sastry; B. Ashok Kumar
347-351N-ALKYLATION OF N-MONOSUBSTITUTED SULFONAMTOES IN IONIC LIQUIDSYi Hu; Zhen-Chu Chen; Zhang-Goo Le; Qin-Guo Zheng
353-359SYNTHESIS OF TETRAHEDRAL CARBOXAMIDE HYDROGEN BOND ACCEPTORSAmy S. Cannon; Tianying Jian; Jun Wang; John C. Warner
361-362IMPROVED SYNTHESIS OF 3-AMINOFURAZAN-4-CARBOXYLIC ACIDKevin G. Meyer
363-366HEXAMETHYL ENETETR AMMONIUM FLUOROCHROMATE. A NEW REAGENT FOR OXIDATION OF ORGANIC SUBSTRATESErsan Turunc; Fatma Aydin
367-370PREPARATION OF TRIAZAPHENAN THRENESCharles F. Nutaitis; Megan Brennan
371-374A CONVERGENT SYNTHETIC ROUTE TO 2-OXOPYRIDO[2,3-a]CARBAZOLES via 2-OXOPYRANO[2,3-a]CARBAZOLES FROM 1-OXO-1,2,3,4-TETRAHYDROCARBAZOLESI. Antony Danish; K. J. Rajendra Prasad
375-379A CONVENIENT METHOD FOR THE PREPARATION OF 2,5-bis-(4-AMINOPHENYL)-1,3,4-OXADIAZOLEMatthew C. Davis; Andrew P. Chafin
380-383AN IMPROVED PROCEDURE FOR THE ETHERIFICATION OF α-HYDROXY ACID DERIVATIVESSanjeev Kumar; Uma Ramachandran
383-386FACILE BECKMANN REARRANGEMENT OF KETOXIMES MEDIATED BY YTTRIUM TRIFLATESurya Kanta De
386-390AN IMPROVED SYNTHESIS OF NEOCRYPTOLEPINERobert Engqvist; Jan Bergman

Volume 36, Issue 3 (2004)

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201-276MOLYBDENUM IN ORGANIC SYNTHESIS. A REVIEWJitender M. Khurana; Sushma Chauhan; Arpita Agrawal
277-279IMPROVED SYNTHESIS OF 3,4-DIHYDRO-2,6-DIMETHYL-4-OXOQUINAZOLINEShiyan Chen; Jimao Lin; Bingjie Qin
279-283PREPARATION OF 3-BROMO-2-(NITROMETHYLENE)PYRROLIDINE AND 3-BROMO-N-METHYL-l-NITRO-l-BUTEN-2-AMINEJ. Geno Samaritoni
283-286A FACILE ONE-POT PREPARATION OF ISOTHIOCYANATES FROM N-FORMAMIDES AND SULFUR POWDER WITH bis(TRICHLOROMETHYL) CARBONATEW. G. Shan; G. F. Bian; W. K. Su; X. R. Liang
287-289AN EFFICIENT ONE STEP CONVERSION OF 3-FORMYLCHROMONES INTO 3-CYANOCHROMONESG. Jagath Reddy; D. Latha; C. Thirupathaiah; K. Srinivasa Rao
289-292AN EFFICIENT SYNTHESIS OF 2,3-DICYANOINDOLETomasz Janosik; Adam C. Lipson; Gordon W. Gribble
292-296SYNTHESIS OF 6-(2,2-DIMETHYL-3,4-DIHYDRO-3-OXO-1,4(2H)-BENZOXAZIN-7-YL)PYRIDAZIN-3-ONESZiaeddin Moussavi; Nicolas Lebegue; Pascal Carato; Said Yous; Pascal Berthelot

Volume 36, Issue 2 (2004)

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99-120HOMOGENEOUS RHODIUM(I)-CATALYZED REDUCTIVE AMINATIONSVitali I. Tararov; Renat Kadyrov; Thomas H. Riermeier; Uwe Dingerdissen; Armin Börner
121-127A NOVEL AND DIRECT METHOD FOR THE PREPARATION OF 4-AMINO-1,1,3,3-TETRASUBSTTTUTED GUANIDINES AND OF [1,2,4]TRIAZOLO-FUSED HETEROCYCLIC DERIVATIVESM. Abdul-Ghan; Sh. N. Khattab; A. M. El-Massry; A. El-Faham; Adel Amer
129-133PREPARATION OF METHYL 2-METHOXYCARBONYLMETHYL-6-OXO-1,6-DIHYDROPYRIDINE-3-CARBOXYLATESong Feng; Xuchang He; Gengli Yu; Yu Xia; Donglu Bai
135-140AN ANOMALOUS HOUBEN-HOESCH REACTION AND SOME APPLICATIONS IN ARYLATION REACTIONSF. Sánchez-Viesca; María R. Gómez; Martha Berros
141-149SYNTHESIS OF URETHANES BY A MODIFIED CURTIUS REACTION WITH ALCOHOLSArmandodoriano Bianco; Francesco Bonadies; Raffaella Napolitano; Giancarlo Ortaggi
151-155SYNTHESIS OF 3-SUBSTITUTED-2-ACYLIMINO-4-THIAZOLIDONES UNDER MICROWAVE IRRADIATIONYanqing Peng; Gonghua Song; Ling Liu
156-161WILLIAMSON REACTION IN IONIC LIQUIDSZhen Yuan Xu; Dan Qian Xu; Bao You Liu
161-163IMPROVED SYNTHESIS OF PHENYLSELENOGLYCOLIC ACIDSHamdi Özkan; Ali Disli; Yilmaz Yildirir
164-166A NOVEL AND SIMPLE SYNTHESIS OF (1S, 2S)-2-AMINO-l-(p-NITROPHENYL)-3-TRITYLOXYPROPANOLJian-Li Yuan; Hui-Fen Dai; Fen-Er Chen
166-170SYNTHESIS OF 2-SUBSTITUTED THIAZOLIDINE-4-CARBOXYLIC ACIDSElena Pini; Donatella Nava; Riccardo Stradi
170-173FACILE ONE-POT SYNTHESIS OF FLUORESCENT BENZOTHIENO[2,3:c]QUINOLINEHarjinder Singh Bhatti; Sambamurthy Seshadri
173-177SYNTHESIS OF PHENYLENE 1,3- AND 1,44bis(METHYLENE)-3-CARBAMOYL PYRIDINIUM BROMIDESFeng Zhou; Chi-Hua Wang; John C. Warner
178-182THE STRUCTURE OF “ITCA”, A URINARY METABOLITE OF CYANIDEHerbert T. Nagasawa; Steven E. Cummings; Steven I. Baskin
182-185A PRACTICAL SYNTHESIS OF ETHYL L-GLUTAMINE (L-Theanine)Haining Gu; Yongxiang Jiang; Jiong Wang
185-187A FACILE AND DIRECT SYNTHESIS OF ALENDRONATE FROM PYRROLIDONEGuangyu Xu; Yuyuan Xie; Xihan Wu
188-191MODIFIED AND CONVENIENT METHODS FOR THE PREPARATION OF SOME NTTRO MUSKSJavad Safaei-Ghomi; Abdolhamid Bamoniri
192-194SYNTHESIS OF 2-CHLORO- AND 2,5-DICHLOROBENZOPHENONESA. G. Pinkus; F. S. Y. Ma; L. Y. C. Meng; T. C. Chang
195-199NEW AND IMPROVED SYNTHESIS OF (±)-4-BROMO-7,8-DIMETHOXY-ISOCHROMAN-3-ONE, A KEY INTERMEDIATE FOR THE ELABORATION OF (±)-cis-ALPININE AND (±)-cis-ALPINIGENINEDaríO A. Bianchi; Teodoro S. Kaufman

Volume 36, Issue 1 (2004)

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1-31PREPARATION OF TETRAMETHYLPIPERDINE-1-OXOAMMONlUM SALTS AND THEIR USE AS OXIDANTS IN ORGANIC CHEMISTRY. A REVIEWNabyl Merbouh; James M. Bobbitt; Christian Brückner
33-59SYNTHESIS AND CHEMISTRY OF TETRONIC ACIDSDavid Tejedor; Fernando García-Tellado
61-67BENZYLATION OF FLAVAN-3-OLS (CATECHINS)Jamal Muskifa; Riaz A. Khan; Ikhlas A. Khan; Daneel Ferreira
69-71AN IMPROVED SYNTHESIS OF 5-(2-FLUOROPHENYL)-1H-TETRAZOLEK. Srinivas; C. K. Snehalatha Nair; S. Ramesh; M. Pardhasaraclhi
71-73A NEW SIMPLIFIED METHOD FOR THE PREPARATION OF N,N'-DIPHENYLUREAKevin Tran; K. Darrell Berlin
74-76MODIFIED SYNTHETIC ROUTE TO 2-HYDROXYIMINO-N-ARYLACETAMIDESA. Paul Krapcho; Sergio A. Cadarmro
76-81A VERSATILE AND CONVENIENT SYNTHESIS OF ALKYL NITROAROMATIC ETHERS BY NUCLEOPHILIC AROMATIC SUBSTITUTIONRichard A. Bunce; Kerry M. Easton
82-86CONVENIENT SYNTHESIS OF 1-AMINOALKYLPHOSPHONATES UNDER SOLVENT-FREE CONDITIONSBabak Kaboudin; Abbas Rahmani
87-91STEREOSELECTIVE SYNTHESES OF THE METHYL ESTERS OF (E)- AND (Z)-2-METHYL-6-OXOHEFT-2-EOIC ACIDMartin G. Banwell; Jasmine C. Jury
92-95A FACILE SYNTHESIS OF 6-ARn-l-METHYL-3-n-PROPn-6,7-DIHYDRO-1H-PYRAZOLO[4,3-d]PYRIMIDIN-7-OMESN. Ram Reddy; G. Mahesh Reddy; P. Pratap Reddy
96-98SYNTHESIS OF 3-ARYL AZO-3-PENTENE-4-OL-2-ONESAli Disli; Volkan Kaya; Ahmet Gülcet; Yilmaz Yildmr

Volume 35, Issue 6 (2003)

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527-581REGENERATION OF CARBONYL COMPOUNDS FROM OXIMES, HYDRAZONES, SEMICARBAZONES, ACETALS, 1,1-DIACETATES, 1,3-DITHIOLANES, 1,3-DITHIANES AND 1,3-OXATHIOLANESAbdol Reza Hajipour; Sepideh Khoee; Arnold E. Ruoho
583-601o-DIACYLBENZENES IN ORGANIC SYNTHESIS. A REVIEWAntigoni Kotali; Philip A. Harris
603-608A RELIABLE MULTIGRAM SYNTHESIS OF (±) DOXAZOSING. Kumaraswamy; A. K. Das; Nivedita Jena
609-613A NEW SYNTHESIS OF FLUMAZENEL SUITABLE FOR FLUORINE-18 LABELINGGianluigi Broggini; Marco Orlandi; Alberto Turconi; Caterina Zoni
613-616A FACILE SYNTHESIS OF DISULFIDES BY OXIDATION OF THIOLS WITH bis(TRICHLOROMETHYL) CARBONATE AND TRIPHENYLPHOSPHINE OXIDEY. S. Li; X. R. Liang; W. K. Su
616-619A MILD AND EFFICIENT METHOD FOR RACEMIZATION OF α-AMINO ESTERSUma Ramachandran; Sudhanshu Kumar; H. P. S. Chawla
620-622CONVENIENT PREPARATION OF A NEW ZWITTERIONIC TOSYLATEMireia Condom; SebastiáN Ondoño; Joan Suades
623-626A DIELS-ALDER SYNTHESIS OF PYRIDINESJ. B. Hendrickson; Jian Wang
627-630A CONVENIENT PROCEDURE FOR INDIRECT OXIDATION OF AROMATIC METHYL GROUPS TO ALDEHYDES AND CARBOXYLIC ACIDSLeslie W. Deady; Shane M. Devine; Michael L. Rogers
631-637INDEXES

Volume 35, Issue 5 (2003)

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445-500TANDEM REACTIONS INVOLVING ORGANOLITHIUM REAGENTS. A REVIEWGraciela V. García; Norma Sbarbati Nudelman
501-507SYNTHESIS OF N-(4-CHLOROBUTYL)BUTANAMIDE, A CHLORINATED AMIDE ISOLATED FROM ALOE SABAEAMatthias D'hooghe; Zsolt Szakonyi; Ferenc Fülöp; Norbert De Kimpe
509-514SYNTHESIS AND REACTIONS OF FURO[3,2-c]QUINOLINES AND FVRO[3,2-c]COUMARINSHisham A. Abd El-Nabi; A. M. Now El-Din
515-520A SIMPLE AND EFFICIENT METHOD FOR THE EPOXIDATION OF α, β-UNSATURATED ALDEHYDES AND KETONES USING AQUEOUS HYDROGEN PEROXIDE-SODIUM ETHOXIDEA. Patra; M. Bandyopadhyay; S. K. Ghorai; D. Mal
520-524AN IMPROVED PREPARATION OF 4-AMINO-3-MERCAPTOBENZOIC ACIDRobert C. Lang; Craig M. Williams; Mary J. Garson
524-525IMPROVED SYNTHESIS OF 1,3-DIAZA-6-ADAMANTANONETimothy A. Lewis; Gurmit Grewal

Volume 35, Issue 4 (2003)

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361-368EFFECT OF CATIONS, SUBSTRATES AND TEMPERATURE ON THE MICROWAVE-ASSISTED SAPONIFICATION OF BENZOIC AND MESITOIC ESTERSLaurence Perreux; André Loupy
369-374TFFH AS A USEFUL REAGENT FOR THE CONVERSION OF CARBOXYLIC ACIDS TO ANILIDES, HYDRAZIDES AND AZIDESA. El-Fahm; M. Abdul-Ghani
375-382SYNTHESIS OF S-ARYL-D,L-CYSTEINES AND INCORPORATION INTO KERATIN SEQUENCESAvram Gold; Tae-Gyu Nam; K. Jayaraj; R. Sangaiah; David G. Happer; Louise M. Ball; John E. French; Leena A. Nylander-French
383-387POLYMER-SUPPORTED 4-(PHENYLSELENO)MORPHOLINE AS A USEFUL α-SELENENYLATING AGENT FOR SATURATED ALDEHYDES. A HIGHLY EFFICIENT ROUTE TO α-HALOALDEHYDES ON SOLID PHASEShou-Ri Sheng; Xian Huang
387-390EFFICIENT SYNTHESIS OF 4-ISOCYANO-2,2,6,6-TETRAMETHYLPIPERIDINE-1-OXYLJerzy Zakrzewski; Jaroslaw Hupko
391-396NEW EFFICIENT SYNTHESIS OF 2-ALKYLTHIO-5-BENZYLJDENE-4H-IMIDAZOLIN-4-ONESMing-Wu Ding; Yong Sun; Xiao-Peng Liu; Zhao-Jie Liu
397-400SYNTHESIS OF THE DASYCARPIDONE SKELETONNesimi Uludag; Tahsin Uyar; Süleyman Patir
401-408SOLVENT-FREE SYNTHESIS OF SPIRO[3H-INDOLE-3,2′-THIAZOLIDINES]Anshu Dandia; Ruby Singh; Kapil Arya
409-411ALTERNATIVE SYNTHESIS OF N,N′-DJPHENYLTHIOUREA AND ITS ANALYSIS BY LC-MSYu-Chun Xiong; Zhi-Min Zong; Fa-Qin Jiang; Xin-Hua Yuan; Xiao-Hua Wang; Ya-Fei Ji; Li Xu; Hong-Zhan Xiao; Lin-Tao He; Chun-Qi Li; Xian-Yong Wei
412-414CHLOROMETHYL METHYL SULFONE BY OXIDATION OF CHLOROMETHYL METHYL SULFIDEMieczyslaw Makosza; Marek Surowiec
414-417SIMPLE METHODOLOGY FOR THE PURIFICATION OF AMINO ACIDSAntonio José Mota; Elena Castellanos; Eusebio Juaristi
418-420A SHORT SYNTHESIS OF ar-TODOMATUIC ACID AND DIHYDRO-ar-TURMERONE BY THE HECK REACTIONS. B. Solabannavar; P. P. Wadgaonkar; U. V. Desai; R. B. Mane
420-422A CONVENIENT SYNTHESIS OF 1,1′- and 1,2′-DINAPHTHYLMETHANONESL. Wu; Z. M. Zong; X. Y. Wei; Y. M. Qin; G. L. Zou
422-425SYNTHESIS OF 2,5- AND 2,6-DINITROFLUOROBENZENES AND RELATED HYDROQUINONESE. J. Behrman; Ssuhen Chen
426-429SYNTHESIS OF 2,5-DISUBSTITUTED 1,3,4-OXADIAZOLES USING DRY MEDIAM. Kidwai; R. Mohan
429-432A NEW APPROACH TO THE SYNTHESIS OF 1,3-AMINOALCOHOLS FROM MESO CYCLIC ACID ANHYDRIDEJia-Hai Ye; You Huang; Ru-Yu Chen
433-438REACTIONS OF INDOLE-2,3-DIONES WITH 3-AMINOPROPANOLAnshu Dandia; Meha Sati; Sangeeta Sanan; R. Joshi
439-443METHYL 2-CHLORO-4-FLUOROPHENYLTRIOACETATE AS A NEW INTERMEDIATE IN THE SYNTHESIS OF PESTICIDESZhenyuan Xu; Xiaohua Du; Jianbo Gu

Volume 35, Issue 3 (2003)

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239-306RECENT ADVANCES IN THE SYNTHESIS OF RETINOIDSBeatriz Domínguez; Rosana Alvarez; Angel R. de Lera
307-360FRAGMENTATION AND CLEAVAGE REACTIONS MEDIATED BY SAMARIUM IODIDE. PART 2: α- AND β-ELIMINATION REACTIONS OF C-X SUBSTRATESD. Bradley; G. Williams; Judy Caddy; Kevin Blann

Volume 35, Issue 2 (2003)

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141-205HETEROSUBSTITUTED CARBOCYCLIC α-AMINO ACIDS. A REVIEWM. L. Gelmi; D. Pocar
207-214FACILE SYNTHESIS OF ISOXAZOLE 4- AND 5-CARBALDEHYDES AND THEIR CONVERSION TO ISOXAZOLYL-1, 4-DIHYDROPYRIDINESY. R. Mirzaei; S. Bavili-Tabrizi; M. Hashemi-Gohare; H. Zare-Neirizi; L. Edjlali
215-219NOVEL SYNTHESIS OF FUNCTIONALIZED 2-PYRROLIDINONES via UNSATURATED IMIDOYL CYANIDESE. Rosas Alonso; K. Abbaspour Tehrani; M. Boelens; A. V. Tkachev; Z. Szakonyi; F. Fülöp; N. De Kimpe
219-222SELECTIVE TRANSESTERIFICATION OF METHYL AND ETHYL β-KETOESTERSB. P. Bandgar; S. S. Pandit; L. S. Uppalla
223-225NEW METHOD FOR SYNTHESIS OF S-METHYL-N-ARYLTHIOCARBAMATESDawei Cui; Zhibin Li; Runhui Liu; Gonghua Song; Xuhong Qian
225-227A HIGH YIELD, SELECTIVE SYNTHESIS OF 1,3,5-TRIMETHOXYBENZENEYa-Fei Ji; Zhi-Min Zong; Xan-Yong Wei
228-231SYNTHESIS OF N- (4-AMINOPHENYL) MONOAZACROWN ETHERSWei Zeng; Ying Du; Hongbo Li; Xiaoxia Lu; Shengying Qm
231-238SYNTHESIS OF α-HYDROXYTAMOXIFEN AND ITS 4-HYDROXY ANALOGM. R. Lashley; C. W. Dicus; K. Brown; M. H. Nantz

Volume 35, Issue 1 (2003)

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1-140CHIRAL ENOLATE EQUIVALENTS. A REVIEWClaude Spino

Volume 34, Issue 6 (2002)

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559-583SYNTHETIC APPROACHES TOWARD THE BENGAMIDE FAMILY OF ANTITUMOR MARINE NATURAL PRODUCTS. A REVIEWFrederick R. Kinder Jr
585-608THE ZINCKE REACTION. A REVIEWWei-Chieh Cheng; Mark J. Kurth
609-642THE BIRCH REDUCTION OF STEROIDS. A REVIEWHélène Pellissier; Maurice Santelli
643-646CONVENIENT SYNTHESIS OF DI(n-OCTADECYL)AMINE AND DI(n-HEXADECYL)AMINELuciano Lattuada; Fulvio Uberti
647-651IODINATION OF AROMATIC COMPOUNDS UNDER MILD AND SOLVENT-FREE CONDITIONSAbdol R. Hajipour; Arnold E. Ruoho
652-655PREPARATION OF 5,10,11,11a-TETRAHYDRO-1H, 3H-THIAZOLO[2,3-c]-AND 5,10,11,11a-TETRAHYDRO-1H, 3H-THIAZOLO[4,3-c]-[1,4]BENZODIAZEPINESAlexey B. Dyatkin; Bruce E. Maryanoff
655-657FACILE PREPARATION OF trans-2,3-bis(-tert-BUTYLAMINOMETHYL) NORBORNENEJ. H. Wynne; W. M. Stalick
658-664SYNTHESIS OF 1-[4-(1,5-DIALKYL-1H-1,2,4-TRIAZOL-3-YL)]BENZYL-1H-INDOLES AND 5,6-DIHALOQUINOLONESYaseen A. Al-Soud; Rana F. Halah; Najim A. Al-Masoudi
665-670A CONVENIENT REDUCTION OF HIGHLY FUNCTIONALIZED AROMATIC CARBOXYLIC ACIDS TO ALCOHOLS WITH BORANE-THF AND BORON TRIFLUORIDE-ETHERATEM. H. Chen; E. Iakovleva; S. Kesten; J. Magano; D. Rodriguez; K. E. Sexton; J. Zhang; H. T. Lee
671-680INDEXES

Volume 34, Issue 5 (2002)

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441-465SYNTHESES OF l-IDURONYL SYNTHONS. A REVIEWHélène Pellissier
467-492RECENT PROGRESS IN THE ASYMMETRIC SYNTHESIS OF α-SUBSTITUTED PROPARGYLAMINESJ. Blanchet; M. Bonin; L. Micouin
493-4992-ALKYLINDOLE-3-CARBOXYLATE ESTERS BY A TANDEM REDUCTION-ADDITION-ELIMINATION REACTIONRichard A. Bunce; Marty H. Randall; Kirby G. Applegate
499-502ONE-POT SYNTHESIS OF SELENOESTERS FROM ALKYNYL ARYL SELENIDESShouri Sheng; Xiaoling Liu
502-507NaBH4-MnCl2, FOR IMPROVED REDUCTION OF β-KETO ESTERS ATTACHED TO A CHIRAL AUXILIARY. COMPARISON WITH Zn(BH4)2P. R. R. Costa; C. V. F. Lima; P. R. Paiva; S. Pinheiro
507-511A FACILE AND EFFICIENT ZINC-PROMOTED ALLYLATION OF CARBONYL COMPOUNDSChinpiao Chen; Wen-Chin Dai; Han-Gen Chang
511-514SYNTHESIS OF N-PROTECTED 1H-INDOLE-5-CARBOXYLIC ACIDS WITH ALDOSE REDUCTASE INHIBITORY POTENTIALIoannis Nicolaou; Nazlaa Zaher; Vassilis J. Demopoulos
514-517PREPARATION OF 3-(TRIFLUOROMElTHYL)COUMARINSWojciech Dmowski; Krystyna Piasecka-Maciejewska
517-520A SIMPLIFIED SYNTHESIS OF ETHYL 5-CHLORO-4-FLUORO-1H-INDOLE-2-CARBOXYLATE AND ETHYL 5-CHLORO-6-FLUORO-1H-H-INDOLE-2-CARBOXYLATERomano Silvestri; Gabriella De Martino; Gianluca Sbardella
521-524A CONCISE SYNTHESIS OF CHIRAL 3-HYDROXYMETHYL-5-ISOPROPYL MORPHOLINES FROM VALINOLLing Huang; Marilyn M. Olmstead; Mark J. Kurth
525-530A NOVEL METHOD FOR THE SYNTHESIS OF FORMYL AND HYDROXYMETHYL DERIVATIVES OF 4H-PYRAN-4-ONEM. Ghandi; Y. Bayat; R. Teimuri-Mofrad
531-537SCALABLE SYNTHESES OF Nα-BENZYLOXYCARBONYL-l-ORNITHINE AND OF Nα-(9-FLUORENYLMETHOXY)CARBONYL-l-ORNITHINEEEłżbieta Masiukiewicz; Stanislaw Wiejak; Barbara Rzeszotarskat
537-540A NOVEL AND EFFICIENT BIOMIMETIC HYDROLYSIS OF OXIRANES TO 1,2-DIOLS CATALYSED BY β-CYCLODEXTRIN IN WATER UNDER NEUTRAL CONDITIONSM. Anjun Reddy; L. Rajender Reddy; N. Bhanumathi; K. Rama Rao
540-543IMPROVED LARGE SCALE SYNTHESIS OF 2-TRIMETHYLSILOXY-1,3-BUTADIENERoy T. Uyeda; Phong Vu; Daniel D. Holsworth
543-545AN EFFICIENT SYNTHESIS OF 1,3-DIMETHYL-4-(PHENYLSULFONYL)-4H-FURO[3,4-b]INDOLEJun Jiang; Gordon W. Gribble
545-549A SIMPLE PREPARATION OF N,N-DIMETHYL-N′-ALKYL (ARYL) SULFONYLFORMAMIDINESA. L. Silva; A. Covarrubias-Zúñiga; L. A. Maldonado
549-552A RAPID SYNTHESIS OF DIISOPROPYL 4-(CHLOROMETHYLBENZYL) AND 4-(BROMOMETHYLBENZYL) PHOSPHONATESBernard Moreau; Paul-Alain Jaffrès; Didier Villemin
552-557SYNTHESIS OF CALIX[4]ARENE DIAZACROWN CONTAINING m-XYLYLENE PHENOL SUBUNITXiao-Bing Wan; Guo-Yuan Lu; Zhu Bo; Chum-Ming Jin; Fang Liu

Volume 34, Issue 4 (2002)

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337-366THE SYNTHESIS OF SUCCINIC ACIDS AND DERIVATIVES. A REVIEWKristjan M. Arason; Stephen C. Bergmeier
367-404SYNTHESES AND TRANSFORMATIONS OF PIPERAZINONE RINGS. A REVIEWChristopher J. Dinsmore; Douglas C. Beshore
405-415AN IMPROVED SYNTHESIS OF (S)- OR (R)-N-BcE-PROTECTED 1,5-BENZOTHIAZEPINE DERIVATIVESMuriel Amblard; Monique Calmès; Virginie Roques; Samuel Tabet; Albert Loffet; Jean Martinez
417-424OPPI BRIEFS SYNTHESIS AND EXTRACTION STUDIES OF A NOVEL TETRA-CALIX[4]ARENEAydan Yilmaz; Shahabuddin Memon; Mustafa Yilmaz
425-429SYNTHESIS OF SPIRO-1-PYRAZOLINES BY THE REACTION OF Z-3-ARYLIDENE-1-THIOFLAVANONES WITH DIAZOMETHANEAlbert Lévai
430-432SYNTHESIS OF 2,4-DIMETHYL-5-IODOBENZALDEHYDEM. R. Akula; J. H. Zhang; G. W. Kabalka
432-435A MULTI-GRAM SYNTHESIS OF 1,2:5,6-DI-O-ISOPROPYLIDENE 3-C-TRIMETHYLSILYLMETHYL-α-D-ALLOFURANOSE. AN IMPROVED PREPARATION OF 3-C-HYDROXYMETHYL-α-D-GLUCO-AND 3-C-METHYL-α-D-ALLOFURANOSE DERIVATIVESMasuo Funabashi; Yukinori Ooshiro
436-440SYNTHESIS OF O-PROTECTED MANDELAMTOE AND ITS ELABORATION TO 5-HYDROXY-l,5-DIPHENYLHYDANTOINA. Papakyprianou; A. W. Parkins; P. D. Prince; J. W. Steed

Volume 34, Issue 3 (2002)

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219-269PREPARATION, PROPERTIES AND SYNTHETIC APPLICATIONS OF 2H-AZIRINES A REVIEWFrancisco Palacios; Ana María Ochoa de Retana; Eduardo Martínez de Marigorta; Jesús Manuel de los Santos
271-319NEW DEVELOPMENTS IN THE USE OF ENANTIOMERICALLY ENRICHED SULFOXIDW IN STEREOSELECTIVE SYNTHESESChing-Cheng Wag; Horng-Chih Huang; David B. Reitz
321-325AN IMPROVED PREPARATION OF 4-AMINOPYRIMIDINES-5-CARBOXALDEHYDEThomas W. Bell; Daniel L. Beckles; Michele Debetta; Brian R. Glover; Zheng Hou; Kar-Yan Hung; Alisher B. Khasanov
326-331CONCISE SYNTHESIS OF N-PROTECTED CARBOXYALKYL ETHER AMINESMaciej Adamczyk; Jeffrey R. Fishpaugh; Mohan Thiruvazhi
332-335REDUCTION OF PYRIDYL CARBINOLS WITH SODIUM BOROHYDRIDE/TRIFLUOROACETIC ACIDCharles F. Nutaitis; Thomas J. Greshock; Stephen R. Houghton; Lynn N. Moran; Melissa A. Walter

Volume 34, Issue 2 (2002)

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109-147SELECTED METHODS FOR THE REDUCTION OF THE AZIDO GROUPD. Amantini; F. Fringuelli; F. Pizza; L. Vaccaro
149-167NUCLEOSIDES WITH A CARBON BRIDGE BETWEEN SUGAR AND NUCLEOBASE: THE CHEMISTRY OF 1′-HOMONUCLEOSIDES AND REVERSED NUCLEOSIDES. A REVIEWClemens Lamberth
169-175DEPROTECTION OF TRIMETHYLSILYL AND OF TETRAHYDROPYRANYL ETHERS AND OF ETHYLENE ACETALS WITH BENZYLTRIPHENYLPHOSPHONIUM CHLOROCHROMATEA. R. Hajipour; S. E. Mallakpour; I. M. Baltorkt; H. Backnezhad
177-182METHYL 6-METHOXY-1-OXOINDAN-4-CARBOXYLATEMartin G. Banwell; Scott G. Stewart
182-187AN EFFICIENT ONE-STEP CONVERSION OF BILIVERDINS TO 14-FORMYLTRIPYRRINONESPeng Wang; Yi Zhang; Qingqi Chen; Jin Shi
187-190A SHORT AND HIGHLY ENANTIOSELECTIVE SYNTHESIS OF (6R)-UNDECYLTETRAHYDROPYRAN-2-ONE, THE PHEROMONE OF VESPA ORIENTALISGrzegorz Juszkiewicz; Janusz Jurczak
190-193AN IMPROVED PREPARATION OF 3-(5-BENZOFURANYL)-L-ALANINEGiorgio Ortar
194-198MICROWAVE-ASSISTED SYNTHESIS OF SUBSTITUTED CYCLOPROPYL, FERROCENYL KETONES BY A SULFUR YLIDE REACTION UNDER SOLID-STATE CONDITIONSQi-Hai Xu; Bao-Hua Chen; Yong-Xiang Ma; Wan-Yi Liu; Yong-Min Liang
198-203A SIMPLE SYNTHESIS OF 1-ARYL-POLYENESElena Pini; Elisabetta Rossi; Giuseppe Celentano; Riccardo Stradi
204-207A GENERAL SYNTHESlS OF MACROCYCLIC ESTERSRyszard Ostaszewski; Pawel Ćwierzyhski; Janusz Jurczak
208-213A NOVEL SYNTHESIS OF 2,2,4,5-TETRASUBSTITUTED-1,3-DITHIOLESJian-Ping Zou; Xiang-Shan Wang; Zhi-Tao Wang; Zhong-E Lu
213-217TETRAHYDROFURAN RING-OPENING WITH ACYLOXYPHOSPHONIUM IODIDE CATALYZED BY SAMARIUM TRIIODIDEYunkui Liu; Yongmin Zhang

Volume 34, Issue 1 (2002)

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1-25RECENT SYNTHESES OF EPIBATIDINE. A REVIEWHoracio F. Olivo; Michael S. Hemenway
27-85RECENT DEVELOPMENTS IN THE SYNTHESIS, CHEMICAL MODIFICATIONS AND BIOLOGICAL APPLICATIONS OF SULFUR MODIFIED NUCLEOSIDES, NUCLEOTIDES AND OLIGONUCLEOTIDESStéphane Chambert; Jean-Luc Décout
87-94SYNTHESIS AND CHARACTERIZATION OF PIPERAZINE-2,6-DIONESTeresa Mancilla; Lourdes Canillo; Luis S. Zamudio-Rivera; Hiram I. Beltrán; Norberto Farán
95-97AMIDES BY MICROWAVE-ASSISTED DEHYDRATION OF AMMONIUM SALTS OF CARBOXYLIC ACIDSYanqing Peng; Gonghua Song
98-102AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1-ARYL-4-HYDROXY-1H-PYRAZOLESClemens Lamberth
103-107SYNTHESIS OF THE FOUR STEREOISOMERS OF 1,1,1-TRIFLUOROBUTANE-2,3-DIOLCarlo F. Morelli; Giovanna Speranza; Lavinia Durì; Paolo Manitto

Volume 33, Issue 6 (2001)

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515-564SYNTHESIS AND SYNTHETIC UTILITY OF 3-ISOXAZOLOLSUlrik S. Sørensen; Povl Krogsgaard-Larsen
565-602FRAGMENTATION AND CLEAVAGE REACTIONS MEDIATED BY SmI2. PART 1: X-Y, X-X AND C-C SUBSTRATESD. Bradley; G. Williams; Kevin Blann; Judy Caddy
603-613SYNTHESIS OF JULOLIDINE DERIVATIVESJoel M. Kauffman; Steven J. Imbesi; Mohammed Abdul Aziz
615-619RUTHENIUM CATALYZED OXIDATION OF HALOINDOLES TO ISATINSGordon W. Gribble; Yanbing Liu
621-623A CONVENIENT PREPARATION OF 4-(t-BUTYLOXYCARBONYLAMINO)ANILINEB. Nageswara Rao; T. Venkateswarlu; P. Gundu Rao; Murali K. Divi
625-632INDEXES

Volume 33, Issue 5 (2001)

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411-454RECENT ADVANCES IN THE SYNTHESIS OF PYRROLESVitor F. Ferreira; Maria Cecília B. V. de Souza; Anna C. Cunha; Letícia O. R. Pereira; Maria L. G. Ferreira
455-476FUNCTIONALIZATION OF THE 18-METHYL GROUP OF STEROIDS. A REVIEWHélène Pellissier; Maurice Santelli
477-485SYNTHESIS OF COELENTERAZINEMaciej Adamczyk; Donald D. Johnson; Phillip G. Mattingly; You Pan; Rajarathnam E. Reddy
487-499SYNTHESIS OF METHYL (E)-4-[2-(2,3-DIHYDRO-3-METHYL-3-HYDROXYMETHYLBENZO[b]THIEN-5-YL)-1-PROPENYL]BENZOATE [(E)-3], METHYL (E)-4-[2-(2,3-DIHYDRO-3-METHYL-3-HYDROXYMETHYL-5-BENZOFURANYL)-1-PROPENYL] BENZOATE [(E)-4], AND METHYL (E)-4-[2-(2,3-DIHYDRO-3,3-DIMETHYL-5-BENZOFURANYL)-3-HYDROXY-1-PROPENYL]BENZOATE [(E)-7] AS POTENTIAL METABOLITES OF SELECTED HETEROAROTINOIDS WITH FUSED FIVE-MEMBERED RINGSJonathan B. Gale; Jozef Klucik; Shankar Subramanian; K. Darrell Berlin
501-505A NOVEL SYNTHESIS OF 2-ACYLPYRIDINES via INVERSE ELECTRON DEMAND DIELS-ALDER REACTION OF 5-ACYL-1,2,4-TRIAZLNESA. Rykowski; E. Olender; D. Branowska; H. C. van der Plas
505-514SYNTHESIS OF HAPTEN PHOSPHORAMIDITESM. Adamczyk; D. D. Johnson; P. G. Mattingly; R. E. Reddy

Volume 33, Issue 4 (2001)

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315-334RECENT PROGRESS IN THE SYNTHESIS AND REACTIVITY OF AZETIDINE-2,3-DIONES. A REVIEWBenito Alcaide; Pedro Almendros
335-340BASE CATALYSIS IN THE WILLGERODT-KIM)LER REACTIONJacques H. Poupaert; Karim Bouinidane; Marc Renard; Didier M. Lambert; Majed Isa
341-349SYNTHESIS AND CHARACTERIZATION OF NEW 2-SUBSTITUTED ISOINDOLINE DERIVATIVES OF α-AMINO ACIDSTeresa Mantilla; Lourdes Carrillo; Luis S. Zamudio-Rivera; Hiram I. Beltrán; Norberto Farfán
351-356ADDITION OF ACETONITRILE ANIONS TO UNSATURATED SYSTEMS UNDER ULTRASONICALLY DISPERSED POTASSIUM SYSTEMYang Gao; Hui Wang; Minghua Xu; Hongzhen Lian; Yi Pan; Yaozeng Shi
357-361IMPROVED SYNTHESIS OF ALKYL DIACETYLACETATESS. J. Bingham; J. H. P. Tyman
361-368SYNTHESIS OF 6-HALO-1,2-BENZISOXAZOLES, CHROMENO-6,7-ISOXAZOLES AND CHROMENO-6,7-OXAZOLESLenuta Cires; Harry Ofenberg; Cotinica Craita
369-371AN IMPROVED SOLVENT-FREE PREPARATION OF 2-IMIDOYLPHENOLSCristina Cimarelli; Gianni Palmieri; Emanuela Volpini
372-375STEREOSELECTIVE SYNTHESIS OF (2E)-CINNAMANILIDES via DESULFONYLATION OF (2E)-α-AMIDO-α, β-UNSATURATED SULFONES BY SAMARIUM/GLACIAL ACETIC ACID/ETHANOL SYSTEMYunkui Liu; Yongmin Zhang
376-379MICROWAWASSISTED SYNTHESIS OF HEXASUBSTITUTED CYCLOTRIPHOSPHAZENESChengfeng Ye; Weimin Liu; Yunxia Chen; Zhongwen Ou
379-381A FACILE SYNTHESIS OF W-BENZYLOXYCARBONYL-(S)-2-AMINO-3-(DIMETHYLAMINO)PROPANOICACIDRyszard Andruszkiewicz; Aleksandra Walkowiak
381-386AN EXPEDITIOUS SOLVENTLESS SYNTHESIS OF ISOXAZOLESM. Kidwai; P. Sapra
386-390TWO-FOLD CYCLOALKYLATIONS OF A BICYCLO[3.3.0]OCTANE-3,7-DIONEEckehard Volker Dehmlow; Hans-Jorg Breyholz; Beate Neumann; Hans-Georg Stammler
391-394A NEW FACILE AND EXPEDITIOUS SYNTHESIS OF N-HYDROXY-N′-PHENYLOCTANEDIAMJDE, A POTENT INDUCER OF TERMINAL CYTODIFFERECNTIATIONAntonello Mai; Monica Esposito; Gianluca Sbardella; Silvio Massa
395-400EFFICIENT SOLVENT-FREE MICROWAVE-ASSISTED ESTERIFICATION OF FUSEL OIL USING p-TsOH AND H3PW12O40 AS CATALYSTSE. R. Pérez; N. C. Carnevalli; P. J. Cordeiro; U. P. Rodrigues-Filho; D. W. Franco
400-405THE PREPARATION OF 1-ALLYLURACIL. N(1)-ALKYLATION OF N(3)-PROTECTED URACIL DERIVATIVESZdzislaw Paryzek; Bartlorniej Tabaczka
405-409CONVENIENT N-PROTECTION OF L-PYROGLUTAMIC ACID ESTERSRahul Jain

Volume 33, Issue 3 (2001)

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203-303NEW TRENDS IN PEPTIDE COUPLING REAGENTSFernando Albeiicio; Rafael Chinchilla; David J. Dodsworth; Carmen Nájera
305-310DRY ARENEDIAZONIUM NITRATES FROM AROMATIC AMINES AND UREAS WITH NITROGEN DIOXIDE ADDUCTS OF DIOXANE AND OF TRIBUTYL PHOSPHATEZ. Zhang; X. Liu; Q. Zhang; S. Zhang; T. Huang
311-313A PRACTICAL SYNTHESIS OF (3aα, 6aα)-1,3-DIBENZYL HEXAHYDRO-1H-THIENO[3,4-d]IMIDAZOL-2(3H)-ONEFen-Er Chen; Ge Meng; Yan-Ping He; Yu Cheng; Xiu-Hong Ling

Volume 33, Issue 2 (2001)

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103-172ASYMMETRIC 1,3-DIPOLAR CYCLOADDITIONS FOR THE CONSTRUCTION OF ENANTIOMERICALLY PURE HETEROCYCLES. A REVIEWStaffan Karlsson; Hans-Erik Högberg
173-179REACTION OF METHACRYLOYL ISOCYANATE WITH SULFONIUM AND PHOSPHONIUM YLIDESTaizo Hatta; Shojiro Ishibashi; Otohiko Tsuge
181-184A NOVEL SYNTHESIS OF 2H-1,4-BENZOSELENAZINES FROM (o-NITROPHENYL)DISELENIDES AND ω-BROMOKETONES PROMOTED BY Sm/TiCl4 SYSTEMWeihui Zhong; Yongmin Zhang; Xiaoyuan Chen
185-187LOW VALENT TITANIUM INDUCED ONE-POT SYNTHESIS OF IMIDAZOLIDINESZhifang Li; Yongmin Zhang
187-190REDUCTIVE COUPLING OF CARBONYL COMPOUNDS TO PINACOLS WITH SAMARIUM/TMSCI SYSTEMMingxin Yu; Yongmin Zhang
190-194A NEW AND CONVENIENT SOLVENT-FREE METHOD FOR THE PREPARATION OF 1,4-DIARYL THIOSEMICARBAZIDESJian-Ping Li; Qian-Fu Luo; Yu-Lu Wang; Hong Wang
194-198SYNTHESIS OF 2-CYANO-3-DIMETHYLAMINO-N-PHENYLACRYLAMIDES USING THE VILSMEER REACTIONS. Selvi; P. T. Perumal
198-201BORON TRIFLUORIDE MEDIATED, ONE-POT SYNTHESIS OF 3-METHYL-1,2-DIHYDRONAPHTHALENESRama R. Malladi; George W. Kabalka

Volume 33, Issue 1 (2001)

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1-58CHEMICAL AND BIOCHEMICAL HYDROXYLATIONS OF STEROIDS. A REVIEWHélène Pellissier; Maurice Santelli
59-74RECENT PROGRESS IN THE SYNTHESIS OF bis-TRIAZENESKeith Vaughan
75-80SYNTHESIS OF 2(3H)-BENZOXAZOLINONE DERIVATIVES AS POTENTIAL MELATONIN RECEPTOR LIGANDSSaid Yous; Frédérique Klupsch; Isabelle Lesieur
81-86SYNTHESIS OF NOVEL TETRAPYRROLES AND THEIR ZINC COMPLEXESYi Zhang; Jin Shi
87-90DIRECT REGENERATION OF CARBONYL COMPOUNDS FORM OXIMES WITH PEG-NO2Xinming Liu; Qingzhi Zhang; Shensong Zhang; Jinming Zhang
91-95PREPARATION OF 2-PHENYL-4-(1H-PYRAZOL-5-YL)QUINOLINESS. P. Grant; D. R. Hurst; T. L. Cordray; C. F. Beam
95-100A PRACTICAL METHOD FOR THE SYNTHESIS OF PHENOPHTHALEIN SPIROLACTAMSMaciej Adamczyk; Jonathan Grote
100-1021,3-DIPOLAR CYCLOADDITIONS OF 3-PHENYLSYDNONE WITH ACETYLENE DICARBOXYLATES IN SUPERCRITICAL CARBON DIOXIDEA. E. McGowin; L. Jackson; L. W. Marshall; K. Tumbull

Volume 32, Issue 6 (2000)

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505-546RECENT PROGRESS IN ISOLATION, BIOACTIVITY EVALUATION AND TOTAL SYNTHESIS OF DIARYLHEPTANOIDSJieping Zhu; G. Islas-Gonzalez; M. Bois-Choussy
547-555A CONTINUOUS PROCEDURE FOR PREPARATION OF para FUNCTION ALIZED AROMATIC THIOLS USING NEWMAN-KWART CHEMISTRYSechoing Lin; Brian Moon; Kenneth T. Porter; Craig A. Rossman; Thomas Zennie; James Wemple
557-561DEHYDRATION OF CEDROL TO α-CEDRENE USING COPPER(II) SULFATE AND OTHER ACIDIC SALTSEdmund J. Eisenbraun; Kirk W. Payne; Jeremy S. Bymaster
563-567UNEXPECTED DIECKMANN CONDENSATION IN THE SYNTHESIS OF METHYL 6-(6-METHOXY-2-NAPHTHYL)-6-OXOHEXANOATE WITH AN ARYLCADMIUM REAGENTCarmen Balo; Franco Fernández; Xerardo García-Mera; Carmen López
567-570REDUCTIVE COUPLING OF KETONES WITH IMINES PROMOTED BY THE TITANIUM TETRACHLORIDE/SAMARIUM SYSTEMYongmin Ma; Yongmin Zhang
571-573A FACILE SYNTHESIS OF ARYL ISOTHIOCYANATES FROM ARYLAMINESZhibin Li; Xuhong Qian; Zhi Liu; Zhong Li; Gonghua Song
573-577SYNTHESIS OF 1,9-DIAMIDINIUMACRIDINE AS A POTENTIAL RECEPTOR FOR PHOSPHATE ESTER RECOGNITIONR. P. Dixon; J. S. Snyder; L. Bradley; J. Linnenbrink
577-580A SYNTHESIS OF (E)-ω-CARBOXY-2-ALKENOIC ESTERSRichard A. Bunce; Demck M. Herrod
581-584A CONVENIENT SYNTHESIS OF cis-UROCANIC ACID, AN ENDOGENOUS IMMUNOSUPPRESSANTTaj Mohammad; Harry Morrison
584-588[2+2] CYCLOADDITIONS OF BENZOFURAN-3(2H)-ONE ENAMINES WITH DIMETHYL ACETYLENEDICARBOXYLATEN. Tunoglu; G. Okay
588-592SELECTIVE CATALYTIC OXIDATION OF ALCOHOLS USING HYDROGEN PEROXIDEJ. H. Wynne; C. T. Lloyd; D. R. Witsil; G. W. Mushrush; W. M. Stalick
593-596A LITHIATION APPROACH TO 5-SUBSTITUTED-1-BENZENESULFONYLPYRAZOLESKenneth Turnbull; Andre P. Brower
596-600SILICA GEL PROMOTED SOLVENT-FREE SYNTHESIS OF ARYLCARBINOLS AND FERROCENYLCARBINOLSWan-Yi Liu; Qi-Hai Xu; Yong-Xiang Ma
600-603SYNTHESIS OF THYMYL ETHERS AND ESTERS USING POLYMER-SUPPORTED THYMOL ANIONP. P. Kumbhar; U. R. Kapadi; D. G. Hundiwale; S. B. Attarde; P. M. Dewang; N. S. Pawar
605-615INDEXES

Volume 32, Issue 5 (2000)

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409-451AN OVERVIEW OF SYNTHETIC STUDIES OF ANTIBIOTICS FROM MYXOBACTERIADavid R. Williams; Jie Jack Li; Richard H. Hutchings
453-459SYNTHESIS OF NEW FURAN-DERIVED N-SUBSTITUTEDAMINOMETHANEPHOSPHONATESJaroslaw Lewkowski; Monika Rzezniczak; Romuald Skowronski
461-468AN IMPROVED SYNTHESIS OF ±18 METHYL EICOSANOIC ACIDDarren J. Cundy; Paul A. Gurr
469-479REACTION OF N-[(TRIMETHYLSILYL)METHYL]CARBODIIMIDES WITH BIFUNCTIONAL NUCLEOPHILESOtohiko Tsuge; Taizo Hatta; Masanori Shinozuka; Hideki Tashiro; Hironori Maeda; Akikazu Kakehi
481-485NEW METHOD FOR SYNTHESIS OF (ω-CHLOROALKYL) PYRROLESBin Tu; Changqi Wang; Jinshi Ma
485-488EFFICIENCY OF THE URUSHIBARA NICKEL CATALYZED ATMOSPHERIC HYDROGENATION IN THE SYNTHESIS OF ANILINE DERIVATIVESX. Liu; T. Jia; J. Chen; Z. Jiang; H. Zhang; X. Huang
488-490AN IMPROVED SYNTHESIS OF α-METHOXY-α-(TRWLUOROMETHYL)-PHENYLACETIC ACID (MOSHER'S ACIDKeith R. Buszek; Nagaaki Sato
491-492IMPROVED SYNTHESIS OF (R)- AND (S)-β-METHYL-γBUTYROLACTONEKeith R. Buszek; Nagaaki Sato
493-497AN EFFICIENT SYNTHESIS OF ENANTIOPURE 3-CHLOROSTYRENE OXIDE via OXAZABOROLIDINJGCATALYZED REDUCTIONOh Kyoung Choi; Byung Tae Cho
498-501A NOVEL SYNTHESIS OF 3-SUBSTITUTED MDAZOLIDIN-2-ONE-1-CARBONYL CHLORIDESWeike Su; Kewei Huang; Yongmin Zhang
502-504IMPROVED SYNTHESIS OF 3,5,6-TRIFLUOROPYRIDIN-2,4-DIOLElsa Anselmi; Jean-Claude Blazejewski; Claude Wakselman

Volume 32, Issue 4 (2000)

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307-330RECENT PROGRESS ON THE SYNTHESIS OF CYATHANE TYPE DITERPENES. A REVIEWDennis L. Wright; Christopher R. Whitehead
331-365ASYMMETRIC CATALYSIS OF ACYL TRANSFER BY LEWIS ACIDS AND NUCLEOPHILES. A REVIEWAlan C. Spivey; Adrian Maddaford; Alison J. Redgrave
367-372SYNTHESIS OF FLUORESCENCE PROBES WITH A 2,6-AMINONAPHTHALENE-CARBONYL CHROMOPHORECarmen Balo; Franco Fernández; Xerardo García-Mera; Carmen López
373-376AROMATIC HYDROXYLATION BY A NEW CUPRIC NITRATE-H2O2-PHOSPHATE BUFFER SYSTEMAayesha Nasreen; Srinivas R. Adapa
376-379A CONVENIENT PREPARATION OF METHYL 4-(2-AMINOETHYL)BENZOATEStephen W. Wright
379-381AN EFFICIENT AND FACILE PREPARATION OF 2,2′,4,4′-TETRABROMODIPHENYLAMINEXiaoxia Wang; Cailan Wang; Xiaoyang Wang; Yulu Wang
381-384AN EFFICIENT AND SCALABLE SYNTHESIS OF METHYL 3-HYDROXYMETHYLBENZOATEM. H. Chen; J. G. Davidson; J. T. Freisler; E. Iakovleva; J. Magano
385-390SYNTHESIS OF 1-(p-NITROBENZYL)AZOLES AND 1-(p-NITROBENZYL)BENZAZOLESCarmen Pardo; Sabine Graf; Mar Ramos; Esther Sesmilo; José Elguero
391-394RAPID AND SELECTIVE REGENERATION OF CARBONYL COMPOUNDS FROM THEIR OXIMES UNDER MILD. NEUTRAL AND SOLVENT-FREE CONDITIONSB. P. Bandgar; S. S. Makone
394-397A CONVENIENT AND EFFECTIVE METHOD FOR THE SYNTHESIS OF TETRAOXAQUATERENESRobert Pajewski; Ryszard Ostaszewski; Janusz Jurczak
398-400AN IMPROVED SYNTHESIS OF 2,3-bis(BROMOMETHYL)-1,4-DIMETHOXYBENZENEJørgen Eskildsen; Trine Christensen; Theis Reenberg; Uffe Larsen; Jørn B. Christensen
401-405PREPARATION OF IMIDAZO[2,1-b]THIAZOLES AND THIAZOLO[3,2-a]-BENZIMIDAZOLES USING S-ETHENYLSULFILIMINESKatsuya Ikeda; So-Ichiroh Hata; Yasuhiro Tanaka; Tamotsu Yamamoto
407CORRIGENDUM

Volume 32, Issue 3 (2000)

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205-234AMINES via NUCLEOPHJLIC 1,2-ADDITION TO KETIMINES. CONSTRUCTION OF NITROGEN-SUBSTITUTED QUATERNARY CARBON ATOMS. A REVIEWArno G. Steinig; Denice M. Spero
235-264RECENT ADVANCES IN THE CHEMISTRY OF OXIMESEdgars Ãbele; Edmunds Lukevics
265-269SYNTHESIS OF (S)-(-)-1-[(9-FLUORENYLMETHOXYCARBONYL)AMINO-5-CARBOXYPENTYL]-3-HYDROXYPYRIDINIUM TRIFLUOROACETATEMaciej Adamczyk; Rajarathnam E. Reddy
269-271MICROWAVE-ASSISTED SYNTHESIS OF TRIARYL PHOSPHATESA. D. Sagar; N. A. Shinde; B. P. Bandgar
272-275SIMPLE AND PRACTICAL SYNTHESES OF DIBENZYL, BENZYL ETHYL AND BENZYL METHYL MALONATESAna Luisa Silva; Adrián Covarrubias-zúñiga; Luis Angel Maldonado
276-279A ONE-POT SYNTHESIS OF PYRAZOLO [3,4-b][1,4]OXAZINESM. A. Raslan; F. M. Abd El-Latif; H. H. Otto; K. U. Sadek
280-283A RAPID METHOD FOR THE CYCLIZATION OF 2′-HYDROXYCHALCONES INTO FLAVONESMukta Gupta; Satya Paul; Rajive Gupta; Andre Loupy
284-287RAPID N-ALKYLATION OF CARBAZOLE, PHENOTHIAZLNE AND ACRIDONE UNDER MICROWAVE IRRADIATIONXingjun Fan; Jinmao You; Tianquan Jiao; Ganzu Tan; Xianda Yu
287-290ESTERIFICATION BY MICROWAVE IRRADIATION ON ACTIVATED CARBONXingjun Fan; Keguo Yuant; Caili Hao; Nan Li; Ganzu Tan; Xianda Yu
290-293SYNTHESIS OF 4-BORONO-2-FLUOROPHENYLALANINEG. W. Kabalka; N. K. Reddy; L. Wang; R. R. Malladi
293-297PREPARATION OF bis-[SPIROFLUORENE-9,4′-(1-AZA-2-CYCLOPENTENE)[1,5-a]INDOLINE-8′-YL]SULFONEE. O. Gogritchiani; H. Dürr; Sh. A. Samsoniya
298-301AN OPTIMIZED PREPARATION OF 2,3-DIHYDRO-1-METHYL-4-OXONAPHTHALENE-1-CARBOXYLIC ACIDA. G. Lo Cascio; G. R. Labadie; M. Gonzalez Sierra; R. M. Cravero
302-306FACILE AND EFFICIENT SYNTHESIS OF α-AMINOPHOSPHONATE DERIVATIVES OF 1,3,4-OXADIAZOLE AND 1,3,4-THIADIAZOLEShui-Ming Lu; Ru-Yu Chen

Volume 32, Issue 2 (2000)

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103-122SYNTHESIS OF 3-AZABICYCLO[3.1.0]HEXANES. A REVIEWGrant R. Krow; Kevin C. Cannon
123-152HYDROGEN PEROXIDE AND AIR AS INEXPENSIVE OXIDANTS IN PHASE-TRANSFER CATALYSIS. A REVIEWSabine Schrader; Eckehard Volker Dehmlow
153-159NOVEL STEREOSELECTIVE SYNTHESIS OF E- ARYL ALDOXIME AND KETOXIME O-ETHERSEdgars Abele; Ramona Abele; Juris Popelis; Edmunds Lukevics
161-167A CONVENIENT SYNTHESIS OF 2H-PYRAN-2-ONES AND OF 3- AND 5- BROMO-2H-PYRAN-2-ONESStamatia I. Kotretsou; Minas P. Georgiadis
169-173IMPROVED PROCEDURE FOR THE LARGE SCALE SYNTHESIS OF 1,2,3,4,4a,9b-HEXAHYDRODIBENZOTHIOPHENEJohn C. Dicesare; L. Brian Thompson; Ryan J. Andersen; John Nail
175-183EFFICIENT AND FACILE ROUTES TO NITRONESAlan R. Katritzky; Xilin Cui; Qiuhe Long; Baozhen Yang; Allan L. Wilcox; Yong-Kang Zhang
185-188RATE ACCELERATION OF THE BAYLIS-HILLMAN REACTION USING CRYSTALLINE CYCLODEXTRIN COMPLEXESL. Rajender Reddy; K. Rama Rao
189-192PREPARATION AND REACTIVITY OF CERTAIN OXAPOLYCYCLIC SYSTEMSMichael Sander; Eckehard Volker Dehmlow
192-196AN EFFICIENT OXIDATION OF LONG CHAIN ALKYL METHYL SULFIDES TO SULFOXIDESTamotsu Yamamoto; Tetsushi Hayakawa; Mugi Yoshino; Soh-Ichiroh Hata; Yorinobu Hirayama
197-201LARGE SCALE PREPARATION OF CELL PERMEABLE, NON-PHOSPHATE-CONTAINING GRB2 SH2 DOMAIN INHIBITORSDing-Guo Liu; Zhu-Jun Yao; Yang Gao; Terrence R. Burke Jr.
202-20310a. A CONVENIENT SYNTHESIS OF 3,5-DI-(t-BUTYL)BROMOBENZENE FROM BENZENEZhengning Li; Zhuo Zheng; Huilin Chen

Volume 32, Issue 1 (2000)

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1-40RECENT ADVANCES IN CLAY-CATALYZED ORGANIC TRANSFORMATIONSMilind D. Nikalje; Prodeep Phukan; Arumugam Sudalai
41-45IMPROVED AND EXPEDITIOUS MICROWAVE SYNTHESIS OF ETHYL 1,3-CYCLOHEXADDEN-1-CARBOXYLATENicolas Tesson; Sandrine Deshayes
47-55A NOVEL METHOD FOR THE SYNTHESIS OF 4H-PYRAN-4-ONE DERIVATIVESA. Shahrisa; R. Tabrizi; H. R. Ahsani
57-61AN IMPROVED SYNTHESIS OF HYPERICIN AND RELATED COMPOUNDSEwa Gruszecka-Kowalik; Leon H. Zalkow
63-67SYNTHESIS OF 4-[4-(BROMOMETHYL)-2-OXAZOLYL]-2,6-bis(1,1-DIMETHYLETHYL)PHENOLJohn R. Rizzo; Benjamin A. Anderson; Lawrence J. Heinz; Richard C. Hoying; Jill A. Panetta
69-74SYNTHESIS OF 6-CHLOROMETHYL BENZOTHIAZOLIN-2-ONE AND OF 6-CHLOROMETHYL BENZOXAZOLIN-2-ONEPascal Carato; Saïd Yous; Patrick Depreux
75-79SYNTHESIS AND CHARACTERIZATION OF ISOMERIC 2,5-DJMETHYL-6-PHENYL-3-CYCLOHEXENE-1-METHANOL ANALOGSGary M. Coppola; Robert E. Damon; Michael J. Shapiro; Karl G. Gunderson; Michael X. Kolpak
81-83SILICA GEL CATALYZED PREPARATION OF CINNAMIC ACIDS UNDER MICROWAVE IRRADIATIONH. M. Sampath Kumar; B. V. Subba Reddy; P. Thirupath Rddy; D. Srinivas; J. S. Yadav
84-88SYNTHESIS AND CHARACTERIZATION OF N-ALKYL HYDROXYACETAMIDESLuis S. Zamudio Rivera; Hurdes Carrillo; Teresa Mantilla
88-91AN IMPROVED SYNTHESIS OF 3-CYANO-4-FLUOROBENZYL BROMIDEGary A. Cain
92-94A NOVEL ROUTE TO THYMOL FROM m-CRESOLK. J. Divakar; V. V. Dhekne; B. D. Kulkami; P. L. Joshi; A. S. Rao
94-96SYNTHESIS OF 4,6-DINITROINDOLEVladimir V. Rozhkov; Alexander M. Kuvshinov; Svyatoslav A. Shevelev
96-99A CONVENIENT SYNTHESIS OF N-Boc-4-FORMYLPIPERINEGary A. Cain; Christopher A. Teleha
99-101A FACILE METHOD WITH IMPROVED YIELDS IN THE SYNTHESIS OF 6-ARYLPYRIDO[2′,3′:4,5]PYRIMIDO[1,6-a]BENZIMIDAZOLESG. Suma; R. H. Bahekar; A. R. R. Rao

Volume 31, Issue 6 (1999)

CEditorial Board Page
579-615SYNTHESIS AND REACTIONS OF SULFINYL CHLORIDES. AN UPDATEAdrian L. Schwan; Rick R. Strickler
617-680SYNTHETIC USES OF ORTHOQUINONE MONOKETALS AND THEIR ORTHOQUINOL VARIANTS. A REVIEWStéphane Quideau; Laurent Pouységu
681-688INVESTIGATION OF THE ALKYLATION OF ALDOXIMES AND KETOXIMES WITH α-EPOXIDESSultan Kurbanov; Abdulkadir Sirit; Nejdet Sen
689-692IMPROVED METHOD FOR THE ESTERIFICATION OF SUGAR ACETALS WITH DICYCLOHEXYLCARBODIIMIDEClarissa C. Perrone; Paulo R. R. Costa; Vítor F. Ferreira
693-694A CONVENIENT PREPARATION OF THIOFORMAMIDE. SYNTHESIS OF THIAZOLE-4-CARBOXYLIC ACIDJ. Rohály; L. Novák; Cs. Szántay
694-697REDUCTIVE OXIDATION OF CARBOXYLIC ACIDS TO ALDEHYDES WITH SODIUM BOROHYDRIDE AND PYRIDINIUM CHLOROCHROMATEJin Soon Cha; Dae Yon Lee; Jong Mi Kim
698-7012-(1-AZETIDINYL)- AND 2-(1-PYRROLIDINYL)PYRIDINE via SNAr REACTIONS OF 2-FLUOROPYRIDINE AND 2-PYRIDINYL TRIFLATEStan V. D'andrea; Jeremiah P. Freeman; Jacob Szmuszkovicz
702-704A FACILE SYNTHESIS OF 3ß-ACETOXYLANOST-8-EN-24-ONE (24-KETOLANOSTERYL ACETATE)Edward J. Parish; Hang Sun; Stephen A. Kizito; Edna S. Kaneshiro
705Corrigendum
707-718INDEXES

Volume 31, Issue 5 (1999)

CEditorial Board Page
467-505STEREOCHEMISTRY OF THE ALKYLATION OF LACTONES. A REVIEWMalika Ibrahim-Ouali; Jean-Luc Parrain; Maurice Santelli
507-536MAIN METHODOLOGIES FOR THE SYNTHESIS OF RADIALENES. AN UPDATEFlorence Geneste; Alec Moradpour
537-541SYNTHESIS OF (+)-OBTUNONE. A NEW ROUTE TO THE CADINANE SKELETONBarry B. Snider; Zheng Chen
543-549SYNTHESIS OF 3,3,5,5-TETRAMETHYLMORPHOLINONES FUNCTIONALIZED AT THE 6-POSITIONDario Lazzari; Mirco Rossi; Massimo Soverini; Marco Mazzega; Ottorino De Lucchi
551-557NEW SYNTHESES OF SUBSTITUTED PYRIDAZIN-6-ONES AND PYRIDAZIN-6-IMINESH. Behbehani; M. M. Abdel-Khalik; M. H. Elnagdi
559-561SUBSTITUTION REACTION OF N,N'-DIPHENYLUREA BY AMINES TO UNSYMMETRIC PHENYLUREASYing Yang; Shiwei Lu
562-564DE(MONOTHIO)ACETALIZATION INDUCED BY HYPERVALENT IODINE AND SODIUM IODIDELing-Ching Chen; Huey-Min Wang
565-570HEMIESTERS OF DEXANABINOL AND THEIR WATER-SOLUBLE SALTSEmil Pop; Ferenc Soti; Stanislaw Rachwal
571-572AN IMPROVED SYNTHESIS OF tert-BUTYL Nα-tert-BUTOXYCARBONYL-L-(S-TRITYL)CYSTEINATEElżb�eta Masiukiewicz; Barbara Rzeszotarska
573-575FERROUS SULFATE PROMOTED CONVERSION OF N,N-DIMETHYLHYDRAZONES AND PHENYLHYDRAZONES TO CARBONYL COMPOUNDSAayesha Nasreen; Srinivas R. Adapa
577Corrigendum

Volume 31, Issue 4 (1999)

CEditorial Board Page
359-377REACTIONS OF CARBON TETRACHLORIDE AND CARBON TETRABROMIDE WITH ANIONS AND CARBANIONS. A REVIEWEdgars Abele; Edmunds Lukevics
379-397THE CHEMISTRY OF 4′,5′-UNSATURATED NUCLEOSIDES. A REVIEWClemens Lamberth
399-405A COMPARISON OF IMINE FORMING METHODOLOGIESBrian E. Love; Tavia S. Boston; Binh T. Nguyen; Jeffrey R. Rorer
407-412ACYLATION AND ALKYLATION OF 2- AND 4-METHYLBENZONITRILERichard A. Bunce; Lara B. Johnson
413-421N-SUBSTITUTED 3-OXA- AND 3-THIA-7-AZABICYCLO[3.3.1]NONANES AS POTENTIAL PRECURSORS OF ANTIARRHYTHMICSSameer Tyagi; Kevin M. Couch; Gregory L. Garrison; K. Darrell Berlin; Benajmin J. Scherlag; Eugene Patterson; Ralph Lazzara
423-425SYNTHESIS OF N-(5-AMINO-2-PYRIMIDn)-N′-[4-(p-FLUOROPHENYL)-4-OXOBUTYL]PIPERAZINE, A USEFUL INTERMEDIATE TO ANTIPSYCHOTIC AGENTSGianluigi Broggini; Gaetano Zecchi
425-429SYNTHESIS OF N-(3-MERCAPTOPROPANOYL)-AZA-18-CROWN-6, N-(4-MERCAPTOBUTANOYL)-AZA-18-CROWN-6 AND THEIR DIMERSXinhao Yang; J. Justin Gooding; D. Brynn Hibbert; Naresh Kumar
429-433NEW N,N′-bis (SUBSTITUTED PHENYLAZO) PIPERAZINES AND THEIR CLEAVAGE REACTIONS IN ACETIC ACIDErkan Yanarates; Ali Disli; Yilmaz Yildirir
433-439PHASE-TRANSFER CATALYZED ALKYLATION OF HYDROXY 9,10-ANTHRAQUINONESDouglas R. Robello; Teresa D. Eldridge; Edward J. Urankar
440-442MULTI-GRAM SYNTHESIS OF DIMYRISTOYL PENTAERYTHRITOLMike E. Lizarzaburu; Ryan M. Jones; Michael H. Nantz; Mark J. Kurth
442-447IMPROVED SYNTHESIS OF cis-9,10-DIHYDRO-9,10,-PHENANTHRENEDICARBOXIMIDES AND 9,10-PHENANTHRENEDICARBOXIMIDESPiotr Grycz; Jacek Gawroński
447-450PREPARATION OF 3-TETRADECYLINDOLEJames H. Wynne; George W. Mushrush; Wayne M. Stalick
450-453A NOVEL METHOD FOR THE SYNTHESIS OF TELLUROESTERSSonglin Zhang; Yongmin Zhang
453-456AN EFFICIENT ONE-POT SYNTHESIS OF α-PHENYLSELENO-α,β-UNSATURATED NITRILES via ARSONIUM SALTSGui-Sheng Deng; Zhi-Zhen Huang; Xian Huang
456-459AN IMPROVED SYNTHESIS OF Nα-BENZYLOXYCARBONYL-L-LYSINEEłżbieta Masiukiewicz; Stanislaw Wiejak; Barbara Rzeszotarska
460-462IMPROVED PREPARATION OF METHYL 4,6-O-BENZYLIDENE-α-D-GLUCOPYRANOSIDERolando A. Spanevello; Damiáh D. Saavedra
462-465A NEW AND EFFICIENT SOLVENT-FREE SYNTHESIS OF bis-ARYL CARBODIAZONESHong Wang; Yulu Wang; Jianping Li; Xiaoyang Wang

Volume 31, Issue 3 (1999)

CEditorial Board Page
245-294SYNTHESIS OF POLYPODAL DIPHENYLPHOSPHINE LIGANDS. A REVIEWDorothée Laurenti; Maurice Santelli
295-304“ONE-POT” SYNTHESIS OF DIMETHYL [1-SUBSTITUTED-5-HYDROXY-1H-PYRAZOL-4-YL]PHOSPHONATESPaula C. Miller; John M. Molyneaux
305-313SYNTHESIS OF NEW CONDENSED 2-AMINO-4H-PYRAN-3-CARBONITRILES AND OF 2-AMINOQUINOLINE-3-CARBONITRILESSaleh M. Al-Mousawi; Yehia M. Elkholy; Mohammad A. Mohammad; Mohammad H. Elnagdi
315-319NITRATION STUDIES ON 4-PHENYL-5-SUBSTIUTED-1,3-DIOXANES AS CHLORAMPHENICOL INTERMEDIATESB. G. Hazra; V. S. Pore; S. P. Maybhate; B. V. Bapat; V. K. Gumaste; A. S. Rao
319-323AN EFFICIENT SYNTHESIS OF MEQUITAZINEYves Guminski; Valerie Fabre; Patrick Lesimple; Thierry Imbert
324-328FRIEDEL-CRAFTS ACYLATION WITH MALONIC ACIDS IN POLYPHOSPHORIC ACIDOlivier Renault; Patrick Dallemagne; Sylvain Rault
328-332SYNTHESIS OF NEW TYPES OF LEWIS ACIDS REARRANGEMENT OF STILBENE OXIDESYoshihiro Ohba; Kazuaki Ito; Tomomi Nagasawa
333-335A NEW, FACILE METHOD FOR DETRIFLUOROACETYLATION OF ESTERS WITH TRIETHYLAMINE PRETREATED SILICA GELLigong Ou; Donglu Bai
335-341BENZYLTRIPHENYLPHOSPHONIUM DICHROMATE AS A MILD REAGENT FOR THE OXIDATION OF ORGANIC COMPOUNDSAbdol Reza Hajipour; Iraj Mohammadpoor-Baltork; Kurosh Niknam
341-346PREPARATION AND CHARACTERIZATION OF NEW SUBSTITUTJED 5-METHOXY-2-STYRYL-4-PYRONESZdenka Stiplošek; Marija Šindler-Kulyk; Krešimir Jakopčić
347-348SIMPLE, HIGH YIELD PREPARATION OF 3-NITRO-1,2-PHENYLENEDIAMINEViktor Milata; Jozef Saloň
349-352IMPROVED SYNTHESIS OF SYMMETRICAL DIPYRROMETHENESBin Tu; Changqi Wang; Jinshi Ma
352-358TRANSFORMATION OF 6-HALOPENICILLANATES INTO 3-HALO-4-OXOAZETIDINE DERIVATIVESIrena Lukić

Volume 31, Issue 2 (1999)

CEditorial Board Page
125-143SYNTHESIS OF α-FLUORO ALDEHYDES AND KETONES. A REVIEWFranklin A. Davis; Parimala V. N. Kasu
145-166SELECTIVE PROTECTION OF THE VARIOUS HYDROXY GROUPS OF CHOLIC ACID AND DERIVATIVES. A REVIEWHongwu Gao; Jerry Ray Dias
167-172ipso-NITRATION OF HEXAMETHOXY[(2.1)3]METACYCLOPHANE, A CALIXARENE ANALOGOUS MACROCYCLIC META CYCLOPHANETakehiko Yamato; Yuko Kinosaki; Fenglei Zhang
173-179SYNTHESIS OF NEW vic-DIOXIME DERIVATIVES OF p-(tert-BUTYL) CALIXARENE AND SOME METAL COMPLEXESHasalettin Deligöz
181-187A NEW REDUCTION OF THE ENONE SYSTEM OF 18B-GLYCYRRHETIC ACIDR. Pellegatat; M. Pinza; G. Pifferi; C. Farina
189-192ADDUCTS OF PIPERAZINE WITH NITRIC OXIDEJoseph A. Hrabie; Joseph E. Saavedra; Keith M. Davies; Larry K. Keefer
193-200REACTION OF bisPHENOL-A DIGLYCIDYL ETHER WITH SUBSTITUTED PHENOLSSylvie Jost; Laurent Vanbellinghen; Philippe Henderson; Jacqueline Marchand-Brynaert
201-203STEREOSELECTIVE SYNTHESIS OF (E)-VINYL ARYL SULFIDES via HYDROZIRCONATION OF TERMINAL ALKYNESXian Huang; Ping Zhong; Wei-Rong Guo
204-207CONVERSION OF ACID CHLORIDES TO ALDEHYDES BY OXIDATION OF ALKOXYALUMINUM INTERMEDIATES WITH PYRIDINIUM CHLOROCHROMATE OR PYRIDINIUM DICHROMATEJin Soon Cha; Jong Mi Kim; Joong Hyun Chun; Oh Oun Kwon; Sang Yong Kwon; Sung Wook Han
207-211EXPEDIENT SYNTHESIS OF (1R,3S)-(+)-3-(TRIFLUOROMETHYL)CAMPHONANIC ACID AND DERIVATIVESWojciech Dmowski; Krystyna Piasecka-Maciejewska
211-214(R)-2-HYDROXY-3-TRIPHENYLMETHYLTHIOPROPANOIC ACID, AN INTERMEDIATE IN THE SYNTHESIS OF HYDROXY ANALOGS OF OXYTOCINKazimierz Wisniewski
214-215PREPARATION OF N-TRITYLPYRROLIDINE AND N-TRITYLPIPERIDINEMurthy R. Akula; George W. Kabalka
216-220PREPARATION OF β-KETOPHOSPHONATES AND THEIR VINYLOGUES BY OXIDATION OF THE CORRESPONDING ALCOHOLSElmar L. Müller; Agnes M. Modro; Tomasz A. Modro
220-222A CONVENIENT REDUCTION OF UNSATURATED BICYCLIC ANHYDRIDESFerenc Csende; Géza Stájer
222-225A SIMPLE PROCEDURE FOR THE ALKYLATION OF 4-HYDROXYCOUMARINS AT C-3 POSITIONG. Tóth; S. Molnár; T. Tamás; I. Borbély
225-227A ONE-STEP SYNTHESIS OF 1-HYDROXY-10-METHYL-9(10H)-ACRIDINONEGary M. Coppola
227-230ISOMERIZATION OF LONGIFOLENE TO ISOLONGIFOLENE CATALYZED BY MONTMORILLONITE CLAYA. R. Ramesha; Shridhar Bhat; Kandikere R. Prabhu
230-231IMPROVED SYNTHESIS OF bis(2,2,2-TRIFLUOROETHYL) PHOSPHOROCHLORIDATERussell A. Bowman; Joseph R. Stock; John A. Jackson
232-236A SIMPLE AND EFFICIENT SYNTHESIS OF γ-AMINOBUTYRIC ACID (GABA) DERIVATIVESV. Dryanska; I. Pashkuleva
237-240SYNTHESIS OF N-PROTECTED 2-AMINOHEXANESULFONIC ACIDVioletta Constantinou-Kokotou
240-243MICHAELIS-BECKER SYNTHESIS OF bis(2,2,2-TRIFLUOROETHYL)PHOSPHONO ESTERSGregory M. Ciszewski; John A. Jackson

Volume 31, Issue 1 (1999)

CEditorial Board Page
1-86RECENT ADVANCES IN THE SYNTHESIS OF INDAN SYSTEMS. A REVIEWBor-Cherng Hong; Sepehr Sarshar
87-97PREPARATION AND PARTIAL DEACETYLATION OF DIHYDROQUERCETIN ACETATESE. Kiehlmann
99-106α-VINYLATION OF TERTIARY ACTIVE HYDROGEN COMPOUNDSRichard A. Bunce; Scott E. Burns
106-109AN IMPROVED LARGE SCALE SYNTHESIS OF 2,3-DIHYDROXYTEREPHTHALIC ACID AND DIMETHYL 2,3-DIHYDROXYTEREPHTHLATEB. -C. Chen; M. S. Bednarz; J. E. Sundeen; Z. J. Zhang; T. J. Caulfield; G. S. Bisacchi
110-111A FACILE SYNTHESIS OF 3-CHLORO-4-(2′,2′,2′-TRIFLUOROETHOXY)BENZONITRILERong Zhang; Xuhong Qian; Weida Zhou
112-116A FACILE AND EFFICIENT METHOD FOR THE REGENERATION OF CARBONYL COMPOUNDS FROM HYDRAZONES AND OXIMES BY OXONE® UNDER HETEROGENEOUS CONDITIONSAbdol Reza Hajipour; Nasrien Mahboubghah
117-119THE REGIOSELECTIVE NITRATION OF α,β-UNSATURATED NITRILES WITH NITROGEN OXIDESArturo Navarro-Ocaña; Eduardo Barzana; Daniel López-González; Manuel Jiménez-Estrada
120-123THE SELENIUM DIOXIDE OXIDATION OF 2,3- AND 3,4-DIMETHYLPYRIDINESA. D. Dunn

Volume 30, Issue 6 (1998)

CEditorial Board Page
603-629RECENT PROGRESS IN THE SYNTHESIS OF p-QUINONES AND p-DIHYDRO-QUINONES THROUGH OXIDATION OF PHENOL DERIVATIVES. A REVIEWShuji Akai; Yasuyuki Kita
631-655ACTIVATION OF CARBOXYLIC ACIDS BY PYROCARBONATES. SCOPE AND LIMITATIONS. A REVIEWV. F. Pozdnev
657-697SUBSTITUTED GLUTACONIC ACIDS AND THEIR ESTERS IN ORGANIC SYNTHESIS. A REVIEWPavel F. Vlad; Miron Z. Krimer
699-702HIGHLY EFFICIENT SYNTHESIS OF FATTY ACID DOPAMIDESZ. Czarnocki; M. P. Matuszewska; I. Matuszewska
703-705SYNTHESIS OF 1,2- AND 1,4-bis[α-(2,4,6-TRINITROANILINO)-ACETAMIDO]BENZENE AS NEW INSENSITIVE EXPLOSIVESB. P. Bandgar; V. R. Damal; S. S. Pandit
706-709MILD AND SELECTIVE METHOD FOR THE OXIDATIVE CLEAVAGE OF ACETALS AND THIOACETALSB. P. Bandgar; Sameer A. Kulkarni; J. N. Nigal
709-713THE SYNTHESIS OF 3-AMINO-2-DIALKYLAMINOPYRIDINESA. D. Dunn
713-716TRIMETHYLAMMONIUM CHLOROCHROMATE (TMACC) ADSORBED ON ALUMINA FOR CLEAVAGE OF CARBON-NITROGEN DOUBLE BONDS UNDER NON-AQUEOUS CONDITIONSGui-Sheng Zhang; De-Hong Yang; Mi-Feng Chen
716-719A FACILE SYNTHESIS OF NEW 2-PHOSPHONOBENZYLOXY-1,3,2-BENZOXAZA(DIOXA OR DIAZA)PHOSPHOLESJia Zhou; Ruyu Chen
721-732INDEXES

Volume 30, Issue 5 (1998)

CEditorial Board Page
489-550RECENT PROGRESS IN SOLID PHASE HETEROCYCLE SYNTHESES. A REVIEWJeffrey W. Corbett
551-600RECENT PROGRESS IN THE SYNTHESIS, PROPERTIES AND REACTIONS OF TRISULFANES AND THEIR OXIDESEdward L. Clennan; Kristina L. Stensaas
601Corrigendum

Volume 30, Issue 4 (1998)

CEditorial Board Page
373-400APPLICATIONS OF TRIMETHYLSILYL HALIDES-OXIDANTS COMBINATIONS IN ORGANIC SYNTHESIS. A REVIEWPadma S. Vankar; M. Venkat Ram Reddy; Yashwant D. Vankar
401-425PHOTOCHEMICAL TRANSFORMATIONS OF 2(5H)-FURANONES. A REVIEWAhmed I. Hashem; Alexander Senning; Abdel-Sattar S. Hamad
427-432A RAPID WILLIAMSON SYNTHESIS UNDER MICROWAVE IRRADIATION IN DRY MEDIUMDariusz Bogdal; Jan Pielichowski; Krzysztof Jaskot
433-437FACILE SYNTHESIS OF 5-(DIHYDROXYBORYL)-2,4-bis(ALKOXY)PYRIMIDINES AND N(1)-SUBSTITUTED 5-(DIHYDROXYBORYL)URACILSHanna Wojtowicz-Rajchel; Krzysztof Golankiewicz
439-446SYNTHESIS AND SPECTRAL DATA OF SOME NEW N-NITROSO-N-PHENYLHYDROXYLAMINE (CUPFERRON) DERIVATIVESAlexandru T. Balaban; Robert E. Garfield; Melanie J. Lesko; William A. Seitz
447-451A FACILE SYNTHESIS OF o-, m-, p-(TRIMETHYLSTANNYL)BENZYL CHLORIDES AND AMINESA. B. Koldobsky; V. E. Vakhmistrov; O. S. Shilova; V. N. Kalinin; K. Abbaspour Tehrani; N. De Kimpe
451-453A NOVEL ROUTE TO 4-ARYLIDENE-2-PHENYL-5(4H)-OXAZOLONESM. Kidwai; R. Kumar
453-455IMPROVED PREPARATION OF FLURBIPROFENM. N. Deshmukh; V. Lakshminarayana
455-460EFFICIENCY OF THE VILSMEIER-HAACK METHOD IN THE SYNTHESIS OF p-AMINOBENZALDEHYDESRyszard Gawinecki; Sylwia Andrzejak; Agnieszka Puchala
460-463IMPROVED PREPARATION OF SURFACTANTS DERIVED FROM SUCROSE WITH ULTRASOUNDJacques Besson; Catherine Fayet; J. Gelas; Christelle Lamazzi
463-466AN EFFICIENT AND FACILE PROCEDURE FOR DEPROTECTION OF 1,1-DIACETATES USING ANHYDROUS FERROUS SULFATET. S. Jin; Y. R. Ma; Z. H. Zhang; T. S. Li
467-469A HIGH YIELDING PREPARATION OF 2,2′-BIPYRIDINE-1-OXIDEF. W. Joachim Demnitz; Maria Betânia D'heni
469-472SURFACE MEDIATED SYNTHESIS OF O-PHOSPHOROTHIOATESK. Ramadas; N. Janarthanan; D. Meera Rani
473-476AN IMPROVED PREPARATION OF S,S'-DIMETHYL N-CYANODITHIOIMINOCARBONATELyndon K. Marble
477-481NEW SYNTHESES OF bis(TETRAMETHYLENE)FLUOROFORMAMIDINIUM HEXAFLUOROPHOSPHATE (BTFFH) AND 1,3-DIMETHYL-2-FLUORO-4,5-DIHYDRO-1H-IMIDAZOLIUM HEXAFLUOROPHOSPHATE (DFIH). UTILITY IN PEPTIDE COUPLING REACTIONSAyman El-Faham
481-484SYNTHESIS OF BENZO[c][2,7]NAPHTHYRIDINES AND 2,13-DIAZABENZO[b]CHRYSENECharles F. Nutaitis; Matthew L. Crawley; Judy Obaza-Nutaitis
485-488PREPARATION OF O-(3,3,8,10,10-PENTAMETHYL-1,2-DITHIA-5,8-DIAZACYCLODECAN-5-YL)ETHYL O-PIVALOYLOXYMETHYL PHENYLPHOSPHONATENicholas Bodor; Katalin Prokai-Tatrai; Emo Koltai; Laszlo Prokai

Volume 30, Issue 3 (1998)

CEditorial Board Page
243-289RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF ISOTHIOCHROMANS. A REVIEWYao-Chang Xu
291-324SYNTHESES OF AVENACIOLIDE AND RELATED bisLACTONES. A REVIEWVictor S. Martín; Carmen M. Rodríguez; TomáS Martín
325-330BORANE-(N-SUBSTITUTED)BENZOTRIAZOLE COMPLEXES AND THEIR ALKYLATION REACTIONSAlan R. Katritzky; Yunfeng Fang; Sergei A. Belyakov
331-337CONVENIENT PREPARATION OF 14-HYDRO-5H-TRIBENZO[a,d,f]CYCLOOCTENESTakehiko Yamato; Naozumi Sakaue; Koji Fujita
339-348CHEMOSELECTIVE SYNTHESIS OF PROTECTED POLYAMINES AND FACILE SYNTHESIS OF POLYAMINE DERIVATIVES USING O-ALKYL-O'-(N-SUCCINIMIDYL) CARBONATESMaciej Adamczyk; Jeffrey R. Fishpaugh; Kevin J. Heuser
349-352NEW SYNTHESIS OF PHENYLTHIOGLYCOLIC ACIDS via RELATED TRIAZENE COMPOUNDSAli Disli; Yilmaz Yildirir
352-356A SIMPLE REGIOSELECTIVE SYNTHESIS OF (R)-10-HYDROXYAPORPHINE DIRECTLY FROM (R)-10,11-DIHYDROXYAPORPHINE [(R)-APOMORPHINE]Jack C. Kim; Sang-Duk Bae; Ji-A Kim; Soon-Kyu Choi
356-359A NEW SYNTHESIS OF 6,7-DICHLORO-DIBENZO[c,f][2,7]-NAPHTHYRIDINES via PHOTOCYCLIZATIONS. Vijayalakshmi; S. P. Rajendran
360-363SYNTHESIS OF DISULFIDES BY THE OXIDATIVE COUPLING OF THIOLS WITH CALCIUM HYPOCHLORITE AND SILICA GEL IN HEXANEMasao Hirano; Shigetaka Yakabe; Nobuteru Uraoka; Takashi Morimoto
363-367NEW SPIROPYRAN-4-YLINDOLIDINE DERIVATIVES FROM THE REACTION OF 2-OXO-3-CYANOMETHYLIDENE-2,3-DIHYDROINDOLES WITH CYCLOHEXANEDIONES AND PHENOLSFatima Al-Omran; Ibrahim El-Ghamry; Mohammed H. Elnagdi
367-372A FACILE SYNTHESIS OF 5-BENZOYLCYTOSINE DERIVATIVESR. B. Toche; M. N. Jachak; T. S. Dalvi; R. W. Sabnis; H. Junek; T. Kappe

Volume 30, Issue 2 (1998)

CEditorial Board Page
121-143THE ASYMMETRIC PAUSON-KHAND REACTION. A REVIEWS. T. Ingate; J. Marco-Contellers
145-176THE DEVELOPMENT AND APPLICATION OF 1,3-DITHIANE 1-OXIDE DERIVATIVES AS CHIRAL AUXILIARIES AND ASYMMETRIC BUILDING BLOCKS FOR ORGANIC SYNTHESIS. A REVIEW
177-181A NOVEL AND FACILE SYNTHESIS OF O-ACYLBENZALDEHYDESAntigoni Kotali; Maria Papapetrou; Vassilios Dimos; Philip A. Harris
183-186AN EFFICIENT PROCEDURE FOR THE PREPARATION OF FMOC-AMINO ACIDSStephen P. Raillard; Adam D. Mann; Ted A. Baer
187-194CYCLOPROPYL AND PYRAZOLYL SELENADIAZOLYL AND THIADIAZOLYL SULFONES AND THEIR REACTIVITYV. Padmavathi; R. P. Sumathi; M. V. Ramana Reddy; D. Bhaskar Reddy
195-202INVESTIGATION OF THE ALKYLATION OF AROMATIC AND HYDROAROMATIC ALDOXIMES WITH HALOHYDRINSErsin Güler; Nejdet Sen; Abdulkadir Sirit; Sultan Kurbanov; Ramazan Mirzaoglu
203-210SYNTHESIS OF SYMMETRICAL AND UNSYMMETRICAL DISUBSTITUTED α-PYRENYLMETHYL AND α-PERYLENYLMETHYL MALONATE AND CYANOACETATE ALLYL ESTERSAlan R. Katritzky; Zhijun Yang; Jamshed N. Lam; Colleen C. Nagel
211-215A NOVEL SYNTHESIS OF 2-AMINO DIARYLKETONE DERIVATIVES AND OF POLYFUNCTIONALLY SUBSTITUTED QUINOLINESFatima Al-Omran; Adel Abou El-Khair; Mohammed Hilmy Elnagdi
215-218PREPARATION OF ALUMINA-SUPPORTED DIMETHYLAMMONIUM CHLOROCHROMATE (DMCC) AND ITS USE IN THE OXIDATION OF ALCOHOLS AND BENZOINSGui-Sheng Zhang; Qi-Zeng Shi; Mi-Feng Chen; Kun Cai
218-222A SIMPLE REGIOSELECTIVE NUCLEAR BROMINATION OF ALKYL PHENYL ETHERSShigetaka Yakabe; Masao Hirano; Takashi Morimoto
222-225SYNTHESIS OF 3,6-DI-(tert-BUTYL)FLUORENE BY NICKEL(0) CATALYZED COUPLING OF ARYL HALIDESGitendra C. Paul; Joseph J. Gajewski
226-229ASYMMETRIC EPOXIDATION OF UNFUNCTIONALIZED OLEFINS via FORMATION OF CRYSTALLINE CYCLODEXTRIN COMPLEXESHidetake Sakuraba; Yoshio Tanaka
230-234LITHIUM HYPOCHLORITE-CLOROX AS A NOVEL OXIDATIVE MIXTURE FOR METHYL KETONES AND METHYL CARBINOLSM. M. Madler; J. Klucik; P. S. Soell; C. W. Brown; S. Liu; K. D. Berlin; D. M. Benbrook; P. J. Birckbichler; E. C. Nelson
235-238[3.3.1]PROPELLANE-2,8-DIONE. SYNTHESIS AND STRUCTUREI. David Reingold; Guido Beckmann; Amanda M. Grannas; Steven R. Brunette; Brian D. Williams; Scott Lovell; Bart E. Kahr
239-241A NOVEL METHOD OF SYNTHESIS OF ALKYL α-CYANOACRYLOYL GLYCOLATESXuelin Yang

Volume 30, Issue 1 (1998)

CEditorial Board Page
1-51BIOMIMETIC AND SYNTHETIC APPROACHES TO MARINE SPONGE ALKALOIDS DERIVED FROM BIS-PYRIDINE MACROCYCLES. A REVIEWNorbert Matzanke; Robert J. Gregg; Steven M. Weinreb
53-612-SUBSTITUTED HEXAHYDROPYRIMIDINES AND THEIR TAUTOMERISMKirill N. Zelenin; Valeriy V. Alekseyev; Ilya V. Ukraintsev; Igor V. Tselinsky
63-70REDUCTION OF ORGANIC COMPOUNDS WITH THEXYL-S-BUTOXYBORANEJin Soon Cha; Seok Won Chang; Jong Mi Kim; Oh Oun Kwon; Joong Hyun Chun; Sung Dong Cho; Hyung Soo Lee
71-78SYNTHESIS OF (1R,3S)-3-AMINO-1,2,2-TRIMETHYLCYCLOPENTYLMETHANOLJosé M. Blanco; Olga Caamaño; Franco Fernández; Xerardo García-Mera; José E. Rodríguez
79-85IMPROVED SYNTHESIS OF 7,7-DIMETHYL-1,4-DIOXO-2,3,4,5,6,7-HEXAHYDROINDEN-2-YL-ACETIC AND PROPIONIC ACID FROM CITRALIstván Kádas; Géza Árvai; Gabriella Horváth
87-90MICROWAVE-PROMOTED SYNTHESIS OF 1-ARYLOXY-3-ALKYLAMINO-2-PROPANOLSBeata Pchelka; Jan Plenkiewicz
90-93FACILE SYNTHESES OF P-(DICYANOMETHYLENE)BENZOQUINONESMasato Nanasawa; Hiroshi Takahashi; Tetsuo Kuwabara
93-96SYNTHESIS AND CYCLIZATION OF 1-(N-NITROAMIDINO)THIOUREAS TO 2,4-DIAMINOTHIAZOLESR. Binu; K. K. Thomas; G. C. Jenardanan; K. N. Rajasekharan
97-99AN EFFICIENT OXIDATION ARYLSEMICARBAZIDES TO THE AZO UREASCailan Wang; Yulu Wang; Xiaoyang Wang; Jianping Li; Hong Wang; Shensong Zhang
100-103A SIMPLE, ONE-POT PROCEDURE FOR THE PREPARATION OF DOPAMINERGIC ALKYLTHIOAPOMORPHINESSándor Berényi; Csaba Csutorás; Susanna Gyulai; Sándor Makleit
103-106REGIOSELECTIVE EPOXIDE RING-OPENING TO THE ENANTIOMERICALLY PURE α-HYDROXY ANALOGUE OF S-TERT-BUTYL CYSTEINEFlorine Cavelier; Anne-Marie Yim
107-109IMPROVED SYNTHESIS OF O-BENZENEDISULFONIMIDEFranklin A. Davis; Gajendran Sundarababu; Hongyan Qi
109-1141-ALKYLIDENE(ARYLIDENE)AMINO-2-AMINOETHANES AND THEIR TAUTOMERIZATION TO IMIDAZOLIDINESKirill N. Zelenin; Ilya V. Ukraintzev
115-116IMPROVED PREPARATION OF 5,6-DICHLOROCYCLOHEX-2-ENE-1,4-DIONEVitor Francisco Ferreira; Francis J. Schmitz
117-120A CONVENIENT SYNTHESIS OF (E)-(1-PROPENYLSULFONYL)BENZENEL. M. Finkielsztein; E. N. Alesso; B. Lantaño; J. M. Aguirre; G. Y. Moltrasio Iglesias

Volume 29, Issue 6 (1997)

CEditorial Board Page
603-629OPTICALLY ACTIVE SELENIUM AND TELLURIUM COMPOUNDS. SYNTHESIS AND APPLICATION FOR ASYMMETRIC SYNTHESIS. A REVIEWToshio Shimizu; Nobumasa Kamigata
631-664THE SYNTHESIS OF ISOCOUMARINS OVER THE LAST DECADE. A REVIEWElio Napolitano
665-669REDUCTION OF CARBOXYLIC ACIDS TO ALDEHYDES BY THEXYLALKOXYBORANESJin Soon Cha; Seok Won Chang; Jong Mi Kim; Oh Oun Kwon; Jae Cheol Lee
671-677SYNTHESIS OF AMINOTOLUENESULFONAMIDE DERIVATIVES USING CONVENTIONAL HEATING OR MICROWAVE-ASSISTED METHODSRolando Pérez; Eduardo R. Pérez; Margarita Suárez; Leandro González; André Loupy; María Luisa Jimeno; Carmen Ochoa
679-685IMPROVED SYNTHESES OF 2,2',3,3',6,6'-HEXACHLOROBIPHENYLStephen C. Waller; Eugene A. Mash
687-689CONDENSATION REACTION OF ACYLOINS WITH UREA WITHOUT SOLVENT UNDER MICROWAVE IRRADIATIONJun-Cai Feng; Qing-Hua Meng; Yang Liu; Li Dai
689-696CHEMICAL TRANSFORMATION OF DIHYDRO- AND TETRAHYDRO-1,5-BENZODIAZEPIN-2-ONES INTO AMIDINESBenedikta Dale Puodziunaite; Lina Vertelyte; Regina Janciene; Zita Stumbreviciute
696-701N-ACETYL-α,β-DEHYDROAMINO ACID N'-METHYLAMIDES AND N',N'-DIMETHYLAMIDESLeszek Smelka; Barbara Rzeszotarska; Malgorzata A. Broda; Zbigniew Kubica
701-706A FACILE SYNTHESIS FOR RACEMIC AND OPTICALLY ACTIVE 1-AMINOINDANSRamy Lidor; Eliezer Bahar; Ora Zairi; Gasan Atili; Dora Amster
707-710SYNTHESIS OF HEXASUBSTITUTED NITROBENZENE DERIVATIVESvia VICARIOUS NUCLEOPHILIC SUBSTITUTION OF HYDROGENM. Makosza; S. Nizamov
711-715A NOVEL ROUTE TO NEW DIBENZO[b,f][1,5]DIAZOCINE DERIVATIVES AS CHEMOSENSITIZERSE. Nonnenmacher; A. Hever; A. Mahamoud; C. Aubert; J. Molnar; J. Barbe
715-719N-BROMOSUCCINIMIDE-CHLOROFORM, A MORE CONVENIENT METHOD TO NUCLEAR BROMINATE REACTIVE AROMATIC HYDROCARBONSReginald H. Mitchell; Yongsheng Chen; Ji Zhang
721-734INDEXES

Volume 29, Issue 5 (1997)

CEditorial Board Page
499-539APPROACHES TO PARTIAL SYNTHESES OF 11-OXO STEROIDS. A BRIEF REVIEWHongwu Gao
541-547[2+2] CYCLOADDITION REACTIONS OF ENAMINES WITH ELECTRON-DEFICIENT ACETYLENESN. Tunoglu; N. Uludag
549-560OPTIMIZED SYNTHESIS OF SOME γ,γ-DISUBSTITUTED ALLYLAMINESUlrich Jordis; Franz Grohmann; Bernhard Küenburg
561-568SYNTHESIS OF FLUORESCEIN PHOSPHATES AND SULFATESJohn Scheigetz; Michael Gilbert; Robert Zamboni
569-571TiCl4-Zn INDUCED REDUCTIVE COUPLING REACTIONS IN THE ABSENCE OF SOLVENTJian Chen; Jing Li; Ming-Hui Yu; Wei-Xing Chen; He-Liang Fu
572-576SYNTHESIS OF 13-ETHYL-11-METHYLENE-18,19-DINOR-17α-PREGN-4-EN-20-YN-17-OLHongwu Gao; Xiangdong Su; Liming Zhou; Zhensu Li
577-579A FACILE SYNTHESIS OF 3-AMINO-1(2)H-PYRAZOLO[3,4-c]PYRIDINEA. D. Dunn
580-583A FACILE SYNTHESIS OF 1-BENZYLOXYCARBONYLAMINO-(SUBSTITUTED)PHENYLMETHYLPHOSPHINATESQing Dai; Ruyu Chen
584-587MICHAEL REACTIONS IN AQUEOUS MICELLES OF CETYLTRIMETHYLAMMONIUM BROMIDEC. D. Mudaliar; K. R. Nivalkar; S. H. Mashraqui
587-589α,β-UNSATURATED SULFONES BY THE WITTIG REACTION OF STABLE YLIDE WITH ALDEHYDES UNDER MICROWAVE IRRADIATIONCong Fu; Caiding Xu; Zhi-Zhen Huang; Xian Huang
590-5932,5-DISUBSTITUTED FURANS BY OXIDATION OF β-DICARBONYL COMPOUNDS IN THE PRESENCE OF FURANAttilio Citterio; Maffezzoni Tino; Maronati Antonietta; Roberto Sebastiano
594-600PREPARATION OF RING-SUBSTITUTED PHENOXYAMINE DERIVATIVESEtsuko Miyazawa; Takeshi Sakamoto; Yasuo Kikugawa
600-601MODIFICATION OF ROUND BOTTOM FLASKS TO ALLOW COMPLETE REMOVAL OF CONTENTS BY SYRINGEBrian E. Love
602CORRIGENDUM

Volume 29, Issue 4 (1997)

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365-407REDUCTIVE CLAISEN REARRANGEMENTS OF ALLYLOXYANTHRAQUINONES. A REVIEWRichard C. Cambie; Jared B. J. Milbank; Peter S. Rutledge
409-458RECENT PROGRESS IN THE USE OF HYPERVALENT IODINE REAGENTS IN ORGANIC SYNTHESIS. A REVIEWTsugio Kitamura; Yuzo Fujiwara
459-464p-CHLOROPHENOL AS A SOLVENT FOR CYCLOADDITION OF CYCLOPENTADIENONES WITH NON-ACTIVATED OLEFINSTamaki Jikyo; Masashi Eto; Toshikazu Matsuoka; Kazunobu Harano
465-470SYNTHESIS OF 6-HYDROXY-3,4,5,6-TETRAHYDRO-2-PYRIDONES AND 3,4-DIHYDRO-2-PYRIDONES BY H2O2/DMSO HYDRATION OF Δ-KETONITRILESAttilio Citterio; Elena Carnevali; Alessandra Farina; Valdo Meille; Stefano Alini; Livius Cotarca
471-473AN IMPROVED ROUTE TO CYCLOALKA[b]PYRROLE 2-CARBOXYLATESC. Balsamini; A. Bedini; G. Tarzia; A. Tontini
473-476SYNTHESES AND STEREOCHEMISTRY OF TETRAHYDROFURAN DERIVATIVES FROM α-PINENEFu-Chu Liu; Zhen-Qi Mei; You-Chu Wang; Jun Lin
477-480SYNTHESIS OF SUBSTITUTED 1-TETRALONESPunit Kumar
480-484DETHIOACETALIZATION OF DITHIOLANES WITH FERRIC NITRATE AND SILICA GEL IN HEXANEMasao Hirano; Ken Ukawa; Shigetaka Yakabe; Takashi Morimoto
485-488SYNTHESIS OF 3-O-BENZYL-3,7-IMINO-1,3,6,7-TETRADEOXY-L-MANNO-HEPTITOL AND OF 3-O-BENZYL-3,7-IMINO-1,3,6,7-TETRADEOXY-D-GLUCO-HEPTITOLFabio Degiorgis; Marco Lombardo; Claudio Trombini
488-494A CONVENIENT SYNTHESIS OF NEW HALOTHIENYL β-AMINOACIDS AS VERSATILE BUILDING BLOCKSOlivier Renault; Patrick Dallemagne; Sylvain Rault
494-496NEW SIMPLE SYNTHESIS OF THE HOUSEFLY SEX ATTRACTANTYao-Pin Yen; Fey-Long Wang
497-498IMPROVED ONE-POT PREPARATION OF TETRAMETHYLFLUOROFORMAMIDINIUM HEXAFLUOROPHOSPHATETomas Vojkovsky; Brian Drake

Volume 29, Issue 3 (1997)

CEditorial Board Page
243-283BRIDGED POLYCYCLIC AROMATIC HYDROCARBONS. A REVIEWRonald G. Harvey
285-292SYNTHESIS OF NEW ARYL AND HETEROAROMATIC SUBSTITUTED PYRIDINES, PYRAZOLES, PYRIMIDINES AND PYRAZOLO[3,4-D]PYRIDAZINESFatima Al-Omran; Nouria Al-Awadi; Adel Abou El-Khair; Mohammed Hilmy Elnagdi
293-299TETRAHYDROPYRANYLOXY-DIRECTED ortho LITHIATION OF AROMATIC SYSTEMS. SYNTHESIS OF o-HYDROXYCINNAMATE ESTERS FROM PHENOLSRichard A. Bunce; Joel D. Moore
300-303A NEW ROUTE FOR THE PREPARATION OF XANTHENE DERIVATIVES USING FRIEDEL-CRAFTS INTRAMOLECULAR CYCLOBENZYLATIONTakehiko Yamato; Masayasu Komine; Yoshiaki Nagano
303-308SYNTHESIS OF (1R,cis)-2-(3-AMINO-2,2-DIMETHYLCYCLOBUTYL)ETHANOL, A PRECURSOR OF CYCLOBUTANE CARBOCYCLIC NUCLEOSIDESJosé E. R. Borges; Franco Fernández; Xerardo García; Antonio R. Hergueta; Carmen López
308-311AN IMPROVED PROCEDURE FOR THE SYNTHESIS OF ANHYDROECGONINE METHYL ESTERC. R. Holmquist; K. R. Parham; J. A. Holleman; F. I. Carroll
311-314SYNTHESIS OF UNSYMMETRICAL α-(N-ARYLCARBONYL)AMINO DIORGANYL SELENIDES via BENZOTRIAZOLE INTERMEDIATES PROMOTED BY SmI2Weiliang Bao; Yongmin Zhang; Yunfa Zheng
315-321REDUCTION OF 1,3-AZOLE AND 1,3-BENZAZOLE CARBINOLS WITH SODIUM BOROHYDRIDE-TRIFLUOROACETIC ACIDCharles F. Nutaitis; Judy Obaza-Nutaitis
321-330ELECTROPHILIC SUBSTITUTION OF 7-tert-BUTYL-1-SUBSTITUTED PYRENES. A NEW ROUTE FOR THE PREPARATION OF 1,3-DISUBSTITUTED PYRENESTakehiko Yamato; Masakazu Fujimoto; Yoshiaki Nagano; Akira Miyazawa; Masashi Tashiro
330-335EFFICIENT SYNTHESIS OF EXO-1-AZABICYCLO[2.2.1]HEPTAN-3-OLStephen D. Barrett; Juan C. Jaen; Bradley W. Caprathe; Anthony J. Thomas; Haile Tecle
335-337TETRAHYDROFURAN RING-OPENING WITH ACID ANHYDRIDES CATALYZED BY SAMARIUM TRIIODIDEWeiliang Bao; Taokai Ying; Yongmin Zhang; Mingxin Yu
338-341THE EFFICIENT SYNTHESIS OF FMOC-L-HOMOGLUTAMINEKazimierz Wiśniewski; Aleksandra S. Kolodziejczyk
341-347ALLYLIC AND PHENOLIC PHOSPHATE ESTERS OF DEXANABINOLEmil Pop; Ferenc Soti; Anat Biegon; Marcus E. Brewster
347-352SYNTHESIS OF 4H-CYCLOPENTA[def]CHRYSENE AND OTHER METHYLENE-BRIDGED POLYCYCLIC HYDROCARBONSWei Dai; Ronald G. Harvey
352-355N-PERFLUOROALKANESULFONYLPHOSPHORAMIDES via AN IMPROVED ATHERTON-TODD REACTIONShizheng Zhu; Jie Zhang; Bin Xu; Chaoyue Qin
355-357A NOVEL SYNTHESIS OF 4-CYANO-2-(2-HYDROXYBENZOYL)PYRIDO[1,2-α]-BENZIMIDAZOLES FROM 3-FORMYLCHROMONEKusukuntla Venkat Reddy; A. V. Subba Rao
358-361AN EFFICIENT SYNTHESIS OF 3-BROMO-2-(BROMOMETHYL)-1-PROPENETheodore Axenrod; Kajal K. Das; Hamid Yazdekhasti; Paritosh R. Dave; Alfred G. Stern
361-364A CONCISE SYNTHESIS OF SYMMETRIC 1,3,5-C3-TRISUBSTITUTED BENZENESM. W. Majchrzak; J. N. Zobel; D. J. Obradovich; G. A. Peterson

Volume 29, Issue 2 (1997)

CEditorial Board Page
137-176SELECTIVE TRANSITION METAL-PROMOTED CARBON-CARBON AND CARBON-HETEROATOM BOND FORMATION. A REVIEWRenzo Rossi; Fabio Bellina
177-183A PRACTICAL PREPARATION OF L-ASPARTYL-D-2-AMINOBUTYRIC ACID (S)-α-PHENYLPROPYLAMIDE, A NEW HIGH-POTENCY SWEETENERGeorge A. King III; James G. Sweeny
185-194SYNTHESIS OF NITRONES FROM 3,4-DIHYDROISOQUINOLINE DERIVATIVES BY OXIDATION WITH m-CHLOROPEROXYBENZOIC ACIDBao-Xiang Zhao; Yang Yu; Shoji Eguchi
195-199AN ALTERNATIVE STRATEGY FOR THE PURIFICATION OF meso-2,4-PENTANEDIOLBarbara Gordillo; Javier Hernández
201-205ADIPOYLATION OF 2-METHOXYNAPHTHALENEC. Balo; F. Fernández; E. Lens; C. López
207-210NEWER ROUTE FOR THE SYNTHESIS OF β-PHENYLTHIO, β-PHENYLSULFINYL AND β-PHENYLSULFONYL NITROETHYLENESV. Ramamoorthy; S. Sivasubramanian; S. Muthusubramanian
211-214A CONVENIENT SYNTHESIS OF OXAZOLO[3,2-a]QUINOLONESHisham A. Abd El-Nabi
214-218SYNTHESIS OF DIETHYL 3-ARYL-3-OXOPROPYLPHOSPHONATESJen-Wen Yu; Steve K. Huang
218-221ASYMMETRIC SYNTHESIS OF (R)-N-(t-BUTOXYCARBONYL)-4-CYANOPHENYLALANINE METHYL ESTERAngelo Pecunioso; Damiano Papini; Bruno Tamburini; Francesco Tinazzi
221-223A FACILE SYNTHESIS OF 3-FLUOROTHIOPHENE-2-CARBOXYLIC ACIDEdward C. Taylor; Ping Zhou
223-226THE ALKYLATION OF COUMARIN AT C-3 OF 4-HYDROXYCOUMARINIbro Tabakovic; Katmerka Tabakovic; Igor Gaon
226-230AN IMPROVED GENERAL METHOD FOR THE PREPARATION OF 4-ARYL SUBSTITUTED bisPYRAZOLO[3,4-b;4,3'-e]PYRIDINESAgnieszka Puchala; Danuta Rasala; Erkki Kolehmainen; Monika Prokesová
231-234AN ALTERNATIVE SYNTHESIS OF ETHYL 3-(2-CHLORO-4,5-DIFLUOROPHENYL)-3-OXOPROPIONATE AND ETHYL 3-(2,6-DICHLORO-5-FLUOROPYRIDIN-3-YL)-3-OXOPROPIONATEFrank J. Urban; Bernard S. Moore; Peter L. Spargo
234-236AN IMPROVED SYNTHESIS OF bis(p-PHENYLENE)-32-CROWN-4Devdatt S. Nagvekar; Harry W. Gibson
237-240IMPROVED SYNTHESES OF 20- AND 26-MEMBERED bis(5-CARBOMETHOXY-1,3-PHENYLENE) CROWN ETHERSDevdatt S. Nagvekar; Harry W. Gibson
240-2425-BENZYLOXYRESORCINOL, A MONOPROTECTED PHLOROGLUCINOLDevdatt S. Nagvekar; Harry W. Gibson

Volume 29, Issue 1 (1997)

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1-32SYNTHETICALLY USEFUL REACTIONS WITH NICKEL BORIDE. A REVIEWJitender M. Khurana; Amita Gogia
33-62ELECTROPHILE MEDIATED HETEROATOM CYCLIZATIONS ONTO C-C π-BONDS. PART 1: HALOGEN AND CHALCOGEN MEDIATED CYCLIZATIONMartyn Frederickson; Ronald Grigg
63-115ELECTROPHILE MEDIATED HETEROATOM CYCLIZATIONS ONTO C-C π-BONDS. PART 2: METAL ION MEDIATED CYCLIZATIONMartyn Frederickson; Ronald Grigg
117-122IMPROVED PROCEDURES FOR PREPARATION OF 4-HYDROXY- AND 2-AMINO-4-METHOXY-2-AMINOPYRIDINESRichard J. Sundberg; Songchun Jiang
123-128A CONVENIENT, LARGE-SCALE SYNTHESIS OF ABIRATERONE ACETATE [3β-ACETOXY-17-(3-PYRIDYL)ANDROSTA-5,16-DIENE], A POTENTIAL NEW DRUG FOR THE TREATMENT OF PROSTATE CANCERGerard A. Potter; Ian R. Hardcastle; Michael Jarman
128-131A CONCISE PREPARATION OF 2,6-DIMETHYL-4-NITROCHLOROBENZENEStephen W. Wright
131-134A FACILE SYNTHESIS OF 9-HYDROXYBENZO[a]PYRENEShoujun Chen; Chunhua Wang; Peter P. Fu
135CORRIGENDUM

Volume 28, Issue 6 (1996)

CEditorial Board Page
641-682RECENT ADVANCES IN THE STEREOSELECTIVE SYNTHESIS OF HYDROXYLATED PYRROLIZIDINES. A REVIEWGiovanni Casiraghi; Franca Zanardi; Gloria Rassu; Luigi Pinna
683-690SYNTHESIS OF SOME NOVEL FUNCTIONALIZED DOUBLE MICHAEL ACCEPTORS BASED ON bis(VINYLSULFONYL)METHANE (BVSM)Andrew S. Kende; Kevin R. Guertin; Edgar E. Riecke; Istvan Kaldor
691-693A CONVENIENT ONE-STEP SYNTHESIS OF DIALKYLBENZO[k]FLUORANTHENES AND TETRAETHYL bis-BENZO[k][k′]FLUORANTHENESShadpour E. Mallakpour; Hossien Nasr-Isfahani
694-699REACTION OF NITRILIUM SALTS WITH 6-AMINOURACILAtef Hamed; Mahmoud Al-Talib
699-701CONSTRUCTION OF THE PYRAZOLO[1,5-a][6,1]BENZODIAZONINE AND PYRAZOLO[1,5-a][7,1]BENZODIAZECINE SKELETONSGianluigi Broggini; Luisa Garanti; Giorgio Molteni; Gaetano Zecchi
702-704AN IMPROVED SYNTHESIS OF 2-(HYDROXYMETHYL)INDENEHasan Palandoken; William T. McMillen; Michael H. Nantz
705-708A SELECTIVE AND CONVENIENT OXIDATION OF SULFIDES TO SULFOXIDES WITH FERRIC NITRATE AND SILICA GELM. Hirano; K. Komiya; S. Yakabe; J. H. Clark; T. Morimoto
709-710EXPEDIENT SYNTHESIS OF N1-TRITYLIMIDAZOLE-4-CARBOXALDEHYDEMichele C. Jetter; Robert E. Boyd; Allen B. Reitz
711-713SYNTHESIS OF Nα-BENZYLOXYCARBONYL-L-HISTIDINE HYDRAZIDE: AN UNDESIRED SIDE-PRODUCTElzbieta Masiukiewicz; Barbara Rzeszotarska
713-716THE LESS FAVORED 1-DERIVATIVES OF DIMETHYLDIHYDROPYRENE BY FORMYLATIONReginald H. Mitchell; Danny Y. K. Lau; Akira Miyazawa
717-729INDEXES

Volume 28, Issue 5 (1996)

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499-543SYNTHESIS OF THE FIRE ANT ALKALOIDS, SOLENOPSINS. A REVIEWSabine Leclercq; Désiré Daloze; Jean-Claude Braekman
545-608CYCLOADDITIONS OF ortho-QUINODIMETHANES DERIVED FROM BENZOCYCLOBUTENES IN ORGANIC SYNTHESIS. A REVIEWPierre-Yves Michellys; Hélène Pellissier; Maurice Santelli
609-612SYNTHESIS AND CONFORMATIONAL PROPERTIES OF 2,2′-DIHYDROXY-9,9′-BIANTHRYLM. Ghiaci; Y. Bayat
613-617SULFATED ZIRCONIA AS AN EFFICIENT CATALYST FOR TETRAHYDRO PYRANYLATION AND ACETALIZATIONAnjana Sarkart; Omprakash S. Yemult; B. P. Bandgar; N. B. Gaikwad; Prakash P. Wadgaonkar
618-622THE MANNICH REACTION OF DIALKYL KETONES, AROMATIC ALDEHYDES AND AROMATIC AMINESJunhua Zou
622-627SYNTHESIS OF o-KETOARYL CARBOXYLIC ESTERS USING PHENYLIODOSO DIACETATEAntigoni Kotali; Alexandros Koulidis; Huey-Min Wang; Ling-Ching Chen
627-634SYNTHESIS OF 7-HYDROXY-4-(ω-CARBOXYALKYL)COUMARINS AND 7-(DIMETHYLAMINO)-4-(ω-CARBOXYALKYL)COUMARINSMaciej Adamczyk; Phillip G. Mattingly; You Pan; Sushil Rege
634-637ISOMER DISTRIBUTION IN THE METHYLATION OF [1]-BENZOTHIENO[2,3-d]TRIAZOLE UNDER PHASE-TRANSFER CATALYTIC CONDITIONSSabine Schrader; Eckehard V. Dehmlow
639CORRIGENDUM

Volume 28, Issue 4 (1996)

CEditorial Board Page
371-409DEALKYLATION OF ETHERS. A REVIEWBrindaban C. Ranu; Sanjay Bhar
411-441SYNTHESIS OF BIUDGEHEAD-SUBSTTTUTED BICYCLO[1.1.1]PENTANES. A REVIEWErnest W. Delia; Ian J. Lochert
443-452SYNTHESIS OF NEW ALLYLIC MTROXIDES via THE WADSWORTH-EMMONS REACTIONTamás Kalai; Zoltán Szabó; József Jekö; Kálmán Hideg
453-462A NEW ROUTE FOR THE SYNTHESIS OF 3-(3-THIENYLOXY)-1,2-PROPANEDIOLS AND 3-(3-THIENYLOXY)-1,2-EPOXYPROPANESR. Donoso; P. Jordan de Urries; J. Lissavetzky
463-467A SIMPLE ONE-POT PREPARATION OF 4-ALKOXY-AND 4-ALKYLTHIO-CATECHOLS AND o-BENZOQUINONESChristopher J. Cooksey; Edward J. Land; Patrick A. Riley
467-469REDUCTION OF AROMATIC SULFONYL CHLORIDES TO DISULFIDESM. H. Zhang; M. Zheng; T. Cheng; S. X. Wang
470-474SYNTHESIS OF PROCAINAMIDE METABOLITES. N-ACETYL DESETHYLPROCAINAMIDE AND DESETHYLPROCAINAMIDEMaciej Adamczyk; James R. Fino
474-477(±)-SEDAMINE AND (±)-ALLOSEDAMINE BY REDUTION OF N-METHYL-2-PHENACYLIDENEPIPER1DINEM. Ghiaci; M. Adibi
478-480AN IMPROVED PREPARATION OF 1-METHYL-4-CYANO-4-PHENYLPIPERIDINEDino Gnecco; J. L. Tera; Raul G. Enríquez; William F. Reynolds; C. Marazano
480-483EFFICIENT IN SITU ESTERIFICATION OF CARBOXYLIC ACIDS USING CESIUM CARBONATEJong Chan Lee; Yoon Seok Oh; Sung Hye Cho; Jung D. Lee
484-486A FACILE LARGE SCALE PREPARATION OF RACEMIC 2.2′-DIHYDROXY-1,1′-BINAPHTHYLH. -J. DeuBen; P. Frederiksen; T. Bjornholm; K. Bechgaard
487-490A TRIPHOSGENE-BASED SYNTHESIS OF (S)-α,α-DIPHENYL-2-PYRROLIDINEMETHANOLTeodoro S. Kaufman; Viviana L. Ponzo; Juan Zinczuk
490-492SYNTHESIS OF PENTACOORDINATE PHOSPHORUS COMPOUNDS BY THE ATHERTON-TODD REACTIONRu-Zhen Cao; Xing-Zhong Zeng; Yan-Nan Liu; Lun-Zu Liu
492-494CONVERSION OF ALCOHOLS TO ALKYL CHLORIDES WITH SILICA CHLORIDEF. Mohanazadeh; A. R. Momeni
495-498DI-tert-BUTYL4-[(2-tert-BUTOXYCARBONYL)ETHYL]-4-AMINOHEPTANEDICARBOXYLATEGeorge R. Newkome; Claus D. Weis

Volume 28, Issue 3 (1996)

CEditorial Board Page
249-288bis-PROTECTED HYDROXYLAMINES AS REAGENTS IN ORGANIC SYNTHESIS. A REVIEWJeffrey L. Romine
289-318THE TRIFLUOROMETHYL GROUP IN ORGANIC SYNTHESIS. A REVIEWAlexander S. Kiselyov; Lucjan Strekowski
319-324SIMPLE PROCEDURES FOR THE PREPARATION OF α,ω-HYDROXYALKANETHIOLSLuis E. Iglesias; Alicia Baldessari; Eduardo G. Gros
325-332SYNTHESIS OF 6H-bis-[1]-BENZOPYRANO[2,3-b:3′,4′-e]PYRIDIN-8(8H)ONES AND 3-(2′-HYDROXYBENZOYL)-5H-[1]BENZOPYRANO[4,3-b]PYRIDINES AND THEIR DERIVATIVESK. Venkat Reddy; G. Sabitha; A. V. Subba Rao
333-338STEREOSPECIFIC ONE-POT SYNTHESIS OF 5-CARBOXY-3,4-DIPHENYLIMIDAZOLIDIN-2-ONE, A USEFUL PRECURSOR TO THE CORRESPONDING 2,3-DIAMINOPROPANOIC ACIDIvanka K. Kavrakova; Maria J. Lyapova
339-344AN UNUSUAL EPIMERIZATION IN THE OXIDATION OF A 4C-(HYDROXYMETHYL)-2,3,4-TRIDEOXY-2-HEXENOPYRANOSIDE USING FETIZON'S REAGENTAndrew G. H. Wee; Lin Zhang
345-347CONVENIENT AND EFFICIENT SYNTHESIS OF IMIDAZOLIUM CYCLOPHANESCheng-He Zhou; Ru-Gang Xie; Hua-Ming Zhao
348-351EFFICIENT PREPARATION OF 4-SUBSTITUTED-6-ACYL-7-METHOXYCOUMARINSM. V. Paradkar; M. S. Kulkarni; S. A. Kulkarni; H. M. Godbole
352-355A COMPARATIVE STUDY OF OXIDANTS ON THIOLSK. Ramadas; N. Srinivasan; N. Janarthanan; R. Pritha
355-359SELECTIVE REDUCTION OF α,β-UNSATURATED ALDEHYDES AND KETONES TO ALLYLIC ALCOHOLS WITH DHSOBUTYLALKOXYALANESJin Soon Cha; Oh Oun Kwon; Sang Yong Kwon
360-3614-CARBOMETHOXYNICOTINIC ACIDB. S. Moore; R. W. McLaughlin; F. J. Urban; G. R. Young
362-365SYNTHESIS OF 2-ARYL[1,2,4]-TRIAZOLO[5,1-b]BENZOTHIAZOLESHuey-Min Wang; Ling-Ching Chen
366-369AN OLIGO VICINAL DIIMINE BY THE EHRLICH-SACHS REACTION OF A β-IMINOKETONE WITH NITROSOBENZENEFrank Millich; Modasser T. El-Shoubary

Volume 28, Issue 2 (1996)

CEditorial Board Page
127-164PROGRESS IN THE MITSUNOBU REACTION. A REVIEWDavid L. Hughes
165-171TOTAL SYNTHESIS OF (±)-SIGMOIDIN-A [3′,4′,5,7-TETRAHYDROXY-2-(γ,γ-DIMETHYLALLYL)FLAVANONE] AND OF ANTIARONEFLianyun Zhao; Yulin Li
173-177AN EFFICIENT ONE POT SYNTHESIS OF N,N-DISUBSTITUTED UNSYMMETRICAL UREAS AND CARBAMATESN. Choy; K. Y. Moon; C. Park; Y. C. Son; W. H. Jung; Ho-Il Choi; C. S. Lee; C. R. Kim; S. C. Kim; H. Yoon
179-183REDUCTIVE ALKYLATION OF α-AMINOAMIDESPaolo Pevarello; Raffaella Amici; Vittorio Pinciroli; Mario Varasi
185-192CONDENSATION OF FORMALDEHYDE WITH PHLOROGLUCINOL AND ITS MONOMETHYL ETHERE. Kiehlmann; E. C. Lathioor; K. W. Lai
193-201SYNTHESIS AND ENZYMATIC RESOLUTION OF A CARBOCYCLIC ANALOGUE OF RIBOFURANOSYLAMINEMichael L. Edwards; James E. Matt Jr.; David L. Wenstrup; Christopher A. Kemper; Rose A. Persichetti; Alexey L. Margolin
203-209SYNTHESES OF α- AND β-DIMERS OF LITHOCHOLIC ACID ESTERSYuexian Li; Jerry Ray Dias
211-214SYNTHESIS OF cis-[4-(AMINOMETHYL)-2-CYCLOPENTENYL]METHANOL FROM NORBORNADIENECarmen Balo; Belen Dominguez; Franco Fernandez; Evangelina Lens; Carmen Lopez
215-216A CONVENIENT SYNTHESIS OF 2(5H)-FURANONERuzhen Cao; Chong Liu; Lunzu Liu
217-221SYNTHESIS OF 7-DESOXY-8-ALLYLCOUMARINSRaghao S. Mali; Ashok S. Walture; Kantipudi N. Babu
221-225EXPEDIENT SYNTHESES OF ESPINTANOL, p-METHOXYCARVACROL AND THYMOQUTNOL DIMETHYL ETHERBjora C. Soderberg; Shari L. Fields
226-230CONDENSATION OF 1,4-DIACETYL-2,5-PIPERAZINEDIONE WITH ALDEHYDES PROMOTED BY ULTRASONICALLY DISPERSED POTASSIUMLi Xin Wang; Yao Zeng Shi; Ming Hua Xu; Hong Wen Hu
230-234SYNTHESIS OF 1,3,6,8-TETRAMETHOXY-cis-4b,5,9b,10-TETRAHYDROINDENO[2,1-a]INDENE-5,10-DIONED. E. Bianchi; E. N. Alesso; G. Y. Moltrasio Iglesias
234-237RAPID OXIDATION OF SULFIDES AND SULFOXIDES WITH SODIUM HYPOCHLORITEJitender M. Khurana; Atulya K. Panda; Abhijit Ray; Amita Gogia
237-241MIXED DISULFIDES OF L-CYSTEINE AND ITS DERIVATIVES WITH 2-MERCAPTOETHANOLHerbert T. Nagasawa; Jonathan F. Cohen; William B. Rathbun
242-2446,6-bis(CARBOXY-2-OXABUTYL)-4,8-DIOXAUNDECANE-I,II-DICARBOXYLIC ACIDGeorge R. Newkome; Claus D. Weis
245-246SYNTHESES OF 2-CHLORO-4,5-DIFLUOROBENZOIC ACIDZhibin Li; Naihua Huang
247CORRIGENDUM

Volume 28, Issue 1 (1996)

CEditorial Board Page
1-64SYNTHESIS OF β-CARBOLINES. A REVIEWBrian E. Love
65-76ACTIVE-SITE-DIRECTED ENZYME-ACTIVATED N-NITROSOAMIDE INHIBITORS OF TRYPSINYulong Chen; Emil H. White
77-81ENANTIOSELECTIVE SYNTHESIS OF N-Boc AND N-Fmoc PROTECTED DIETHYL 4-PHOSPHONO(DIFLUOROMETHYL)-L-PHENYLALANINE (F2Pmp)Mark S. Smyth; Terrence R. Burke Jr.
83-90A CONVERGENT AND STEREOSELECTIVE SYNTHESIS OF CEMBRENENE PRECURSOR-4,10-DIMETHYL-7-ISOPROPENYL-14-OXO-3Z,5E,10E-PENTADECATRIENALWeidong Li; Yulin Li; Ying Li
91-95AN IMPROVED SYNTHESIS OF HIGH-PURITY FELODIPINESai-Hay Yiu; Edward E. Knaus
97-101BENZOTRIAZOLE-MEDIATED SYNTHESIS OF N-ALKYL-N,N′-DIARYLHYDRAZINESAlan R. Katritzky; Sergei V. Verin; Baozhen Yang
103-109REGIO- AND STEREOSELECTIVE OXIDATIONS OF THE EXOCYCLIC SULFUR ATOM OF TWO ENDOCYCLIC KETENE DITHIOACETALSRobert D. Walkup; Dan W. Knight; Simon G. Bott
111-115SYNTHESIS OF (±)-3-BROMOMETHYL-1,5-HEXADIENE AND (±)-3-BROMOMETHYL-3-METHYL-1,5-HEXADIENERichard A. Bunce; Brian J. Murray
115-117A FACILE PREPARATION OF BUSPIRONE N-OXIDE USING DAVIS' REAGENTBang-Chi Chen; Derron R. Stark
117-120A FACILE METHOD FOR DEBROMINATION OF vic-DIBROMIDESMing Zheng; Mei-Hua Zhang; Jian-Guo Shao; Qi Zhong
121-123RAPID N-ALKYLATION OF BENZOXAZINONES AND BENZOTHIAZINONES UNDER MICROWAVE IRRADIATIONZhi-Zhen Huang; Liu-Sheng Zu
123-125IMPROVED PREPARATION OF SOME NITROINDOLINESMichael B. Mortensen; Fadhil S. Kamounah; Jørn B. Christensen

Volume 27, Issue 6 (1995)

CEditorial Board Page
603-612CYCLOADDITIONS OF AZIDOALKYLCARBOXYLATES TO ACETYLENES AND ENAMINES. REGIOSELECTIVE SYNTHESIS OF SUBSTITUTED TRIAZOLESF. Palacios; A. M. Ochoa de Retana; J. Pagalday; J. M. Sánchez
613-619NOVEL SYNTHESIS OF SOME PYRIDINETHIONE NUCLEOSIDES RELATED TO 3-DEAZAUREDINEAdel M. E. Attia; Elsayed I. Ibrahim; Fouad E. A. Hay; Mohammed M. A. Abbasi; Hanaa A. E. Mansour
621-624PRACTICAL SYNTHESIS AND CHARACTERIZATION OF 7-BENZYLIDENENALTREXONE (BNTX)Anita H. Lewin; Melanie R. Nilsson; Jason P. Burgess; F. Ivy Carroll
625-6351,3-DIPOLAR CYCLOADDITION OF AZIDOALKYLPHOSPHONATES AND CARBOXYLATES TO MALEIMIDE AND NAPHTHOQUINONEF. Palacios; A. M. Ochoa de Retana; J. Pagalday
637-644A SYNTHESIS OF 4-α-GUANIDINO-2-DEOXY-2,3-DIDEHYDRO N-ACETYLNEURAMINIC ACIDJohn Scheigetz; Robert Zamboni; Michael A. Bernstein; Bruno Roy
645-650REGIOSELECTIVE BROMINATION OF CARDANOL DERIVATIVESO. A. Attanasi; S. Buratti; P. Filippone
651-652IMPROVED SYNTHESIS OF 2H-1,3(3H)-OXAZINE-2,6-DIONE (OXAURACIL)Gretchen M. Rehberg; Brian M. Glass
652-656DIBROMANTIN AS A REAGENT FOR THE AROMATIC BROMINATION OF POLYALKYLBENZENESXavier Herault; Pakorn Bovonsombat; Edward Mc Nelis
657-659AN IMPROVED SYNTHESIS OF 1-(2-HYDROXYETHYL)URACILBaijayantimala Garnaik
660-663SRN1 REACTIONS IN LIQUID AMMONIA AT ROOM TEMPERATUREP. G. Manzo; S. M. Palacios; R. A. Alonso; R. A. Rossi
663-667FACILE SYNTHESIS OF 3-CHLOROCOUMARINSRaghao S. Mali; Jyoti V. Deshpande
668-670PREPARATION OF NEW 4′,5′-DISUBSTITUTED BENZOCROWN ETHERSHaluk Akkus; Ahmet Gül
671-674PREPARATION OF 2(2-HYDROXYMETHYL-6-METHYL)PHENYLETHANOLD. G. Tombari; A. G. Moglioni; G. Y. Moltrasio Iglesias
674-678A CONVENIENT SYNTHESIS OF δ-CONICEINENorbert De Kimpe; Elena Stanoeva; Angelina Georgieva; Marian Keppens; Oleg Kulinkovich
678-682SYNTHESIS OF PYRAZINO(3,2,1-J,K)CARBAZOLE DERIVATIVESK. J. Rajendra Prasad; C. S. Vijayalakshmi; D. Sowmithran
682-684AN EFFICIENT SYNTHESIS OF (S)-(+)-2-TRIDECANOL ACETATE, AN AGGREGATION PHEROMONE OF DROSOPHILA MULLERIFranz Bracher; Brigitte Schulte
685-690SYNTHESES OF 3-AND 3,3′-SUBSTITUTED 1,1′-BI-2-NAPHTHOLSJing Li; Weidong Li; Ying Li; Yulin Li; Shiyan Yang
691-694SYNTHESIS OF A SPIROCYCLIC OXENDOLE ANALOGUE AS A PUTATIVE REPLACEMENT FOR PR02-PRO3-GLY4-PHE5 IN BRADYKININ ANTAGONISTSR. Richard Goehring

Volume 27, Issue 6 (1995)

695-697A PRACTICAL SYNTHESIS OF 4-BROMO-2-CYANO-3-METHYL-2-BUTENENITRILELinda S. Newton; Samantha Chan; Barbara J. Sitter; Steven J. Brenek; Jeffery W. Raggon; Tamim F. Braish
697-700NEW METHOD FOR THE PREPARATION OF GUANYLTHIOUREASPeter Tari; Antal Gajary
700-703AN IMPROVED SYNTHESIS OF 3-(2,5-DIMETHOXYBENZYL)PYRROLEChristina Aquino-Binag; Naresh Kumar; Paul Pigram
703-706OXIDATION OF VARIOUS ALCOHOLS WITH IN SITU GENERATED MONTMORILLONITE K10-SUPPORTED FERRIC NITRATE REAGENT IN AN APROTIC SOLVENTMasao Hirano; Kan Komiya; Takashi Morimoto
707-709AN IMPROVED SYNTHESIS OF DIMETHYLTITANOCENEJoseph F. Payack; David L. Hughes; Dongwei Cai; Ian F. Cottrell; Thomas R. Verhoeven
709-713(±)-3,4,4a,5,6,7-HEXAHYDRO-4a,7,7-TRIMETHYL-1(2H)-NAPHTHALENONERichard A. Bunce; R. Shawn Childress
715CORRIGENDA
717-734INDEXES

Volume 27, Issue 5 (1995)

CEditorial Board Page
519-540RECENT ADVANCES IN THE REACTIONS OF HYDRAZINES AND HYDROXYLAMINES WITH (α,β-UNSATURATED AND β-DICARBONYL COMPOUNDSKirill N. Zelenin
541-545B-HYDROXYDIISOPINOCAMPHEYLBORANE AS A MILD, CHEMOSELECTIVE REDUCING AGENT FOR ALDEHYDESJin Soon Cha; Eun Ju Kim; Oh Oun Kwon; Sang Yong Kwon; Wone Woo Seo; Seok Won Chang
547-550SYNTHESIS OF [1]BENZOPYRANO[3,4-h]BENZO[b]-1,6-NAPHTHYRIDINE-6-ONESK. Rajendra Prasad; Malleshwar Darbarwar
550-552AN IMPROVED SYNTHESIS OF FENBUFENRafael Castillo; Margarita Suárez-Herrera; Mayra Aparicio; Francisco Hernández-Lui; Alicia Hernández
552-555IMPROVED SYNTHESIS OF PHENYLACETAMIDES BY THE WILLGERODT REACTION WITH MICROWAVE HEATINGChristopher R. Strauss; Robert W. Trainor
555-559A CHEMOENZYMATIC SYNTHESIS OF (R)-2-(1-HYDROXYETHYL)-1,3-DITHIANEFranz Bracher; Thomas Litz
559-561CHALCONES BY THE WITTIG REACTION OF A STABLE YLIDE WITH ALDEHYDES UNDER MICROWAVE IRRADIATIONCaiding Xu; Guoying Chen; Xian Huang
561-564A NEW, VERY SHORT PREPARATION OF 3-BENZOYLCYCLOHEXANONE, A KEY BUILDING BLOCK IN KETOPROFEN SYNTHESISRoberto Ballini; Giovanna Bosica
564-566ULTRASONICALLY ACCELERATED SYNTHESES OF FURAN-24-DICARBALDEHYDE FROM 5-HYDROXYMETHYL-2-FURFURALLouis Cottier; Gérard Descotes; Jaroslaw Lewkowski; Romuald Skowroñski
567-568IMPROVED PREPARATION OF tris-(2-FURYL)PHOSPHINEAntonio J. Zapata; Ana C. Rondon
569-570AN IMPROVED PROCEDURE FOR THE PREPARATION OF 3-METHYL-2-CYCLOPENTEN-1-ONEMatthew L. Karpinski; Dale Nicholas; John C. Gilbert
571-572ONE-POT SYNTHESIS OF 4-[2-(3, 4-DICHLOROPHENOXY)ETHYL]-1-PENTYLPIPERIDINE HYDROCHLORIDE (SB 201823-A)Oskar Axelsson; Dan Peters
572-574THE SYNTHESIS OF TRIMETHYLSILYLMETHOXYMETHYL CHLORIDEArthur G. Schultz; Yongwen Wang
574-575A CONVENIENT LARGE-SCALE PREPARATION OF endo-2-METHYLBICYCLO[2.2.1]HEPT-5-ENE-exo-2-CARBOXYLIC ACIDAlan R. Katritzky; Qingmei Hong; Zhijun Yang; Darren J. Cundy; Katherine Brown-Wensley
576-579SONICATION AND ALUMINUM AMALGAM IN THE LEIMGRUBER-BATCHO REACTION. AN IMPROVED PREPARATION OF 6-AMINOINDOLEF. Dean Toste; I. W. J. Still
579-581A NOVEL SYNTHESIS OF TRIARYLBISMUTH DISULFONATESLi-Ming Jiang; Zhi-Zhen Huang; Xian Huang

Volume 27, Issue 5 (1995)

582-586A CONCISE SYNTHESIS OF PELLITORINEJ. Edward Semple
586-590A LARGE SCALE PREPARATION OF 1-ETHYNYLCYCLOPENTENE AND 1-HEXEN-4-YNEEnrico Davin; Matteo Giongo; Mario Riocci
590-592TRIMETHYLSILYL TRICHLOROACETATE AS A CHLOROFORM ALTERNATIVE FOR THE SYNTHESIS OF α-(TRICHOLOROMETHYL)-3-NITROBENZYL ALCOHOLSteven A. Weissman
592-595SYNTHESIS OF 1,3-DIMETHYLAZULENENicholas M. Irvine; Marek Majewski
595-600SYNTHESIS OF ACETOXYLATED AND HYDROXYLATED NITROBENZO[a]PYRENE AND NUROBENZO[e]PYRENEM. -J. Lee; J. -S. Lai; E. Cheng; P. P. Fu
600-602LARGE SCALE SYNTHESIS OF 2-CHLORO-5-FLUOROPYRIMIDINEAudrey Dunaiskis; Tom Staigers; Tom Keltonic; Tom Chappie; Cliff Meltz; Robert Dugger; Mark A. Sanner

Volume 27, Issue 4 (1995)

CEditorial Board Page
383-456ACYL MAIN GROUP METAL AND METALLOID DERIVATIVES IN ORGANIC SYNTHESIS. A REVIEWCarmen Nájera; Miguel Yus
457-462ALTERNATE PREPARATION OF α-KETO ESTERS FROM ACID CHLORIDESAlan R. Katritzky; Zuoquan Wang; Adam P. Wells; Peter J. Steel
463-467REACTION OF 3-SULFOLENES WITH CONJUGATED ALDEHYDES AND KETONESR. Padmakumar; T. Subramanian; S. V. Bhat
469-473AN EFFICIENT SYNTHESIS OF DAGOP. Anantha Reddy; James P. Hayes; Anita H. Lewin; George A. Brine
475-479SYNTHESIS OF NEW POLYMTROSTILBENESXinhua Peng; Tianyun Chen; Chunxu Lu; Rongkang Sun
480-482OXIDATIVE CLEAVAGE OF KETOXIMES WITH BENTONITIC CLAY-SUPPORTED COPPER (II) NITRATER. Sanabria; P. Castaneda; R. Miranda; A. Tobón; F. Delgado; L. Velasco
483-487A CONVENIENT PREPARATION OF 1-HYDROPEROXY-(1-p-NITROPHENYL)ETHANOL BY THE ACID-CATALYZED OXIDATION OF p-NITROACETOPHENONE WITH HYDROGEN PEROXIDELázaro F. R. Cafferata; Juan C. Autino
487-492NEW CONDENSATION PRODUCTS OF DIAMINES WITH 3-UREIDOMETHYLENECOUMARINM. Hamdi; R. Sakellariou; V. Spéziale
492-494A NOVEL SYNTHESIS OF ORGANIC DISELENIDESZhi-Zhen Huang; Fei-Yan Liu; Jing-Xing Du; Xian Huang
495-498A CONVENIENT PREPARATION OF DIBENZO[a,e]CYCLOOCTATRIENE USING FRIEDEL-CRAFTS INTRAMOLECULAR ACYLATIONTakehiko Yamato; Hisataka Inoue; Maki Fukumoto; Masashi Tashiro
499-500IMPROVED PREPARTION OF 2,5-DIMETHYL-1,3-CYCLOHEXANEDIONEDelphine Joseph; Maria-Joao Queiroz; Gilbert Kirsch
500-503AN IMPROVED SYNTHESIS OF 4-HYDROXY AND 4′-METHOXYBIPHENYL-2-CARBOXYLIC ACIDSGeneviève Estenne; Pierre Dodey; Patrice Renaut; Gérard Leclerc
503-5061-(BENZENESULFONYL)PYRROLE-3-CARBOXALDEHYDEDong Xiao; Daniel M. Ketcha
507-510LIPOSOMES PREPARED FROM 2-[bis-(2-HEXACOSA-10, 12-DIYNOLOXYETHYL)AMINO]ETHANESULFONIC ACIDMark T. Holtzapple; Frank C. VanDuker Jr.; Ki Y. Nam; James J. Lalond
510-513A SUPERIOR SYNTHESIS OF CHOLINERGIC ANABASEINEJohn A. Zoltewicz; Michael P. Cruskie Jr.
513-516A PRACTICAL SYNTHESIS OF 4-(3′,4-DIHYDROXYLPHENYL)-1,2,3,4-TETRAHYDROKOQUINOLINEXumiao Zhao; Xiuying Wan
517CORRIGENDUM

Volume 27, Issue 3 (1995)

CEditorial Board Page
243-272RECENT PROGRESS IN THE SYNTHESIS OF NITROPOLYARENES. A REVIEWBongsup P. Cho
273-303SYNTHETIC AND ANALYTICAL ASPECTS OF THE CHEMISTRY OF PIRACETAM-TYPE SUBSTITUTED PYRROLIDINES. A REVIEWAlex Haahr Gouliaev; Jane Binau Mønster; Mette Vedsø; Alexander Senning
305-346NATURALLY OCCURRING β-LACTONES: OCCURRENCE, SYNTHESES AND PROPERTIES. A REVIEWChristopher Lowe; John C. Vederas
347-354THE PREPARATION OF SOME ANALOGUES OF MYRISTOYL CoARatna Pankayatselvan; Frank S. Guziec Jr.; Aravamudan S. Gopalan; Ramesh Raghavachari; Lynn James Guziec; Dongchu Wei; Ronald L. Felsted; Constance J. Glover
355-359SYNTHESIS OF 1-ARYLCYCLOPROPANECARBONITRILES UNDER PHASE-TRANSFER CATALYTIC CONDITIONSMichal Fedorynski; Andrzej Jonczyk
361-366PREPARATION OF THIOL ACIDS, THIOL ESTERS AND AMIDES BY REACTIONS OF CARBONYL SULFIDE WITH GRIGNARD REAGENTSAlan R. Katritzky; Jean-Luc Moutou; Zhijun Yang
367-372THE NICKEL(I) CATALYZED COUPLING OF A DIARYLZINC WITH AN ARYL CHLORIDE IN THE SYNTHESIS OF XENALIPINJohn F. Eaddy
373-374FACILE OXIDATIVE DECARBOXYLATION OF AROMATIC α-HYDROXY ACIDS BY SODIUM METAPERIODATE IN THE PRESENCE OF DIBENZO-[18]-CROWN-6 AND PTCA. R. Kore; A. D. Sagar; M. M. Salunkhe
375-377SOLID-PHASE SYNTHESIS OF A PEPTIDE COMPRISING THE 605-611 DISULFIDE LOOP OF GP41, TRANSMEMBRANE GLYCOPROTEIN OF HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 (HIV-1)G. G. Gevorkian; M. Viveros; F. Zamudio; C. Larralde
378-380A SIMPLE PREPARATION OF MONO-tert-BUTYL BENZYLOXYCARBONYL-L-GLUTAMATESMichal Kempny; Barbara Rzeszotarska; Krzysztof Pawelczak
381-382FURTHER APPLICATIONS OF THE NOVEL SYNTHESIS OF ARYLTHIOGLYCOLIC ACIDSY. Yildirir; A. Disli

Volume 27, Issue 2 (1995)

CEditorial Board Page
127-160PALLADIUM- AND/OR COPPER-MEDIATED CROSS-COUPLING REACTIONS BETWEEN 1-ALKYNES AND VINYL, ARYL, 1-ALKYNYL, 1,2-PROPADIENYL, PROPARGYL AND ALLYLIC HALIDES OR RELATED COMPOUNDS. A REVIEWRenzo Rossi; Adriano Carpita; Fabio Bellina
161-169PHOSPHORYLATED ADENINE DERIVATIVES AS POTENTIAL SYNTHONS FOR ANTIVIRAL AGENTSMarwan El Masri; K. Darrell Berlin
171-178“ONE POT” SYNTHESIS OF β-FUNCTIONALIZED VINYL AZIDES THROUGH ADDITION OF TETRAMETYLGUANIDINIUM AZIDE TO ACETYLENIC AND ALLENIC COMPOUNDSF. Palacios; D. Aparicio; J. M. de los Santos; I. Perez de Heredia; G. Rubiales
179-184PERFORMANCE FLUIDS AS AN INERT MEDIUM FOR THE PREPARATION OF BENZOTRIAZOLE DERIVATIVESAlan R. Katritzky; Dorin Toader; Jinlong Jiang
185-212SYNTHESIS OF AMINOCYCLOBUTANE MONO- AND DICARBOXYLIC ACIDS AND DERIVATIVES THEREOF FROM (PHENYLSULFONYL)BICYCLOBUTANESYehiel Gaoni
213-216A NOVEL SYNTHESIS OF α-ARYLSELENOPHOSPHORANESLi Wang; Zhi-Zhen Huang; Hang Li; Xian Huang
216-219COUPLING OF THIOLS AND SELENOLS CATALYZED BY TRIS[TRTNITRATOCERIUM (IV)]PARAPERIODATEN. Iranpoor; P. Salehi; F. Shiriny
219-221AN IMPROVED PROCEDURE FOR THE PREPARATION OF ARYLOXIRANESLeslie W. Deady; José Desneves
221-224SYNTHESIS OF ALDIMINES BY DEOXYGENATION OF NITRONESS. Sivasubramanian; V. Ramamoorthy; G. Balasubramanian
224-228IMPROVED PREPARATIONS OF SYMMETRIC PORPHYRINSLingjiang Cheng; Jinshi Ma
229-232SIMPLE AND CONVENIENT PROCEDURE FOR THE PREPARATION OF ACID CHLORIDES OF PENICILLINSErnesto G. Mata; Carlos E. Boschetti; Oreste A. Mascaretti
233-236PREPARATION OF 4-CHLORO-2-THIOPHENECARBOXYLIC ACID via SELECTIVE BISULFITE SALT ADDITION PROCEDUREJeffrey W. Raggon; Jennifer M. Welborn; Jane E. Godlewski; Sarah E. Kelly; Thomas G. Lacour
236-239A NEW EFFICIENT SYNTHESIS OF 3-AMINO-1-PHENYLPYRROLEFrédéric Fabis; Patrick Dallemagne; Sylvain Rault; Max Robba
239-242A PRACTICAL METHOD FOR THE SYNTHESIS OF N-FLUORENYLMETHOXYCARBONYL DIAMINESMaciej Adamczyk; Jonathan Grote

Volume 27, Issue 1 (1995)

CEditorial Board Page
1-31SYNTHESIS AND CHEMISTRY OF MELATONIN AND OF RELATED COMPOUNDS. A REVIEWHelmut M. Hugel; David J. Kennaway
33-74TRIFLUOROMETHYL AND PERFLUOROALKYL DERIVATIVES OF AZOLES. A REVIEWJosé Elguero; Alain Fruchier; Nadine Jagerovic; Andreas Werner
75-80SYNTHESIS OF HALOGENATEDISOXAZOLYL NAPHTHOQUINONESV. G. Dabbene; M. C. Briñón; M. M. De Bertorello
81-83EFFICIENT REDUCTION OF NTTROARENES TO AMINES BY SODIUM BOROHYDRIDE AND CUPROUS BROMIDE-DIMETHYL SULFIDEHimatkumar V. Patel; Kavita A. Vyas; Sudhanshu P. Pandey; Peter S. Fernandes
84-86IODINATION OF NAPHTHOQUINONES AND COUMARIN CATALYZED BY CERIC AMMONIUM AND MERCURIC NITRATESJ. Sharma; P. K. Singh; K. P. Singh; R. N. Khanna
87-91THE SYNTHESIS AND CHARACTERIZATION OF NOVEL bis(FORMAZANS)Yasar Gok; H. Basri Senturk
92-95INVERSE-ELECTRON DEMAND DIELS-ALDER CYCLOCONDENSATIONS IN THE SYNTHESIS OF 5-8-5 FUSED RING SYSTEMSJ. Gabriel Garcia; Mark L. McLaughlin
95-98TRANSFORMATION OF CARBOXYLIC ESTERS TO ALDEHYDES WITH SODIUM tris(DIETHYLAMINO)ALUMINUM HYDRIDEJin Soon Cha; Jong Mi Kim; Min Kyoo Jeoung; Oh Oun Kwon; Eun Ju Kim
99-102SYNTHESIS OF ALLYL ETHENYL ETHERS USING S-ETHENYLSULFILIMINESTamotsu Yamamoto; Shigeru Fujita; Kei Sugawara; Tsuyoshi Watanabe
103-106SYNTHESIS OF 2-SUBSTITUTED 3,4-DIHYDROOXAZOLES USING S-ETHENYLSULFILIMINESKatsuya Ikeda; Hiroyuki Honda; Takanori Matsuo; Tamotsu Yamamoto
107-108SYNTHESIS OF (S)-(+)PANTOLACTONEMonique Calmes; Jacques Daunis; Robert Jacquier; Francois Natt
109-113SYNTHESIS OF 5-ALKYLAMINO- AND 5-DIALKYLAMINO-5-DEOXYTHYMIDINE AND 5′-DEOXY-XYLO-THYMIDINE ANALOGSWojciech Urjasz; Lech Celewicz; Krzysztof Golankiewicz
113-117SYNTHESIS OF 3-VINYLINDOLES FROM 3-ALKYLIDENEINDOL-2(3H)-ONESE. M. Beccalli; A. Marchesini
117-120A SAFE AND CONVENIENT PROCEDURE FOR THE SYNTHESIS OF POLYAMBSES via AZIDE INTERMEDIATESVladimir V. Martin; Laszlo Lex; John F. W. Keana
120-122IMPROVED PREPARATION OF 2,5-DIMETHYL-1,4-CYCLOHEXANEDIONEMaria-Joao Queiroz; Delphine Joseph; Gilbert Kirsch
122-125SYNTHESIS OF 5-BROMO-3,3-DIPHENYL-1-PENTENERichard A. Bunce; R. Shawn Childress

Volume 26, Issue 6 (1994)

CEditorial Board Page
617-644RECENT PROGRESS IN THE SYNTHESIS OF AVERMECTINS AND MILBEMYCINS. A REVIEWTimothy A. Blizzard
645-670SYNTHESIS OF α,ω-ALKANEDIOLS. A REVIEWSarita A. Patwardhan
671-674AN EFFICIENT SYNTHESIS OF (2R, 5R)- AND (2R, 5S)-2-METHYL-5-HYDROXYHEXANOIC ACID LACTONESMing-Jung Wu; Jiann-Yih Yeh
674-677SIMPLIFIED CONDITION FOR SYNTHESIS OF CURCUMIN I AND OTHER CURCUMINOIDSK. V. D. Babu; K. N. Rajasekharan
677-680A HIGH-YIELD SYNTHESIS OF 3-PENTADECYLPYRIDINEWayne M. Stalick; Joseph H. Murray
680-682AN IMPROVED ELECTROSYNTHETIC PREPARATION OF THE FEMALE HOUSEFLY SEX PHEROMONEE. A. Marquez; A. J. Zara; J. Tércio; B. Ferreira; L. O.de; S. Bulhões
682-684THE SYNTHESIS OF 6-PROPYL-2-SELENOURACIL, THE SELENIUM ANALOGUE OF THE ANTI-THYROID DRUG PTUWei-Xiao Hu; Frank S. Guziec Jr.
685-687A CONVENIENT DIRECT PREPARATION OF 2-CYANOPYRIMIDINEWei-Xiao Hu; Ratna Pankayatselvan; Frank S. Guziec Jr.
687-690ANALOGS OF TRYPTOPHANEmil Pop; Katalin Prókai-Tátrai; Marcus E. Brewster; Nicholas Bodor
691-695PRODUCT SELECTIVITY IN THE SYNTHESIS OF THREE NOVEL PHOSPHORUS-CONTAINING HETEROCYCLES FROM ACYCLIC PRECURSORS BY SELECTION OF BASE STRENGTHCharles C. Orji; A. G. Pinkus
696-701MONOSUBSTITUTED 2,2′-BIPYRIDINESMilon Sprecher; Ronald Breslow; Orly Uziel; Todd M. Link
702-705SYNTHESIS OF R-(+)-1,3-DITHIANE 1-OXIDE
706-711PREPARATION OF METABOLITES OF IMIPRAMINE AND PHENYTOINMaciej Adamczyk; Jeffrey R. Fishpaugh; John C. Gebler; Kevin J. Heuser
713-726INDEXES

Volume 26, Issue 5 (1994)

CEditorial Board Page
499-531RECENT DEVELOPMENTS IN TETRAZOLE CHEMISTRY. A REVIEWSteven J. Wittenberger
533-538SYNTHESIS OF A S-4-CARBOXYPHENYLALANINE DERIVATIVE FOR USE IN PEPTIDE SYNTHESISRobert G. Franz; Joseph Weinstock; Raul R. Calvo; James Samanen; Nambi Aiyar
539-547PREPARATION OF TRIOLS AND ETHERS RELATED TO PODOPHYLLOTOXINM. A. Castro; M. Gordaliza; J. Miguel del Corral; A. San Feliciano
549-551A CONVENIENT SYNTHESIS OF 3-(2-METHYLPYRIDYL)ACETIC ACID METHYL ESTER, A PYRITHIAMINE INTERMEDIATEMilena E. Ivanova; Vanya B. Kurteva; Maria J. Lyapova
551-554CONVENIENT SYNTHESIS OF 2,3-DIHYDROXY-2-METHYLPROPANAMIDE via 2,3-EPOXY-2-METHYLPROPANAMIDEJ. F. Pilichowski; G. Mailhot; M. Bolte
555-557SYNTHESIS OF ALKYL ISOTHIOCYANATES FROM PRIMARY ALKYL AMINES USING DICYANDIAMIDE AS A DEHYDROSULFURIZING AGENTTamotsu Yamamoto; Atsushi Terada; Takashi Muramatsu; Katsuya Ikeda
557-560AN IMPROVED SYNTHESIS OF 9-CHLORO-1,8-p-MENTHADIENETeodoro S. Kaufman; Ranjan P. Srivastava; Robert D. Sindelar
560-5675-NITRO-2-FURYL DIIMIDOYL DISULFIDES BY IODINE OXIDATION OF N-ARYL-5-NITRO-2-THIOFURAMIDESAna Dunja Mance; KrešImir Jakopčić
567-570RESOLUTION OF 5-VINYL-2-PYRROLIDINONE. A PRACTICAL SYNTHESIS OF (S)- AND (R)-VIGABATRINZ. Y. Wei; Edward E. Knaus
571-573FACILE SYNTHESIS OF PHEROMONE OF Dichocrocis Punctiferalis, A SERIOUS PEST OF SPICESS. A. Hassarajani; A. S. Subaraman; V. R. Mamdapur
573-577USEFUL SYNTHESES OF PYRANO- AND PYRIDOINDOLESRaghao S. Mali; Anita Manekar-Tilve
578-580AN IMPROVED SYNTHESIS OF Nε-FMOC-L-LYSINE AND Nδ-FMOC-L-ORNITHINEMaria Henczi; Donald F. Weaver
580-583AN EFFICIENT AND CONVENIENT PROCEDURE FOR ESTER HYDROLYSISJ. M. Khurana; Arti Sehgal
583-588CONVERSION OF AROMATIC NITRILES TO ALDEHYDES BY SODIUM tris (DIALKY-LAMINO) ALUMINUM HYDRIDESJin Soon Cha; Min Kyoo Jeoung; Jong Mi Kim; Oh Oun Kwon; Jae Cheol Lee
588-593SYNTHESIS AND REACTIONS OF PHOSPHINIMINES USING HYDRAZONOYL HALIDESHamdi M. Hassaneen; Nehal M. Elwan; Hyam A. Abdelhadi; Monther T. Fouad; Mohammed S. Algharib
593-595OXIDATION OF 3β-ACETOXY-5α-LANOST-8-ENE WITH CHROMYL CHLORIDE. THE PREPARATION OF 5α,8β-LANOST-9(11)-EN-7-ONE DERIVATIVESK. Staliński; Z. Paryzek
595-598A SIMPLE PROCEDURE FOR THE PREPARATION OF 2-PHOSPHORYLATED FURANOSESClemens Lamberth

Volume 26, Issue 5 (1994)

599-602SYNTHESIS OF 1,3-DIAMINESVioletta Constantinou-Kokotou; George Kokotos
602-605A CONVENIENT PREPARATION OF 4-VINYLPHENYLACETIC ACID AND ITS METHYL ESTERStephen W. Wright; Lester D. McClure
605-608IMPROVED SYNTHESIS OF FLUOROMETHYL PHENYL SULFONEDonald P. Matthews; Rose A. Persichetti; James R. McCarthy
608-610AN EFFICIENT ONE STEP SYNTHESIS OF tert-BUTYL GLYCINATE AND tert-BUTYL SARCOSINATEFlorine Cavelier; Marc Rolland; Jean Verducci
611-614A CONCISE SYNTHESIS OF 8-PHENYLOCTADECANOIC ACIDRajiv Sharma; Victor E. Marquez
615CORRIGENDUM

Volume 26, Issue 4 (1994)

CEditorial Board Page
393-420SYNTHESIS OF CARCINOGENIC OXYGENATED DERIVATIVES OF BENZ[c]ACRIDINES. A REVIEWNoboru Motohashi; Masami Kawase; Jahangir Emrani
421-428SYNTHESIS OF 4-(NITROBENZYL- AND BENZOYL)PIPERIDINE DERIVATIVES BY NITRATION OF ARYLALKYLPIPERIDINESSiya Ram
429-438SYNTHESIS OF IMIDAZOQUINOLINES AND IMIDAZOISOQUINOLINES FROM AZANAPHTHALENE CARBOXYLIC ACIDSKevin C. Langry
439-444AN ALTERNATIVE SYNTHESIS OF ARYL AND HETEROARYL BROMIDES FROM ACTIVATED ARYL HYDROXY COMPOUNDSAlan R. Katritzky; Jianqing Li; Christian V. Stevens; David J. Ager
445-457A CONVERGENT SYNTHESIS OF (±)-SARCOPHYTOL-A BENZYL ETHERWeidong Li; Jianmin Mao; Ying Li; Yulin Li
459-464REDUCTION OF ORGANIC COMPOUNDS WITH SODIUM ALUMINUM HYDRIDE IN THEORETICAL AMOUNTJin Soon Cha; Herbert C. Brown
465-468SYNTHESIS OF SEVERAL N-SUBSTITUTED AMINO-2-PYRIDONESGalal E. H. Elgemeie; Samia R. El-Ezbawy; Hosny A. Ali; Abdel-Kader Mansour
469-471IMPROVED ALKYLATION OF ETHYL ACETOACETATE AND DIETHYL MALONATEDidier Barbry; Catherine Faven; Aziz Ajana
471-472IMPROVED PREPARATION OF 4-CHLOROMETHYLPHENYL ACETATEJørn B. Christensen
473-476SYNTHESIS AND COMPETITIVE N- AND O-ALKYLATION OF 10-METHYLPYRIDO[3,2-g]QUINOLINE-4,6-DIONEA. Mahamoud; J. -P. Galy; J. Barbe
476-478A CONVENIENT PREPARATION OF 9H-FLUORENE-9-ACETIC ACIDR. Richard Goehring
479-482REGIOSELECTIVE SYNTHESIS OF 10-HYDROXY-11-METHOXYAPORPHINE FROM (RS)-10,11-DIHYDROXYAPORPHINEJack C. Kim; Won-Woo Park
482-484A SHORT SYNTHESIS OF TRIDEC-12-EN-2-ONE, THE MINOR CONSTITUENT OF THE BARK OF LITSEA ELLIPTICA (LAURACEAE)S. Mithran; A. S. Subbaraman; V. R. Mamdapur
485-488TREATMENT OF CONJUGATED AZOALKENES WITH N-ACYL-N'-TOSYLHYDRAZIDES. A USEFUL ENTRY TO ASYMMETRIC bis-ACYLHYDRAZONESOrazio A. Attanasi; Stefania Santeusanio; Franco Serra-Zanetti
488-491A HIGHLY STEREOSELECTIVE TRANSFORMATION OF β-SANTALENE TO (E)-β-SANTALOLP. A. Unnikrishnan
491-494A SUPERIOR METHOD FOR THE SYNTHESIS OF 7a-METHYL-2,3,7,7a-TETRAHYDRINDEN-5(6H)-ONEH. Surya Prakash Rao; K. Subba Reddy
494-497A SIMPLE AND SHORT SYNTHESIS OF 2(2′-AMINOBENZYLAMINO)BENZYL ALCOHOL, A CONSTITUENT OF JUSTICIA GENDARUSSA BURM LEAVESVijayendra P. Kamat; Janardan K. Kirtany
498ADDENDUM. A SIMPLE, EFFICIENT PREPARATION OF 1,1-bis(TRIMETHYLSILOXY)-1,3-BUTADIENE

Volume 26, Issue 3 (1994)

CEditorial Board Page
257-290RECENT PROGRESS IN THE USE OF SULFONYL RADICALS IN ORGANIC SYNTHESIS. A REVIEWMichèle P. Bertrand
291-320THE SYNTHESIS AND REACTIONS OF PRISMANES. RECENT DEVELOPMENTSMark A. Forman; William P. Dailey
321-326FACILE AND HIGH-YIELD SYNTHESIS OF NEW 4-PHOSPHORANYLIDENE-4,5-DIHYDROPYRAZOL-5-ONES BY REACTION OF CONJUGATED AZOALKENES WITH PHOSPHINESOrazio A. Attanasi; Paolino Filippone; Daniela Giovagnoli
327-330A SIMPLE AND EFFICIENT PREPARATION OF METHOXYMETHYL ESTERS OF PENICILLINS AND CEPHALOSPORINSJacek Pankowski; Jerzy Winiarski
331-335A SIMPLE SYNTHESIS OF THE HETEROCYCLIC S,S-DIPHENYLSULFILIMINESOlga G. Vlasova; Oleg A. Rakitin; Lenor I. Khmelnitski
337-341AN ALTERNATE METHOD FOR THE SYNTHESIS OF SECONDARY NITRAMINESZ. Daszkiewicz; A. Domański; J. B. Kyziol
343-346AN EFFICIENT, LARGE-SCALE SYNTHESIS OF IDOXIFENE {(E)-1-[4-[2-(N-PYRROLIDINO)ETHOXY]PHENYL]-1-(4-IODOPHENYL)-2-PHENYL-1-BUTENE}Raymond McCague; Gerard A. Potter; Michael Jarman
347-349SINGLE-STEP SYNTHESIS OF 2,3-DIHYDRO-2,2DIMETHYL-1H-PHENOTHIAZIN-4(10H)-ONESV. Gupta; A. Gupta; R. S. Rathore; R. R. Gupta
349-352AN IMPROVED SYNTHESIS OF THIENO(2,3-B)QUINOLINES via S-OXIDESS. P. Rajendran; P. Shanmugam
353-355OXIDATIVE REARRANGEMENT OF THE PURINE RING USING MAGNESIUM MONOPERPHTHALATEAdel Amer
355-357AN ECONOMICAL PREPARATION OF 2-(2-BROMOETHYL)-1,3-DIOXANEJorn B. Christensen; Anne Schluter
357-360SYNTHESIS OF N-PHOSPHORYLUREAS BY REACTION OF PHOSPHORYLAMIDES WITH N-SUBSTITUTED TRICHLOROACETAMIDESJan Petrov; I. Atanassova; V. Ognyanova
360-362SYNTHESIS OF 3-ACETOACETYL-7-METHYL-2H,5H-PYRANO[4,3-B]PYRAN-2,5-DIONEB. Boutemeur-Kheddis; A. Bendaas; M. Hamdi; R. Sakellariou; V. Spéziale
362-366A NEW APPROACH TO ALKYL 2-OXOQUINOLINE-3-ACETATES BY TRIPHENYLPHOSPHINE-INDUCED CYCLIZATION OF ALKYL O-FORMYLMALEANILATESN. P. Argade; S. M. Babar; V. Balasubramaniyan
366-370EFFICIENT REGIOSELECTIVE ALKYLATION OF 2-CARBOXAMIDOPIPERAZINE. APPLICATION TO THE SYNTHESIS OF THE NMDA COMPETITIVE ANTAGONIST (�)-CPPP. Pevarello; G. Scappi; M. Varasi
370-373PURIFICATION OF 1,2-DIHYDRONAPHTHALENE- AN IMPORTANT INTERMEDIATE IN THE HYDROPROCESSING OF NAPHTHALENEMike D. Cagle; Sharbil J. Firsan; E. J. Eisenbraun

Volume 26, Issue 3 (1994)

374-376THE PREPARATION OF Δ2 STEROIDS. AN IMPROVED PROCEDUREP. Nowak; K. Blaszczyk; Z. Paryzek
377-378AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1,3-DITHIANEHarish K. Patney
379-382PREPARATION OF REDOX DERIVATIVES OF 3α-HYDROXY-5α-PREGNANE-11,20-DIONEEmil Pop; Marcus E. Brewster; Katalin Prókai-Tátrai; Nicholas Bodor
383-385SYNTHIESIS OF PYRAZOLO (3,4-b)QUINOLINES AND THEIR 1-PHENYL DERIVATIVESS. P. Rajendran; M. Manonmani; S. Vijayalakshmi
386-389OXIDATION OF AMINES BY DICHLORODICYANOQUINONE (DDQ) WITH TRAPPING BY TRIMETHYLSILYL CYANIDER. J. Sundberg; M. -H. Theret; L. Wright
391-392CORRIGENDUM

Volume 26, Issue 2 (1994)

CEditorial Board Page
129-158REAGENT-CONTROLLED ASYMMETRIC DIELS-ALDER REACTIONS. A REVIEWTaeboem Oh; Michael Rally
159-192o-HYDROXYARYL KETONES IN ORGANIC SYNTHESIS. A REVIEWAntigoni Kotali; Philip A. Harris
193-235ASYMMETRIC REDUCTIONS OF CARBON-NITROGEN DOUBLE BONDS. A REVIEWQi-Cong Zhu; Robert O. Hutchins; Marygail K. Hutchins
237-241CONVENIENT SYNTHESIS OF 2,3,5-TRIARYL-5-OXOPENTANOIC ACIDS AND OF THEIR t-BUTYL ESTERSV. Dryanska; A. Popovich
243-248AN EFFICIENT ONE-POT CONVERSION OF α-AMINO ACID ESTERS TO γ-AMINO-α,β-UNSATURATED CARBOXYLATESZ. Y. Wei; E. E. Knaus
249-255β-TRIFLUOROACETYLATION OF LACTAMS AND BENZOLACTAMSJ. P. Bouillon; C. Atès; C. Maliverney; Z. Janousek; H. G. Viehe

Volume 26, Issue 1 (1994)

CEditorial Board Page
1-84FURANOSESQUITERPENE SYNTHESIS. AN UPDATED REVIEWAngela J. Allen; Valerie Vaillancourt; Kim F. Albizati
85-100ORGANOTIN ENOLATES IN ORGANIC SYNTHESIS. A REVIEWIkuya Shibata; Akio Baba
101-109AN IMPROVED METHOD FOR THE PREPARATION OF 4-ARYL-2,6-DIPHENYLPYRYLIUM PERCHLORATES AND THEIR REACTION WITH AMMONIA AND METHYLAMINETomasz Bak; Danuta Rasala; Ryszard Gawinecki
111-113PREPARATION OF O-[2-(2-PYRIDYL)ETHYL]- AND O-[2-(TRIMETHYLSILYL)ETHYL]HYDROXYLAMINESToshiyuki Henmi; Takeshi Sakamoto; Yasuo Kikugawa
114-118A cis-1,2-DIAMINE FROM THE STEREOSELECTIVE REDUCTION OF AN α-AMINO ENAMINEStan V. D'andrea; Shikai Zhao; Stephen A. Mizsak; Jeremiah P. Freeman; Jacob Szmuszkovicz
118-120AROMATIC NITRATION OF 2-PHENYLHYDRAZONES OF 1,2-DICARBONYL COMPOUNDS USING CERIUM(IV) AMMONIUM NITRATEHimatkumar V. Patel; Kavita A. Vyas; Sudhanshu P. Pandey; Peter S. Fernandes
121-123A STRAIGHTFORWARD SYNTHESIS OF O-PROTECTED 3-HYDROXYPROPANAL DERIVATIVESDenis Barbier; Jean-Paul Salvi; Nadia Walchshofer; Joëlle Paris
123-125SIMPLE AND FACILE OXIDATION OF ALDEHYDES TO CARBOXYLIC ACIDSB. Ramesh Babu; K. K. Balasubramaniam
125-127OXIDATION OF FLAVANONES WITH LEAD TETRAACETATE, TRIMETHYL ORTHOFORMATE AND PERCHLORIC ACIDMahavir S. Khanna

Volume 25, Issue 6 (1993)

CEditorial Board Page
607-632PROGRESS IN THE FISCHER INDOLE REACTION. A REVIEWDavid L. Hughes
633-637SYNTHESIS OF DIMETHYL 1,4-DIHYDROXY-5,6,8-TRIMETHOXYNAPHTHALENE-2,3-DICARBOXYLATE, A KEY INTERMEDIATE FOR FREDERICAMYCIN ARaghao S. Mali; Prakash G. Jagtap
639-647SYNTHESIS OF 2-0-PROTECTED GLYCEROL DERIVATIVESJ. Michael Chong; Kenneth K. Sokoll
649-657SYNTHESIS OF FUNCTIONALIZED ACRYLATESMichele Curci; Jean-Luc Mieloszynski; Daniel Paquer
659-663ONE-POT SYNTHESIS PF NOVEL 10-ARYL[1,2,4]TRIAZOLO[3′,4′:2,3][1,3,4]-THIADIAZEPINO[6,7-c]QUINOLIN-6(5H)-ONESA. Jayashree; Malleshwar Darbarwar
665-671PREPARATIVE SYNTHESIS OF RL-252 VANADYL COMPLEXMichael W. Wilson; John C. Hodges
673-679PREPARATION OF OPTICALLY ACTIVE NEW MERCAPTO CHIRAL AUXILIARIES DERIVED FROM CAMPHORDong-Sheng Lee; Shung-Ming Hung; Ming-Chun Lai; Han-Yang Chu; Teng-Kuei Yang
681-683A NEW METHOD FOR THE SYNTHESIS OF DIACYL SELENIDESYongmin Zhang; Xueshun Jia; Xunjun Zhou
683-686SYNTHESIS OF N-METHYLATED QUINOLONESJ. N. Domínguez; J. Charris
687-689A FACILE SYNTHESIS OF β-DAMASCONEP. A. Unnikrishnan
690-693A SIMPLE PROCEDURE FOR THE PREPARATION OF (METHYL- AND PHENYLTHIO)ARYLOXYACETONITRILESAndrzej Jończyk; Essa-Hassan Muttar
693-695A CONVENIENT METHOD FOR THE SYNTHESIS OF FLAVANONES BY THE SELECTIVE OXIDATION OF FLAVAN-4-OLS WITH HYPERVALENT IODINEOm V. Singh
696-698CHLOROFORM-MEDIATED DDQ OXIDATION OF N-METHOXYSEPTORINOL, A SUBSTANCE ISOLATED FROM THE FUNGUS SEPTORIA NODORUM BERKM. Devys; M. Barbier; J. F. Bousquet; A. Kollmann
698-703SYNTHESIS OF CARBENOXOLONE ANALOGS FROM ARGENTATIN BRoberto Martínez; Ma. del Rosario Arellano-García; Mariano Martínez-Vazquéz; A. Gallegos Julian
703-704SIMPLE AND CONVENIENT PROCEDURE FOR THE PREPARATION OF 1-METHYL-4-NITROBENZIMIDAZOLEViktor Milata; Dusan Ilavský
705-706PREPARATION OF SOME 2,3-DIHYDROBENZOTHIAZOLE-2-CARBOXAMIDESH. P. Penner; Racine Gamer; Edgar L. Scott III
707-708AN IMPROVEMENT IN THE SYNTHESIS OF 1,2,4,9-TETRAHYDROCARBAZOL-3-ONEWilliam A. Boulanger; Victoria Dolsen
708-710A SIMPLE PREPARATION OF 4-AMINO-5-ARYL-2H-IMIDAZOL-2-ONESMadhu Srivastava; Ram Lakhan
711CORRIGENDUM
713-727INDEXES

Volume 25, Issue 5 (1993)

CEditorial Board Page
481-513PREPARATION AND REACTIONS OF INDOLIN-2(3H)-ONES. A REVIEWGary M. Karp
515-556THE LATERAL METALATION OF ISOXAZOLES. A REVIEWNicholas R. Natale; Yousef R. Mirzaei
557-562PREPARATION OF PHENYLGLYCOLIC ACIDS AND SODIUM p-(N,N-DIALKYLAMINO)PHENYLGLYCOLATESAlan R. Katritzky; Barbara Galuszka; Stanislaw Rachwal; Doreen Lynch
563-568FACILE LARGE SCALE SYNTHESIS OF 5-ALKYLURACILSHenryk Koroniak; Aleksander Jankowski; Miroslaw Krasnowski
569-575SYNTHESIS OF 2-ARYL-4,5,6,7-TETRAHYDRO-6,6-DIMETHYL-2 H-BENZO[D][1,2,3]TRIAZOL-4-ONESH. Abdel Hamid; A. Mousaad; M. Sayed; E. S. H. El Ashry
577-579AN IMPROVED SYNTHESIS OF 5-(3,4-DIMETHOXYPHENYL)-3-HYDROXY-4-NITROCYCLOHEXENEA. F. Ibañez; A. R. Martinez; G. Y. Moltrasio Iglesias
579-581AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1,6-DICARBOXYHEX-3-ENEPradeep T. Deota; Sugra Abid
581-583A FACILE SYNTHESIS OF bis(3-ARYL-3-OXO-1-PROPENYL)BENZENESJian-Guo Shao; Jing-Feng Zhou; Chang-Qing Liu; Qi Zhong
583-585AN IMPROVED SYNTHESIS OF 2-METHALLYLOXYPHENOLV. B. Deodhar; V. S. Dalavoy; U. R. Nayak
585-587SYNTHESIS OF 1-HYDROXY-7-PHENOXYNAPHTHALENEAlan R. Katritzky; Marudai Balasubramanian; Michael Siskin
588-590FACILE SYNTHESIS OF 2-ARYL-4H-3,1-BENZOXAZIN-4-ONESD. V. Ramana; E. Kantharaj
590-592PREPARATION OF bis(2,2,2-TRIFLUOROETHYL)SELENIDE AND TELLURIDE AND OF BIS(2,2,2-TRIFLUOROETHYL)DISELENIDE AND DITELLURIDEK. K. Bhasin; Vijay Gupta; R. Khajuria; R. P. Sharma
592-594SYNTHESIS OF PENTAFLUOROPHENYL-4-(N-MALEIMIDOMETHYL) CYCLOHEXANE-1-CARBOXYLATE (FMCC)Maciej Adamczyk; Donald Johnson
595-597A SIMPLE, EFFICIENT PREPARATION OF 1,1-BIS(TRIMETHYLSILOXY)-1,3-BUTADIENEGregory S. Welmaker
597-599A ONE-STEP PREPARATION AND HETERO-DIELS-ALDER DIMERIZATION OF 2-PHENYLPROPENALTarja Laitalainen; Pirjo Kuronen; Antti Hesso
600-601A SIMPLE AND PRACTICAL APPROACH TO UNSYMMETRICAL PHENYLUREASKrishnamurthy Ramadas; Natarajan Srinivasan
602-606THIOPHENO[3,2][1]BENZAZEPINE, BENZO[3,4]CYCLOHEPTA[2,1-b]THIOPHENES, THIAZOLO[5,4-d][1]BENZAZEPINE AND BENZO[3,4]CYCLOHEPTA[2,1-d]THIAZOLESV. Peesapati; N. Lingaiah

Volume 25, Issue 4 (1993)

CEditorial Board Page
373-401SYNTHESIS OF 9-SUBSTITUTED GUANINES. A REVIEWFinn Priess Clausen; Jørgen Juhl-Christensen
403-435RECENT PROGRESS IN THE PREPARATION AND SYNTHETIC USES OF THE REACTIONS OF 3H-PYRAZOLES. A REVIEWToshikazu Nagai; Masashi Hamaguchi
437-443AN IMPROVED PREPARATION OF (S)-N-(BOC)-CYCLOHEXYLALANINAL. THE MOFFAT-SWERN OXIDATION OF α-AMINOALCOHOLSD. J. Krysan; A. R. Haight; J. E. Lallaman; D. C. Langridge; J. A. Menzia; B. A. Narayanan; R. J. Pariza; D. S. Reno; T. W. Rockway; T. L. Stuk; J. H. Tien
445-448SYNTHESIS OF 5,5′DIFLUORO-BAPTA-AM, A USEFUL IN VIVO PROBE FOR CALCIUM DETERMINATIONPhilip E. Morris Jr.
449-456SYNTHESES OF TETRASUBSTITUTED CYCLOPENTANESKenichi Somekawa; Masafumi Nomura; Shoichi Aoki; Shinji Noma; Tetsuro Shimo
457-461AN EFFICIENT SYNTHESIS OF BOC-AMINOACETALDEHYDE AND ITS APPLICATION TO THE SYNTHESIS OF N-(2-BOC-AMINOETHYL)GLYCINE ESTERSKim L. Dueholm; Michael Egholm; Ole Buchardt
463-466LIPASE-CATALYZED TRANSACYLATION REACTIONS IN AZEOTROPIC DISTILLATIONGialih Lin; Shih-Huang Liu
466-469THEXYL- AND ISOPINOCAMPHEYLHALOBORANES AS STEREOSELECTIVE REDUCING AGENTSJin Soon Cha; Soo Jin Min; Jong Mi Kim; Oh Oun Kwon; Min Kyoo Jeoung
469-473BROMOACETALDEHYDE AND IODOACETALDEHYDE BY OZONOLYSIS OF ALLYL BROMIDE AND ALLYL IODIDEMadhukar Jachak; Martin Mittelbach; Hans Junek
473-477SYNTHESIS OF SPIN-LABELED TRIAZENESZahary Raikov; Vesselina Gadzheva; Mario Koch; George Kolar
478-480AN IMPROVED LARGE-SCALE PREPARATION OF 3,3′,4,4′-TETRAAMINODIPHENYL ETHERAlan R. Katritzky; Zhijun Yang; Darren J. Cundy

Volume 25, Issue 3 (1993)

CEditorial Board Page
259-292SYNTHESIS OF CARCINOGENIC BENZ[c]ACRIDINES. A REVIEWNoboru Motohashi; Jahangir Emrani; Roger Meyer; Masami Kawase
293-299SYNTHESIS OF NEW SUBSTITUTED PYRIDAZINESA. H. H. Elghandour; M. K. A. Ibrahim; I. S. A. Hafiz; M. H. Elnagdi
301-307SYNTHESIS OF POTENTIALLY BIOLOGICALLY ACTIVE COMPOUNDS via THE STOBBE CONDENSATIONVictorine B. Baghos; S. H. Doss; E. F. Eskander
309-314MACROCYCLE SYNTHESES: CYCLIC KETONES, KETOALKENES, DIKETONES AND DIENES OF RING SIZE C21 TO C26Malcolm D. E. Forbes; Yi Dang
315-3191,1′-CARBONYLDIBENZOTRIAZOLE AND 1,1′-SULFONYLDIBENZOTRIAZOLE. VERSATILE REAGENTS FOR THE DEHYDRATION OF ALDOXIMES AND AMIDES TO NITRILESAlan R. Katritzky; Gui-Fen Zhang; Wei-Qiang Fan
321-325ENANTIOSELECTIVE SYNTHESIS OF (4R)-4-NONANOLIDE AND (5R)-5-DECANOLIDE FROM A COMMON INTERMEDIATEH. Rama Mohan; A. S. Rao
327-330REACTION OF PIVALOYLACETONITRILE WITH AROMATIC ALDEHYDESK. Popandova-Yambolieva; T. Iossifova
330-333A CONVENIENT SYNTHESIS OF (±)-10-METHYL-2-TRIDECANONE, THE PHEROMONE OF SOUTHERN CORN ROOTWORMA. Sharma; A. Pawar; S. Chattopadhyay; V. R. Mamdapur
333-336A SHORT SYNTHESIS OF (11Z, 15Z)-EICOSADIENOIC ACID, A COMPOUND OF MARINE SPONGE ORIGINB. A. Kulkarni; A. Chattopadhyay; V. R. Mamdapur
336-338CONVENIENT SYNTHESIS OF 2-PHENETHYL ALCOHOL BY HYDROLYSIS OF 2-BROMOETHYLBENZENE UNDER PHASE TRANSFER CONDITIONSHayder A. Zahalka; Yoel Sasson
338-341IMPROVEMENT OF THE VILSMEIER-HAACK REACTIONDenis Blaser; Monique Calmes; Jacques Daunis; François Natt; Anne Tardy-Delassus; Robert Jacquier
341-344SYNTHESIS OF 2-HYDROXY-3-METHYLCYCLOPENT-2-EN-1-ONE FROM LINALYL ACETATEMaria Lucilia dos Santos; Gouvan C. de Magalhães
344-346A SIMPLE SYNTHESIS OF BRASSILEXIN, A CRUCIFERAE PHYTOALEXINMichel Devys; Michel Barbier
347-352VILSMEIER REACTION OF 3-METHYL-N-(4′-SUBSTITUTED)-AZOBENZENESULFONAMIDO)-2-QUINOXALINONE DYESI. M. A. Awad
353-355NEW CHEMICAL CONVERSIONS OF 5-HYDROXYMETHYLFURFURAL AND THE ELECTROCHEMICAL OXIDATION OF ITS DERIVATIVESRomuald Skowronski; Grzegorz Grabowski; Jaroslaw Lewkowski; Géard Descotes; Louis Cottier; Claire Neyret
356-360SYNTHESIS OF PYRAZOLINE AND ISOXAZOLINE DERIVATIVES OF ANDROSTANE SERIESA. U. Siddiqui; D. Ramesh; Y. Satyanarayana; M. Srinivas; A. H. Siddiqui
360-362ASYMMETRIC INDUCTIVE SYNTHESIS OF α-AMINOARYLACETIC ACIDS IN THE PRESENCE OF β-CYCLODEXTRINWeiliang Xu; Yongmin Zhang
363-365A NEW SYNTHESIS OF SYMMETRIC PIPERAZINES DERIVATIVESJean-Charles Lancelot; Bertrand Letois; Max Robba
365-368SAMARIUM TRIIODIDE CATALYZED DITHIOACETAL AND DITHIOKETAL FORMATIONYongmin Zhang; Yongping Yu; Ronghui Lin
368-371A CONVENIENT SYNTHESIS OF 7-HYDROXY-3-HYDROXYMETHYL-4-PHENYL-2-NAPHTHOIC ACID, LACTONE FORMJoseph F. Payack; Dean R. Bender
373CORRIGENDUM

Volume 25, Issue 2 (1993)

CEditorial Board Page
141-208THE USE OF ISOCYANIDES IN HETEROCYCLIC SYNTHESIS. A REVIEWStefano Marcaccini; Tomás Torroba
209-213AN EFFICIENT, LARGE-SCALE SYNTHESIS OF TRIISOPENTADECANOINThomas A. Foglia; Peter D. Vail
215-222SELENIUM OXIDE OXIDATION OF ABIETA-7,13-DIENES IN METHANOLA. San Feliciano; J. M. Miguel del Corral; M. Gordaliza; M. A. Salinero
223-228CONVENIENT SYNTHESIS OF 6-METHYL, 8-METHYL AND 6,8-DIMETHYL DERIVATIVES OF 5-HYDROXY-1,2,3,4-TETRAHYDRO-2-QUINOLINONEDominique Blondet; Francette Laure; Jean-Claude Pascal
229-231IMPROVED PREPARATION OF AMINOMETHYLENEMALONIC ACID DERIVATIVES BY TIN-PROMOTED ADDITION OF DIETHYL MALONATES TO NITRILESMarco Nicolini; Attilio Citterio
232-233IMPROVED AND CONVENIENT SYNTHESIS OF DISULFIDES IN THE ABSENCE OF SOLVENT CATALYZED BY CLAYFENHarshadas M. Meshram
234-237SYNTHESIS OF 2-DIMETHYLAMINO-5-(α-CHLOROALKENYL)-13-OXAZIN-6-ONESEgle M. Beccalli; Alessandro Marchesini
237-240THE SYNTHESIS OF TWO BICYCLO[4.3.0]NONANE DERIVATIVESC. W. Bird; R. Cooper
241-243MICHAEL REACTION OF FLUORENE AND INDENE BY PHASE-TRANSFER CATALYSISYan Chaoguo; Lu Wenxing; Wu Jitao
243-246PREPARATION OF THE RACEMATE AND ENANTIOMERS OF 3-HYDROXY-5,5-DIMETHYLHEXANOIC ACIDWayne J. Brouillette; Ahmed S. Abuelyaman; Carla A. Hosmer; Robert N. Comber; Ashraf Saeed
247-249AN EFFICIENT PREPARATION OF 2H-[5,4-b]-PYRIDOISOTHIAZOLONEStephen W. Wright; Ronald L. Corbett
249-251AN IMPROVED SYNTHESIS OF 1-(t-BUTYLOXYCARBONYL)-3-(BROMOMETHYL)INDOLET. K. Venkatachalam; S. Mzengeza; M. Diksic
252-255SYNTHESIS OF 3,6-DIMETHOXY-2-NAPHTHALDEHYDEAdel M. Moussa; Jun-Rui Yang; Margaret E. Langmuir
255-258A PRACTICAL PROCEDURE FOR THE SYNTHESIS OF 5-SUBSTITUTED γ-LACTAMSZ. Y. Wei; E. E. Knaus

Volume 25, Issue 1 (1993)

CEditorial Board Page
1-14SYNTHETIC APPLICATIONS OF DIARYL ETHER PHOTOCHEMISTRY. A REVIEWRenée Pollard; Peter Wan
15-40CHEMISTRY OF N-METHOXY-N-METHYLAMIDES. APPLICATIONS IN SYNTHESIS. A REVIEWMukund P. Sibi
41-81HOMOENOLATES AND OTHER FUNCTIONALIZED ORGANOMETALLICS. A REVIEWMichael T. Crimmins; Philippe G. Nantermet
83-90THE REACTIONS OF SOME ALKOXYCARBONYL ISOTHIOCYANATES WITH ALCOHOLS, PHENOLS AND AMINESAlan R. Katritzky; Marek K. Bernard; Qiu-He Long; Linghong Xie; Nageshwar Malhotra; Morton Beltzer
91-97A SIMPLE SYNTHESIS OF 1-HYDROXYALKYL-1,2,3,4-TETRAHYDROISOQUINOLINESLászló Lázár; Ferenc Fülöp; Gábor Bernáth; Jorma Mattinen
99-105ACETYLATION OF 4-AMINO-44-DIHYDRO-1H-1,2,4-TRIAZOL-5-ONESAykut A. Ikizler; Haydar Yüksek
105-108SYNTHESIS OF SOME BENZOTHIAZOLOBENZOTRIAZEPINESM. V. Deshmukh; D. S. Deshpande
108-110A NEW ROUTE FOR THE SYNTHESIS OF Z-11-HEXADECEN-1-OL, A SEX PHEROMONE OF CHILO INFUSCATELLUS (SNELL)S. Narasimhan; K. Ganeshwarprasad
110-115SYNTHESIS OF C-24 THIAZOLIDINONE AND OXAZOLIDINONE DERIVATIVES OF BILE ACIDSA. U. Siddiqui; A. H. Siddiqui; T. Sundara Ramaiah
116-117AN IMPROVED SYNTHETIC ROUTE TO TRIFLUOROMETHYL-6-SUBSTITUTED-2(1H)-PYRIDONESB. Narsaiah; A. Sivaprasad; R. V. Venkataratnam
118-121A CONVENIENT ONE-POT SYNTHESIS OF NOVEL FUNCTIONALIZED TERPHENYLSV. V. Suresh; H. M. Chawla
122-125A CONVENIENT SYNTHESIS OF 2-AMINOALKYL ALLYL ETHERSAlexander Dobrev
125-130PREPARATION OF LOW MOLECULAR WEIGHT, OPTICALLY ACTIVE ALLYLIC ALCOHOLS FROM (S)-(-)-ETHYL LACTATEJohn C. McKew; Mark J. Kurth
130-133AN IMPROVED PREPARATION OF 2,4-DINITROPHENYL THIOETHERS FROM THIOLCARBONIC ESTERSKazunobu Harano; Masashi Eto; Shoji Kubota; Takuzo Hisano
133-137A CONVENIENT PREPARATION OF N-DEMETHYLDILTIAZEM AND ITS CONVERSION TO A DILTIAZEM HOMOLOGJose Alexander
137-139THE ONE-STEP SYNTHESIS OF p-tert-BUTYLCALIX[5]ARENEDonald R. Stewart; C. David Gutsche

Volume 24, Issue 6 (1992)

CEditorial Board Page
623-647SYNTHETIC OXIDATIONS WITH HYPOCHLORITES. A REVIEWJacek Skarzewski; Renata Siedlecka
649-654SYNTHESES OF 2,3-DIHALO-1-(PHENYLSULFONYL)INDOLESGordon W. Gribble; Brett D. Allison; Samuel C. Conway; Mark G. Saulnier
655-659SELECTIVE NITROSATION OF DIALKYLUREAS CONTAINING A BASIC β-NITROGENJoseph E. Saavedra; David W. Farnsworth
661-665CONVENIENT PREPARATION OF 1-ADAMANTANOL FROM ADAMANTANE INDUCED BY A HYDRIDE TRANSFERM. Gami; R. Jalal; R. Gallo
665-669FORMATION OF A 1,2-DIHYDROPYRAZINE USING AN AMINO ACID AND D-GLUCOSEC. W. Yuan; J. Beauhaire; C. Marty; J. L. Fourrey; H. Richard
670-672AN IMPROVED SYNTHESIS OF 2,3,4,6,7,8-HEXAHYDROQUINOLINESElmar Schuster; Gerhard Jas; Dieter Schumann
673-675A FACILE PREPARATION OF 2,3,4,4a,5-6-HEXAHYDROQUINOLINEBodo Juhnke; Gerhard Jas; Dieter Schumann
675-678A CONVENIENT SYNTHESIS OF SOME NEW PYRANO[2,3-d]PYRIMIDINESV. K. Ahluwalia; Rakesh Kumar; Renu Aggarwal
679-681SYNTHESIS OF 2(N-ALKYLAMINO)ISOBUTYRALDEHYDESNorbert De Kimpe; Marc Boeykens; Mark Boelens; Kurt De Buck; Johan Cornelis
682-684SIMPLE SYNTHESIS OF ARYLALIPHATIC DIKETONESAdama Saba; Faustin Sié Sib; Jean-Pierre Aycard
685-687A CONVENIENT SYNTHESIS OF cis-(1R)-N-BENZYL-(2S)-(HYDROXYMETHYL)CYCLOHEXYLAMINEB. Vanderplas; C. W. Murtiashaw; T. Sinay; F. J. Urban
687-690STUDY IN CROSSOVER FRIES MIGRATIONR. N. Khanna; K. P. Singh; Jyotsana Sharma
690-692AN IMPROVED SYNTHESIS OF 2,4-DIMETHOXYPHENYLACETIC ACIDE. N. Alesso; J. M. Aguirre; G. Y. Moltrasio Lglesias
692-694A CONVENIENT SYNTHESIS OF (4-NITROPHENYL) (4-PIPERIDINYL) KETONEMichel Monclus; André Luxen
695-696A CONVENIENT PROCEDURE FOR THE PREPARATION OF 2-BROMO-1-PHENYLETHANOLS. S. Bhosale; P. L. Joshi; A. S. Rae
696-698A CONVENIENT PREPARATION OF 4-CYCLOPROPYLPHENOLBruce W. Horrom; H. Mazdiyasni
698-701A NEW SYNTHESIS OF 3-AMINO-1-IMIDAZOLIN-4-ONES BY THE HYDRAZINOLYSIS OF 5-OXAZOLONESVinod K. Ahluwalia; Mukesh K. Sharma; Rashmi Sharma
701-704IMPROVED PREPARATION OF WHYDROXYPROGESTERONEM. O. Violeta Benedetti; Gerardo Burton
705-717INDEXES

Volume 24, Issue 5 (1992)

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501-507PREPARATION OF NOVEL 2-AMINOADAMANTYL- AND 4-AMINOPROTOADAMANTYLCARBONITRILESKata Mlinaríc-Majerski; Mira Kaselj; Danko Škare
509-516IMPROVED SYNTHESIS OF 3-HALO- AND 3-METHOXYPHENANTHRENESAna Eirín; Franco Fernández; Carmen González; Carmen López
517-520METHYL CYCLOPROPENE-3-CARBOXYLATES BY DIRECT CATALYTIC CYCLOPROPENATION OF ACETYLENES WITH METHYL DIAZOACETATEE. A. Shapiro; A. V. Kalinin; O. M. Nefedov
520-522A FACILE SYNTHESIS OF 2-(2′-SUBSTITUTED VINYL)BENZOXAZOLESJian-Guo Shao; Qi Zhong; Hai-Ping Liao; Chang-Qing Liu; Jing-Feng Zhou
523-525FACILE SYNTHESIS AND AANTIMICROBIAL ACTIVITY OF SPIROBICYCLO[3.2.1]OCTANE-2′,3-(4H)-[2H]-THIAZOLO[3,2-B]-s-TETRAZINESJag Mohan
525-527SYNTHESIS OF EVERNIPENTANONE BY ADDITION OF n-BUTYLLITHIUM ON ETHYL EVERNINATEM. Devys; E. Desnoës; M. Barbier
527-532SYNTHESIS OF β- AND γ-ALKOXY AND β-DIMETHYLAMINO 1- AND 2-SUBSTITUTED-1,3-CYCLOPENTADIENESWilliam S. Rees Jr.; Kerstin A. Dippel
532-536SYNTHESIS OF MODELS RELATED TO TASPINEM. L. Scarpati; A. Bianco; R. Lo Scalzo
536-539A CONVENIENT METHOD FOR THE PREPARATION OF cis-3,4,8,8a-TETRAHYDRO-6H-[1,3]-DIOXEPINO[5,6-d]OXAZOLESMiljenko Dumć; Ivan Butula; Mladen Vinković; Boris Kamenar
540-543FORMATION OF 1-CHLORO-1-ALKYNES FROM 1,1-DICHLORO-1-ALKENES UNDER PHASE-TRANSFER CONDITIONS WITHOUT SOLVENTPeter Vinczer; Szilvia Sztruhar; Lajos Novak; Csaba Szantay
543-546SYNTHESIS OF TWO METHYLBENZOSUBERONES AND A DIMETHYLBENZOCYCLOHEPTENEArthur G. Anderson Jr; Harry F. Richards
546-548SYNTHESIS OF ESTRIOL 16α-4′,5′-DEHYDROGLUCURONIDEMaciek Adamczyk; Yon-Yih Chen; Jeffrey R. Fishpaugh
548-551SYNTHESIS OF CYCLOPROPANES USING S-ETHENYLSULFILIMINESKatsuya Ikeda; Hiroshi Satoh; Tamotsu Yamamoto
553-582RECENT PROGRESS IN THE CHEMISTRY OF ACYLSILANES. A REVIEWPier F. Cirillo; James S. Panek
583-621RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF SUBSTITUTED PIPERIDINES. A REVIEWChia-Lin J. Wang; Mark A. Wuonola

Volume 24, Issue 4 (1992)

CEditorial Board Page
369-435USES OF THE FRIES REARRANGEMENT FOR THE PREPARATION OF HYDROXYARYLKETONES. A REVIEWRobert Martin
437-462SELECTIVE FUNCTIONALIZATION AND CONFORMATIONAL PROPERTIES OF CALIX[4]ARENES, A REVIEWJ. -D. van Loon; W. Verboom; D. N. Reinhoudt
463-467PREPARATION OF 6-, 7- AND 8-MEMBERED SULTAMS BY FRIEDEL-CRAFTS CYCLIZATION OF ω-PHENYLALKANESULFAMOYL CHLORIDESAlan R. Katritzky; Jing Wu; Stanislaw Rachwal; Bogumila Rachwal; David W. Macomber; Terrance P. Smith
469-473A CONVENIENT ONE-POT SYNTHESIS OF 2-CINNAMOYLCOUMARAN-3-ONES FROM 2-CINNAMOYLOXYACETOPHENONES USING THALLIUM(III) p-TOLUENESULFONATEMahavir S. Khanna; Chandra P. Garg; Ram P. Kapoor
475-478A NOVEL ROUTE TO N-(BENZOTRIAZOL-1-YLMETHYL)AMIDESAlan R. Katritzky; Barbara Galuszka; Yongmin Zhang; Stanislaw Rachwal
478-484SYNTHESIS OF POTENTIAL PRECURSORS OF HEPTABOWTIENE, A NOVEL NON-BENZENOID HYDROCARBONArthur G. Anderson Jr.; Barry T. Murphy
484-488AN IMPROVED SYNTHESIS OF 4,7-DIMETHOXY-1H-INDOLEH. D. Hollis Showalter; Gerd Pohlmann
488-492LARGE-SCALE PREPARATION OF THE SULFUR-TRANSFER REAGENT 3H-1,2-BENZODITHIOL-3-ONE 1,1-DIOXIDEJ. B. Regan; L. R. Phillips; S. L. Beaucage
492-496SYNTHESIS OF 4-AROYL-[(5-PHENYL-2(2H)-TETRAZOLYL)-1-OXOETHYL]- THIOSEMICARBAZIDES AND 4-AROYL-5-[(5-PHENYL-2(2H)-TETRAZOLYL)METHYL)-1,2,4-(4H)-TRIAZOLE-3-THIONEFeng Xiaorning; Chen Rong; Cai Shaoyin
497-499A NEW SYNTHETIC ROUTE TO 2-CARBOMETHOXYCYCLOPENT-2-ENONE via RHODIUM(II)-MEDIATED DECOMPOSITION OF DIAZOESTERSPaolo Ceccherelli; Massimo Curini; Maria Carla Marcotullio; Ornelio Rosati

Volume 24, Issue 3 (1992)

CEditorial Board Page
245-284BIOSYNTHETIC, BIOMIMETIC AND RELATED EPOXIDE CYCLIZATIONS. A REVIEWStephen K. Taylor
285-307“CESIUM ION EFFECT” AND MACROCYCLIZATION. A CRITICAL REVIEWCarlo Galli
309-325ELECTROCATALYTIC HYDROGENATION ON HYDROGEN-ACTIVE ELECTRODES. A REVIEWJean-Claude Moutet
327-330ONE-POT CONVERSION OF CARBOXYLIC ACIDS TO ALDEHYDES BY TREATMENT OF ACYLOXY-9-BORABICYCLO[3,3,1]NONANES WITH LITHIUM tris(DIETHYLAMINO)ALUMINUM HYDRIDEJin Soon Cha; Jae Cheol Lee; Heung Soo Lee; Sung Eun Lee
331-334SELECTIVE CONVERSION OF AROMATIC NITRILES TO ALDEHYDES BY LITHIUM tris(DIHEXYLAMINO)ALUMINUM HYDRIDEJin Soon Cha; Sung Eun Lse; Heung Soo Lee
335-337TRANSFORMATION OF CARBOXYLIC ESTERS TO ALDEHYDES WITH LITHIUM tris(DIETHYLAMINO)ALUMINUM HYDRIDEJin Soon Cha; Soo Jin Min; Jae Cheol Lee; Heung Soo Lee; Sung Eun Lee
338-339AN IMPROVED PROCEDURE FOR THE ISOLATION OF 2-(N,N-DIETHYJAMINOMETHYL)-4-NITROPHENOLM. C. B. V. de Souza; A. M. R. Bernardino; M. C. Soares; M. G. Retzlaff
339-342SYNTHESIS OF 4-trans-[1-[4-[2-(5-CHLORO-2-METHOXYBENZAMIDO)ETHYL] BENZENESULFONYL]UREIDO]CYCLOHEXANOL HEMISUCCINATE ESTERRobert L. Stephont; R. Sam Niedbala; Keith J. Schrayt; Ned D. Heindel
342-345SYNTHESIS OF 1-(2-(2,4-DICHLOROPHENYL)-2-[(2-THIENYL)METHOXY]ETHYL]-lH-IMIDAZOLE AND 1-[2-(2,4-DICHLOROPHEL)-2-[(2-FURYL)METHOXY]ETHYL]-1H-IMIDAZOLE, TWO NEW MICONAZOLE ANALOGUESRaymundo Cruz-Almanza; Teresa Hemández; Francisco Pérez; Cristina Lemini
346-349ONE-POT SYNTHESIS OF ISOTHIOCYANATES FROM PRIMARY AMINES SYNTHESIS USING CYANAMIDE?Tamotsu Yamamoto; Susumu Sugiyama; Kenji Akimoto; Kiyoshi Hayashi
349-351AN IMPROVED SYNTHESIS OF 2,4-HEXADIEN-l-OLPeter Vinczer; Lajos Novak; Csaba Szantay
352-354CONSTRUCTION OF THE PYRAZOLO[1,5-a] [4,1]BENZOTHIAZEPINE SYSTEM BY INTRAMOLECULAR NITRILIMINE CYCLOADDITIONGianluigi Broggini; Luca Bruché; Gaetano Zecchi
355-358SYNTHESIS OF STEROIDAL HETEROCYCLIC COMPOUNDS FROM A CLAISEN CONDENSATION PRODUCT OF A 6-KETO STEROLA. U. Siddiqui; U. M. Rao; M. Srinivas; A. H. Siddiqui
358-362NEW HETEROCYCLES FORMING REACTIONS OF ACYL THIOFORMANILIDESZhong E. Lu; Da Qing Sun; Tian Lin Xu; Jun Wan; Le Cun Xu; Ke Qian Chen
363-365OXIDATION OF ALCOHOLS USING TRIPHOSGENEI. A. Rivero; R. Somanathan; L. H. Hellberg
365-368A STUDY ON CYANOACETIC ACID HYDRAZIDEA. Aykut Ikizler; Aysun Lkizler; Neslihan Uzunismail

Volume 24, Issue 2 (1992)

CEditorial Board Page
121-126A NEW SYNTHESIS OF AN AMINO ACID BASED SWEETENERAlan R. Katritzky; N. Shobana; Philip A. Harris; John B. Hill; David J. Ager
127-133NEW AND RENEWED SYNTHESES OF 10-PHENYLANTHRONE AND 10-HYDROXY-10-PHENYLANTHRONEStephen E. Branz; Kate Jin; Yanzhou Liu; Tram N. Dao
135-141A CONVENIENT SYNTHESIS OF ISOPHYTOL BY CROSS-COUPLING REACTION OF A GRIGNARD REAGENT AND A PROTECTED ALLYLIC CHLORIDETetsuo Miyakoshi; Mitsuhiro Hagimoto
143-146PREPARATION OF BENZO[c-2,7]NAPHTHYRIDINECharles F. Nutaitis; Mark W. Ledeboer
147-157N-SULFONYL LACTAMS via SULFONATION OF LACTIM ETHERSJennline Sheu; Michael B. Smith; Thomas R. Oeschger; Jacqueline Satchell
159-163IMPROVED PREPARATION OF 14β-HYDROXYPROGESTERONEJohn F. Templeton; Yulin Yan
165-167ONE-POT REDUCTIVE DICHLOROCARBENE ADDITION TO ARYL KETONES. A NEW GENERAL METHOD FOR THE SYNTHESIS OF 2-ARYLPROPIONIC ACIDSE. F. Llama; C. del Campo; J. V. Sinisterra
168-171EFFICIENT SYNTHESIS OF TRICYCLIC ANTIDEPRESSANT NORMETABOLITESMaciek Adamczyk; Jeffrey R. Fishpaugh; Donald Johnson
171-175SYNTHESIS OF PYRAZOLO[3,4-d]PYRIDAZINE, PYRAZOLO[3,4-d]PYRIMIDINE AND IMIDAZO[1,2-a]PYRIDINE DERIVATIVES USING HYDRAZONYL BROMIDESHamdi M. Hassaneen; Ahmad S. Shawali; Nehal M. Elwan; Nada M. Abounada
176-181SYNTHESIS OF NOVEL meta-BROMOPHENOLIC COMPOUNDSChun-Shan Wang; Yih-Min Sun; A. Mendoza
181-185REDUCTION OF 3- AND/OR 5-UNSUBSTITUTED 2-ETHYLPYRAZOLIUM SALTS WITH COMPLEX METAL HYDRIDES. SYNTHESIS OF PYRAZOLIDINESLuis A. Bañuelos; Purificaciön Cuadrado; Ana M. González; Francisco J. Pulido
185-188A CONVENIENT PREPARATION OF 5,5-DIALKYL MELDRUM'S ACIDSBang-Chi Chen; Ping Lue
188-191SYNTHESIS OF N-SUBSTITUTED 2-ALKYL-4-ARYLOXAZOLE-5-CARBOXAMIDESRicardo Bossiot; Stefano Marcaccini; Roberto Pepho; Cecilia Polo; Tomas Torroba
191-194A ONE-POT SYNTHESIS OF NαBENZYLOXYCARBONYL Nω-t-BUTOXYCARBONYL-L-ORNITHINE AND L-LYSINEElzbieta Masiukiewicz; Barbara Rzeszotarska; Jaroslaw Szczerbaniewicz
194-197SYNTHESIS OF DIFLUORODURENE AND DIFLUOROPYROMELLITIC ACIDWojciech Dmowski; Krystyna Piasecka-Maciejewska
197-200PREPARATION OF SOME PHOSPHOLIPID-TARGETED METRONIDAZOLE DERIVATIVESR. A. McClelland; T. A. Modro
200-2044-PIPERIDINOPYRIDINE AS AN EFFECTIVE CATALYST FOR THIONE-THIOL REARRANGEMENT OF XANTHATESKazunobu Harano; Hidetoshi Nakagawa; Hideo Kiyonaga; Takuzo Hisano
204-208A NOVEL SYNTHESIS OF 2,3-DIHYDRO[1,5]BENZOTHIAZEPIN-4(5H)-ONESJean-Charles Lancelot; Bertrand Letois; Carmela Saturnono; Paolo De Caprariis; Max Robba
209-243THE AZA-WITTIC REACTION IN HETEROCYCLIC SYNTHESIS. A REVIEWShoji Eguchi; Yuji Matsushita; Keizo Yamashita

Volume 24, Issue 1 (1992)

CEditorial Board Page
iIMPORTANT NOTICE TO AUTHORS
1-5SYNTHESIS OF SOME TETRAHYDRO-3,3′-BISQUNAZOLIN-4,4′-DIONESA. K. D. Bhavani; P. S. N. Reddy
7-12REDUCTIVE DECYANATION vs ADDITION OF GRIGNARD REAGENTS WITH HINDERED NITRILESStuart S. Kulp; Anthony Romanelli
13-20RING OPENING OF SOME SUBSTITUTED STYRENE OXIDESUlhas P. Dhokte; A. Somasekar Rao
21-26SYNTHESIS OF SOME SPIRO-ISOXAZOLIDINE-3,5-DIONESD. Bhaskar Reddy; V. Padmavathi; B. Seenaiah; M. V. Ramana Reddy
27-32SYNTHESIS OF FURANO BENZOSUBERONES AND FURANO TETRALONES via CLAISEN REARRANGEMENTV. Peesapati; N. Lingaiah
33-37SYNTHESIS OF NEW SUBSTITUTED PYRIDINES, PYRANO[2,3-d]IMIDAZOLES AND PYRROLO[2,1-b]QUINAZOLINESO. H. Hishmat; A. A. Magd El Din; N. A. Ismail
39-43AN IMPROVED PROCEDURE FOR THE PREPARATION AND RESOLUTION OF dl-2,3-DIMETHYLSUCCINIC ACIDScott C. Sutton; Michael H. Nantz; Shawn R. Hitchcock
45-48PREPARATION OF N-BENZOYL-1-(5,6-DIMETHOXYINDANYLMETHYLAMINE) FROM 5,6-DIMETHOXYINDANONED. G. Tombari; A. G. Moglioni; F. P. Dominici; G. Y. Moltrasio de Iglesias
48-51STEREOSELECTIVE REDUCTION OF PIVALOYLOXYMETHYL (2S,5R,6S)-6-ACETYL-3,3-DIMETHYL-7-OXO-4-THIA-1-AZABICYCLO[3.2.0]HEPTANE-2-CARBOXYLATE WITH SODIUM BOROHYDRIDEDaniele Donati; Carla Marchioro; Bruno Tamburini; Antonella Ursini
52-54CONVENIENT SYNTHESIS OF NIESHOUTIN (CYCLOOBLZQUETIN), A FUROCOUMARIN ISOLATED FROM THE HEARTWOOD OF Ptaeroxylon obliquumR. S. Mali; Anita R. Manekar; S. G. Tilve
55-57A NEW, MILD PREPARATION OF 2,4,6-TRINITROFLUOROBENZENEJulian M. Dust; Richard A. Mandeville
57-60AN IMPROVED SYNTHESIS OF MONOESTERS OF PHOSPHORIC ACIDAgnes M. Modro; Tomasz A. Modro
60-63REACTION OF THIONYL BROMIDE WITH KETONESS. M. Al-Mousawi; I. Bhatti; S. D. Saraf
64-66A CONVENIENT SYNTHESIS OF METHYL 4-AMINO-5-CHLORO-2-MTHOXYBENZOATERichard L. Ehrenkaufer; James G. Scripko; Patricia L. Hoffman
66-67IMPROVED SYNTHESIS OF DIMETHYLAMINOTHIOACETAMIDEKenneth P. Moder; Frank R. Busch; David C. Richter
67-70A NEW ROUTE FOR SYNTHESIS OF 1-TRIACONTANOLB. V. S. K. Rao; R. Supharao
71-73SYNTHESIS OF NOVEL 9-ARYL-2,8-DIMETHYL-9H-PURIN-6-AMINES BASED ON STERICALLY HINDERED o-BROMOANILINESS. V. Eswaran; S. K. Sajadian

Volume 24, Issue 1 (1992)

73-76SYNTHESIS OF 2,3-DIDEOXY-d-arabino-HEPTONO-1,4-LACTONE via A WITTIG REACTION ON UNPROTECTED d-ARABINOSEJohn W. Lyga
76-77AN IMPROVED SYNTHESIS OF α-CHLORODIPHENYLACETIC ACIDJ. B. Maciel; R. A. S. San Gil; A. C. Neto
78-80PREPARATION OF 1,4-BIS(2,4,5-TRIMETHOXYPHENYL) BUTANEEmile Al-Farhan; Rosemary Amofah; Philip M. Keehn; Robert Stevenson
81-83ONE-POT SYNTHESIS OF 2-SPIROTHIAZOLIDIN-4-ONE DERIVATIVESMaher F. El-Zohry
83-87PHASE TRANSFER CATALYZED N-ALKYLATION OF sym-N,N′-DIARYLUREASU. R. Kalkote; A. R. Choudhary; N. R. Ayyangar
87-91THE RESOLUTION OF RACEMIC AMINES BY THE FORMATION OF DIASTEREOMERIC AMIDES WITH AMINO ACIDSClara K. Miao; Ronald Sorcek; Jürgen H. Nagel
91-93A CONVENIENT METHOD FOR THE GENERATION OF NITRILE OXIDE AND ITS APPLICATION TO THE SYNTHESIS OF 2-ISOXAZOLINESK. M. Lokanatha Rai; N. Linganna; Alfred Hassner; C. Anjanamurthy
95-118OXIDATIVE REARRANGEMENT OF FURYLCARBINOLS TO 6-HYDROXY-2H-PYRAN-3(6H)-ONES, A USEFUL SYNTHON FOR THE PREPARATION OF A VARIETY OF HETEROCYCLIC COMPOUNDS, A REVIEWMinas P. Georgiadis; Kim E. Albizati; Taxiarchis M. Georgiadis
119CORRIGENDUM

Volume 23, Issue 6 (1991)

CEditorial Board Page
683-711APPLICATIONS OF MICROWAVE ENERGY IN ORGANIC CHEMISTRY. A REVIEWRudolph A. Abramovitch
713-720SYNTHESIS OF 1,1′-BIS(2-SULFOETHYL)PURPURATE(BISEP) TRISODIUM AND TRIPOTASSIUM SALTS. MEMBRANE IMPERMEANT CALCIUM INDICATORS FOR MUSCLE CONTRACTION STUDIESPhilip L. Southwick; Allan S. Wagman; Alan S. Waggoner
721-728THE SYNTHESIS OF N-CYANO-O-METHYLPSEUDOUREAS AND SOME OF THEIR FURTHER TRANSFORMATIONSJ. Zmitek; B. Jenko; D. Milivojevic; J. Anzel
729-734SYNTHESIS OF SOME ISOTHIOCYANATOPHENYLBORONIC ACIDSKondareddiar Ramalingam; David P. Nowotnik
735-739NEW SYNTHESIS OF 1-AZABICYCLO[5.3.0]DECANEGerald B. Hammond; Raymond G. Plevey
741-747HYDROXYMETHYLATION OF FLAVONESGyörgy Litkei; Tamás Patonay; László Szilágyi; Zoltán Dinya
749-752SYNTHESIS OF SUBSTITUTED 3-CHLORO-5-ARYLPENTA-2,4-DIEN-1-ALS AND OF 3-CHLORO-5-(5-FORMYLARYL)PENTA-2,4-DIEN-1-ALS BY THE VILSMEIER REACTIONM. Venugopal; P. T. Perumal
753-754A SIMPLE SYNTHESIS OF O-ISOPROPOXYPHENOLV. B. Deodhar; V. S. Dalavoy; U. R. Nayak
754-757SYNTHESIS OF METHOXYTAMOXIFENHoda A. El-Wakil
757-760TWO IMPROVED SYNTHESES OF N,N'-bis(3,3-DIETHOXYPROPYL)SUCCINAMIDEJohn T. Hortenstine; John E. Mills
760-762HEPTAFLUOROISOPROPOXIDE ION IN AROMATIC SUBSTITUTIONKeith E. Peterman; Wojciech Dmowski
762-764SYNTHESIS OF 5-HYDROXYMETHYL-1,4-DIOXAN-2-ONEGianluigi Broggini; Gaetano Zecchi
764-766CONVENIENT ONE-POT PROCESSES FOR THE PREPARATION OF CHLOROACETALDEHYDE DIALKYL ACETALSM. S. Malik; N. K. Sangwan; O. P. Malik; K. S. Dhindsa
767CORRIGENDA
769-781INDEXES

Volume 23, Issue 5 (1991)

CEditorial Board Page
571-5921,2-bis(ARYLSULFONYL)ALKENES. A REVIEWSergio Cossu; Ottorino De Lucchi; Davide Fabbri; Giulia Licini; Lucia Pasquato
593-610THE CHEMISTRY OF 1,3-DIOXIMES. A BRIEF REVIEWAntigoni Kotali; Vassilios P. Papageorgiou
611-616A ONE-POT PREPARATION OF DIMETHYL N-ALKYLIMINODITHIOCARBONATESC. Alvarez-Ibarra; M. L. Quiroga; E. Martinez-Santos; E. Toledano
617-620A CONVENIENT PREPARATION OF DIPHENYLMETHANES FROM BROMOBENZENES USING THE GRIGNARD CROSS-COUPLING REACTIONTakehiko Yamato; Naozumi Sakaue; Kazuaki Suehiro; Masashi Tashiro
621-626NITRO DERIVATIVES OF BENZOCOUMARINS. KEY INTERMEDIATES IN THE SYNTHESIS OF BENZOCOUMARIN-BASED FLUORESCENT REAGENTS FOR BIOLOGICAL APPLICATIONSJun-Rui Yang; Carol A. Lambert; Margaret E. Langmuir; Richard Laura
627-631AN ALTERNATE SYNTHESIS OF 3,4-DIAMINOBEZOPHENONE AND OF MEBENDAZOLEN. R. Ayyangar; R. J. Lahoti; Thomas Daniel
633-638SYNTHESIS OF (E,E)-BIS(ARYLCYCLOPROPYL) SULFONES FROM NOVEL (E,E)-BIS(STYRYL) SULFONESM. V. Ramana Reddy; D. Bhaskar Reddy; P. V. Ramana Reddy; S. Vijayalakshmi
639-643SYNTHESIS OF PRIMIN AND MICONIDIN AND THEIR 3-METHOXY ISOMERSSunday S. Arogba
645-650NOVEL SYNTHESIS OF PYRIDINE-2(1H)THIONES, N-AMINO-2-PYRIDONES AND PYRIDAZINE DERIVATIVESG. H. Elgemeie; S. R. El-Ezbawy; M. M. Ramiz; O. A. Mansour
651-654OXIDATION OF ADAMANTANE TO 1-ADAMANTANOL USING TETRA-N-BUTYLAMMONIUM OXONERajkumar Kumarathasan; Norman R. Hunter
655-658SYNTHESIS OF 2-HALO-4,5-DIFLUOROBENZOIC ACIDSTamim F. Braish; Darrell E. Fox
658-660AN IMPROVED PREPARATION OF QUINUCLIDIN-3-THIOLS. D. Aster; S. S. Yang; G. D. Berger
660-665THE REACTION OF NINHYDRIN WITH ACETIC ACIDJack B. Campbell; Edward R. Lavagnino; Charles W. Ryan
665-667FACILE CHROMONE RING-OPENING OF KHELLINEmile Al-Farhan; Philip M. Keehn; Robert Stevenson
667-670A NEW METHOD FOR THE SYNTHESIS OF 3β-HYDROXY-4α-BROMOCARANE AND OF cis-3-CARENE EPOXIDEMilind D. Choubal; Joseph Y. Bassett
670-672A NOVEL CLASS OF OXAZOLE DERIVATIVES. 4-ACYL-2-ARYLTHIO-5-ETHOXYOXAZOLESRicardo Bossio; Stefano Marcaccini; Roberto Pepino; Cecilia Polo; Tomás Torroba
673-676THE MANNICH REACTION OF CYCLIC KETONES, AROMATIC ALDEHYDES AND AROMATIC AMINESYi Lin; Zou Junhua; Lei Huangshu; Lin Xiaomei; Zhang Mingxiao
676-679IMPROVED SYNTHESIS OF A 2-ARYLBENZO[B]FURAN-3-CARBOXYLIC ACIDMichel Barbier
679-682SYNTHESIS OF NOVEL TRIAZOLO[2,3,b]-1,3,4-THIADIAZOLIUM SALTSZhu Zheng-Hua; Chen Shu-Ling; Yao Zu-Guang

Volume 23, Issue 4 (1991)

CEditorial Board Page
399-402N-ALKYLATION OF HINDERED SECONDARY AROMATIC AMINES WITH 2-IODOBUTANEAlan R. Katritzky; Jing Wu; Stanislaw Rachwal
403-411REDUCTION OF HETEROCYCLIC ALCOHOLS WITH SODIUM BOROHYDRIDE-TRIFLUOROACETIC ACID. PREPARATION OF bis-HETEROCYCLIC METHANESCharles F. Nutaitis; Richard Patragnoni; Greg Goodkin; Beth Neighbour; Judy Obaza-Nutaitis
413-418SYNTHESIS OF THIENO[3,2-e]-1,2,4-TRIAZOLO[a]PYRIMIDINESS. Tumkevicius; J. Mickiene
419-424THE BROMINATION OF 2,5-DIMETHOXYBENZALDEHYDE. STRUCTURAL PROOF OF THE 6-BROMO ISOMER via 3,6-DIMETHOXYBENZOCYCLOBUTENEManik S. Sardessai; Hanley N. Abramson
425-4272,4-DI-t-BUTYLBROMOBENZENE BY SILVER ION-ASSISTED BROMINATION OF 1,3-DI-t-BUTYLBENZENEAlbeit J. Fry; Shastra Solomon
427-431REDUCTION CLEAVAGE OF AROMATIC CYCLIC ACETALS WITH ZIRCONIUM CHLORIDE-LITHIUM ALUMINUM HYDRIDEWu Shaozu; Ren Tianhui; Chen Ning; Zhang Yulan
432-434SYNTHESIS OF cis6-OCTALIN-1,4-DIONE bis-ACETALSStan V. D'Andrea; Jeremiah P. Freeman; Jacob Szmuszkovicz
435-438PREPARATION OF N-UNSUBSTITUTED THIOAMIDES BY A MODIFIED WILLGERODT-KINDLER REACTIONQi-Dong You; Hou-Yuan Zhou; Qi-Zhou Wang; Xing-Han Lei
438-441SOLVENT EFFECT ON THE GOMBERG-BACHMANN-HEY ARYLAPON OF PYRIDINEMarek Gurczynski; Piotr Tomasik
441-442IMPROVED SYNTHESIS OF 2,4-HEXADIENOIC ACIDPéter Vinczer; Lajos Novák; Csaba Szántay
443-447APPLICATION OF POTASSIUM t-BUTOXIDE IN TOLUENE AS A BASE IN THE WITTIG REACTION IN LARGE-SCALE PHEROMONE SYNTHESESPéter Vinczer; Lajos Novák; Csaba Szántay
447-450A CONVENIENT SYNTHESIS OF 2,5-DIAMINO-1,4-BENZENEDIOLMuthiah Inbasekaran; Robert Strom
450-455REACTION OF 4-[BIS(ALKYLTHIO)METHYLENE]-2-PHENYL-2-OXAZOLIN-5-ONES WITH AMBIDENT NUCLEOPHILESJalpana Roy; N. S. Rawat
455-457A RAPID PREPARATION OF 2,2′-DIMERCAPTOBIPHENYLSergio Cossu; Giovanna Delogu; Davide Fabbri; Paola Maglioli
458-459PREPARATION OF TETRAETHYL (OXYDI-2,1-ETHANEDIYL)BISPHOSPHONATE AND 1,2-BIS[2-(DIETHYLPHOSPHONO)ETHOXY]ETHANEBalram Dhawan; Derek Redmore
460-463SYNTHESIS OF A HEXAALKYNYLHEXAPHENYLBENZENEJohn A. Hyatt
465-543TAXANE DITERPENE SYNTHESIS STRATEGIES. A REVIEWCharles S. Swindell
545-568RECENT DEVELOPMENTS IN THE AREA OF ANNDLATED FURANS. A REVIEWAlbert Padwa; S. Shaun Murphree
569CORRIGENDA

Volume 23, Issue 3 (1991)

CEditorial Board Page
273-320THE CHEMISTRY OF PYRAZOLIDINONES. A REVIEWRosa María Claramunt; José Elguero
321-356CONVERSION OF RESIN ACIDS INTO STEROIDAL COMPOUNDS. A REVIEWAntonio Abad; Consuelo Agulló; Manuel Arnó; Luis R. Domingo; Ramón J. Zaragozá
357-363AN IMPROVED FISCHER SYNTHESIS OF NITROINDOLES. 1,3-DIMETHYL-4-, 5- AND 6-NITROINDOLESAlan R. Katritzky; Stanislaw Rachwal; Shibli Bayyuk
365-372A FACILE SYNTHETIC ROUTE TO HYDROXY METABOLITES OF TRICYCLIC ANTIDEPRESSANTSMaciek Adamczyk; Yon-Yih Chen; Jeffrey R. Fishpaugh
373-374A FACILE SYNTHESIS OF ACYL-PROTECTED FORMALDEHYDE CYANOHYDRINSJeffrey H. Byers; Robert C. Baran; Molly E. Craig; John T. Jackman
375-376AN IMPROVED PREPARATION OF N-BENZYLOXYCARBONYL-L-LYSINE METHYL ESTER HYDROCHLORIDEZoltan Balajthy
377-378PREPARATION OF 1-(o-AMINOBENZOYL)-1-METHYLHYDRAZINESFerenc Fülöp; Kalevi Pihlaja
379-382CONVERSION OF 3-AROYLMETHYL-5-ARYLMETHYLENE-2,4-DIOXO-1,3-THIAZOLIDINES INTO 6-ARYL-4,5-DIHYDRO-1,2,4-TRIAZIN-3(2H)-ONESMohamed T. Omar; Ali M. Youssef
382-385SYNTHESIS OF NEW bis(m-PHENYLENE)-32-CROWN-10 DERIVATIVESYadoiiah Delaviz; Harry W. Gibson
386-387AN IMPROVED SYNTHESIS OF 3-PHENYL- AND 3-METHOXYQUINALDINEM. R. Akula; M. W. Wolowyk; E. E. Knaus
388-390CARBON-CARBON COUPLING ON ATTEMPTED HYDROLYSIS OF BROMOMALEIMIDESV. Balasubramaniyan; G. K. Laddha; N. P. Argade
390-392A CONVENIENT SYNTHESIS OF 5,7-DIHYDROXYCHROMONEGayland F. Spencer
392-394AN IMPROVED PREPARATION OF A TRICYCLIC LACTONE, A POTENTIALLY USEFUL PRECURSOR OF HIGHLY FUNCTIONALIZED TERPENOIDSJ. Zinczuk; J. A. Bacigaluppo; M. P. Mischne; M. I. Colombo; E. A. Rúveda
395-396A NEW AND CONVENIENT PREPARATION OF 3-BROMO-4-CHLORONITROBENZENEKantilal Kosandal; A. K. S. Bhujanga Rao; C. Gundu Rao; B. B. Singh
396-397A CONVENIENT SYNTHESIS OF (2S)-2-AMINO-3-PHENYLPROPANOLRamalinga Dharanipragada; Arled Alarcon; Victor J. Hruby

Volume 23, Issue 2 (1991)

CEditorial Board Page
133-138AN EFFICIENT SYNTHESIS OF α-ASARONEFrancisco Díaz; Leticia Contreras; Rosa Flores; Joaquín Tamariz; Fernando Labarrios; Germán Chamorro; Héber Muñoz
139-146β-KETONITROSAMINES AS SYNTHETIC EQUIVALENTS OF α-METHYLENE ALKANOLAMINO ANIONSJoseph E. Saavedra; David W. Famsworth
147-151PREPARATION AND SOME SIMPLE REACTIONS OF 1-SUBSTITUTED IMIDAZOLE-2,4,5-TRIONESBehzat Altural; Yunus Akcamur; Gert Kollenz
153-156ALKYLATION OF PHENYLACETONITRILE USING POTASSIUM CARBONATE AS A BASEChengzhi Xu; Xiangjun Mao; Hongbo Shen; Wenquiang Chen
157-162A FACILE ONE POT SYNTHESIS OF 3-SUBSTITUTED-1,2,4-TRIAZOLO[4,3-B][4,1,2]BENZOTHIADIAZINE-8-ONESB. Radha Rani; M. F. Rahman; U. T. Bhalerao
163-172AN IMPROVED SYNTHESIS OF NAPHTHO[2,3-d]-1,3-DIOXOLE-5-METHOXY-6-CARBOXYLIC ACIDJordan Zjawiony; John R. Peterson
173-180AN EFFICIENT LARGE SCALE PREPARATION OF (S)-1,1,2-TRIPHENYLETHANEDIOL 2-ACETATEA. Millar; L. W. Mulder; K. E. Mennen; C. W. Palmer
181-185SYNTHESIS OF bis-ISOXAZOLYLNAPHTHOQUINONESC. S. Ortiz; M. R. Longhi; M. M. De Bertorello; M. C. Briñon
186-188SYNTHESIS AND THERMOLYSIS OF CYCLOALKENYL AZIDES. A SIMPLE ROUTE TO POLYCYCLIC ISOXAZOLESMd. Izhar Sami; Gandhi K. Kar; Jayanta K. Ray
188-190AN IMPROVED SYNTHESIS OF 5-METHYLPYRAZINE-2-CARBOXYLIC ACIDI. Iovel; Yu. Goldberg; M. Shymanska
191-192OPTIMAL CONDITIONS FOR ACETYLATION OF AROMATIC TERTIARY ALCOHOLSL. Sipos; M. Zsuga; T. Kelen
193-195A CONVENIENT PREPARATION OF trans-3,4-DIPHENYLAND trans, trans-2,3,4-TRIPHENYLVALEROLACTONESJean A. Stanley; Susan Dakin; Linda Szabo; Leila Posaw; Christine Lee; Wen Min Hou
196-197FACILE SYNTHESIS OF HOMOTRIPTYCENES via ADDITION OF BENZOCYCLOPROPENE AND ANTHRACENESKatsuhiro Saito; Kazuaki Ito; Kensuke Takahashi; Shinzo Kagabu
198-200A NOVEL SYNTHESIS OF SOME ARYLTHIOGLYCOLIC ACIDSY. Yildirir; G. Okay
200-203AN OPTIMIZED SYNTHESIS OF DIMETHYL 2,2′-DIHYDROXY-1,1′-BINAPHTHALENE-3,3′-DICARBOXYLATE AND OF METHYL 2,2-DIHYDROXY-1,1′-BINAPHTHALENE-3-CARBOXYLATEMartin Hovorka; Jirí Závada
204-206EXPEDITIOUS ROUTES TO SYMMETRICALLY AND ASYMMETRICALLY SUBSTITUTED PYRIDINES FROM CHELIDAMIC ACIDPaolo Scrimin; Paolo Tecilla; Umberto Tonellato

Volume 23, Issue 2 (1991)

207-208SYNTHESIS OF DIALLYL SELENIDES. V. Amosova; V. A. Potapov; V. V. Nosyreva; A. F. Klimchuk
208-210O-METHYLATION OF POLYMER-SUPPORTED PHENOXIDES WITH DIMETHYL SULFATEA. Sarkar; B. Ram
211-213AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1-FERROCENYL-1-PHENYLMETHYLAMINEMarek Topolski; Janusz Rachon
214-216AN IMPROVED SYNTHESIS OF 6-(O-PHOSPHORYLCHOLINE)HYDROXYHEXANOIC ACIDPawel Knopik; Karol S. Bruzik; Wojciech J. Stec
217-235REGIOSPECIFIC ALKYLATION OF CYCLOHEXENONES. A REVIEWKenneth F. Podraza
237-272RECENT ADVANCES IN o-QUINODIMETHANE CHEMISTRYNazario Martin; Carlos Seoane; Michael Hanack

Volume 23, Issue 1 (1991)

CEditorial Board Page
1-65SYNTHESIS OF REACTIVITY OF λ5-PHOSPHAZENES. USES AS SYNTHETIC INTERMEDIATESJosé Barluenga; Francisco Palacios
67-92PYRROLOQUINOLINESDavid St. Clair Black; Naresh Kumar
93-101SYNTHESIS OF ETHYL N-CARBOBENZOXYTYROSYL-S-BENZYLCYSTEINYLGLYCINATEM. Dymicky; D. M. Byler
103-110SYNTHESIS OF cis AND trans-4-AMINOCYCLOHEXYL-D-ALANINE DERIVATIVES AND DETERMINATION OF THEIR STEREOCHEMISTRYPemmaraju N. Rao; Dorothy M. Peterson; C. Kirk Acosta; Martin L. Bahr; Hyun K. Kim
111-113SYNTHESIS OF A NEW AZATETRACYCLODECANE RING SYSTEM via INTRAMOLECULAR ADDITION OF AZIDE ON DOUBLE BONDS. Berényi; Gy. Gulyás; Gy. Batta; S. Makleit
114-115SYNTHESIS OF 1-(2-PYRIDINE-1-OXIDE)-2-(1-METHYL-2-PYRIDINIUM)-ETHANE CHLORIDEAi Jeng Lin
116-118A ONE-STEP SYNTHESIS OF CLOMID INTERMEDIATEMohammed I. Al-Hassan
119-122A FACILE SYNTHESIS OF rac-1-O-ALKYLGLYCEROLSB. V. S. K. Rao; A. Gangadhar; R. Subbarao; G. Lakshminarayana
122-125N-(DIPHENYLMETHYLENE)-α,β-DIDEHYDROAMINO ACID ESTERS. THERMAL AND LEWIS ACID INDUCED DIMERIZATIONSCesarino Balsamini; Giorgio Tarzia; Gilberto Spadoni; Americo Salvatori; Lamberto Staccioli
126-127A ONE-STEP SYNTHESIS OF OCIMIN BY A bis-WITTIG REACTIONDipti S. Khasnis; Ramchandra B. Mane
127-130A DIRECT APPROACH TOWARD THE SYNTHESIS OF ANALOGS OF ERBSTATINTerrence R. Burke Jr.
130-132AN IMPROVED SYNTHESIS OF 9-CHLORO-2-METHOXYACRIDINELynn James Sanfilippo

Volume 22, Issue 6 (1990)

CEditorial Board Page
655-706ARGININE, HISTIDINE AND TRYPTOPHAN IN PEPTIDE SYNTHESIS. THE INDOLE FUNCTION OF TRYPTOPHANBarbara Rzeszotarska; Elzbieta Masiukiewicz
707-746RECENT PROGRESS IN THE SYNTHESIS AND REACTIVITY OF NITROKETONES. A REVIEWGoffredo Rosini; Roberto Ballini; Marino Petrini; Emanuela Marotta; Paolo Righi
747-753ONE-STEP SYNTHESIS OF TRIFLUOROMETHYL- AND OF METHOXY-SUBSTITUTED BENZYNE PRECURSORSGary L. Grunewald; Aldean J. Kolar; Moorthy S. S. Palanki; Vidyadhar M. Paradkar; Thomas J. Reitz; Daniel J. Sall
755-760THE FRIEDEL - CRAFTS REACTION OF PHENOLS WITH CARBETHOXY ISOTHIOCYANATETadeusz Jagodziński
761-764AN IMPROVED SYNTHESIS OF (R)- AND (S)-2-METHYLPIPERAZINEJohn S. Kiely; Stephen R. Priebe
764-766TRANSFORMATION OF SOME β-TETRALONES TO 1,3-DIFORMYL-2-CHLORONAPTHALENESS. L. Evans; H. A. Lloyd; D. Lebeau; E. B. Sokoloski
766-768A CONVENIENT PREPARATION OF ETHYL 3,3 DIMETHYL-3H-INDOLE-2-CARBOXYLATEColin W. G. Fishwick; Andrew D. Jones; Michael B. Mitchell
769-780INDEXES

Volume 22, Issue 5 (1990)

CEditorial Board Page
547-574REARRANGEMENTS OF EPOXY ALCOHOLS AND RELATED COMPOUNDS. A REVIEWGöran Magnusson
575-578DIRECT ALKYLATION OF NITROARENES via VICARIOUS NUCLEOPHLIC SUBSTITUTION OF HYDROGENZbigniew Wrobel; Mieczyslaw Makosza
579-588SYNTHESIS OF 2-CHLORO-3-ALKYL- AND ARYLQUINOLINESFerenc Korodi; Zoltan Cziaky
589-595SYNTHESIS OF α-CHLORO-α,β-UNSATURATED ALDIMINES AND OF α-CHLORO-α,β-UNSATURATED ALDEHYDESChristian Stevens; Norbert De Kimpe
597-603THE PREPARATION OF Nα-t-BOC-2,3-DIAMINOPROPIONIC ACID (DPR) AND OF Nα-t-BOC-2,4-DIAMINOBUTYRIC ACID (DBR) DERIVATIVES SUITABLE FOR SOLID PHASE PEPTIDE SYNTHESISC. Freeman Stanfield; Arthur M. Felix; Waleed Danho
605-611CONVENIENT C-3 OXIDATION OF DEOXY AND AMINODEOXY SUGARSMária Mádi-Puskas; Pál László; István F. Pelyvás; Ferenc Sztaricskai
613-618A SIMPLE AND CONVENIENT SYNTHESIS OF 5-SUBSTITUTED BENZOXAZOLESKenneth R. Kunz; Ethan Will Taylor; Harold M. Hutton; Barry J. Blackburn
619-622CONVENIENT PREPARATION OF METABOLITES OF 6-n-PROPYLTHIOURACILF. S. Guziec Jr.; Lynn James Sanfilippo; Loide Mayer Wasmund
623-626A FACILE SYNTHESIS OF 5-DEOXY-D-RIBONIC ACID LACTONE AND OF 5-DEOXY-D-RIBOSEG. M. Escandar; L. F. Sala
627-629A SYNTHESIS OF (±)-3-ACETOXY-2,6-DIMETHYL-1,5-HEPTADIENE, THE SEX PHEROMONE OF THE COMSTOCK MEALYBUGSuk-Ku Kang; Choong-Sil Park
630-632IMPROVED METHOD FOR BISALLYLATION OF cis-BICYCLO [3.3.0]OCTANE-3,7-DIONE via THE CLAISEN REARRANGEMENTK. Sambasivarao; J. M. Cook
632-636BIOMIMETIC MODELING OF ASYMMETRIC SYNTHESIS OF ARYLALKYL SULFOXIDES USING β-CYCLODEXTRIN COMPLEXESK. Rama Rao; H. M. Sumpath Kumar; N. Bhanumathi; P. B. Sattur
636-638DIMETHYL 4-NITROPHENYLMALONATEM. A. E. Bowman; R. E. Bowman
639-641AN IMPROVED SYNTHESIS OF 3-NITROFLUORENEJ. R. Moran; G. Emmett
641-643AN IMPROVED SYNTHESIS OF 4′,5′-DIAMINOBENZO-15-CROWN-5Yasar Gök
643-645PREPARATION OF AN o-SUBSTITUTED BENZAMIDINE BY THE PINNER METHOD. A LITERATURE CLARIFICATIONC. C. Cheng
645-648AN IMPROVED SYNTHESIS OF 4,8,9,10-TETRAARYL-1,3-DIAZAADAMANTANESS. Sivasubramanian; M. Sundaravadivelu; N. Arumugam
648-650AN IMPROVED OZONOLYTIC APPROACH TO 6-OXOHEPTANALM. R. Karim; P. Sampson
651-654A CONVENIENT PREPARATION OF (+)-5(S)-METHYL-2(5H)-FURANONE. SYNTHESIS OF (S)-(+)-SULCATOLSuk-Ku Kang; Dong-Ha Lee; Sung-Gyu Kim

Volume 22, Issue 4 (1990)

CEditorial Board Page
399-484SYNTHESIS OF α-AMINOALDEHYDES AND α-AMINOKETONES. A REVIEWLawrence E. Fisher; Joseph M. Muchowski
485-493IMPROVED PROCEDURES FOR THE PREPARATION OF BENZO[c]CINNOLINE, ITS N-OXIDE AND SOME BROMO DERIVATIVES AND SYNTHESIS OF PYRROLIDINO, PIPERIDINO, AND MORPHOLINOBENZO[c]CINNOLINESEmine Kilic; Celal Tüzün
495-500IMPROVED SYNTHESIS OF 1,2-DIMETHOXY-3-ISOPROPYLBENZENE AND GENERAL SYNTHESIS OF 3-SUBSTITUTED-1,2-DIMETHOXYBENZENESLorraine M. Deck; Eugenia M. Brazwell; David L. Vander Jagt; Robert E. Royer
501-506IMPROVEMENTS IN THE SEMMLER-WOLF REARRANGEMENT OF 19-NORTESTOSTERONE OXIMEWilliam B. Smith; Milind P. Sant
507-511A NOVEL METHOD FOR HANDLING ORGANIC REACTIONS IN A BOMB TUBEG. Csanády; G. Knapp
511-514AN IMPROVED SYNTHESIS OF ALKYL 1-ALKYL-3-METHYL-2-PYRAZOLINE-5-ONE-4-DITHIOCARBOXYLATESAlfonso Oliva; Gerardo Léon; René Maurelia
514-518A SIMPLE ROUTE TO SOME SPIROIMIDAZOLONESC. del Campo; E. F. Llama
519-521SYNTHESIS OF 4,4-bis(2-METHOXYETHYL)CYCLOHEXANONE AND OF 4,4-bis(2-METHOXYETHYL)-2-CYCLOHEXEN-1-ONEElaine N. Cheeseman
522-525EFFECTIVE AND PREFERENTIAL TRANSFORMATION OF COMPOUNDS HAVING 2-HALOETHYL GROUPS ON POSITIVE SULFUR INTO ETHENYL COMPOUNDS UNDER PTC CONDITIONSY. Shimizugawa; T. Takahashi; M. Ishii; T. Yamamoto
526-528A FACILE SYNTHESIS OF NATURAL MHPG, A METABOLITE OF NOREPINEPHRINEM. Adamczyk; Y. Y. Chen; J. F. Fishpaugh
528-531ULTRASOUND-PROMOTED SODIUM BOROHYDRIDE REDUCTION OF PENTACYCLO[5.4.0.02,6.03.10.05,9]UNDECANE-8,11-DIONE (PCUD-8,11-DIONE) AND OF 4,4-DIMETHOXY-2,3,5,6-TETRACHLORO-PCUD-8,11-DIONEAlan P. Marchand; G. Madhusudhan Reddy
532-534AN IMPROVED SYNTHESIS OF DIMETHYL DIACETOXYFUMARATE AND ITS CONDENSATION WITH HETEROCYCLIC AMINESM. Tisler; R. Zupet
534-537DEOXYGENATION OF EPOXIDES WITH ALUMINUMPeter W. D. Mitchell
538-540ARYL HYDROGEN PHTHALATESP. C. Crofts; M. Ghahhary; M. Tajbakhsh-Jadidi
540-543IMPROVED PREPARATION OF DI-O-ISOPROPYLIDENE-1,2;5,6-D-MANNITOLC. Morpain; B. Nasser; B. Laude; N. Latruffe
544-546PREPARATION OF 4-THIAZOLIDINONE-1-OXIDESJ. B. Lee; S. Y. Yergatian; B. C. Crowther; I. M. Downie

Volume 22, Issue 3 (1990)

CEditorial Board Page
269-314ORGANOMETALLIC CARBOXAMIDATION. A REVIEWConstantinos G. Screttas; Barry R. Steele
315-397N-DIENYL AMIDES AND LACTAMS: PREPARATION AND DIELS-ALDER REACTIVITYMichael B. Smith

Volume 22, Issue 2 (1990)

CEditorial Board Page
131-165DIELS-ALDER REACTIONS OF CYCLOALKENONES IN ORGANIC SYNTHESISFrancesco Fringuelli; Aldo Taticchi; Ernest Wenkert
167-201CARBON-CARBON BOND CLEAVAGE BY THE HALLER-BAUER AND RELATED REACTIONS A REVIEWJohn P. Gilday; Leo A. Paquette
203-208ASYMMETRIC SYNTHESIS OF 2-,3-, AND 4-METHYLOCTANOIC ACIDSPhilip E. Sonnet; Joseph Gazzillo
209-213A ONE-POT PROCEDURE FOR THE PREPARATION OF PHOSPHONIC ACIDS FROM ALKYL HALIDESAlan R. Katritzky; Boguslaw Pilarski; Jack W. Johnson
215-227SYNTHESIS AND REACTIONS OF β-SILYLOXYACYLCYCLOPROPANES TRIMETHYLSILYL HALIDE-ZINC HALIDE INDUCED CYCLOPROPYLCARBINYL REARRANGEMENTA. M. Moiseenkov; B. A. Czeskis; N. M. Ivanova; O. M. Nefedov
229-2332,10-DICHLORO-6-(SUBSTITUTED ARYLOXY)DIBENZO[d,g][1,3,6,2]DIOXATHIA-PHOSPHOCIN 6-OXIDES. SYNTHESIS AND SPECTRAL CHARACTERISTICSC. Devendranath Reddy; K. Anuradha; K. Darrell Berlin; Prasanna S. Sunthankar; Satish V. Mulekar
235-244SYNTHESIS OF SOME 3,4-DIHYDRO-2H-1-BENZOTHIOPYRAN-4-OLSVicki L. Pruitt; K. Darrell Berlin; Kenneth S. Hirsch
245-253AN EFFICIENT SYNTHESIS OF 2′,3′-DIDEOXYADENOSINE via THE COREY-WINTER REACTIONRussell L. K. Carr; Thomas A. Donovan Jr.; Mahendra N. Sharma; C. Daniel Vizine; Michael J. Wovkulich
255-264THE PREPARATION OF AMIDE DERIVATIVES OF 3-AZABICYCLO-[3.3.1]NONANES AS NEW POTENTIAL ANTIARRHYTHMIC AGENTSStan A. Zisman; K. Darrell Berlin; B. J. Scherlag
265-268SYNTHESIS OF 2′,3′-DIDEOXY-5-METHYLCYTIDIN-2-ENE, A CYTIDINE ANALOG OF 3′-DEOXYTHYMIDIN-2′-ENE (d4T)Tai-Shun Lin; Jing-Hua Yang

Volume 22, Issue 1 (1990)

CEditorial Board Page
1-36RECENT ADVANCES IN THE USE OF ACYLIUM SALTS IN ORGANIC SYNTHESIS. A BRIEF REVIEWMahmoud Al-Talib; Hasan Tashtoush
37-45SYNTHESIS OF 1,4-DIMETHOXYBENZ[a]ANTHRACENES AND OF 7,10-DIMETHOXYCHOLANTHRENESMelvin S. Newman; A. R. Choudhary; A. Kumar
47-55SYNTHESIS OF MANNICH COMPOUNDS FROM FLAVANONESGyörgy Litkei; Tamás Patonay; Jenó Kardos
57-61REGIOSPECIFIC 5′-SILYLATION OF NUCLEOSIDESVasu Nair; Greg S. Buenger
63-70AN INEXPENSIVE AND CONVENIENT PREPARATION OF METHOXYMETHYL AND PHENYLTHIOMETHYL ETHERSR. Karl Dieter; Ravindra Datar
71-76A CONVENIENT SYNTHESIS OF N-[2-[[[5-[(DIMETHYLAMINO)METHYL]-2-FURANYLMETHYL]THIO]ETHYL]THIENO-[3,4-d]ISOTHIAZOL-3-AMINE-1,1-DIOXIDE HYDROCHLORIDE, A POTENT GASTRIC ACID ANTISECRETORY AGENTArthur A. Santilli; Robert L. Morris; Anthony C. Scotese; Donald P. Strike
77-84COMPETITIVE BIMOLECULAR REDUCTION IN THE SYNTHESIS OF KETONES MICHAEL ADDITION OF GRIGNARD REAGENTS TO α-ENONESC. Alvarez-Ibarra; M. S. Arias-Pérez; E. Moya; M. A. Rodríguez-Barranco
85-87A NEW ROUTE TO NITRO-AND BENZOYLPHTHALIDESWenjeng Guo; Y. F. Duann
87-94SYNTHESIS OF 3-QUINUCLIDINYL BENZILATE DERIVATIVESG. W. Kabalka; S. B. Mathur; Y. -Z. Gai
94-97AN EFFICIENT SYNTHESIS OF α,β-UNSATURATED CARBOXYLIC ACIDS AND NITRILESChang Kiu Lee; Jeung Yeop Shim
97-99SYNTHESIS OF N-DESMETHYL MESORIDAZINET. Mohammad; E. M. Hawes; K. K. Midha
99-102MONOMETHYLATION OF 3,4-DIHYDROXYBENZALDEHYDE AS AN ALTERNATE ROUTE TO ISOVANILLINAndre Loupy; Mustapha Majdoub
102-104A CONVENIENT SYNTHESIS OF 2,3-DIBROMOANTHRACENEMurthy R. Akula
104-105THE PREPARATION OF 5-CHLORO-2-INDOLINONE BY DIRECT CHLORINATION OF 2-INDOLINONEPaul Pranc
106-108BENZIMIDAZOLE ANTIVIRALS. REGIOSPECIFIC SYNTHESIS OF ARYL BENZIMIDAZOYL KETONES BY SULFONAMIDE ANION DISPLACEMENT OF AROMATIC FLUORIDESamuel J. Dominianni
109-1112,2-DIMETHYL-6-[(TRIPHENYLPHOSPHORANYLIDENE)METHYL]-4H-1,3-DIOXIN-4-ONE. A FOUR-CARBON HOMOLOGATING AGENT REQUIRING NO ACTIVATIONChristina Bodurow; Michael A. Carr; Larry L. Moore
112-113A CONVENIENT ONE-POT SYNTHESIS OF 2-METHYL-2-BENZYLTHIOPROPANALGerald S. Jones Jr.; David R. Elmaleh

Volume 22, Issue 1 (1990)

113-117IMPROVED SYNTHESIS OF NITRO DERIVATIVES OF N-PHENYLGLYCINEK. U. B. Rao; R. K. Bhongle; S. R. Yoganarasimhan
117-119AN EFFICIENT METHOD FOR THE SYNTHESIS OF N-(p-AMINOBENZOYL)AMINO ACIDSA. Panduranga Reddy; C. Kasi Reddy
119-121A FACILE SYNTHESIS OF BIOTIN N-HYDROXYSUCCINIMIDE ESTERK. N. Parameswaran
122-123A SIMPLE AND SHORT SYNTHESIS OF (Z)-13-EICOSEN-10-ONE, THE SEX PHEROMONE OF THE PEACH FRUIT MOTHSuk-Ku Kang; Dong-Ha Lee
124-128SYNTHESIS OF POTENTIAL 1-[1-(2-THIENYL)CYCLOHEXYL]PIPERIDINE METABOLITESGeorge A. Brine; David K. Sawyer; F. Ivy Carroll
128-130AN ALTERNATIVE METHOD FOR TOLNAFTATEN. R. Ayyangar; R. D. Wakharkar; V. H. Deshpande; B. Rai

Volume 21, Issue 6 (1989)

CEditorial Board Page
659-704PREPARATION AND REACTIONS OF 4-OXOCARBONYL COMPOUNDS. A REVIEWTetsuo Miyakoshi
705-749MICHAEL ADDITION OF ORGANOLITHIUM COMPOUNDS. A REVIEWDavid A. Hunt
751-756METHYLATION OF BIDENTATE NITROGEN-CONTAINING HETEROCYCLES WITH METHYL IODIDE AND POTASSIUM HYDROXIDE IN DIMETHYL SULFOXIDEElisabetta Giorgini; Lucedio Greci; Giorgio Tosi; Vittorio Bocchi
757-761A SIMPLE PROCEDURE FOR THE SYNTHESIS OF LABILE ARYL OXIRANES BY EPOXIDATIONFrancesco Fringuelli; Ferdinando Pizzo; Raimondo Germani; Gianfranco Savelli
763-770SYNTHESIS OF 7-HYDROXY-4-BENZOFURANACETIC ACIDS. J. Kesten; I. C. Pattison; O. P. Goel
771-776CYCLIC CARBONATE ESTER OF 4-NITROCATECHOL. REACTIONS WITH AMINESDaniel A. Laufer; Kenneth Doyle; Xiaodong Zhang
777-788INDEXES

Volume 21, Issue 5 (1989)

CEditorial Board Page
521-618SYNTHESIS OF QUASSINOIDS. A REVIEWKenji Kawada; Moonsun Kim; David S. Watt
619-627SYNTHESIS OF CHROMOPHORIC ANALOGS OF ACETYLCHOLINE HALIDESLeroy H. Klemm; Warner L. Peticolas; Kori L. Clement; K. Jeffry Wilson
629-632A FACILE PREPARATION OF 2(Z), 5(Z), 8(Z)-TETRADECATRIEN-1-OL, A KEY INTERMEDIATE FOR EICOSANOID SYNTHESISDomenico Badone; Roberto Pagliarin; Massimo Sisti; Paolo Tavecchia
633-641PREPARATION OF AZULENE DERIVATIVES: AN AMINOACID, DICARBOXYLATES, AN ISOTHIOCYANATE, AND RELATED COMPOUNDSLeRoy H. Klem; Bruce S. Hudson; Jennifer J. Lu
643-645AN IMPROVED SYNTHESIS OF 1-(4-NITROBENZYL)-1.2-ETHYLENEDIAMINE, PRECURSOR OF THE CORRESPONDING ETHYLENEDIAMINETETRAACETIC ACIDRene C. Gaudreault; Antoine A. Noujaim
645-648SYNTHESIS OF 2-HEXYLNAPHTHALENEB. Dewprashad; E. J. Eisenbraun
649-652THE 2- AND 4-NITRO AND 2- AND 4-ACETAMIDO 5,6,7,8,9,10-HEXAHYDRO DERIVATIVES OF CYCLOHEPTA[b]INDOLEArthur G. Anderson Jr.; Harry F. Richards; Ralph D. Haddock
653-6552,3,4,5,6,7-HEXAHYDROCYCLOPENTA-1,4-THIAZINE AND THE 8,9-DIHYDRO-, 4-ACETYL AND l-OXO - 4-ACETYL DERIVATIVESArthur G. Anderson Jr.; Russell A. Labar; Ralph D. Haddock
655-656A FACILE REDUCTION OF 1,8-NAPHTHALIMIDE TO 1,2,3,4-TETRAHYDRO-1,8-NAPHTHALIMIDEMichael D. Crenshaw; C. C. Cheng
657CORRIGENDUM

Volume 21, Issue 4 (1989)

CEditorial Board Page
393-450ARGININE, HISTIDINE AND TRYPTOPHAN IN PEPTIDE SYNTHESIS. THE IMIDAZOLE FUNCTION OF HISTIDINEBarbara Rzeszotarska; Elzbieta Masiukiewicz
451-477RECENT DEVELOPMENTS IN THE SYNTHESIS OF ALDEHYDES BY REDUCTION OF CARBOXYLIC ACIDS AND THEIR DERIVATIVES WITH METAL HYDRIDES. A REVIEWJin Soon Cha
479-484REACTIONS OF SOME AROMATIC AMINES WITH CINNAMOYL ISOTHIOCYANATEA. H. H. Elghandour; M. M. M. Ramiz; M. K. A. Ibrahim; M. R. H. Elmoghayar
485-491SYNTHESIS OF 2,6-DIPHENYL-9-METHYLENE-1-AZA-7-OXASPIRO[4.5]DECAN-8-ONEST. Mohamed Ikramudden; N. Chandrasekara; K. Ramarajan; K. Selvaraj; Satish V. Mulekar; K. Darrell Berlin
493-500SYNTHESIS OF PURPURATE-1,1′-DIACETIC ACID (PDAA) TRIPOTASSIUM SALT. A NEW CALCIUM INDICATOR FOR BIOLOGICAL APPLICATIONSPhilip L. Southwick; Alan S. Waggoner
501-504IMPROVED PROCEDURE FOR THE ONE-STEP SYNTHESIS OF α-KETOESTERSJanak Singh; Thomas P. Kissick; Richard H. Mueller
505-508A CONVENIENT PROCEDURE FOR THE PREPARATION OF t-BUTYLDIMETHYLSILYL ETHERS OF HYDROXYAMINO ACIDSF. Orsini; F. Pelizzoni; M. Sisti; L. Verotta
509-511AN IMPROVED PROCEDURE FOR THE PREPARATION OF 1,1,1-TRICHLORO-4-METHYL-3-PENTEN-2-YL DIAZOACETATEA. R. A. S. Deshmukh; B. M. Bhawal; D. G. Panse; G. H. Kulkarni
511-514FACILE SYNTHESIS OF 2-METHOXYISOBUTYLISONITRILEK. Ramalingam
514-515AN IMPROVED SYNTHESIS OF 2-ISOCYANATOBENZONITRLEDieter Sicker; Frauke Fiebig; Gerhard Mann
515-517A CONVENIENT “HYDROGEN TRANSFER” HYDROGENATION OF TESTOSTERONEDimitris M. Spyriounis; George Ikonomidis; Vassilis J. Demopoulos
517-519TEREPHTHALOHYDROXIMOYL CHLORIDEAbrahim Karatas; Celal Tuzum

Volume 21, Issue 3 (1989)

CEditorial Board Page
257-296USE OF SUBSTITUTED 3-SULFOLENES AS PRECURSORS FOR 1,3-BUTADIENESTa-Shue Chou; Hsi-Hwa Tso
297-301CYCLZATION OF ω-HALONITRILES WITH ORGANOLITHIUMSVincent Gallulo; Liberty Dimas; Charles A. Zezza; Michael B. Smith
303-308SYNTHESIS OF TWO PHOTOLABILE BENZYL MANGANESE DERIVATIVES INCORPORATING A GEOMETRICALLY INACCESSIBLE RADICAL TRAPJohn F. W. Keana; Sovitj Pou
309-314SYNTHESIS OF (±)-NOROORALYDINE AND (±)-TETRAHYDROPALMATINEKazuhiko Orito; Tsutomu Matsuzaki; Hiroshi Suginome
315-319A SIMPLIFIED PROCEDURE FOR PREPARING THE CHOLINERGIC NEUROTOXIN 1-ETHYL-1-(2-EYDROXYETHYL)AZIRIDINIUM ION (AF64A)Walter H. Moos; Robert E. Davis; Roy D. Schwarz
321-326ACYLATION OF 1,2,4,5-TETRAHYDRO-3-MEIHYL-3H-3-BENZAZEPIN-2-ONE IN THE PRESENCE OF SODIUM HYDRIDEKazuhiko Orito; Harumi Kaga; Hiroshi Suginome
327-335SYNTHESIS OF 2,6-DIARYLTETRAHYDROPYRAN-4-ONESTimothy M. Fakler; K. Darrell Berlin
337-339SYNTHESIS OF 1,3-bis(2-BROMOPHENYL)PROPANERichard A. Bunce; Vicki L. Taylor; Henry D. Reeves
340-341A PRACTICAL SYNTHETIC METHOD FOR N-METHYL-o-TOLUIDINEAlan R. Katritzky; Kunihiko Akutagawa
341-3434-(2-ARYLALKENYL)-3-CYANO-2H-1-BENZOPYRAN-2-ONESY. Anghelova; E. Dimitrova
344-346AN IMPROVED SYNTHESIS OF 5-HYDROXYPENTANALPeter Vinczer; Zoltan Juvancz; Lajos Novak; Csaba Szantay
346-348A SIMPLE SYNTHESIS OF (+)-trans-VERBENYL PROPIONATE, A PHEROMONE ANALOG OF AMERICAN COCKROACH USING LEAD(IV) PROPIONATEPeter Vinczer; Maria Kajtar-Peredy; Zoltan Juvancz; Lajos Novak; Csaba Szantay
348-351SYNTHESIS OF (2-BUTYL-3-BENZOFURANYL)[4-[2-(DIETHYLAMINO)ETHOXY]-3,5-DIIODOPHENYL)METHANE DERIVATIVESGeorge W. Kabalka; Thomas P. Kennedy; Naganna M. Goudgaod; Rajender S. Varma
351-353L-DOPA-3-0-SULFATE BY THE PERSULFATE OXIDATION OF L-TYROSINEE. J. Behrman; J. M. Bidinger
354-355A FACILE SYNTHESIS OF DIARYLACETONITRILE FROM DIARYKETONES AND TRIMETHYLSILYL CYANIDEKatsuhiro Saito; Shinzo Kagabu; Yoichi Horie; Kensuke Takahashi
355-358AN IMPROVED PROCEDURE FOR THE DICHLOROACETYLATION OF PRIMARY AND SECONDARY AMINESBraja G. Hazra; V. S. Pore; S. P. Maybhate
359-360THE LITHIATION OF 1,4-DIMETHOXYNAPHTHALENE AND CARBOXYLATION OF THE PRODUCTSMelvin S. Newman; Anil R. Choudhary
360-363AN EFFICIENT PREPARATION OF 1,2-DIHYDROCYCLOBUTA[a]NAPHTHALENEDavid A. Hunt

Volume 21, Issue 3 (1989)

364-366THE SYNTHESIS OF THE DIIMINE AND THE RADICAL CATION CHLORIDE OF N,N′-DIPHENYL-p-PHENYLENEDIAMINEMukarram H. Zaghal; Mazin Y. Shatnawi
366-368HETEROGENEOUS SYNTHESIS OF REISSERT COMPOUNDS UTILIZING POTASSIUM CYANIDE ADSORBED ON AMBERLITE XAD RESINSFrank D. Popp; Frederick F. Duarte
368-371TRANSFORMATION OF SOME ARYL, BENZYL KETONES TO 2-ARYL-1,3-DICHLOROINDENES BY VILSMEIER REAGENTI. W. Elliott; S. L. Evans; L. T. Kennedy; A. E. Parrish
371-373AN IMPROVED SYNTHESIS OF (S)-3-METHYL-γ-BUTYROLACTONEPatrizia Ferraboschi; Paride Grisenti; Alberto Fiecchi; Enzo Santaniello
373-375A SIMPLE REDUCTION OF ARALKYL KETONES TO ALCOHOLSA. S. Radhakrishna; K. R. K. Prasad Rao; S. C. Nigam; R. Bakthavatchalam; B. B. Singh
375-376A CONVENIENT SYNTHESIS OF TOSYLLACTONITRILE AND ITS REACTION WITH BENZENEA. S. Radhakrishna; R. Bakthavatchalam; K. R. K. Prasad Rao; B. B. Singh
377-380CHEMOSELECTIVE CATALYTIC HYDROGENATION OF CARBONYL CONJUGATED DOUBLE BONDS IN THE PRESENCE OF STYRENOID BONDS IN BICYCLO[3.3.1]NONADIENONESR. Chakraborti; B. C. Ranu; U. R. Ghatak
380-383PREPARATION OF NOVEL 2-ARYL-4H-NAPHTH[2,1-e]-1,3,4-OXADIAZINE- 6-OL DERIVATIVESR. Ashok Kumar; C. K. Kokate; M. S. Rao; T. V. Padmanabha Rao
383-385A CONVENIENT ONE-STEP SYNTHESIS OF AROYL CYANIDES FROM AROMATIC ALDEHYDESSuk-Ku Kang; Houng-Kyu Sohn; Sung-Gyu Kim
386-388PREPARATION OF 1-ETHYNYL-7-METHOXYNAPHTHALENEJane A. Moore; James W. Roche; Philippe Prince; Richard D. Gandod; Frank R. Fronczek
388-390REDUCTION OF SULFONYL CHLORIDES WITH SODIUM CYANOBOROHYDRIDEShinzo Kagabu
390-392A CONVENIENT SYNTHESIS OF DIETHYL (MERCAPTOMETHYL)PHOSPHONATEG. K. Farrington; Alok Kumar; F. C. Wedler

Volume 21, Issue 2 (1989)

CEditorial Board Page
129-133SYNTHESIS OF BRANCHED LONG CHAIN ALIPHATIC PRIMARY ALKYL BROMIDESAlan R. Katritzky; Adam Bieniek; Long Chiang
135-139THE PREPARATION OF 1-(α-AMINOALKYL) - BENZOTRIAZOLES IN AQUEOUS SOLUTIONAlan R. Katritzky; Boguslaw Pilarski; Laszlo Urogdi
141-146A SIMPLE PREPARATION OF 2-UNSUBSTITUTED 4-AMINOOXAZOLESRam Lakhan; Ram Lakhan Singh
147-156REGIOSELECTTVE SYNIHESIS OF CHOLESTANE-3β,5α,6α-TRIOL-7-ONE 3-ACETATE AND EIGHT STEREOISOMERIC CHOLESTANE-3β,4,5α,6 AND OF 3β,5α,6,7-TETROL TRIACETATESJames Warren; Stephen O'brien; Harold R. Nace
157-162CONVENIENT LARGE SCALE PREPARATION OF 5-METHYL- AND 4-NITRO- 2-IODOSOBENZOIC AND OF 4-NITRO-2-IODOXYBENZOIC ACIDSAlan R. Katritzky; G. Paul Savage; John K. Gallos; H. Dupont Durst
163-171SYNTHESIS OF NOVEL 1,2,4-TRIAZOLOQUINAZOLINE RING SYSTEMSJózsef Reiter; László Pongo
173-178SYNTHESIS OF ANALOGS OF PROPRANOLOL HYDROCHLORIDEJames S. Farina; Steven A. Jackson; Corbin L. Cummings
179-217RECENT PROGRESS IN TEE CONTROL OF CARBON VERSUS OXYGEN ACYLATION OF ENOLATE ANIONST. Howard Black
219-221A SHORT SYNTHESIS OF cis-1,7,7-TRIMETHYLBICYCLO[4.4.0]DEC-3-ENEWilliam A. Donaldson; Joseph W. Strohbach
221-223A FACILE SYNTHESIS OF 3,4-DIHYDRO-1,5-BENZODIOXEPIN-2-ONESM. S. Reddy; G. L. D. Krupadanam; G. Srimannarayana
223-225A SIMPLE PREPARATION OF 1-HYDROXYPYRENERaj K. Sehgal; Subodh Kumar
225-228AN IMPROVED SYNTHESIS OF (1R, 2R)-(-)-a-(1-ISOPROPYLAMINOETHYL)BENZYL ALCOHOLDuy H. Hua; Roch Chan-yu-King; Robert A. Ostrander; Jeffrey A. McKie
228-230A FACILE SYNTHESIS OF BENZYL ISOTHIOCYANATES BY USE OF 18-CROWN-6 ETHERS. Muthusamy; V. T. Ramakrishnan
230-232A NEW METHOD FOR THE CONVERSION OF ALDOXIMES INTO NITRILES WITH ZEOLITESM. Narayana Rao; Pradeep Kumar; Kamini Garyali
232-237SIMPLE SYNTHESIS OF ALKYNES FROM 1,2-DIBROMOALKANES USING PTC CONDITIONSPeter Vinczer; Terez Kovacd; Lajos Novak; Csaba Szantay
237-240REDUCTION OF 1,3,5-TRISUBSTITUTED 2-ALKYLPYRAZOLIUM SALTS WITH COMPLEX METAL HYDRIDES. SYNTHESIS OF 3-PYRAZOLINESAngel Alberola; Luis A. Banuelos; Purification Cuadrado; Ana Ma Gonzalez; Fco. Jose Pulido
241-242A SIMPLE ONE-STEP SYNTHESIS OF 5-ACETOXY-6-CHLORO-2-HEXANONENaresh K. Sangwan; Kuldip Singh Dhindsa

Volume 21, Issue 2 (1989)

243-245USE OF 5,8-DIMETHOXYQUINOLINES IN THE SYNTHESIS OF NOVEL 5,12-DIHYDROXY-6,11-DIOXO-1-AZANAPHTHACENESP. N. H. Nizar; S. M. S. Chauhan
245-248A CONVENIENT SYNTHESIS OF POLYFLUORINATED α, ω-DIAMINESThomas F. Ball; Robert N. Henrie II
249-251NITRATION OF 2-CARBONYL-3,4-DICHLOROFURAN DERIVATIVESK. Yamamoto; J. Koyanagi; A. Tanaka; I. Horie; M. Ichikawa; S. Swaminathan; J. F. Hatcher; G. T. Bryan
251-253FACILE PREPARATION OF L-2-OXOTHLUOLIDINE-4-CARBOXYLIC ACID (OTC)T. Kömives
253-254A CONVENIENT PREPARATION OF ETIWL 7-BROMOHEPTANOATEStefano Canonica; Marinella Ferrari; Massimo Sisti
255-256AN IMPROVED SYNTHESIS OF (1α,6α)-8,8-DIOXABICYCLO[4.3.0]NONA-2,4-DIENEMartin G. Banwell

Volume 21, Issue 1 (1989)

CEditorial Board Page
1-46SYNTHETIC CHEMISTRY OF NATURALLY OCCURRING OLIGOPEPTIDE ANTIBIOTICS AND RELATED LEXITROPSINSJ. William Lown
47-65SYNTHESIS OF LARGE CONDENSED POLYCYCLIC AROMATIC HYDROCARBONS. A REVIEWJohn C. Fetzer
67-74PREPARATION OF N-1-BUTYLOXYCARBONYL-Oω-9-FLUORENYLMETHYL ESTERS OF ASPARTIC AND GLUTAMIC ACIDSD. R. Bolin; C. -T. Wang; A. M. Felix
75-82LOWER ALIPHATIC 2-OXOACIDS AND THEIR ETEYL ESTERS FROM ETHYL ESTERS OF 2-HYDROXY ACIDSRoman Kozłowski; Zbigniew Kubica; Barbara Rzeszotarska; Leszek Smełka; Grzegorz Pietrzyński
83-90PREPARATION OF CARBOBENZOXY-L-TYROSINE METHYL AND ETHYL ESTERS AND OF THE CORRESPONDING CARBOBENZOXY HYDRAZIDESM. Dymicky
91-104PREPARATION OF α,α-DIALKYL-β-HALOKETONESPaul Sulmon; Norbert De Kimpe; Niceas Schamp
105-108PREPARATION OF NEW 5-CYANO AND 5-CARBAMOYLIMIDAZOLES FROM 5-NITROIMIDAZOLES BY PHOTOCYANATIONMichel P. Crozet; Patrice Vanelle; Olivier Jentzer; José Maldonado
109-118RACEMIC TOTAL SYNTHESES OF ISOAUSTROBAILICNAN-1 AND OF SOME RELATED ARYLTETRALIN LACTONESRobert Dhal; Khalid Lalami; Eric Brown
119-124SYNTHESIS OF PYRAZOLES AND 2-PYRAZOLINES FROM C-PHENYLAMINOCARBONYL-N-ARYLFORMOHYDRAZIDOYL CHLORIDESHamdi M. Hassaneen; Abdelgawad A. Fahmi; Ikhlas M. Abbas; Ahmad S. Shawali
125-128PREPARATION OF 3-CHLORO-6-(TRIPHENYLMETHYLAZO) PYRIDAZINECarlo Farina; Riccardo Monguzzi; Mario Pinza

Volume 20, Issue 6 (1988)

CEditorial Board Page
533-584RECENT APPLICATIONS OF OXOCHROMIUMAMINE COMPLEXES AS OXIDANTS IN ORGANIC SYNTHESIS. A REVIEWFrederick A. Luzzio; Frank S. Guziec Jr.
585-590A NEW SYNTHETIC METHOD FOR THE 2-SUBSTITUTION OF PYRROLEAlan R. Katritzky; Kunihiko Akutagawawa
591-592OXIDATIVE NITROMETHYLENATION (SNH SUBSTITUTION) IN PYRIDINIUM SALTSDick J. Buurman; Henk C. van der Plas
593-597SYNTHESIS OF 7-OXO ALCOHOLS via ENAMINEG. Pratap; K. L. Shanatha; V. S. Bhaskar Rao
598-599SYNTHESIS OF NITROALKANES FROM BROMOALKANES BY PHASE-TRANSFER CATALYSISPramodchandra V. Sane; Man Mohan Sharma
600-602SYNTHESIS OF PHENYLACETYL-L-CYSTEINYL-D-VALINE DISULFIDE. A BIOSYNTHETIC PRECURSOR OF PENICILLINGJ. M. Luengo; M. T. Alemany; M. J. Arin; M. T. Diez; F. Salto
603-616INDEXES

Volume 20, Issue 5 (1988)

CEditorial Board Page
427-464ARGININE, HISTIDINE AND TRYPTOPHAN IN PEPTIDE SYNTHESIS. THE GUANIDINO FUNCTION OF ARGININEBarbara Rzeszotarska; Elzbieta Masiukiewicz
465-474THE CYANAMIDO MOIETY AS A NOVEL LEAVING GROUPJözsef Reiter
475-483AN IMPROVED SYNTHESIS OF (E)-9-DODECEN-1-YL ACETATE, THE SEX PHEROMONE OF RHYACIONIA BUOLIANAF. Szurdoki; L. Novák; C. S. Szántay; E. Baitz-gács; M. Tóth
485-491SYNTHESIS OF URACIL-5-PHOSPHINIC AND 5-THIOPHOSPHONIC ACIDSTokumi Maruyama; Shuhei Kimura; Mikio Honjo
493-496EFFICIENT SYHTHESIS OF α-CHLOKOVIHYL PHEHYL SULFONEKrzysztof Wojciechowskl
497-503IMPROVED PREPARATION OF PENICILLIN N AND ISOPENICILLIN NGeorge W. Huffman
505-510A FACILE SYNTHESIS OF ARYLAZOSELENAZOLES AND OF AROYLSELENADIAZOLESHamdi M. Hassaneen; Ahmed M. Farag; Mohammed S. Algharib; Ahmad S. Shawali
511-519A ONE-POT PREPARATION OF SUBSTITUTED BIS-1, 3, 5-TRIAZINIUM SALTSHasan Tashtoush; Mahmoud Al-Talib
521-526SYNTHESIS AND REACTIONS OF C-(2-THENOYL)-N-ARYLFORMHYDRAZIDOYL BROMIDESAhmed M. Farag; Mohamed S. Algharib
527-532SYNTHESIS OF MICROMINUTIN AND 4-METHYLMICROMINUTINR. D. Wakharkar; V. H. Deshpande; A. B. Landge; B. K. Upadhye

Volume 20, Issue 4 (1988)

CEditorial Board Page
317-369SYNTHESIS AND REACTIONS OF FUNCTIONALIZED SILYLENOL ETHERS. A REVIEWJean-Marie Poirier
371-376AN EFFICIENT LARGE SCALE PREPARATION OF D, L-2-AMINO-5-PHOSPHONOPENTANOIC ACID (D, L-AP5)Paul L. Ornstein
377-383A CONVENIENT SYNTHESIS OF 3, 5-DIMETHYL-4-ISOXAZOLYL AND OF 3, 5-DIMETHYL-4-ISOTHIAZOLYLKETONESAngel Alberola; Purificacion Cuadrado; Ma Carmen Sañudo; Tomás Torroba
385-392SYNTHESES OF CARCINOGENIC β-KETONITROSAMINES FOUND IN MOLDY MILLET, WHEAT FLOUR AND CORNBREADJoseph E. Saavedra; Guo-Kui Pei; David W. Farnsworth
393-399AN EFFICIENT SYNTHESIS OF 5-BROMO-2-HYDROXYCYCLOHEPTA-2, 4, 6-TRIEN-1-ONE AND ITS METHYL ETHERMartin G. Banwell; John N. Lambert; Monica E. Reum; René Onrust
401-404SYNTHESIS OF ISOXAZOLYL 2-PYRAZOLINESG. Venkateshwarlu; E. Rajanarendar; C. J. Rao; A. Krishna Murty
405-408ALDEHYDES FROM ACYLHYDRAZINES BY REDUCTION WITH SODIUM BOROHYDRIDE IN THE PRESENCE OF CUPRIC CHLORIDEOrazio A. Attanasi; Franco Serra-Zanetti; Giorgio Tosi
408-414SYNTHESIS OF UNUSUAL CONJUGATED AZOALKENESOrazio A. Attanasi; Mario Grossi; Amedeo Mei; Franco Serra-Zanetti
414-418SYNTHESIS OF N-PYRROLYL ACIDSA. Negro; M. T. Diez; M. T. Alemany
419-422A PROCEDURE FOR THE LARGE-SCALE PREPARATION OF METHYL IMINO (METHYLTHIO) METHYL CARBAMATEC. Someswara Rao; M. Rambabu; N. L. Mistry
423-425PREPARATION OF 4-NITROPHTHALIC ANHYDRIDE FROM N-METHYL-4-NITROPHTHALIMIDERomas J. Kazlauskas

Volume 20, Issue 3 (1988)

CEditorial Board Page
199-204A SHORT SYNTHESIS OF (±)-α-CHAMIGRENEEmil R. Koft; Thomas A. Broadbent
205-211PREPARATION OF STYRYL BENZYLSULFONES AND 1, 2-BIS (STYRYLSULFONYLMETHYL)-4, 5-DIMETHYLBENZENESD. Bhaskar Reddy; N. S. Reddy; S. Reddy; H. V. R. Reddy; S. Balasubramanyan
213-222SYNTHESIS OF ACENAPHTHO[1, 2-b]BENZO[d]THIOPHENEGandhi K. Kar; Basanta G. Chatterjee; Jayanta K. Ray
223-230THE SYNTHESIS OF PEROPYRENE-TYPE POLYCYCLIC AROMATIC HYDROCARBONSJ. C. Fetzer; W. R. Biggs
231-2364-PHENYL-Δ3-DIHYDROPYRANS BY REDUCTION OF PYRILIUM SALTS WITH SODIUM BOROHYDRIDE IN ACETIC ACIDTeodor-Silviu Balaban; Alexandru T. Balaban
237-243SYNTHESIS OF ALKYL INDOLIZINES FROM PYRYLIUM SALTSAntonie Dinculescu; Teodor-Silviu Balaban; Alexandru T. Balaban
245-252SYNTHESIS OF 4-HYDROXY-4-(2-THIENYL)PENTAMIDER. Cruz-Almanza; F. García; B. Ramírez; M. Ordoñez
253-260SYNTHESIS OF THE ANTIHYPERTENSIVE AGENT 1-(1-METHYLETHYL)-2-(2-[4-(3-TRIFLUOROMETHYLPHENYL)-1-PIPERAZINYL]ETHYL)-1H-NAPHTH[1, 2-d] IMIDAZOLE CITRATEE. Toja; A. Trani
261-269APPROACH TO THE SYNTHESIS OF AN OPTICALLY ACTIVE POLYNUCLEOTIDE ANALOGMing-Jye Lan; C. G. Overberger
271-274S, S-DIARYL- AND S-(2-SUBSTITUTED ETHYL)-S-PHENYL-N-TOSYLSULFILIMINES FROM CHLORAMINE T UNDER PTC CONDITIONSTamotsu Yamamoto; Daisaburo Yoshida
275-279A SIMPLE PREPARATION OF 1-ALKOXY-1-ALKYN-3-OLSWayne M. Stalick
279-284“ONE POT” FISCHER SYNTHESIS OF (2, 3, 3-TRIMETHYL-3-H-INDOL-5-YL)-ACETIC ACID. DERIVATIVES AS INTERMEDIATES FOR FLUORESCENT BIOLABELSPhilip L. Southwick; Jennifer G. Cairns; Lauren A. Ernst; Alan S. Waggoner
285-289SYNTHESIS OF 3- AND 4-CHLORO-1H-PYRROLO[3, 2-c]PYRIDIN-4(5H)-ONEG. Cristalli; P. Franchetti; M. Grifantini; E. Nasini; S. Vittori
289-292PREPARATION OF 2, 6-DIMETHYL-4-PHENYLPYRYLIUM SULFOACETATET. S. Balaban; A. Dinculescu; A. T. Balaban
293-295LARGE SCALE PREPARATION OF 1, 3-DIMETHYLADAMANTANEThomas J. Dooley; William Rowe
295-298A CONVENIENT SYNTHESIS OF 10, 10′-DIMETHYL-9, 9′-BIACRIDYLIDENEMarion R. Surgi; Julian Tirado-Rives
299-302AN IMPROVED SYNTHESIS OF ETHYL 4-HYDROXY-3-METHYLBENZOFURAN-2-CARBOXYLATEP. C. Bélanger; C. Dufresne; C. K. Lau; J. Scheigetz
302-305IODIDE SALTS OF NITROGEN HETEROCYCLES BY BROMIDE-IODIDE EXCHANGEIn-Sook Han Lee; Chang Kiu Lee; In Sup Han
305-311SYNTHESIS OF 3-METHYL- AND 3-tert-BUTYLPHENANTHRENER. C. Bansal; S. A. Samad; J. S. Thomson; E. J. Eisenbraun
311-316SYNTHESIS OF 2-[4-METHOXY-2-[2-(METHYLSULFINYL)ETHOXY]PHENYL]-1H-IMIDAZO[4, 5-b]PYRIDINE, A POTENT NONGLYCOSIDE INHIBITOR OF Na+, K+-ATPASEDavid W. Robertson; Joseph H. Krushinski

Volume 20, Issue 2 (1988)

CEditorial Board Page
105-108A NEW PROCEDURE FOR THE SELECTIVE α-OXYALKYLATION OF HETEROAROMATIC BASES BY CYCLIC ETHERS AND HYDROGEN PEROXIDEE. Vismara; F. Fontana; F. Minisci
109-115SYNTHESES OF N-CARBOXYMETHYL DIPEPTIDES via N-CARBOXY α-AMINO ACID ANHYDRIDES (NCA) INTERMEDIATESJerry W. Skiles; James D. Warus; John T. Suh
117-121HOMOLYTIC ALKYLATIONS OF 3, 6-DICHLOROPYRIDAZINEJack G. Samaritoni
123-128SYNTHESES OF OXYGENATED DERIVATIVES OF 3-METHYLCHOLANTHRENEHongmee Lee; Ronald G. Harvey
129-134A FACILE STEREOCONTROLLED SYNTHESIS OF 3-DEOXY-1, 2-0-ISOPROPYLIDENE-β-L-THREO-PENTOFURANOSE FROM DIACETONE GLUCOSERobert D. Walkup; Raymond T. Cunningham
135-143REGIOSELECTIVE FORMATION OF β-KETOAMIDES IN THE DIBENZOCYCLOOCTANE FAMILYJ. A. Moore; T. D. Mitchell
145-172NOVEL SYNTHETIC REACTIONS WITH 2-PYRIDYL RELATED REAGENTS. A REVIEWSunggak Kim
173-177PREPARATION OF 4-(CARBETHOXY)-5-ALKYL- AND 5-PHENYL FURAN-2-ACETIC ACIDS AND ITS METHYL ESTERSFrancisco Yuste; Hermila Vergel; Héctor Barrios; Benjamin Ortíz; RubéN Sánchez-obregón
177-180A SIMPLIFIED SYNTHESIS OF LOWER ALKYL BROMIDESR. Kozlowski; Z. Kubica; B. Rzeszotarska
180-184A CONVENIENT SYNTHESIS OF t-BUTYL ESTERS OF AMINO ACIDSG. Csanàdy; K. Medzihradszky
184-187A CONVENIENT SYNTHESIS OF β-KETO DIESTERSHans-Werner Schmidt; Manfred Klade
187-191SYNTHESIS OF METHYL trans-2-PHENYLCYCLOPROPANE CARBOXYLATESJames A. Beres; Robert David Crouch Jr.
191-195AN IMPROVED SYNTHESIS OF 1, 2-DEHYDRO-N-ACETYLDOPAMINEHemalata Dali; Manickam Sugumaran
196-198A SYNTHESIS OF 5, 10-DIANISYLPERHYDROPHENAZINEJeremiah P. Freeman; Jacob Szmuszkovicz

Volume 20, Issue 1 (1988)

CEditorial Board Page
1-51WHARTON FRAGMENTATIONS OF CYCLIC 1, 3-DIOL DERIVATIVES. A REVIEWDrury Caine
53-62SYNTHESIS OF THREE NEW ANALOGS OF DL-THYROXINEGeorge A. Brine; Karl G. Boldt; Michael L. Coleman
63-72SYNTHESES OF ω-ALKYNYL ALDEHYDES AND KETONES via OXIDATION OF ω-ALKYNYL ALCOHOLS WITH PYRIDINIUM DICHROMATEDonald E. Bierer; George W. Kabalka
73-82SYNTHESIS OF STEREOISOMERS 2-PHENYLIMINO-3, 1-PERHYDRO-BENZOXAZINES AND 3, 1-PERHYDROBENZOTHIAZINESFerenc Fülöp; Gábor Bernáth; György Csirinyi
83-86A FACILE METHOD FOR THE SYNTHESIS OF 1, 2, 3-TRIAROYLCYCLOPROPANES UNDER PHASE-TRANSFER CONDITIONSO. Bhaskar Reddy; V. M. Subramanyam; V. Padmavathi
87-91SYNTHESIS OF DIBENZOHEPTALENE BISLACTONES via A DOUBLE INTRAMOLECULAR CANNIZZARO REACTIONJ. A. Moore; Douglas R. Robello; Julius Rebek Jr.; R. Gadwood
93-95AN IMPROVED PROCEDURE FOR THE PREPARATION OF ETHYL α-CARBETHOXY-β-(ARYLAMINO)ACRYLATESA. K. S. Bhujanga Rao; Arakali S. Radhakrishna; C. Gundu Rao; Bajrang Bali Singh; Surendra P. Bhatnagar
96-99RACEMIZATION-FREE PREPARATION OF Boc-Tyr(Et)-OH ACTIVE ESTERSO. Nyéki; A. Rill; L. Klsfaludy
100-101AN IMPROVED METHOD FOR THE SELECTIVE HYDROLYSIS OF 1-ACETYL-5-BROMO-4-CHLOROINDOXYL ACETATE TO 1-ACETYL-5-BROMO-4-CHLOROINDOXYLJerry W. Misner
102-103A CONVENIENT PREPARATION OF 3-CARBETHOXY-2, 4-DIMETHYLQUINOLINE HYDROCHLORIDEL. A. M. Bastlaansen; J. A. M. v. Schijndel; H. M. Buck

Volume 19, Issue 6 (1987)

CEditorial Board Page
427-432SIMPLE PHASE-TRANSFER ALKYLATION OF O-(TETRAHYDROPYRAN-2-YL) ARYLALDEHYDE CYANOHYDRINSHéctor Barrios; Consuelo Sandoval; Benjamín Ortíz; Rubén Sánchez-Obregón; Francisco Yuste
433-435S-ALKYLATION OF THIOACRIDONE DERIVATIVES USING SOLID-LIQUID PHASE TRANSFER CATALYSIS WITHOUT SOLVENTMircea Vlassa; Maria Kezdi
435-438SYNTHESIS OF γ, δ-UNSATURATED KETONESThomas C. McKenzie
439-442SYNTHESIS OF R,S-2-(3-BENZO[b]THIENYL)GLYCINE USING IMPROVED AMIDOALKYLATION METHODOLOGYJ. P. Gardner; B. G. Jackson
442-446REDUCTIVE DEHALOGENATION OF HALOACETOPHENONES WITH RANEY ALLOYS IN ALKALINE SOLUTIONMasashi Tashiro; Hiroshi Nakamura; Kouji Nakayama
447-449INTRA- AND INTERMOLECULAR ACYLATION OF 2-BENZYLSUCCINIC AND 2-BENZYLGLUTARIC ANHYDRIDESIwao Hashimoto; Masashi Tashiro
450-455SYNTHESIS OF NEW HETEROCYCLOCOUMARINS FROM 3,4-DIAMINO- AND 4-CHLORO-3-NITROCOUMARINSM. Trkovnik; V. Kalaj; D. Kitan
455-457α,α-DIBROMODESOXYBENZOIN FROM THE REACTION OF THIONYL BROMIDE WITH BENZOINS. D. Saraf; Fatima Al-Omran
457-461A SIMPLE PREPARATION OF 4-SUBSTITUTED-6,7-DIMETHOXYISOQUINOLINESC. S. Giam; Swee Yong Lee; Deborah L. Ambrozich
461-465A SHORT AND CONVENIENT SYNTHESIS OF 12-OXO-E-10-DODECENOIC ACID (TRAUMATIN)Bruce J. Gaede
466-467A CONVENIENT PROCEDURE FOR THE PREPARATION OF TRIETHYLAMINE-SULFUR TRIOXIDEVijay Nair; Seymour Bernstein
468-470A CONVENIENT SYNTHESIS OF DIFLUOROACETIC ACIDM. Cecilia Luz; William P. Dailey
471-475MICHAEL REACTION OF NITROMETHANE WITH β,β-DISUBSTITUTED ACRYLATE ESTERSRichard A. Bunce; Raymond E. Drumright
477-486INDEXES

Volume 19, Issue 4-5 (1987)

CEditorial Board Page
263-268A NEW SYNTHETIC METHOD FOR ortho-SUBSTITUTED BENZANILIDESAlan R. Katritzky; Wei-Qiang Fan
269-276SYNTHESIS OF 6,7,12-TRIMETHYLBENZ[a]ANTHRACENE 6,7-, AND 6,12-DIHETHYLBENZ[a]ANTHRACENEGuido H. Daub; Lorraine M. Deck; Alberto A. Leon
277-282AN IMPROVED SYNTHESIS OF 2-METHYLBENZ[a]ANTHRACENELorraine M. Deck; Guido H. Daub; Alberto A. Leon
283-328SYNTHESES AND SELECTED REDUCTIONS OF CONJUGATED NITROALKENES. A REVIEWGeorge W. Kabalka; Rajender S. Varma
329-426α-HALONITROSO COMPOUNDS. A REVIEWGünter Kresze; Bernhard Ascherl; Heinz Braun; Helena Felber

Volume 19, Issue 2-3 (1987)

CEditorial Board Page
83-159RECENT SYNTHETIC APPLICATIONS OF N-NITROSAMINES AND RELATED COMPOUNDSJoseph E. Saavedra
161-166FORMATE ESTERS BY CANNIZZARO-TISHCHENKO REACTION OF GRIGNARD AND SODIUM ALKOXIDES WITH FORMALDEHYDERichard A. Bunce; A. Joe Shellhammer Jr.
167-172A NEW AND CONVENIENT SYNTHESIS OF 4-AMINO-3-NITROBENZOPHENONE AND 2-AMINO-5-NITROBENZOPHENONE AND THEIR N-ALKYL DERIVATIVESN. R. Ayyangar; R. J. Lahoti; K. V. Srinivasan; Thomas Daniel
173-180REGIOSELECTIVE DEOXYGENATION OF CHLORAMPHENICOL AND OF (1R,2R)-(+)-2-AMINO-1-PHENYL-1,3-PROPANEDIOLP. Ramaiah; A. S. Rao
181-186SYNTHESIS OF DIIMINES FROM 1,2-DICARBONYL COMPOUNDS BY DIRECT CATALYZED CONDENSATIOND. Armesto; P. Bosch; M. G. Gallego; J. F. Martin; M. J. Ortiz; R. Perez-Ossorio; A. Ramos
187-195PREPARATION OF THE 9-cis, 13-cos-. AND ALL trans-ISOMERS OF α- AND β2-RETINALMichael F. Vaezi; Cynthia Y. Robinson; Kenneth D. Hope; Wayne J. Brouillette; Donald D. Muccio
197-208SYNTHESIS OF BIOLOGICAL MARKERS IN FOSSIL FUELS 5. A SYNTHESIS OF 5α-CHOLAN-24-OIC ACIDAyhan S. Demir; Mark R. Sabol; Alwarsamy Jeganathan; Eric Kurt Dolence; David S. Watt; J. Michael Moldowan
209-214A CONVENIENT SYNTHESIS OF (dl)-1-AMINO-4-CARBOXYCYCLOHEXANE-1-13C-CARBOXYLIC ACIDN. Dale Ledford; Cathy R. Cutcliff; H. Blair Wood Jr.; Michael Barfield
215-248RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF TETRAZINES. A BRIEF REVIEWMichael J. Hearn; Fiona Levy
249-250A SIMPLE PREPARATION OF 6-CHLORO-5, 8-QUINOLINEDIONEArthur Haber
251-252ONE-STEP PREPARATION OF 4-BROMOMETHYL-2,3,5,6-TETRABROMOPHENOLWenjeng Guo; George Wu
252-255[2-CARBOXY-2′-CHLORO-4,4′, 5.5′-TETRA(BENZYLOXY)] AZOBENZENE FROM THE BENZYNE DECOMPOSITION OF 2-CARBOXY-4, 5-DIBENZYLOXYBENZENEDIAZONIUM CHLORIDEFrank W. Muellner; Ashraf N. Abdel-Sayed; Ludwig Bauer; James N. Shoolery
255-257THREE NEW PRODUCTS FROM METHYL 3,4-DIPHENYL-5-NITRO-2-FUROATE BY CATALYTIC REDDCTIONK. Yamamoto; A. Tanaka; M. Ichikawa; S. Swaminathan; G. T. Bryan
258-260THE IODINATION OF FLUORENE TO 2,7-DIIODOFLUORENER. C. Bansal; E. J. Eisenbraun; R. J. Ryba
261OPPI-CORRIGENDUM

Volume 19, Issue 1 (1987)

CEditorial Board Page
1-7SELECTIVE REDUCTION OF THE FORMYLATED BILE ACIDS TO THE CORRESPONDING FORMYLATED BILE ALCOHOLS ANALOGSA. A. Malik; C. M. Sharts
9-16SYNTHESIS OF MEBENDAZOLE AND ENVIROXIME. ACYLATION OF 2-AMINO-5-BENZOYLBENZIMIDAZOLET. Ravindranathan; R. D. Wakharkar; A. B. Landge
17-24THE PREPARATION OF SOME DIIMINESPaul Sulmon; Norbert De Kimpe; Niceas Schamp
25-38SYNTHESIS OF β, β-DISUBSTITUTED ACYCLIC α-ENONES WITH AN ASYMMETRIC CARBONC. Alvarez Ibarra; M. S. Arias Pérez; J. M. Esteban; E. Moya
39-44AN IMPROVED SYNTHESIS OF 1,3-BIS(5-t-BUTYL-2-SUBSTITUTED PHENYL)PROPANESTakehiko Yamato; Akihiko Tsuge; Keizo Koya; Kazumasa Kobayashi; Hiroshi Sakamoto; Masashi Tashiro
44-48A SIMPLE SYNTHESIS OF 3-(1-PYRROLYL) FLAVONOIDSGyörgy Litkei; Tamas Patonay; Erzsobet Peli
48-52AN IMPROVED PREPARATION OF 1,2,5-TRIMETHYL-3-NITROPYRROLE. FRIEDEL-CRAFTS ACYLATION WITH 2-FLUOROBENZOYL CHLORIDEM. R. Pavia
52-56A SIMPLE SYNTHESIS OF SOME NOVEL OXIME ETHERSYunus Akcamur; Gert Kollenz
57-60AN IMPROVED SYNTHESIS OF 1,4-BIS(2′-METHYL-6′-KIHYLANILINO)ANTHRAQUINONEF. Ivy Carroll; John F. Sherrill; Dale E. Stelz; Wilson M. Whaley
61-63AN EFFICIENT SYNTHESIS OF 2-(3,4-DIMETHOXYPHENYL) SUCCINIMIDEFrancesco Claudi; Ugo Gulini; Vincenzo Perlini
64-66AN IMPROVED SYNTHESIS OF γ-L-GLUTAMYL-TAURINEJ. Gulyas; F. Sebestyen; J. Hercsel-Szepespataky; A. Furka
67-71AN IMPROVED SYNTHESIS OF DIMETHYL (E)-5-METHOXYCARBONYL-2-ENEDIOATE AND DIMETHYL (E)-6-METHOXYCARBONYL-2-ENEDIOATERichard A. Bunce; Joey D. Pierce
71-74DIIMIDE REDUCTION OF SUBSTITUTED STYRENES AND OF PHENYL-1,3-BUTADIENESTakeshi Negoro; Yoshitsugu Ikeda
75-78SYNTHESIS OF N,O-DIMETHYLHYDROXYLAMINE HYDROCHLORIDEO. P. Goel; U. Krolls
78-80A CONVENIENT SYNTHESIS OF t-BUTYL N-(2-BROMOETHYL)CARBAMATEV. G. Beylin; O. P. Goel
80-82CHLORINATION OF PYRIDAZINONES WITH CHLOROCARBONYL ISOCYANATET. N. Srinivasan; K. Rama Rao; P. B. Sattur

Volume 18, Issue 6 (1986)

CEditorial Board Page
369-427SELENIUM AND TELLURIUM ISOLOGUES OF CARBOXYLIC ACID DERIVATIVESShinzi Kato; Toshiaki Murai; Masaru Ishida
429-439INDEXES

Volume 18, Issue 5 (1986)

CEditorial Board Page
iANNOUNCEMENTS
iiNOTICE
299-327CONJUGATED AZOALKENES: ATTRACTIVE PRODUCTS AND VERSATILE INTERMEDIATESOrazio A. Attanasi; Luciano Caglioti
329-343SYNTHESIS OF 3-SELENA-7-AZABICYCLO[3.3.1]NONANES AND CERTAIN DERIVATIVESM. Daniel Thompson; Gary S. Smith; K. Darrell Berlin
345-352SELECTIVE PROTECTION OF THE SIDE CHAIN HYDROXY GROUP IN BILE ALCOHOL DERIVATIVESA. A. Malik; R. J. Cormier; C. M. Sharts
353-360SYNTHESIS AND SINGLE CRYSTAL X-RAY DIFFRACTION CHARACTERIZATION OF [2-AMINO-N-(2,6-DIMETHYLPHENYL)-ACETAMIDATO-N2] DICHLOROETHYLSELENIUM, A SELENIUM-CONTAINING LIDOCAINE MIMICM. Daniel Thompson; K. Darrell Berlin; Gary S. Smith; Dick van der Helm; Steve W. Muchmore; Krzysztof A. Fidelis
361-363IMPROVED HIGH-YIELD CONVERSION OF DINITROMESITYLENE TO NITROMESIDINERajan Ramaswami; A. G. Pinkus
363-3681,2-DINITROCYCLOHEXENEJoseph H. Boyer; Philip F. Pagoria

Volume 18, Issue 4 (1986)

CEditorial Board Page
219-226α,β-UNSATURATED ALDEHYDES BY ONE-STEP VINYLOGATION OF CARBONYL COMPOUNDSLucette Duhamel; Gérard Plé; Béatriz Contréras
227-236SYNTHESIS OF OXYGEN HETEROCYCLES FROM 2-ARYLIDENE-1,3-D1 KETONESJ. A. Ciller; N. Martín; M. Quinteiro; C. Seoane; J. L. Soto
237-244SYNTHESIS AND OPTICAL RESOLUTION OF 1-(1-NAPHTHYL)-2-DIMETHYLAMINOETHANOLLeroy H. Klemm; Jennifer J. Lu
245-252REACTION OF 2,7-DI-t-BUTYL-2,4,5,7,9,10-HEXACHLORO-trans-10b,10c-DIMETHYL-2,7,10b,10c-TETRAHYDROPYRENE WITH ALCOHOLS AND WATER AND THE CHEMISTRY OF THE PRODUCTS OBTAINEDTakehiko Yamato; Kazumasa Kobayashi; Masashi Tashiro
253-262SYNTHESIS OF ANTIFUNGAL ISOCOUMARINSH. Kaji; M. Yamada; K. Nozawa; K. Kawai; S. Nakajima
263-268A CONVENIENT SYNTHESIS OF (d1)-o-CARBOXY13C-PHENYLALANINEN. Dale Ledford; Pamala C. Gibbs; H. Blair Wood Jr.; Michael Barfield
269-272A FACILE SYNTHESIS OF N-CHLORO FATTY AMIDESW. A. Henderson Jr.; L. W. Chang
272-275SYNTHESIS OF 1,3,4-THIADIAZOLYL UREASE. V. P. Tao; Stanislaw Rolski
275-2781-METHYL-4-NITRO-5-IMIDAZOLYL SULFONESNed D. Heindel; C. Jeffrey Lacey; Belle A. Mease; David V. Woo
278-281A CONVENIENT SYNTHESIS OF PYRROLE-3-CARBOXALDEHYDEVassilis J. Demopoulos
281-283DIRECT PREPARATION OF 1,3,5-TRIAZA-1,3,5-TRINITROCYCLOHEXANE FROM HEXAMETHYLENETETRAMINEJohn W. Fischer; Ronald L. Atkins
283-285A FACILE AND EFFICIENT SYNTHESIS OF PYRROLE-3-CARBOXYLIC ACID FROM PYRROLECarlos Cativiela; Jose I. Garcia
286-289SYNTHESIS OF 3-CARBOXYTHIOPHENE-2-ACETIC ACID AND ITS DERIVATIVESReinhold Bender; Dimitri Sarantakis
290-295AN IMPROVED SYNTHESIS OF TRIBENZO[a,cd,1m]PERYLENEJ. C. Fetzer; W. R. Biggs
295-2973-METHYLSUCCINIMIDE AND 3-METHYLPYRROLIDINER. S. Budhram; N. Pourahmady; A. -S. Syed; E. J. Eisenbraun

Volume 18, Issue 3 (1986)

CEditorial Board Page
145-148A FACILE SYNTHESIS OF 3-BENZYLOXY-5-METHOXYPHENOLRubén Sánchez-Obregón; Gerardo Hurtado; Héctor Barrios; Benjamín Ortíz; Francisco Yuste
149-155AN IMPROVED PREPARATION OF m- AND p-TETRAMETHYLXYLYLENEDIISOCYANATESWm. A. Henderson Jr.; Vazken A. Alexanian
157-178SYNTHESIS AND REACTIONS OF β-SULTAMS. A REVIEWJosette Chanet-Ray; Roger Vessiere
179-201THE OXIDATION OF ELECTRON DONORS WITH SULFONYL PEROXIDESRobert V. Hoffman
203-205SYNTHESIS OF PHENACYL ESTERS via POLYMER SUPPORTED REAGENTSM. Thorat; R. Mane; M. Jagdale; M. Salunkhe
206-209PREPARATION OF METHYL a-ALKYL FUMARATESMichael Dymicky
209-212A SELECTIVE SYNTHESIS OF 5-p-AMINOPHENYLBARBITURIC ACIDFrank V. Bright; Richard A. Bunce; Linda B. McGown
213-215A CONVENIENT SYNTHESIS OF 5-TRIFLUOROMETHYLSALICYLIC ACIDJose Alexander
217CORRIGENDUM

Volume 18, Issue 2 (1986)

CEditorial Board Page
79-84β-IODOTRIMETHYLSILYLENOL ETHERS AND α-IODOALDEHYDES AND KETONES FROM α-CHLORO AND α-BROMOCARBONYL COMPOUNDSJean-Marie Poirier
85-93HYDROXYCYCLOHEXANONES FROM THE REACTION OF α-BENZOYLCINNAMONITRILES WITH ETHYL ACETOACETATE. A LITERATURE CORRECTIONM. Quinteiro; J. Chicharro; N. Martin; J. A. Cillar; C. Seoane; J. L. Soto
95-98PREPARATION OF 2-CHLORO- AND 2-AMINO-5-BENZOYLBENZIMIDAZOLEST. Ravindranathan; R. D. Wakharkar; A. B. Landge
99-103A MODIFIED SYNTHESIS OF AMINOBICYCLO[n.1.0]ALKANES FROM ENAMINOSULFONIUM SALTSJürgen Maischein; Christine Roth; Elmar Vilsmaier
104-108PHOTOHALOGENATION OF LAWSONE AND PREPARATION OF 3-SUBSTITUTED 5H-NAPHTHO-[2,3-e]-s-TRIAZOLO[3,4-b][1,3,4]THIADIAZINE-6,11-DIONEM. S. Rao; V. Rajeswar Rao; T. V. Padmanabha Rao
109-112ETHYL 3-CHLORO-2-ETHOXY-5-FORMYL-6-HYDROXY-4-METHYLBENZOATEKau-Ming Chen; Madeleine M. Joullié
113-116A CONVENIENT SYNTHESIS OF DIBENZOBARRELENEPeter W. Rabideau
117-144THE CHEMISTRY OF METHANETRICARBOXYLIC ESTERS. A REVIEWGeorge R. Newkome; Gregory R. Baker

Volume 18, Issue 1 (1986)

CEditorial Board Page
iANNOUNCEMENT
1-5EFFECT OF METAL IONS IN ORGANIC SYNTHESIS. PART XXVIII SYNTHESIS OF NEW 1-AROYLAMINO-3-AMINOCARBONYLPYRROLESOrazio Attanasi; Mario Grossi; Franco Serra-Zanetti
7-10A SYNTHETIC APPROACH TO THE AB-RING SYSTEM OF FORSKOLINYashwant S. Kulkarni; Barry B. Snider
11-12A CONVENIENT REGIOSPECIFIC AND STEREOSELECTIVE SYNTHESIS OF [2,4-2H2]METHYL-trans-4-OXO-2-BUTENOATEM. Saljoughian
13-15SYNTHESIS OF t-BUTYL ESTER OF 7-AMINOCEPHALOSPORANIC ACIDAlberto Mangia; Angelo Scandroglio; Paola Del Buttero
17-78SYNTHETIC APPROACHES TO BINAPHTHALENES. A REVIEWMiha Tišler

Volume 17, Issue 6 (1985)

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385-390CONJUGATED AZOALKENES. PART I SYNTHESIS OF SOME AROYLAZOALKENESOrazio Attanasi; Mario Grossi; Franco Serra-Zanetti
391-3995-SUBSTITUTED INDOLES via SODIUM INDOLINE-2-SULFONATE. A REEXAMINATIONHenry F. Russell; Brenda J. Harris; Darryl B. Hood; Errol G. Thompson; Aldriche D. Watkins; Robin D. Williams
401-407SYNTHESIS OF erithro-α-METHYLEPINEPHRINE HYDROCHLORIDEHoward E. Smith; Jon R. Neergaard; David Robertson
409-410A CONVENIENT SYNTHESIS OP 4-HTDROXY-3-NITROPYBIDINEDanuta Rasala; Ryszard Gawinecki
410-415A CLEAN AND REPRODUCIBLE SYNTHESIS OF 1-BROMO-2-ETHOIYETBANEWayne M. Stalick; Ali Khorrami
416-419IMPROVED SYNTHESIS OF SOME o-BSTERS OF N-PKOTECTED L-GLUTAMIC ACIDK. Pawelczak; L. Krzyzanowski; B. Rzeszotarska
419-422SYNTHESIS OP 8-HrDROXY-1-NAPHTHALDEHYDECarl A. Elliger
422-423OXIDATION OF 2,3DICHLOSO-5,6-DICYANOHYDROQUINONE TO 2,3-DICHLORO-5,6-DICYANOBENZOQUINONEMelvin S. Newman; Vinod K. Khanna
425-436INDEXES

Volume 17, Issue 4-5 (1985)

CEditorial Board Page
239-249APPLICATION OF SPIN LABELING TO DRUG ASSAYS. IV. SPIN- AND RADIOLABELED LIDOCAINEYul Yost; Jordan L. Holtzman
251-253A NEW CERIUM(III)-CATALYSED ROUTE TO CINNAMYL ALCOHOLSK. V. Lakshmy; P. G. Mehta; J. P. Sheth; G. K. Trivedi
254-256A CONVENIENT ONE-POT PREPARATION OF N-SUBSTITUTED HYDROXYLAMINESRajender S. Varma; George W. Kabalka
256-261THE SYNTHESIS OF SOME GUANIDINE DERIVATIVESJ. Zmitek; B. Jenko; A. Kosak; D. Milivojevic
261-264SYNTHESIS OF DIBENZHYDRYLNITROSAMINEJack E. Baldwin; Stephen E. Branz
264-267PREPARATION OF THE PALMITATES OF KAHWEOL AND CAFESTOLLuke K. T. Lam; L. W. Wattenberg
267-270SYNTHESIS OF 3,4-DIPHENYL-1,2,3,4-TETRAHYDROISOQUINOLINESNaseem Peerzada
270-274A MODIFIED PROCEDURE FOR THE PREPARATION OF 5H, 7H-DIBENZO[c,e]SELENEPINDaniel J. Williams; Patrick K. Macy; David R. Hezs
275-315REACTIONS OF THIOCARBONYL COMPOUNDS WITH CHLORINE AND WITH SULFUR DICHLORIDES. A REVIEWHolger C. Hansen; Alexander Senning
317-384SODIUM BOROHYDRIDE IN CARBOXYLIC ACID MEDIA. A REVIEW OF THE SYNTHETIC UTILITY OF ACYLOXYBOROHYDRIDESGordon W. Gribble; Charles F. Nutaitis

Volume 17, Issue 3 (1985)

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155-162REDUCTIVE CLEAVAGE OF N-NITROSOOXAZOLIDINES TO AMINES WITH Al-Ni ALLOY. REDUCTION TO SECONDARY N-ALKYLALKANOLAMINESJoseph E. Saavedra
163-167SYNTHESIS OF 3-MERCAPTOTHIOPHENE-2-AND 4-CARBOXYLIC ACIDSC. Corral; J. Lissavetzky; A. S. Alvarez-Insúa; A. M. Valdeolmillos
169-173AN IMPROVED SYNTHESIS OF 5,5,9,9-TETRAMETHYL-5H, 9H-QUINO[3,2,1-DE]ACRIDINEJohn L. Fox; Chin H. Chen; John F. Stenberg
175-181AN EFFICIENT SYNTHESIS OF D,L-CARNITINE HYDROCHLORIDE via THE ACYLATION OF AN α-AMINOKETONERobert N. Comber; Wayne J. Brouillette
183-186A MODIFIED STRECKER SYNTHESISKhuong Mai; Ghanshyam Patil
187-190A FACILE SYNTHESIS OF 6,7-DIHYDRO-5H-DIBENZO[a,c]CYCLOHEPTENEG. William Griffin; Keith A. Horn
190-192ORGANIC SONOCHEMISTRY. A FACILE SYNTHESIS OF 1-METHYLISOQUINOLINEJ. Ezquerra; J. Alvarez-Builla
192-194STEROIDAL ALLYLIC OXIDATION WITH CHROMIUM TRIOXIDE IN THE PRESENCE OF PYRAZOLEEdward J. Parish; Sarawanee Chitrakorn; Kenneth L. Todd III
195-198A NEW SYNTHESIS OF 2-BROMO-1-(9-PHENANTHRYL)ETHANEMagid Abou-Gharbia; Bruce R. Hoffman
198-203SYNTHESIS OF SOME 2-PYRAZOLIN-5-ONE DERIVATIVES STRUCTURALLY RELATED TO CERTAIN ANALGESIS AND ANTIPYRETIC DRUGSM. A. Metwally; A. A. Fadda; H. M. Hassan; E. Afsah
203-205OXIDATION OF FURFURALDEHYDES WITH SODIUM CHLORITEJ. A. Moore; Emmett M. Partain III
206-210SYNTHESIS OF THIADIAZINE AND ARYLMETHINEAZOTHIAZOLONE DERIVATIVES OF COUMARINR. Djudjic; M. Trkovnik; D. Kitan
210-212AN EFFICIENT SYNTHESIS OF N-(2,4-DIFLUOROPHENYL)-N-METHYL-2,4-DINITRO-6-(TRIFLUOROMETHYL)ANILINEE. V. P. Tao; H. A. Corbitt
212-214A CONVENIENT, TWO-STEP SYNTHESIS OF BICYCLO[3,3,0]OCT-1(5)-ENEPaul J. Okarma; Joseph J. Caringi
215-218AN IMPROVED SYNTHESIS OF METHYL [5-BENZOYL- AND 5-p-FLUOROBENZOYLBENZIMIDAZOL-2-YL]CARBAMATESSiya Ram; Dean S. Wise; Leroy B. Townsend
219-223REACTIVE ALUMINUM POWDERS FOR THE REDUCTION OF HALOARENES. APPLICATION OF THE “PLANNING OF EXPERIMENTS” METHOD FOR THE OPTIMISATION OF OBTAINING REACTIVE METAL POWDERA. Akagah; J. -C. Poite; M. Chanon
223-227A CONVENIENT PREPARATION OF 9-DIMETHYLAMINO-10-CARBOMETHOXYANTHRACENEAndrew T. Brown; Geoffrey Hallas
227-230MILD SELECTIVE OXIDATION OF SULFIDES TO SULFONESSuzanne T. Purrington; Anne G. Glenn
230-235INDIRECT IODINATION WITH 2-(3,5-DIIODO-4-METHOXYPHENYL)-1,3,4-OXADIAZOLE AS A PRECURSOR OF AN AROYL HYDRAZINENed D. Heindel; Marcian Van Dort
235-238A CONVENIENT SYNTHESIS OF N-5-(1,1-DIMETHYLETHYL)-3-ISOXAZOLYL-N,N-DIMETHYLUREAE. V. P. Tao; G. S. Staten

Volume 17, Issue 2 (1985)

CEditorial Board Page
83-89SYNTHESIS OF N-(p-CARBOBENZOXYAMINOBENZOYL)-L-GLUTAMIC ACID α-BENZYL ESTERLeszek Krzyzanowski; Barbara Rzeszotarska
91-97AN IMPROVED PREPARATION OF (±) 3-HYDROXY-2-PYRROLIDINONEO. P. Goel; U. Krolls; E. P. Lewis
99-105PREPARATION OF β-BROMOTRIMETHYLSILOXYENOLETHERS FROM α-BROMOCARBONYL COMPOUNDSLucette Duhamel; Francis Tombret; Jean-Marie Poirier
107-114ACTIVATED NITRILES IN HETEROCYCLIC SYNTHESIS. NOVEL SYNTHESES OF PYRIMIDINES AND PYRIDINESN. M. Abed; N. S. Ibrahim; S. M. Fahmy; M. H. Elnagdi
115-120PREPARATION OF 6-SUBSTITUTED-6H-7-AZA-INDENO[1,2-c] ISOQUINOLINE-5, 11-DIONESS. Wawzonek; M. C. Chen
121-131PREPARATION OF n-MONOALKYL MALEATES AND n-MONO- AND DIALKYL FUMARATESMichael Dymicky; Robert L. Buchanan
133-137CHEMISTRY OF COUMARINS. ANNELATION OP COUMARIN SING via REACTIONS OF 3-AMINO-4-HYDROXYCOUMARINI. Tabakovic; K. Tabakovic; M. Trkovnik; Z. Stunic
138-1401,2,3,4-TETRAHYDRO-1,4,d2-NAPHTHALENE-1,4.5,6,7.8.-d6Mark H. Gaston; Duane R. Skidmore
140-142ONE-POT SYNTHESIS OF NITROSTYRENE OXIDESKarim Rafizadeh; Keith Yates
143-146LOW TEMPERATURE OZONOLYSIS OF METHYL O-METHYL PODOCARPATEEdward J. Parish; Garvis G. McKeen; D. Howard Miles
146-151SYNTHESIS AND ELECTROPHILIC SUBSTITUTION REACTIONS OF FLUORINE CONTAINING ARYLGLYOXAL 2-ARYLHYDRAZONESKrishna C. Joshi; Vijai N. Pathak; Sharda Sharma
152-1543-ARYL-1,2,5-THIADIAZOLES FROM THE REACTION OF TETRASULFUR TETRANITRIDE WITH ARYL METHYL KETONESShuntaro Mataka; Kazufumi Takahashi; Masashi Tashiro

Volume 17, Issue 1 (1985)

CEditorial Board Page
1-9EFFICIENT PREPARATION OF THE CHIRAL AUXILIARIES SAMP and RAMP. N-AMINATION via HOFMANN DEGRADATIOND. Enders; P. Fey; H. Kipphardt
11-16REACTIONS OF SODIUM BOROHYDRIDE IN ACIDIC MEDIA. XIV. REDUCTIVE CLEAVAGE OF CYCLIC ACETALS AND KETALS TO HYDROXYALKYL ETHERSCharles F. Nutaitis; Gordon W. Gribble
17-22SYNTHESIS OF CARBON-13 LABELLED DIALKYLCARBINOLS AND DIALKYLKETONESGeorge W. Kabalka; Mohammad Mohammadi; Sastry A. Kunda; Ronald D. Finn
23-47RECENT SYNTHETIC APPLICATIONS OF NITRONES. A REVIEWN. Balasubramanian
49-52A NEW TYPE OF α-N-AMIDOALKYLATION OF HETEROAROMATIC BASES. MECHANISM OF THE OXIDATION OF THE N-ACYLAMINOETBANOLS BY PEROXYDISULFATEC. Giordano; F. Minisci; V. Tortelli; E. Vismara
53-56A SYNTHESIS OF ACEANTHRYLENER. Sangaiah; A. Gold
56-60SELECTIVE HALOGENATION OF FLAVONOLS BY HYDROHALOGENIC ACIDS IN OXIDATION SYSTEMMasataka Ichikawa; Satoshi Hibino; Mizuo Onishi; James F. Hatcher; A. Mahir Pamukcu; George T. Bryan
60-62AN IMPROVED SYNTHESIS OF WINTERS' PYRIDINE REISSERT ANALOGJohn V. Cooney; George W. Mushrush; Robert N. Hazlett
62-64ONE-STEP PREPARATIONS OF ISOMERIC (2,6-DIOXACYCLOHEXYL)PHENOLSJulian Tirado-Rives; Richard O. Gandour
65-67HOFFMAN REACTION OF 1-PHENYLNAPHTHALENE-2,3-DICARBOXIMIDES. Wawzonek; M. C. Chen
68-70NEW HALO ACETAMIDO AND BENZAMIDOMETHYLPYRIDINESFrank L. Setliff
70-75ACTIVATED NITRILES IN HETEROCYCLIC SYNTHESIS. NOVEL SYNTHESIS OF PYRAZOLES, PYRIDONES AND PYRROLO[2.3-b]PYRIDONESE. M. Zayed; A. A. A. Elbannany; S. A. S. Ghozlan
75-80SYNTHESIS OF 2-ALKOXY-5-NITROBENZAMIDES BY PHASE-TRANSFER CATALYZED NUCLEOPHILIC SUBSTITUTION OF 2-CHLORO-5-NITROBENZAMIDESD. Nisato; R. Sacilotto; M. Frigerio; S. Boveri; G. Boccardi; G. Palmisano; G. Lesma
80-82A PREPARATIVE AVICEL-CELITE TLCNobutaka Suzuki; Toshio Goto

Volume 16, Issue 6 (1984)

CEditorial Board Page
393-400PREPARATION OF SUBSTITUTED 1, 6-DIAMINO-2-OXOPYRIDINESCarlos Seoane; José L. Soto; Pilar Zamorano
401-405O-ALKYL-N-ARYLHYDROXYLAMINES N-ALKOXY-2,4,6-TRI- AND -2,6-DINITROANILINESGabriela Stanciuc; Alexandra T. Balaban
407-4102,4,6-TRIPHENTLPYRYLIUM HYDROGEN SULFATEAntonie Dinculescu; Alexandra T. Balaban
411-425AN IMPROVED MEDIUM-SCALE PREPARATION OF DIBENZO[a, e] CYCLOOCTEN-5(6h), 11(12h)DIONEJ. A. Moore; T. D. Mitchell
427-437INDEXES

Volume 16, Issue 5 (1984)

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299-307IMPROVED SYNTHESIS OF POLYAZOLYLMETHANES UNDER SOLID-LIQUID PHASE-TRANSFER CATALYSISSebastián Juliá; José Ma del Mazo; Luis Avila; José Elguero
309-314STUDIES IN THE SYNTHESIS OF HALOGENATED ANTHRAQUINONES. II. A FACILE PREPARATION, OF 1,4-DICHLORO-5,6,8-TRIHYDROXY-9,10-ANTHRACENEDIONE (5,8-DICHLOROPURPURIN)H. D. Hollls Showalter; Jeanne M. Hoftiezer
315-319A SIMPLE PROCEDURE FOR THE CYCLIZATION OF 2′-HYDROXYCHALCONES INTO FLAVANONESTamas Patonay; György Litkei; Miklós Zsuga; Anikó Kiss
321-328A CONVENIENT SYNTHESIS OF ISOMERICALLY PURE 1-METHYL-2-VINYLCYCLOHEXENE AND 1-VINYLCYCLOHEXENEGeorge W. Kabalka; Mohammad Mohammadi; Mark Hylarides; Ronald D. Finn
329-333IMPROVED PREPARATION OF 2-CHLORO-6-METHYLANTHRAQUINONE, A PRECURSOR FOR THE CORRESPONDING 6-CARBOXYLIC ACID ESTERS AND 2-CHLORO-6,9,10-TRIMETHYLANTHRACENEV. S. Prabhu; John F. W. Keana
335-372AMINE BORANES AS SELECTIVE REDUCING AND HYDROBORATING AGENTS. A REVIEWRobert O. Hutchins; Keith Learn; Behrooz Nazer; David Pytlewski; Andrew Pelter
373-376METHYL 2-(5-ISOPROPYL-3-ISOXAZOLYL) BENZOATERobert K. Howe; Becky R. Shelton
376-379CHLORINATION OF 5,13-DI-t-BUTYL-8,16-DIMETHYL[2.2]METACYCLOPHANEMasashi Tashiro; Takehiko Yamato
379-383PREPARATION OF HROMOBENZOIC ACIDS FROM THE CORRESPONDING BROMOTOLUENES VIA THE KROHNKE METHODMasashi Tashiro; Kouji Nakayama
384-387AN IMPROVED SYNTHESIS OF METHIL- AND BENZYL-ESTERS AS WELL AS HYDRAZIDE OF L-PYOGLUTAMYL-L-HISTIDYL-L-TRYPTOPHANB. Rzeszotarska; E. Masiukiewicz
388-391PARTIAL DEPROTECTION OF 1.2.5.6-DI-O-ISOPROPYLIDENE-D-GLUCOFURANOSESRatnasamy Somanathan; Lars H. Hellberg

Volume 16, Issue 3-4 (1984)

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xix-xlviUNITED STATES DISTRICT COURT DISTRICT OF MASSACHUSETTS
149-153SYNTHESIS OF (±)-EREMOFRULLANOLIDEP. A. Zoretic; R. J. Chambers; C. Bhakta
155-164A PREPARATIVE ROUTE TO ALKOXYPHENOLS USING t-BUTYL FUNCTION AS A POSITIONAL PROTECTIVE GROUPMasashi Tashiro; Takashi Itoh; Haruo Yoshiya; Gouki Fukata
165-169D-α-AMINOADIPIC ACID FROM CEPHALOSPORIN CConstantine Sklavounos
171-198REDUCTION OF SULFOXIDES. A REVIEWJ. Drabowicz; H. Togo; M. Mikołajczyk; S. Oae
199-277RECENT PROGRESS IN THE SYNTHESIS AND REACTIONS OF 1,2,3- AND 1,2,4-TRIAZINESMichael J. Hearn; Fiona Levy
279-285SYNTHESIS OF 6-SUBSTITUTED 3-DEUTEROBENZO[A]PYRENEP. P. Fu; M. W. Chou; L. E. Unruh; J. P. Freeman; D. W. Miller; F. E. Evans; R. Roth
286-289A FACILE SYNTHESIS OF N-BENZOYLBENZIMIDAZOLES BY PHASE-TRANSFER CATALYSIST. J. Dennis; K. Akshaya Kumar; G. Srimannarayana
289-291SYNTHESIS OF 2-NITROCYCLOOCTANONERoberto Ballini; Pietro Sorrenti
292-294A VERY MILD AND EFFICIENT PREPARATION OF δ-VALEROLACTONEAndré Loupy; Farchid Vaziri-Zand
294-297AN IMPROVED SYNTHESIS OF β-TETRALONEDavid C. Hunden

Volume 16, Issue 2 (1984)

CEditorial Board Page
79-83THIOCARBONYL-ACTIVATED TRANSAMINATION. A FACILE SYNTHESIS OF N4-MONO AND N4,N4-DISUBSTITUTED THIOSEMICARBAZONESDaniel L. Klayman; Ai J. Lin
85-89STUDIES IN THE SYNTHESIS OF HALOGENATED ANTHRAQUINONES. I. A CONVENIENT PREPARATION OF 1,4-DICHLORO-5-HYDROXY-9,10-ANTHRACENEDIONEJudith L. Johnson; H. D. Hollis Showalter
91-96A RAPID AND EFFICIENT SYNTHESIS OF 2H-1,4-BENZOXAZINE-3(4H)-THIONES AND 2H-1,4-BENZOTHIAZINE-3(4H)-THIONESD. R. Shridhar; M. Jogibhukta; V. S. H. Krishnan
97-114THE REACTION OF AMINES WITH METHYLENE CHLORIDE. A BRIEF REVIEWJohn E. Mills; Cynthia A. Maryanoff; Robin M. Cosgrove; Lorraine Scott; David F. McComsey
115-119PHASE-TRANSFER CATALYZED DOUBLE MICHAEL CONDENSATION. PREPARATION OF 7,11-BISARYLSPIRO[5,5]UNDECANE-1,9-DIONESD. Loganathan; T. Varghese; G. K. Trivedi
119-125A SYNTHESIS OF THE SIDEROPHORE 1,3,5-TRIS(N,N′,N-2,3-DIHYDROXYBENZOYL)AMINOMETHYLBENZENEPaul F. Schuda; Catherine M. Botti; Michael C. Venuti
126-130SELECTIVE PREPARATION. 41. CONVERSION OF 2,2′-DIHYDROXY-3,3′-DI-t-BUTYL-5,5′-DIMETHYLBIPHENYL TO SOME NOVEL DIBENZOFURANMasashi Tashiro; Haruo Yoshiya
130-136SYNTHESIS OF N-ARYL ENAMINOSULFONES AND IMPROVED PREPARATION OF N-SUBSTITUTED ENAMINONITRILESTatsuo Yamamoto; Motowu Muraoka
136-139SYNTHESIS OF t-BUTOXYCARBONYL AND BENZYLOXYCARBONYL AMINO ACID AMIDESB. Rzeszotarska; M. Makowski; Z. Kubica
140-143SYNTHESIS OF A NEW POLYMER POLY(4′-VINYLDIBENZO-14-CROWN-4)T. C. Kuan; S. J. Wang
144-148THE FRIEDEL-CRAFTS ACYLATION AND BENZOYLATION OF PYRENERonald G. Harvey; John Pataki; Hongmee Lee

Volume 16, Issue 1 (1984)

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1-10REACTIONS WITH HETEROCYCLIC AMIDINES. SYNTHESIS OF SOME NEW AZOLYLTHIOUREA DERIVATIVESM. R. H. Elmoghayar; M. K. A. Ibrahim; F. M. Darwish
11-24PREPARATION OF PYRIDINE-2(1H)-THIONES FROM CHALCONESJ. L. Soto; C. Seoane; M. J. Rubio; J. M. Botija
25-30LARGE-SCALE CYCLOPROPANATIONOljan Repič; Paul G. Lee; Urs Giger
31-36A FACILE PREPARATION OF E-ALKYL ENAMINONESCataldo A. Maggiulli; Ping-Wah Tang
37-41N-SUBSTITUTION OF SACCHARIN UNDER PHASE-TRANSFER CONDITIONSCelso F. Perez; Edgardo L. Calandri; Maria R. Mazzieri; Beatriz Arguello; Angela R. Suarez; Martin J. Fumarola
42-47PHASE-TRANSFER CATALYSED SYNTHESIS OF 4-BENZYLOXY-2-BUTANONESG. Guillaumet; G. Coudert; M. Mpassi
49-77SYNTHESIS AND REACTIONS OF SULFAMIDES. A REVIEWSéan D. McDermott; William J. Spillane

Volume 15, Issue 6 (1983)

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371-377SYNTHESIS OF 4-(4′-HYDROXYPIPERIDINO)-4-PHENYLCYCLOHEXANOL, A DIHYDROXY PHENCYCLIDINE METABOLITEGeorge A. Brine; Karl G. Boldt; Michael L. Coleman; F. Ivy Carroll
379-385DIRECT SYNTHESIS OF Nα-BENZYLOXYCARBONYL-Nε-t-BUTYLOXY-CARBONYL-L-LYSINE FROM L-LYSINEEdgar P. Heimer; Ching-Tso Wang; Theodore J. Lambros; Arthur M. Felix
387-424LANTHANIDES IN ORGANIC SYNTHESISNicholas R. Natale
425-435INDEXES

Volume 15, Issue 5 (1983)

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297-302THE VON BRAUN REACTION BETWEEN N-t-BUTYLAMIDES AND PHOSPHORUS OXYCHLORIDE. A CONVENIENT NITRILE SYNTHESISRobert B. Perni; Gordon W. Gribble
303-313SYNTHESIS OF URACIL, 6-METHYLURACIL AND SOME DIHYDROURACILSK. S. Bhat; A. S. Rao
315-319AN IMPROVED METHOD FOR THE PREPARATION OF 2-SUBSTITUTED 1,2-BENZISOTHIAZOL-3 (2H)-ONES. NOVEL CYCLIZATION OF N-SUBSTITUTED 2-CARBAMOYLBENZENESULFENYL BROMIDES ON ACTIVATED BASIC ALUMINANobumasa Kamigata; Satoshi Hashimoto; Michio Kobayashi
321-327SYNTHESIS OF SOME BICOUMARYL SULPHIDES AND SULPHONESJ. R. Merchant; N. M. Koshti
329-333SUGAR 1,3,4-OXADIAZOLES VII. CYCLIZATION OF ACETATES OF SUGAR AROYLHYDRAZONES USING LEAD TETRAACETATEMahmoud A. M. Nassr
335-340SYNTHESIS OF 3-HYDROXYDIBENZ [a,c] ANTHRACENERonald G. Harvey; Jayanta K. Ray; Kutikat B. Sukumaran
341-348SYNTHESIS OF 6-BROMO-, 8-BROMO- AND 6, 8-DIBROMOCATECHINEberhard Kiehlmann; Pieter J. Van der Merwe; Hans K. L. Hundt
349-359PREPARATION OF 11-HYDROXYMETHYL-2, 3-NAPHTHO-18-CROWN-6 AND ITS CONVERSION INTO A HIGHLY LIPOPHILIC CROWN CARBOXYLIC ACIDBronislaw Czech; Anna Czech; Richard A. Bartsch
361-364THE SYNTHESIS OF HIGH PURITY Nα-BENZYLOXYCARBONYL Nε-t-BUTYLOXYCARBONYL-L-LYSINES. T. Chen; K. T. Wang
365-367A SIMPLIFIED, ONE STEP SYNTHESIS OF CHOLEST-5-EN-3-ONEEdward J. Parish; Sarawanee Chitrokorn
368-369A FACILE SYNTHESIS OF 2, 2′-BIPYRIDYL-3, 3′-DICARBOXYLIC ACIDFranz L. Wimmer; Smita Wimmer

Volume 15, Issue 4 (1983)

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225-231AN ALTERNATIVE TO THE LEUCKART METHOD FOR THE CONVERSION OF PRIMARY AMINES INTO THIOLSSayed Mahmoud M. Elshafie
233-238PREPARATION OF MONOMETHYL FUMARATEMichael Dymicky
239-242A CONVENIENT SYNTHESIS OF 3-HYDROXYTROPONEAnna M. Becker; Rodney W. Rickards
243-249A FACILE SYNTHESIS OF DOPAMINE-4-SULFATEScott L. Harbeson; Daniel J. Kerkman; John F. Debernardis
251-260THE REACTION OF trans-3-HEXENEDIOIC ACID WITH ETHYLENEDIAMINES. A SIMPLE ROUTE TO THE TETRAHYDRO-1H-PYRROLO[1,2-d][1,4]DIAZEPINE RING SYSTEME. R. Lavagnino; C. W. Ryan
261-264THE SYNTHESIS OF SOME BENZO[b]THIOPHENE SUBSTITUTED ARYLACETIC ACID ESTERSD. W. H. Macdowell; D. M. Ondeyka
265-268PHOTOCHEMICAL SYNTHESIS OF 2-(2-ARYL-5-OXAZOLYL) BENZOATESKou-Chang Liu; Robert K. Howe
268-270NEW HYDRAZONOYL BROMIDES AND AZOMETHYLENE PHOSPHORANESR. S. Tewari; P. D. Dixit; P. Parihar
271-275PREPARATION OF 4,4′-DI-t-BUTYLBIPHENYL DERIVATIVESMasashi Tashiro; Yasuhisa Fukuda; Gouki Fukata
276-278SELECTIVE PREPARATION. 44. PREPARATION OF 4-HYDROXYPHENYL PHENYL THIOETHER USING t-BUTYL FUNCTION AS A POSITIONAL PROTECTIVE GROUPMasashi Tashiro; Haruo Yoshiya
278-280SYNTHESIS OF 3-ACETOXY-1-METHYL AND 1-ETHYLINDOLESRoy W. Daisley; Zaha A. Elagbar
280-282PREPARATION OF 3-BROMO-4-NITROPYRIDINE 1-OXIDERoy W. Daisley; Jafar R. Hanbali
283-287NEW SYNTHESIS OF DIASTEREOMERIC (±)-13,17,21-TRIMETHYLPENTA- AND (±)-13,17,21-TRIMETHYLHEPTATRIACONTANESH. A. Tolstikov; V. N. Odinokov; W. R. Achunova; A. M. Moiseenkov; A. V. Semenovsky
288-291E AND Z-CYANOACRYLAMIDES FROM DIAMINOMALEONITRILEJoseph H. Boyer; V. T. Ramakrishnan; T. P. Pillai
292-295THE SYNTHESIS OF KNORR'S PYRROLE BY INVERSE ADDITIONJohn V. Cooney; Erna J. Beal; Robert N. Hazlett
296ERRATUM

Volume 15, Issue 3 (1983)

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137-144EFFICIENT SYNTHESIS OF DL-THYROXINE-p-HYDROXYPHENYL ETHERKarl G. Boldt; George A. Brine
145-148PREPARATION OF 1,2,3,4-TETRAHYDRO-6-METHOXY-5-METHYLNAPHTHALENE-2-ONEMing Shen; Arthur G. Schultz
149-152PRACTICAL SYNTHESIS OF 3,3,4,4-TETRAMETHYLCYCLOPENTANONEPaul A. Aristoff; Cynthia L. Nelson
152-153PREPARATION OF MONOALLYL ETHYLENE GLYCOLSSteven J. Jungk; Richard D. Gandour
154-1565α-HYDROXY-3α-CHOLESTANECARBOXYLIC LACTONELars H. Hellberg; Rodney G. Stoddard; Peter Wintersdorf
157-160A CONVENIENT SYNTHESIS OF 2,3-DICHLORO-1,4-NAPHTHOQUINONE-1-14C USING A NOVEL CHLORINATION PROCEDUREKenneth W. Ehler; Ronald S. Pardini
161-163SYNTHESIS OF 8-(D-GLUCO-PENTA-O-HYDROXYLPENTYL)-7-OXABICYCLO[4.2.0]OCTANEJack C. Kim; Min Sook Kim; Roy L. Whistler; A. K. M. Anisuzzaman
165-198ORGANIC THIONITRITES AND RELATED SUBSTANCES. A REVIEWShigeru Oae; Kōichi Shinhama
199-223POTASSIUM HYDRIDE IN ORGANIC SYNTHESIS. A REVIEWHarold W. Pinnick

Volume 15, Issue 1-2 (1983)

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1-5EFFECT OF METAL IONS IN ORGANIC SYNTHESIS. PART XII A NEW SYNTHESIS OF N-(α-CHLOROBENZYLIDENE)-N'-PHENYLHYDRAZINE BY REACTION OF PHENYLAZOSTILBENE AND COPPER(II) CHLORIDEOrazio Attanasi; Paolo Battistoni; Gabriele Fava
7-15BROMINE OXIDATION OF THE DIPOTASSIUM SALT OF α,α′-DINITROSUCCINONITRILE INTO THE POTASSIUM SALT OF NITROKETOSUCCINONITRILET. P. Pillai; J. H. Boyer
17-28PREPARATION OF IMIDAZOLE AND IMIDAZOLIUM 2-CARBALDEHYDESFiore Ricciardi; Madeleine M. Joullié
29-34PREPARATION OF 3,6-DIOXA-4-(BENZYLOXYMETHYL)-1,8-OCTANEDIOL, A VERSATILE INTERMEDIATE FOR THE SYNTHESIS OF FUNCTIONALIZED CROWN ETHERSBronislaw Czech; David A. Babb; Richard A. Bartsch
35-40SYNTHESIS OF [S-(R*,R*)] – ETHYL α–[(1–CARBOXYETHYL) AMINO]–BENEZENEBUTANOATE, AN IMPORTANT INTERMEDIATE IN THE SYNTHESIS OF ANGIOTENSIN CONVERTING ENZYME INHIBITORSJames S. Kaltenbronn; Dana Dejohn; Uldis Krolls
41-48PREPARATION OF 3-ARYL-3-OXO-2-TOSYLOXYIMINOPROPANENITRILESJ. L. Soto; C. Seoane; J. A. Valdés; F. J. Fernández
49-55NOVEL CYANOHYDRIN FORMATION AND ISOLATION IN THE SYNTHESIS OF 5-IODONOREPINEPHRINEJanice T. Gordon; Kenneth L. Kirk; Mary B. Dratman
57-62THE SYNTHESIS OF α-ACETOXYBENZYLBENZYLNITROSAMINERobert E. Lyle; Valerie E. Gunn; Myron K. Jacobson; William Lijinsky
63-67PREPARATION OF ω-BROMOALKAN-1-OLS FROM α,ω-ALKANEDIOLS BY THE CONTINUOUS EXTRACTION METHODF. Camps; J. M. Casamor; J. Coll; A. Guerrero; M. Riba
67-68AN IMPROVED PROCEDURE FOR THE OXIDATION OF 2,5- AND 5,6-DIHALO-3-METHYLPYRIDINESF. L. Setliff; W. R. Huie; R. L. Adams
69-70SYNTHESIS OF ALKALI AND ALKALINE-EARTH METAL ADDUCTS OF SUCROSELaurence Poncini; Vijaya Chand
71-135REACTIVITY OF β-HALOENAMINES. A REVIEWNorbert De Kimpe; Niceas Schamp

Volume 14, Issue 6 (1982)

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373-380REACTIVITY OF ACETYLMETHYLENE TRIPHENYLARSORANEYaozeng Huang; Yuanyao Xu; Zhong Li
381-392SYNTHESIS OF PSEUDOPEPTIDESNancy Acton; Akira Komoriya
393-395AN IMPROVED PREPARATION OF TRINITROPHLOROGLUCINOLA. A. Defusco; A. T. Nielsen; R. L. Atkins
396-399A SIMPLE ‘ONE-POT’ CONVERSION OF CARBOXYLIC ACIDS INTO NITRILESA. D. Dunn; M. J. Mills; W. Henry
399-403AN EFFICIENT SYNTHESIS OF N'-(o-ALKOXYPHENYL)-PYRIDINECARBOXAMIDINE DERIVATIVESTakuzo Hisano; Masanobu Tasaki; Toshikazu Matsuoka; Masataka Ichikawa
403-406A SYNTHESIS OF FUSED PYRIMIDINESR. Madhav
406-409ANHYDRIDE ACYLATION REACTIONS OF 2,4-DINITROPHENYLHYDRAZINEMichael J. Hearn; Lori Defurio; Wendy Hurst; Carolyn Koss; Marilyn Licthman; Laura Lucas; Patricia Mabrouk; Sally Teng; Catherine Waud
409-414NEW PREPARATION OF N-METHYLIMIDAZOLE-4,5-DICARBOXALDEHYDES AND SOME OF ITS REACTIONSM. El Borai; M. Hassanein
414-417SYNTHESIS OF 7-HYDROXYBENZO[a]PYRENERonald G. Harvey; Peter P. Fu
418-4241,1'-DIHYDROXY-2,2'-DIPHENYL-4,4'BINAPHTHYLJoseph H. Boyer; Jayanti Patel
426-435INDEXES

Volume 14, Issue 5 (1982)

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309-317THE SYNTHESIS OF PHENOLIC ANTIOXIDANTS. 3,5-BIS(3,5-DI-TERT-BUTYL-4-HYDROXYBENZYL)-2,3,6-TRIMETHYLBENZYL DERIVATIVESLuke K. T. Lam; Alex Chung; Alan V. Fladmoe; Lee W. Wattenberg
319-326SYNTHESIS OF 2-AROYL-4-CYANO-4-CARBETHOXY-1,3,5-TRIARYLCYCLOHEXANOLSJ. L. Soto; C. Seoane; A. M. Mansilla; M. Quinteiro
327-331A CONVENIENT SYNTHESIS OF ETHYL α-CARBETHOXY-β-(ARYLAMINO) ACRYLATES AND RELATED COMPOUNDSNagaraj R. Ayyangar; Rajgopal J. Lahoti; Thomas Daniel
333-336AN IMPROVED PREPARATION OF 2,3,4-TRIMETHOXYBENZSUBER-6-ONEJoseph G. Cannon; Basil J. Demopoulos
337-3427-ETHOXY-6-METHOXY-2,2-DIMETHYL-2H-1-BENZOPYRANE. Kiehlmann; J. E. Conn; J. H. Borden
343-346A CONVENIENT SYNTHESIS OF 1-BENZYLINDOLESRobert B. Perni; Gordon W. Gribble
347-349SYNTHESIS OF (2R,3R) 0,0-DIPIVALOYLTARTARIC ACID (DPTA) AND OF (2R,3R) 0,0-DI(ADAMANTANE-1 CARBONYL) TARTARIC ACID (DATA), USEFUL CHIRAL REAGENTS FOR ASYMMETRIC PROTONATIONSL. Duhamel; J. C. Plaquevent
350-353SYNTHESIS OF 4'-ALKYLDIBENZO CROWN ETHERSC. S. Chen; S. J. Wang; S. C. Wu
354-356A SIMPLIFIED APPARATUS FOR GENERATION OF DIAZOMETHANEMilos Hudlicky
357-359NITROSYLSULFURIC ACID HYDROLYSIS OF PRIMARY AMIDESL. G. Wade Jr.; William B. Silvey
359-362SYNTHESIS OF ARYL HALIDES via ORGANOBORANE CHEMISTRYGeorge W. Kabalka; Kunda A. R. Sastry; Usha Sastry; Vishwanatha Somayaji
362-365FACILE OXIDATIVE CLEAVAGE OF CARBON-CARBON MULTIPLE BONDS WITH CHROMIUM(V) REAGENT [(BiPy)H2CrOCl5]T. K. Chakraborty; S. Chandrasekaran
365-369O-CYANOMETHYLOXIME OF NITROGLYOXYLONITRILET. Perumal Pillai; Joseph H. Boyer
369-372A SIMPLE, INEXPENSIVE SYSTEM FOR PERFORMING HIGH PRESSURE REACTIONSPhilip Deshong; C. Michael Dicken; Joseph J. Perez; Robert M. Shoff

Volume 14, Issue 4 (1982)

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225-232ALKYL PHOSPHITES AND PHOSPHONATES AS ALKYLATING AGENTS FOR 1,3,4-THIADIAZOLIDINE-2,5-DITHIONESM. M. Sidky; M. R. Mahran; M. F. Zayed; W. M. Abdou; T. S. Hafez
233-240TRANSFORMATION OF A 3-BROMOMETHYL-CEPHEM INTO 3-ACETOXYMETHYL-CEPHEM DERIVATIVESI. Miskolczi; F. Sztaricskai; R. Bognár
241-247THE SYNTHESES OF PHENOLIC ANTIOXIDANTS. 1,3,5-TRIS(4-HYDROXYPHENOXYMETHYL)MESITYLENE AND RELATED COMPOUNDSLuke K. T. Lam; Chester Yee; Ramdas P. Pai; Lee W. Wattenberg
249-264SYNTHESIS AND USES OF β-KETO ACIDS. A BRIEF REVIEWLauren Oshry; Stuart M. Rosenfeld
265-307HYDROXYLAMINE-O-SULPHONIC ACID. ITS USE IN ORGANIC SYNTHESIS. A REVIEWRaymond G. Wallace

Volume 14, Issue 3 (1982)

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157-162SYNTHESIS OF γ-L-GLUTAMYL-TAURINE (GLUTAURINE)Arthur M. Felix
163-168SYNTHESIS OF 6-SUBSTITUTED-6H-INDENO[1,2-c]ISOQUINOLINE-5,11-DIONESStanley Wawzonek
169-175A MODIFIED APPROACH IN THE SYNTHESIS OF 5- AND 6-METHYLBENZ[a]ANTHRACENESPeter P. Fu; Frederick E. Evans; Dwight W. Miller; J. P. Freeman; Shen K. Yang
177-181A GENERAL METHOD FOR THE PREPARATION OF FORMATESM. Dymicky
183-187A CONVENIENT METHOD FOR THE SYNTHESIS OF KAEMPFEROLMasataka Ichikawa; A. Mahir Pamukcu; George T. Bryan
189-194ALKOXYETHYNYL KETONESG. Himbert; L. Henn
195-197A GENERAL AND CONVENIENT SYNTHESIS OF 2H-1,4-BENZOXAZIN-3(4H)-ONESD. R. Shridhar; M. Jogibhukta; V. S. H. Krishnan
197-198AN UNUSUAL SYNTHESIS OF 2,6-Di-t-BUTYL-4-ISOPROPENYLPHENOLLajos Avar
199-200PREPARATION OF ISATOIC ANHYDRIDE FROM PHTHALIMIDEY. R. Rao; M. Bapuji; S. N. Mahapatra
200-202HIGH-YIELD, ONE STEP PHOTOCHEMICAL SYNTHESIS OF 3- AND 4-BROMOMETHYLBENZOIC ACIDSRavi Subramanyam; A. G. Pinkus
202-203SYNTHESIS OF BENZ(a)ANTHRACENE-5,6-DIONEDominic T. C. Yang; W. M. Trie
204-205SYNTHESIS OF 2-CHLORO-4-FLUORANILINEJeffery B. Press; Corris M. Hoffman
206-2082,4-BIS(BROMOMETHYL)-5-METHYL-N-ACETYL BENZYLAMINE AND 2,4-BIS(CYANOMETHYL)-5-METHYL-N-ACETYLBENZYLAMINENitya G. Kundu; James Peck; Dennis W. Evangelatos
208-213PHOTOCHEMICAL SYNTHESIS OF BULLVALENEDIONET. Miyashi; Y. Takahashi; K. Okada; T. Mukai
213-215AN IMPROVED SYNTHESIS OF TRIALKYLKETENIMINESN. De Kimpe; R. Verhé; L. De Buyck; N. Schamp
216-219METACYCLOPHANES AND RELATED COMPOUNDS. 2. NITRATION AND ACETYLATION OF 2,7-DI(t-BUTYL)-trans-10b,10c-DIMETHYL-10b,10c-DIHYDROPYRENEMasashi Tashiro; Takehiko Yamato
220-224SYNTHESIS OF α-AMINOKETONES BY CATALYTIC HYDROGENATION OF BENZILMONOIMINESBenito Alcaide; Gerardo Escobar; Rafael Pérez-Ossorio; Joaquin Plumet

Volume 14, Issue 1-2 (1982)

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1-8SYNTHESIS OF (±)-NIRANTHINGail E. Schneiders; Robert Stevenson
9-20A VERSATILE METHOD FOR THE CONVERSION OF KETONES TO ALDEHYDESJoseph A. Virgilio; Emanuel Heilweil
21-29SYNTHESES OF FURO-, PYRROLO- AND THIENO[3,2-c]COUMARINSM. Trkovnik; R. Djudić; I. Tabaković; M. Kuleš
31-38PREPARATION OF 2,3,4,6-TETRAMETHYLPYRYLIUM PERCHLORATE AND OF 2,3,4,6-TETRAMETHYLPYRIDINEAlexandru T. Balaban; Anisia Bota
39-442,4,6-TRIMETHYLPYRYLIUM SULFOACETATEAntonie Dinculescu; Alexandru T. Balab
45-89SYNTHESIS OF SULFOXIDES. A REVIEWJózef Drabowicz; Marian Mikołajczyk
91-155REACTIONS OF ACETYLENES WITH HYDRAZINES. A REVIEWWolfgang Sucrow

Volume 13, Issue 6 (1981)

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389-393SYNTHESES OF (S)-(-)-N-METHYLPROLINOLCharles G. Chavdarian; Edward B. Sanders
395-399THE ELECTROCHEMICAL OXIDATIVE HYDROLYSIS OF KETONE OXIMESM. R. van de Mark; A. M. Scornavacca
401-408SYNTHESIS OF 8,12-SECOPROSTAGLANDIN F, AN EICOSENOIC ACID ANALOGUEP. A. Zoretic; J. L. Ferrari
409-414FORMATION OF A NEW TYPE OF 1:2 ADDUCT FROM THE REACTION OF 2,3-LUTIDINE N-OXIDE WITH PHENYL ISOCYANATET. Hisano; M. Ichikawa; T. Matsuoka; K. Muraoka; M. Hamana
414-418TETRACHLOROCYCLOPROPENE, A HIGHLY REACTIVE REAGENT FOR 4 (1H)-PYRIDINONE SYNTHESISM. L. Deem
419-421AN IMPROVED SYNTHESIS OF 2-AMINOCARBAZOLEJ. B. Kyziol; A. Domanski
421-424REACTIONS OF N-AMINOPHTHALIMIDE WITH ELECTROPHILES. PREPARATION AND PROPERTIES OF SOME NEW TRIACYLHYDRAZINESMichael J. Hearn; Stephanie B. Prisch
424-425ONE-POT PROCESS FOR BENZOCAINE FROM p-NITROBENZOIC ACIDS. C. Basa; C. Srinivasulu
426-428THE SYNTHESIS OF METHYL 2-HYDROXY-5-METHOXY-3-METHYLBENZOATEMelvin S. Newman; Ving Gon Lee
429-432THIOPHENE ANALOGUES OF SENDAVERINEJ. M. Barker; P. R. Huddleston
433-444INDEXES

Volume 13, Issue 5 (1981)

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315-322NEW SELECTIVE SYNTHESIS OF 3-BROMOMETHYL-3-CEPHEM ESTERSI. Miskolczi; F. Sztaricskai; R. Bognár
323-330SYNTHESIS OF (±)-ISO-OTOBAPHENOLPralhad A. Ganeshpure; Robert Stevenson
331-336A SIMPLE ONE-STEP SYNTHESIS OF 2-PYRIDONES FROM BENZYLIDENEACETOPHENONESJosé L. Soto; Carlos Seoane; Ana M. Mansilla
337-3478,12-SECOPROSTAGLANDINS. 8-AZADINOR ANALOGSP. A. Zoretic; D. Sarna; N. D. Sinha
349-352A CONVENIENT PREPARATION OF 1-BROMO-2-FLUORONAPHTHALENEGordon W. Gribble; Craig S. LeHoullier; Robert W. Allen; Jeffrey J. Gilbertson
353-356DEALKYLATION OF N-PYRIDYLETHYL-2-ARYLBENZIMIDAZOLES BY ALUMINUM CHLORIDEMasataka Ichikawa; Chiyuki Yamamoto; Takuzo Hisano
356-360A STEREOSELECTIVE SYNTHESIS OF endo-7-PHENYL-2-OXABICYCLO[4.1.0]HEPTANEGregory D. Hobbs; James D. Woodyard; John R. Curtis
360-363A CONVENIENT SYNTHESIS OF 2-PHENYL-2-THIAZOLIN-5-ONESNobutaka Suzuki; Yasuji Izawa
363-365PREPARATION OF 2-ISOCYANATO-5-CHLOROBENZOYL CHLORIDEB. K. Misra; Y. R. Rao; S. N. Mahapatra
365-367A NEW SYNTHESIS OF 4-BROMOMETHYLBENZAL BROMIDE AND 1,4-bis(DIBROMOMETHYL)-BENZENES. D. Saraf
368-371AN IMPROVED SYNTHESIS OF 2-ANTHRALDEHYDEPalanisamy Arjunan; K. Darrell Berlin
371-374A TWO-STEP PREPARATION OF 1-BENZYLPYRAZOLE-2-15NMurtedza bin Mohamed; John Parrick
374-378SYNTHESIS OF A NOVEL ASARONE DIMERC. Lemini; R. Cruz; I. H. Sanchez
379-3824-AMINOPYRAZOLO[3,4-d]PYRIMIDINESBalram Dhawan; Philip L. Southwick
383-387STEROIDAL ADAMANTYLAMIDES AND CARBAMATES. POTENTIAL ANTIVIRAL AGENTSJosef E. Herz; Tomasa Corro; Maritza Velarde; Julieta A. Herz

Volume 13, Issue 3-4 (1981)

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179-184THE STEREOSELECTIVITY OF THE REDUCTION OF HOMOPROPARGYLIC ALCOHOLS TO HOMOALLYLIC ALCOHOLSR. E. Doolittle
185-188A CONVENIENT NEW METHOD FOR THE PREPARATION OF DIMETHYL 3-METHOXYPHTHALATEJose Alexander; Ashok V. Bhatia; L. A. Mitscher
189-196SYNTHESIS OF 5-ALKOXYANTHRANILIC ACIDSJefferson W. Tilley; James Kudless; Richard W. Kierstead; Percy S. Manchand
197-201AN EFFICIENT PREPARATION OF TETRAMETHYLALLENEDonald M. Hilvert; Marcia D. Jacobs; Thomas Hellman Morton
203-207NEW SYNTHESIS OF 2-AMINOBIPHENYLSA. N. Kost; R. S. Sagitullin; A. A. Fadda
209-216trans-1-CHLORO-5(ETHOXYETHOXY)-2-PENTENECornelus G. M. Janssen; Erik F. Godefroi
217-223SYNTHESIS OF FUNCTIONALIZED N-ALKYLMALEIMIDES AS POTENTIAL THIOL-DIRECTED ENZYME INHIBITORSFausto Ramirez; Hiroshi Okazaki; James F. Marecek; Harvey M. Levy
225-240UTILITY AND APPLICATIONS OF BORANE DIMETHYLSULFIDE IN ORGANIC SYNTHESIS. A REVIEWRobert O. Hutchins; Frank Cistone
241-313THE SYNTHESIS OF β-HALOGENATED ENAMINESNorbert de Kimpe; Niceas Schamp

Volume 13, Issue 2 (1981)

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71-79MICHAEL ADDITION OF DITHIOBENZOIC ACID TO α,β-UNSATURATED KETONES. A NEW SERIES OF DITHIOESTERSJayalakshmi Ramachandran; S. R. Ramadas; C. N. Pillai
81-86SYNTHESIS OF 4-ARYL-5,6-BIS (CARBOMETHOXY)-2H-THIOPYRAN-2-THIONES. A NEW SERIES OF CYCLIC DITHIOESTERS OR α-DITHIOPYRONESJayalakshmi Ramachandran; S. R. Ramadas; C. N. Pillai
87-92POLYETHERS. 2. PREPARATION OF ω,ω′-DISUBSTITUTED POLYARYLETHERSMasashi Tashiro; Haruo Yoshiya; Gouki Fukata
93-96STUDIES ON FRIEDEL-CRAFTS CHEMISTRY. 5. THE AlCl3-CH3NO2-CATALYZED FRIEDEL-CRAFTS REACTIONS OF BIS (BROMOMETHYL) BENZENES WITH BENZENEShuntaro Mataka; Yuhsuke Tsuda; Kazufumi Takahashi; Masashi Tashiro
97-101MILD PREPARATION OF PYRROLE-2-CARBOXALDEHYDESJ. A. de Groot; G. M. Gorter-La Roy; J. A. van Koeveringe; J. Lugtenburg
103-108ISOMER-SELECTIVE SYNTHESES OF 2,6-DICHLORO-4-NITROTOLUENE AND 2,4-DIFLUOROANILINELeonard M. Weinstock; Anthony M. Demarco; Roger J. Tull; Ichiro Shinkai
109-112A GENERAL SYNTHESIS OF UNSUBSTITUTED POLYCYCLIC ARENE IMINES. 3-METHYLCHOLANTHRENE 11,12-IMINEIrene Yona; Jochanan Blum
112-115PREPARATION OF p-TOLUENESULFONYL AZIDE. A CAUTIONARY NOTEThomas J. Curphey
116-1183-CHLOROMETHYL-2,4,6-TRIMETHYLBENZOIC ACIDF. H. C. Stewart
118-123SYNTHESIS OF p-BIS (DIMETHYLHYDROXYSILYL) BENZENEH. Matsumoto; K. Shono; Y. Nagai
123-126THE SYNTHESIS OF 3-R-7-CARBOMETHOXYMETHYLENE-7H-1,2,4-TRIAZOLO[3,4-b]-1,3,4-THIADIAZIN-6-ONESNed D. Heindel; Jack R. Reid
126-129REDUCTION OF 5-HYDROXYMETHYL-1-AZA-3,7-DIOXABICYCLO[3.3.0]OCTANE AND OF 2-PHENYL-4,4-DIMETHYLOXAZOLIDINE WITH FORMIC ACIDS. Wawzonek
129-134REACTION OF DIAZOMETHANE WITH N-NITROSO-4-PIPERIDINONESJoseph E. Saavedra
134-136LEWIS ACID CATALYZED PREPARATION OF TETRAMETHYLHEXATHIOADAMANTANEC. S. Giam; R. L. Tabor; T. E. Goodwin
137-140A CONVENIENT PREPARATION OF ALKYL- AND ARYLSULFONYLPYRIDINESC. S. Giam; K. Kikukawa; D. A. Trujillo
140-144A CONVENIENT PREPARATION OF cis-DIHYDROIONONECrist N. Filer; James C. Pugliese; John C. Morrison; David G. Ahern
144-149A CONVENIENT PREPARATION OF α,α-DIPHENYLACETOPHENONEN. Sbarbati Nudelman; A. A. Vitale
149-151AN IMPROVED PREPARATION OF CORONENEA. G. Holba; E. J. Eisenbraun

Volume 13, Issue 2 (1981)

152-155SYNTHESIS OF BENZO[a]PYRENE-12-OLPeter P. Fu; Ronald G. Harvey
155-163SYNTHESIS OF NEW NAPHTHALENE DERIVATIVES WITH POSSIBLE SCHISTOSOMICIDAL EFFECT. PART XS. H. Doss; S. S. A. Dimitry
163-170SULTAM DERIVATIVES WITH POSSIBLE SCHISTOSOMICIDAL ACTIVITY. NAPHTHOSULTAMS Part XIVS. H. Doss; M. Hamed
170-172EFFECT OF METAL IONS IN ORGANIC SYNTHESIS. PART VIII CONVERSION OF ACYLHYDRAZINES AND N-ACYL-N′-TOSYLHYDRAZINES TO AMIDES IN THE PRESENCE OF CUPRIC CHLORIDEOrazio Attanasi; Franco Serra-Zanetti
172-175ETHYL 3,4-DIHYDROXY-5-METHOXYBENZOATE, AN INTERMEDIATE PRODUCT FOR THE SYNTHESIS OF 3,4-DIHYDROXY-5-METHOXYBENZOIC ACIDYosisige Kato
175-178A DETAILED PROCEDURE FOR SYNTHESIS OF 2,3-DIHYDROXYBENZALDEHYDECharles F. Hoyng

Volume 13, Issue 1 (1981)

CEditorial Board Page
1-7SELECTIVE PREPARATION 29. PREPARATION OF 2,6-BIS(CHLOROMETHYL)- AND OF 2,6-BIS(MERCAPTOMETHYL)-4-SUBSTITUTED-TERT-BUTYLBENZENESMasashi Tashiro; Takehiko Yamato
9-12A SIMPLE STEREOSELECTIVE METHOD FOR THE PREPARATION OF (E)-2,5-DIMETHYL-1,3,5-HEXATRIENES. R. Ramadas; R. Ehrencron; J. W. J. Gielen; H. J. C. Jacobs
13-18SYNTHESIS OF 1,1-BIS(HYDROXYMETHYL) CYCLOPROPANESR. Verhe; D. Courtheyn; N. De Kimpe; L. De Buyck; R. Thierie; L. Van Caenegem; N. Schamp
19-22THE SYNTHESIS OF TRIACONTANOL, SODIUM TRIACONTYL SULFATE AND DIHYDROGEN TRIACONTYL PHOSPHATENorman R. Hunter; James L. Charlton; Nancy A. Green; Werner J. Fritz; Brenda M. Addison
23-38BUILDING BLOCKS FOR THE SYNTHESIS OF MAYTANSINOIDSErwin Götschi; Fernand Schneider; Hans Wagner; Karl Bernauer
39-48TWO EFFICIENT SYNTHESES OF INDOLE-3-PROPIONIC ESTERS AND ACIDS. FURTHER APPLICATIONS OF MELDRUM'S ACIDDiane S. Farlow; Michael E. Flaugh; Sharon D. Horvath; Edward R. Lavagnino; Paul Pranc
49-54SYNTHESIS OF OCIMINPralhad A. Ganeshpure; Robert Stevenson
55-58PREPARATION OF 2-HYDROXYETHYLDIMETHYLAMINE ACYLIMIDESRobert J. Small
59-70SYNTHESIS OF SATURATED γ-LACTONES. A REVIEWRaphael Ikan; Vera Weinstein; Uzi Ravid

Volume 12, Issue 6 (1980)

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327-336SYNTHESIS OF PHENOXYPHENYLATED 4,4″-DICARBOXY-p-TERPHENYLSK. S. Y. Lau; F. E. Arnold
337-344CONVENIENT SYNTHESES OF SELECTED 14C- AND 3H-LABELED AROMATIC HYDROXYLAMINESM. R. Thissen; R. W. Roth; W. P. Duncan
345-350CONVENIENT DEALKYLATION OF QUATERNARY AMMONIUM SALTSGeorge R. Newkome; Veronica K. Majestic; Joe D. Sauer
351-356NEW ROUTES TO 4,5-DISUBSTITUTED FLUORENESItamar Willner; Mordecai Rabinovitz
357-360AN IMPROVED SYNTHESIS OF BICYCLO[2,1,1]HEXANE-1-CARBOXYLIC ACIDRawyani S. Abeywickrema; Ernest W. Della
361-391ORGANIC REDUCTIVE COUPLING WITH TITANIUM AND VANADIUM CHLORIDES. A REVIEWYee-Hing Lai
393-400INDEXES

Volume 12, Issue 5 (1980)

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iPrefaceJ. -P. Anselme; J. A. Moore
ii-viCharles G. Ouerberger
265-268SUBSTITUTED PYRAZINES FROM THE CATALYTIC REDUCTION OF α-AZIDOKETONESM. Nakajima; C. A. Loeschorn; W. E. Cimbrelo; J. -P. Anselme
269-274THE SYNTHESIS OF SOME NEW 1,2-BENZOTHIAZINESJoseph G. Lombardino
275-281REACTIONS OF CYCLIC DERIVATIVES OF URACIL AND THYMINEYoshiaki Inaki; Hidekazu Futagawa; Kiichi Takemoto
283-288THE EFFECT OF SOME ARYLOXY SUBSTITUENTS ON THE PREPARATION OF ARYLOXY PHOSPHAZENE TRIMERS AND ON THEIR STRUCTURAL CHARACTERISTICSBogumil Laszkiewicz; Jacek Dutkiewicz
289-295SYNTHESIS OF PURE ALKALI METAL LACTAMATESJ. Šebenda; A. Stiborová; L. Lochmann; Z. Bukač
297-304THE SYNTHESIS OF β-HYDROXYTRYPTAMINESHerbert A. Friedman; Wolfgang H. Vogel
305-308LEAD TETRAACETATE OXIDATION OF CIS- OR TRANS-TETRAHYDROFURAN-2,5-DICARBOXYLIC ACIDSJ. A. Moore; E. M. Partain III
309-326SYNTHETIC APPLICATIONS OF ISOUREAS. A REVIEWLon J. Mathias

Volume 12, Issue 3-4 (1980)

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181-184THIOL ESTERS OF Nα-TOSYL-L-ARGININET. R. Herrin; J. J. Plattner; J. W. Cole; M. R. Shaffar
185-189S-CARBOXYMETHYL DERIVATIVES OF L-CYSTEINYLGLYCINE AND GLYCYL-L-CYSTEINEMarvin D. Armstrong
191-195A PREPARATIVE SCALE SYNTHESIS AND CHROMATOGRAPHIC SEPARATION OF METHOTREXATE-α AND γ-MONOBUTYL ESTERSJ. D. Warren; R. B. Angier; George Morton; Andre Rosowsky
197-200DINITRONATE SALTS OF SUCCINONITRILEEdward F. Witucki; Walter Maya; Milton B. Frankel
201-202A CONVENIENT SYNTHESIS OF p-HYDROXYBENZAL DEHYDESC. W. Bird; Y. -P. S. Chauhan
203-206AN IMPROVED PROCEDURE FOR THE CONVERSION OF 2H-(1, 4)-BENZO-THIAZIN- AND 2H-(1, 4)-BENZOXAZIN-3(4H)-ONES INTO 3(4H)-THIONESD. R. Shridhar; C. V. Reddy Sastry; L. C. Vishwakarma; G. K. A. S. S. Narayan
207-212A GENERAL, HIGHLY EFFICIENT SYNTHESIS OF ACETYL AMINO ACID ETHYL ESTERSM. Dymicky
213-218SYNTHESIS OF α,α′-DIFUNCTIONAL CONJUGATED ENYNESJean-Paul Charpentier; Danielle Mesnard; Léone Miginiac
219-223A FACILE BASE CATALYZED CONDENSATION FOR THE SYNTHESIS OF FUSED PYRIMIDINE-2-CARBOXYLIC ACID ESTERSSusumu Nakanishi; Stephen S. Massett
225-228A NEW RAPID ESTERIFICATION PROCEDURE UTILIZING EXCEPTIONALLY MILD REACTION CONDITIONSC. Gundu Rao
229-230AN IMPROVED METHOD FOR THE SYNTHESIS OF DISULFONYLMETHYL THIOLSULFONATESNils Henning Nilsson; Alexander Senning
230-232SYNTHESIS OF dl-2-METHYL-2-(4-METHYL-3-PENTENYL) 5-OXYMETHYLENEMETHOXY-2H-BENZOPYRAN. A CANNABICHROMENE HOMOLOGUEF. Garcia; R. Laureles; R. Cruz
233-2343-ARYL-5-CARBOMETHOXY-5-CARBOMETHOXYMETHYL-1,4,2-OXATHIAZOLESNed D. Heindel; Gail K. Friedrich; Maria C. Tsai
234-237IMPROVED PREPARATION OF PYRIDO[3′,4′(4′,3′):4,5]IMIDAZO [1,2-c] [1,2,3]BENZOTRIAZINESJessie Lee; Anne Guthrie; Madeleine M. Joullié
238-242IMPROVED SYNTHESES OF 9-HYDROXY- AND 9-BUTOXY-1-PHENALENONEK. D. Franz; R. C. Haddon
242-243t-BUTYL PHENYL CARBONATEJohn W. Scott; David Parker
243-244AN IMPROVED SYNTHESIS OF 2,2′-DIPYRIDYL-1-OXIDEWillem Sont; Howard Alper
244-24613C-LABELLED ALIPHATIC NITRILES AND KETONESGert Kollenz; Hans Waldenberger

Volume 12, Issue 3-4 (1980)

246-249AN EFFICIENT SYNTHESIS OF 5-SULFOSALICYLALDEHYDE SODIUM SALTGarry W. Kirker
249-251A CONVENIENT METHOD FOR THE PREPARATION OF 1-ACYL-2-PHENYLHYDRAZINESMichael J. Hearn; Julia E. Grimwade
251-2532-FLUORO-1,4-NAPHTHALENEDIONER. S. Thomas Loeffler; Carolyn S. James
253-255AN IMPROVED PROCEDURE FOR THE SYNTHESIS OF SALICYLALDEHYDE HYDRAZONECharles F. Hoyng
255-259OXIDATION OF AMINO ALCOHOLS TO AMINO KETONESRobert E. Lyle; John R. Maloney; Roger J. White
259-260SOME 5,6- AND 2,5-DIHALONICOTINAMIDESFrank L. Setliff; John F. Hill
261-262A STEREOSELECTIVE APPROACH TO Z-ALLYLIC ALCOHOLSPeter A. Netland
263-264AN IMPROVED SYNTHESIS OF PHTHALAZINE REISSERT COMPOUNDSomsak Ruchirawat; Pongtip Thepchumrune

Volume 12, Issue 1-2 (1980)

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1-6THE EFFECT OF SOLVENTS AND CHELATING AGENTS ON THE REACTION ALKYNYL LITHIUM REAGENTS WITH OXIRANESR. E. Doolittle
7-11FACILE CATALYTIC SYNTHESES OF SQUALANEJohn W. Scott; Donald Valentine Jr.
13-48HYDROSILANES AS REDUCING AGENTS. A REVIEWYoichiro Nagai
49-180REACTIVITY OF α-HALOGENATED IMINO COMPOUNDSNorbert De Kimpe; Roland Verhé; Laurent De Buyck; Niceas Schamp

Volume 11, Issue 6 (1979)

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271-274RECOMMENDED SYNTHESES FOR 7–METHYLBENZ[a]ANTHRACENE, 12–METHYLBENZ[a]ANTHRACENE AND 7,12–DIMETHYLBENZ[a]ANTHRACENEMelvin S. Newman; J. M. Khanna; Kenneth C. Lilje
275-280A SIMPLE PROCEDURE FOR THE PREPARATION OF PURE MONOALKYL PHENYLACETONITRILESA. Jończyk; M. Ludwikow; M. Makosza
281-284SYNTHESIS OF A DIBENZYLBUTYROLACTONE LIGNAN EXTRACTIVE OF CINNAMOMUM CAMPHORARichard P. Duffley; Robert Stevenson
285-286AN IMPROVED METHOD FOR THE PREPARATION OF 5-HYDROXY-2-PYRROLIDONEBerkeley W. Cue Jr.; Nancy Chamberlain
287-292SYNTHESIS OF A 3α,12β-DIMETHOXY-11-KETO DERIVATIVE OF CHOLIC ACIDBahman Nassim; Jerry Ray Dias
293-311ISOCYANIDES IN ORGANIC SYNTHESIS. A REVIEWM. P. Periasamy; H. M. Walborsky
312THE SYNTHESIS OF OLIVETOL. TRIMETHYLSILYLATION AS A PROTECTIVE GROUP DURING GRIGNARD REACTIONSS. A. Barker; R. L. Settine
313-319INDEXES

Volume 11, Issue 5 (1979)

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201-246CYANOBOROHYDRIDE. UTILITY AND APPLICATIONS IN ORGANIC SYNTHESIS. A REVIEWRobert O. Hutchins; Nicholas R. Natale
247-249BENZO[1,2-b:4,5-b′]DITHIOPHENEN. Aggarwal; D. W. H. MacDowell
249-251SYNTHESIS OF THE ETHYLNITRONE OF ACETALDEHYDEH. F. Schmitthenner; K. S. Bhatki; R. A. Olofson; Julian Heicklen
251-253CONVENIENT SYNTHESIS OF 2-TRIMETHYLSILYLOXYPYRIDINESM. V. Prostenik
253-255SIMULTANEOUS PREPARATION OF BROMOACETIC ACID AND ACETYL CHLORIDEJanusz Swietoslawski; Aleksander Ratajczak
255-2591,7-DIMETHYLINDANE. H. Vickery; J. D. Weaver; E. J. Eisenbraun; A. R. Taylor; M. C. Hamming; G. W. Keen
259-261AN IMPROVED SYNTHESIS OF BENZO[k]FLUORANTHENEE. Harold Vickery; Edmund J. Eisenbraun
261-263BENZO[c]PHENANTHRENEE. H. Vickery; E. J. Eisenbraun
264-26511 H-11-OXO-5,10-DIPHENYLBENZO[b]FLUORENE FROM THE REACTION OF BENZYNE WITH INDANOCYCLONEP. Balasubramanian; S. Jayaraman; K. Narasimhan
265-267STUDIES OF COMPOUNDS RELATED TO AZINES. 11. THE REACTION OF DIETHYL PHENACYLPHOSPHATE KETAZINES WITH 2,2-DIFORMYLBIPHENYLOtohiko Tsuge; Gouki Fukata; Masashi Tashiro
267-270PREPARATION OF 3-(9,10-DIHYDRO-1-ANTHRYL)PENTANE-2,4-DIONEY. Nakano; H. Hiura

Volume 11, Issue 3-4 (1979)

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103-106PREPARATION OF TERTIARY PHOSPHINES USING A CONVENIENT FORM OF LITHIUM DIPHENYLPHOSPHIDEPeter W. Clark
107-110A PRACTICAL PROCEDURE FOR THE PREPARATION OF HINDERED α-HALOEPOXIDES AND α-HALOALDEHYDESJean Gralak; Jean-Yves Valnot
111-114STEREOSELECTIVE REDUCTION OF 2-QUINOLIZIDINONES WITH LITHIUM TRI-s-BUTYLBOROHYDRIDEJames Quick; Clifford Meltz; Ramavana Ramachandra
115-199THE SYNTHESIS OF α-HALOGENATED IMINO COMPOUNDSNorbert De Kimpe; Niceas Schamp

Volume 11, Issue 2 (1979)

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53-61A MILD METHOD FOR DEHYDRATING SOME CARBINOLS TO ALKENES. 1,1-DIARYLAMINOALKENES AS ANALGESICSRobert Bruce Moffett; Gerald N. Evenson
63-66BENZOCYCLOHEPTENE DERIVATIVES FROM THE HOESCH REACTIONJoseph G. Cannon; Jonathan P. Pease
67-70N-PHTHALOYL-L-GLUTAMIC ANHYDRIDE (2-PHTHAL IMIDOGLUTARIC ANHYDRIDE)J. A. Elberling; R. T. Zera; S. D. J. Magnan; H. T. Nagasawa
71-76PREPARATION AND REACTIONS OF 10-SPIROCYCLOPROPYLANTHRONEJ. Eynon; R. LaFauci; S. M. Rosenfeld
77-86SYNTHESIS OF ANTIFUNGAL ISOCOUMARINS (I)S. Nakajima; S. Sugiyama; M. Suto
87-92THE SYNTHESIS OF OLIVETOL. TRIMETHYLSILATION AS A PROTECTIVE GROUP DURING GRIGNARD REACTIONSSteven A. Barker; R. L. Settine
93-95IMPROVED PREPARATION OF SUCCINYLCHOLINE CHLORIDECheng-Hsia Wang; Hsi-Hua Tso; Chao-Tung Chen
95-96AN IMPROVED SYNTHESIS OF FLUORENONE METHYLNITRONEMagid A. Abou-Gharbia; Madeleine M. Joullié
97-991,4-ADDITION TO CITRALMeyer Schwarz; N. Wakabayashi; Eric G. Thing
100-101THE MONOALKYLATION OF DIBENZOYLMETHANEN. Kalyanam; J. W. Karban; J. L. McAtee Jr.

Volume 10, Issue 6 (1978)

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255-260SYNTHESIS OF HINDERED AROMATIC DIKETONES—BY FRIEDEL-CRAFTS ACYLATIONA. G. Pinkus; N. Kalyanam
261-266SYNTHESIS OF γ-UNSATURATED METHYLKETONESFrancis Barbot; Danielle Mesnard; Léone Miginiac
267-272AN EFFICIENT SYNTHESIS OF 4,5-DIMETHOXYBENZOCYCLOBUTENE via THE PARHAM CYCLIALKYLATION REACTIONCharles K. Bradsher; David A. Hunt
273-278SYNTHESIS OF 8-AZA-8,12-SECOPROSTAGLANDIN E2P. A. Zoretic; N. D. Sinha; P. Soja
279-283SYNTHESIS OF THE TRIPEPTIDE AMIDE CARBOBENZOXY-L-PROLYL-TRIFLUORO-DL-LEUCYL GLYCINAMIDEN. H. Pardanani; N. Muller
285-288SIMPLE PREPARATION OF AMINOMETHANEPHOSPHONIC ACIDJaroslav Kahovec; František Ŝvec; Milan Marhol
289-290PREPARATION OF SELENA- AND TELLURA PHTHALIC ANHYDRIDEJan Bergman; L. Engman
291-293SYNTHESIS OF AROYL CHLORIDES FROM SUBSTITUTED BENZOTRICHLORIDEST. Nakano; K. Ohkawa; H. Matsumoto; Y. Nagai
293-295AN IMPROVED SYNTHESIS OF s-TRIAZOLO[1,5-x]AZINESB. Vercek; B. Stanovnik; M. Tisler; Z. Zrimsek
295-297A SIMPLE APPARATUS FOR THE SAFE HANDLING OF PALLADIUM BLACK CATALYSTManuel H. Jimenez
298-300SUBSTITUTED 3,4-DIHYDROXYCINNOLINESManuel Lora-Tamayo; Berta Marco; Carmen Sender
300-304X-RAY CRYSTAL STRUCTURE ANALYSES OF ISOMERIC CYCLOADDUCTS OF 3-PICOLINE-N-OXIDE WITH p-CHLOROPHENYL ISOCYANATETakuzo Hisano; Toshikazu Matsuoka; Masataka Ichikawa; Keiji Muraoka; Tetsuya Komori; Kazunobu Harano; Yoshiteru Ida; Arild T. Christensen
304-306SELECTIVE REACTIVITY OF THE BISENAMINE OF PIPERAZINE-CYCLOHEXANONE WITH BENZOYL CHLORIDERobert E. Lyle; Brian P. Coppola; Jose E. Saavedra; Gloria G. Lyle
307SYNTHESIS OF METHYL 11,12-SECO-2,3-DINOR-10-OXAPROSTAGLANDIN E1P. A. Zoretic; T. Shiah
309-317INDEXES

Volume 10, Issue 5 (1978)

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201-204FORMYLATION OF ARENES BY α,α-DICHLOROMETHYL METHYL ETHER. AN IMPROVED EXPERIMENTAL PROCEDUREA. H. Lewin; S. R. Parker; N. B. Fleming; F. I. Carroll
205-209ACIDIC PROPERTIES OF BENZIMIDAZOLES AND SUBSTITUENT EFFECTS. III.: THE SUBSTITUENT EFFECT ON THE IMIDAZOLE CYCLIZATION FROM N-(m-SUBSTITUTED-PHENYL) PICOLYLAMIDINESMasataka Ichikawa; Shuichi Nabeya; Keiji Muraoka; Takuzo Hisano
211-214SYNTHESIS OF 2-DEOXYALDONONITRILES BY CHAIN ELONGATION OF MONOSACCHARIDE DIETHYL DITHIOACETALSPal Herczegh; Rezso Bognar; Erzsebet Timar
215-220STUDIES ON 4-HYDROXYCOUMARIN. 38. SYNTHESES OF 3-SUBSTITUTED DERIVATIVES. α-BROMOACYL AND 2-AMINOTHIAZOLO AND OF 4H-FURO-[3,2-c][1]-BENZOPYRAN-3-[2H],4-DIONEM. Trkovnik; N. Zivkovic; M. Kules; R. Djudjic
221-224A CONVENIENT SYNTHESIS OF β-KETOESTERSEdward C. Taylor; Ignatius J. Turchi
225-253THE SRN1 REACTION IN ORGANIC SYNTHESIS. A REVIEWJames F. Wolfe; David R. Carver

Volume 10, Issue 4 (1978)

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159-162A NEW SYNTHESIS OF N-BENZYL-2,3-DIHYDRO-4(1H)-ISOQUINOLONEDavid A. Walsh; Dwight A. Shamblee
163-166A CONVENIENT METHOD FOR THE PREPARATION OF 6-CARBOXYMETHYLFLAVONED. R. Shridhar; C. R. Sarma; R. R. Krishna; R. S. Prasad; Y. P. Sachdeva
167-172AN IMPROVED SYNTHESIS OF 3-N-PENTADECYL CATECHOL (3-PDC)Charles R. Dawson; Gilbert P. Ng
173-176A ONE-STEP SYNTHESIS OF 1,4-BENZENEDIETHANOLPeter W. Clark; Eric J. O'reilly
177-180SYNTHESIS OF 9-(P-VINYLPHENYL)-ANTHRACENES. Nozaki; H. Okada; Y. Matsumoto; A. Hagitani; A. Muko
181-194HALOGENATION TABLESMilos Hudlicky
195-196FERROCENYLPHOSPHINES BY A REVISED PROCEDUREArnold W. Smalley
197-200SYNTHESIS OF METHYL 11,12-SECO-2,3-DINOR-10-OXAPROSTAGLANDIN E1P. A. Zoretic; T. Shiah

Volume 10, Issue 3 (1978)

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105-111SYNTHESIS OF 3-SUBSTITUTED 1,4-BENZODIAZEPINE-2-ONESWajid A. Khan; Prithipal Singh
113-121THE T-BUTYL GROUP AS A POSSIBLE PROTECTIVE GROUP IN THE SYNTHESIS OF OLIGO [HYDROXY-1,3-PHENYLENE]METHYLENESV. Böhmer; D. Rathay; H. Kämmerer
123-131SYNTHESIS OF 1,1-DIMETHYLINDANE DERIVATIVES HAVING SYNTHETICALLY USEFUL SUBSTITUENTS AT THE 5- AND 6-POSITIONSJames G. Smith; M. Patricia Massicotte
133-136THE SYNTHESIS OF 4,7-DIHYDRO-1,3-DITHIEPINDavid N. Harpp; Kosta Steliou; Barry T. Friedlander
137-1425,6-DIMETHOXY-2-ISOPROPENYLBENZOFURAN AND 2-ISOPROPENYL-5,6-METHYLENEDIOXYBENZOFURANFred G. Schreiber; Robert Stevenson
143-148ALCL3-CH3NO2 CATALYZED T-BUTYLATION OF BIPHENYL, NAPHTHALENE AND SOME PHENOL DERIVATIVES WITH 2,6-DI(T-BUTYL)-P-CRESOLMasashi Tashiro; Takehiko Yamato
149-156FUNCTIONAL GROUP TRANSFORMATION. CONVERSION OF ALDEHYDES INTO AMIDES VIA α-CYANOENAMINESNobert De Kimpe; Roland Verhé; Laurent De Buyck; Jan Chys; Niceas Schamp
157SYNTHESIS OF TRICYCLIC AND TETRACYCLIC THIAZOLOIMIDAZOLE ACETIC ACIDSA. S. Radhakrishna; K. D. Berlin

Volume 10, Issue 2 (1978)

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55-58SYNTHESIS OF CHLOROALKANE-α,ω-DIOIC ACIDST. Nakano; H. Arai; H. Matsumoto; Y. Nagai
59-62A NOVEL METHOD FOR THE PREPARATION OF SUBSTITUTED 5-AMINO-1,2,3,4-THIATRIAZOLES BY AZA TRANSFER REACTIONB. Stanovnik; M. Tišler; B. Valenčič
63-66ALKYLATION OF PHENAZINE WITH N-CHLOROAMINESA. Citterio; T. Crolla
67-72SYNTHESIS OF α-(DIMETHYLAMINOMETHYLENE) KETONES BY USE OF METHOXYBIS (DIMETHYLAMINO) METHANE (BREDERECK'S REAGENT)Gregory B. Bennett; Robert B. Mason
73-77CONVENIENT ROUTES FOR THE PREPARATION OF 2-ISOPROPYL-5-METHYL CYCLOPENTANONEB. S. Kulkarni; A. S. Rao
79-82THE USE OF PIVALOYL CHLORIDE IN THE SELECTIVE SYNTHESIS OF 3-(T-BUTYL)-4-METHOXYPHENOL – A BHA ISOMERLuke K. T. Lam; Kelly Farhat
83-842-FLUORO-5-NITRO-3-PICOLINE AND 6-FLUORO-5-NITRO-3-PICOLINE BY CHLORIDE-FLUORIDE EXCHANGEF. L. Setliff; D. J. Defoggi
85-902-SUBSTITUTED-3-METHYLQUINOLINESHassan A. El-Sayad; Robert L. McKee
91-94DIRECT CONVERSION OF ALCOHOL TETRAHYDROPYRANYL ETHERS TO ALDEHYDESPhilip E. Sonnet
94-96REDUCTION OF 2-FUROIC ACID WITH METAL-AMMONIA SOLUTIONSH. R. Divanfard; M. M. Joullié
97-100SYNTHESIS AND PHOTOSTABILITY OF SOME N-ALKYL-N,N'-DIARYLFORMAMIDINESJoseph A. Virgilio; Emanuel Heilweil
101-102SYNTHESIS OF PYRUVATE ESTERS BY THE REACTION OF SODIUM PYRUVATE WITH ORGANIC HALIDES IN DMSOPatrick J. Boyle; John F. W. Keana

Volume 10, Issue 1 (1978)

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1-4THE PREPARATION OF (E)-2-PENTENALR. M. Waters; D. J. Voaden; A. Shani; J. Klug
5-8A PREPARATION OF (Z,E)-8,10-TRIDECADIEN-1-OL ACETATER. M. Waters; D. J. Voaden; J. D. Warthen Jr.
9-11A DRY MEDIUM SYNTHESIS OF 1-CYCLOHEXENE CARBOXALDEHYDEJ. L. Hogg; T. E. Goodwin; D. W. Nave
13-16THE SYNTHESIS OF 2,4[1H,3H]QUINAZOLINEDIONE AND SOME OF ITS 3-ARYL SUBSTITUTED DERIVATIVESM. Michman; S. Patai; Y. Wiesel
17-20A NEW ROUTE TO THE SYNTHESIS OF NITROXIDE CARBOXYLIC ACIDSGerald M. Rosen; Elmer J. Rauckman
21-27SYNTHESIS OF (R)-5-ALKYL-5-(1'-METHYL-3'-CARBOXYPROPYL) BARBITURIC ACIDS AND (R)-ALKYL-5-(1'-METHYL-3-CARBOXYPROPYL)-2-THIOBARBITURIC ACIDSF. Ivy Carroll; Abraham Philip
29-321,3-PROPANEDIOLS FROM KETONES BY FORMYLATION AND REDUCTIOND. E. Pearson; John D. Weaver
33-38SYNTHESIS OF AN AZAPROSTAGLANDIN ANALOGP. A. Zoretic; N. D. Sinha
39-44SYNTHESIS OF TRICYCLIC AND TETRACYCLIC THIAZOLOIMIDAZOLE ACETIC ACIDSJ. P. Anselme; A. S. Radhakrishna; K. D. Berlin
45-46AN IMPROVED PROCEDURE FOR SYNTHESIS OF 2-ACETYL-3-(2-METHYL-4-AMINOPYRIMIDIN-5-YL)METHYL-3A-METHYLPERHYDROFURO[2,3-D]THIAZOLEKhashayar Karimian; G. E. Risinger
46-48A CONVENIENT METHOD FOR THE PREPARATION OF 2-AMINO-3',4,4',5-TETRACHLOROBIPHENYLSunil K. Chaudhary; Phillip W. Albro
48-53SULTAMS WITH POSSIBLE SCHISTOSOMICIDAL ACTIVITY. PART VS. H. Doss; A. B. Sakla; M. Hamed

Volume 9, Issue 6 (1977)

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257-262CONVENIENT ONE-STEP CONVERSIONS OF ALCOHOLS OR PHENOLS TO N,N-DIPROPYL ALKOXYACETAMIDESIrving J. Borowitz; Ven-Shun Li; Irwin Gross
263-266DEOXYGENATION OF QUINOXALINE 1,4-DIOXIDES WITH TITANIUM TRICHLORIDEBerkeley W. Cue Jr.; John P. Dirlam; Edward A. Glaser
267-270SUGAR 1,3,4-OXADIAZOLES. IV: THE SYNTHESIS OF SUGAR 1,3,4-OXADIAZOLINE DERIVATIVESM. A. E. Shaban; M. A. M. Nassr; E. H. El. Ashry; V. N. Reinhold
271-276A CONVENIENT N-ACETYLATION OF INDOLESGordon W. Gribble; Laurence W. Reilly Jr.; Jerry L. Johnson
277-280AN IMPROVED SYNTHESIS OF 1-BENZOYL-4-KETO-1,2,2A,3,4,5-HEXAHYDROBENZ [cd]INDOLEDavid E. Nichols; J. Michael Robinson; George S. Li; John M. Cassady; Heinz G. Floss
281-284PREPARATION OF 2-PHENYLPERHYDROAZEPINES. Wawzonek; J. M. Shradel
285-288A SIMPLE SYNTHESIS OF 4-CYCLOHEXENE-1,2-cis-DIOL AND ITS USE AS THE PRECURSOR OF A FUNCTIONALIZED CYCLOHEXENONE SYNTHONGrant R. Krow; Richard Carmosin; Anthony Mancuso
289-296SYNTHESIS OF NITROXYL DERIVATIVES OF BENZO[a]PYRENEH. Schlude
297-299REDUCTIVE ALKYLATION OF ANILINE WITH 2-INDANONE AND 2-TETRALONEJack B. Campbell; E. R. Lavagnino
299-303SULTAMO-STEROIDS IIS. H. Doss; S. S. A. Dimitry
303-307ETHYL 2-(4-AMINOPHENYL) PROPIONATEM. Perchinunno; A. Guerrato; F. Pregnolato
309OPPI-CORRIGENDUM
311-318INDEXES

Volume 9, Issue 5 (1977)

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209-256PHOSPHORUS, ARSENIC, SILICON AND METAL DERIVATIVES OF THIOUREA. A REVIEWHerbert A. Friedman

Volume 9, Issue 4 (1977)

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159-164PREPARATION OF AN 8-AZAPROSTAGLANDIN SYNTHONP. A. Zoretic; B. Branchaud; N. D. Sinha
165-172SYNTHESIS OF SULTAM DERIVATIVES WITH POSSIBLE SCHISTOSOMICIDAL ACTIVITY. PART XII. SYNTHESIS OF KETOSULTAMSS. H. Doss
173-207USES OF THE TRIFYL GROUP IN ORGANIC SYNTHESIS. A REVIEWJames B. Hendrickson; Kenneth W. Bair; Raymond Bergeron; Aziz Giga; Paul L. Skipper; Daniel D. Sternbach; James A. Wareing

Volume 9, Issue 3 (1977)

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103-108AN EFFICIENT, GENERAL SYNTHESIS OF SPIROALKENES AND RELATED DERIVATIVESNicholas R. Natale; Robert O. Hutchins
109-115STUDIES DIRECTED TOWARD SYNTHESIS OF QUASSINOIDS - IV. D-RING CLEAVAGE OF CHOLIC ACID DERIVATIVES - 2Jerry Ray Dias; R. Ramachandra
117-124REACTIONS OF AROYLHYDRAZONES. III: OXIDATIVE CYCLIZATION OF CYCLOHEXANE-1,2-DIONE BIS(AROYLHYDRAZONES) TO SUBSTITUTED 1,2,3-TRIAZOLESM. Shaban; M. Nassr; E. El Ashry; M. Mustafa
125-130IMPROVED SYNTHESIS OF 2,6-DI-t-BUTYL-4-METHYLPYRYLIUM CHLOROSTANNATE AND PERCHLORATE AND OF 2,6-DI-t-BUTYL-4-METHYLPYRIDINEAlexandru T. Balaban
131-147CATECHOLBORANE IN ORGANIC SYNTHESIS. A REVIEWGeorge W. Kabalka
149-150PREPARATION OF PERDEUTERO 9,10-DIHYDROANTHRACENEG. M. Gorter-La Roij; J. Lugtenburg
151-153THE AlCl3 CATALYZED t-BUTYLATION OF HALOBENZENES WITH 2,6-DI-(t-BUTYL)-p-CRESOLM. Tashiro; T. Yamato
153-154SYNTHESIS OF 3-(2-METHYLPHENOXY)-AND 3-(2,6-DIMETHYLPHENOXY)PROPYNER. A. Malzahn; C. M. Peek; J. D. Woodyard
155-157A SIMPLE PREPARATION OF TRAUMATIC LACTONE. A PROSTANOID SYNTHONV. B. Deodhar; V. S. Dalavoy; U. R. Nayak
158OPPI-CORRIGENDUM

Volume 9, Issue 2 (1977)

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49-52SYNTHESIS OF THE SELECTIVE BLADDER CARCINOGEN, N-(n-BUTYL)-N-(3-CARBOXYPROPYL)NITROSAMINE (BCPN)William Gaffield; Larry K. Keefer; Peter P. Roller
53-56USE OF SODIUM CYANOBOROHYDRIDE IN THE SYNTHESIS OF BIRADICAL NITROXIDESElmer J. Rauckman; Gerald M. Rosen; W. Winn Hord
57-62COMPARISON OF SYNTHETIC ROUTES TO DL-CANALINETimo Korpela; Juhani Lundell; Paavo Pasanen
63-83DEXYGENATION OF SULFOXIDES. A REVIEWJozef Drabowicz; Tatsuo Numata; Shigeru Oae
85-87AN IMPROVED SYNTHESIS OF 5β-CHOLEST-3-ENED. T. C. Yang; G. W. Kabalka
87-89IMPROVED PROCEDURE FOR THE PREPARATION OF “OXAURACIL”, 2H-1,3(3H)-OXAZINE-2,6-DIONEJohn H. Macmillan
89-91NOVEL ACID HYDROLYSIS OF 2,3,5,6-DIEPOXY-2,5-DIMETHYL-1,4-BENZOQUINONEAspi B. Daruwala
91-94A RAPID AND MILD PROCESS FOR THE OXIDATION OF 2,3-DICHLORO-5,6-DICYANOBENZOQUINONE (DDQ) FROM 2,3-DICHLORO-5,6-DICYANOHYDROQUINONE (DDHQ)John W. Scott; David R. Parrish; Fred T. Bizzarro
94-96A BRIEF PREPARATION OF THIAN-4-CARBOXYLIC ACID 1,1-DIOXIDEE. Carlon; R. W. Draper; R. Friary
96-98AN EFFICIENT SYNTHESIS OF 4-HYDROXYBENZOTRIFLUORIDEE. R. Lavagnino; B. B. Molloy; J. W. Paschal
99-101SYNTHESIS OF NOPALINE AND ISO-NOPALINED. Cooper; J. L. Firmin

Volume 9, Issue 1 (1977)

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1-4N-DEMETHYLATION OF APOMORPHINE USING METHYL CHLOROFORMATEJack C. Kim
5-8A CONVENIENT METHOD FOR THE PREPARATION OF N-SUBSTITUTED 2(1H)-PYRIDONESC. S. Giam; Albert E. Hauck
9-11IMPROVED SYNTHESIS OF 3-DIMETHYLAMINOPYRIDINEC. S. Giam; Albert E. Hauck
13-14AN IMPROVED PROCEDURE FOR THE DISSOLVING METAL REDUCTION OF TWO BROMONITROPICOLINESF. L. Setliff; J. S. Greene
15-18SYNTHESIS OF SOME SPIRO α-METHYLENE-γ-LACTONESK. Ramalingam; K. D. Berlin
19-25SYNTHESIS OF 3-SUBSTITUTED-2,5-DIMETHYL-6-PYRROLIDINE-1,4-BENZOQUINONESAspi B. Daruwala; Ulfert Hornemann
27-33SYNTHESIS OF SULTAM DERIVATIVES WITH POSSIBLE SCHISTOSOMICIDAL ACTIVITY. PART IVS. H. Doss
35-38A NEW ROUTE TO 1,2-INDANEDIONEH. Harry Szmant; Raghunath Nanjundiah
39-41IMPROVED SYNTHESIS AND PURIFICATION OF N4-ETHYL-L-ASPARAGINER. W. Dineen; D. O. Gray; J. -P. Anselme
41-44AN IMPROVED SYNTHESIS OF 2-HETEROARYL-3-PHENYL-4(3H)-QUINAZOLINONEST. Hisano; K. Muraoka; M. Ichikawa
45-48NOVEL 1,3-DIARYLPYRAZOLINES AND PYRAZOLO[3,4-d]PYRIDAZINESF. Sauter; U. Jordis

Volume 8, Issue 6 (1976)

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245-248HALOGEN AS A READILY CLEAVABLE PROTECTIVE GROUP FOR REACTIVE POSITIONS IN PHENOLS AND PHENOLIC COMPOUNDSH. Kämmerer; G. Happel; V. Böhmer
249-262THE PREPARATION OF ALKYLPHENOLS USING t-BUTYL FUNCTION AS A POSITIONAL PROTECTIVE GROUPM. Tashiro; G. Fukata; T. Yamato; H. Watanabe; K. Oe; O. Tsuge
263-266THE t-BUTYLATION OF AROMATIC COMPOUNDS WITH 2,6-DI(t-BUTYL)-p-CRESOL. THE SELECTIVE SEPARATION OF p-XYLENE FROM C8 AROMATICSM. Tashiro; G. Fukata; T. Yamato
267-270C-ALKYLATION OF PHENOLS BY 2-HYDROXYBENZYLAMINE DERIVATIVESJ. Arct; J. Hetmanek
271-278APPROACHES TO THE SYNTHESIS OF 1-DIPHEIWLCYCLOPROPENYLIDENE-4-(CYCLOPEIMTADIENYLIDENE)-2,5-CYCLOHEXADIENET. Niem; M. D. Rausch
279-282THIENOQUINOLINES. PART V. AN IMPROVED SYNTHESIS OF 2,3-DIHYDROTHIENO[2,3-b]QUINOLINE AND ITS DERIVATIVESP. Shanmugam; T. K. Thiruvengadam; N. Soundararajan
283-2852-ETHYL-2-(3-NITRO-4-HYDROXYPHENYL)-GLUTARIMIDE AND 2-ETHYL-2-(4-HYDROXYPHENYL)-GLUTARIMIDEB. D. Andresen; M. D. Long; R. H. Hammer; H. L. Panzik
287-292HETEROCYCLES DERIVED FROM THE CONDENSATION OF HOMOPHTHALIC ANHYDRIDE WITH ETHYLENEDIAMINEHoracio Grinberg; Samuel Lamdan; Carlos H. Gaozza
293-297OXIDATIVE DEMETHYLATION OF 4,7-DIMETHOXYINDOLES. SYNTHESIS OF 4,7-INDOLOQUINONES FROM 4,7-DIMETHOXYINDOLESYunus A. Shaikh
299-302SYNTHESIS OF 2-BROMOSTYRENEY. Halpern; D. Meidar
302-305NEW 5-SUBSTITUTED-2-FURALDEHYDESD. R. Shridhar; C. V. R. Sastry; M. Jogibhukta; S. R. Moorty; N. K. Vaidya; P. G. Reddy
306-3077-SUBSTITUTED-2,4-DIPHENYL-3H-1,5-BENZODIAZEPINESRonald L. Amey; Ned D. Heindel
309-317INDEXES

Volume 8, Issue 5 (1976)

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205-210THE SYNTHESIS OF 1-AMIDINO-4-AROYLPIPERAZINESPhilip L. Southwick; Balram Dhawan
211-214MILD METHOD FOR ENAMINE FORMATIONP. A. Zoretic; F. Barcelos; B. Branchaud
215-217ELECTROLYTIC PREPARATION OF bis-DIMETHYL-2-HYDROXYPROPYLAMINEAZOBENZIMIDESS. Wawzonek; D. Aelony; W. J. McKillip
219-222N-ACETYL-L-TYROSINE ETHYL ESTERM. Dymicky
223-225IMPROVED PROCEDURE FOR THE DISSOLVING METAL REDUCTION OF INDOLE AND CARBAZOLEJ. W. Ashmore; G. K. Helmkamp
227-230DIRECT CONVERSION OF TRIMETHYLSILYLOXYALKANES TO ALKANOIC ESTERSDenys J. Voaden; Rolland M. Waters
231-236THE REDUCTIVE DEBROMINATION OF BROMOPHENOLSMasashi Tashiro; Gouki Fukata
237-239DICARBOXYLIC ACIDS FROM THE OXIDATIVE OZONOLYSIS OP HYDROXYMETHYLENE KETONES. AN IMPROVED PROCEDURED. T. C. Yang
239-241SIMPLE SYNTHESIS OF 3-t-BUTYLGLUTARIC ACIDM. Tlchy
241-243PARTIAL TRANSALKYLATION OF 3,3′,5,5′-TETRA-t-BUTYL-4,4′-DIHYDROXYBIPHENYLM. Tashiro; G. Fukata
243-2442-INDENECARBOXAMIDED. Tabak; P. A. M. de Oliveira

Volume 8, Issue 4 (1976)

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i-iiiHENRY GILMAN
149-153A CONVENIENT PREPARATION OF D(-)-p-HYDROXYPHENYLGLYCINER. F. Eizember; A. S. Ammons
155-158A SUPERIOR METHACYCLINE SYNTHESIS BY PHOSPHINE OR PHOSPHITE DEHALOGENATIONH. Faubl
159-161THE USE OF TRIMETHYLSULFONIUM IODIDE IN THE SYNTHESIS OF BIOLOGICALLY ACTIVE NITROXIDESElmer J. Rauckman; Gerald M. Rosen; Mohamed B. Abou-Donia
163-168REDUCTIVE METHYLATION OF HYDROXYBIPHENYL WITH ALUMINA AND METHANOLLeroy H. Klemm; Dennis R. Taylor
169-177SYNTHESIS OF 1, 3-DIVINYLAZULENESJ. O. Currie Jr.; R. A. Labar; R. D. Breazeale; A. G. Anderson Jr.
179-183SYNTHESIS OF α-GUAIACONIC ACID (FUROGUAIACIN)Robert Stevenson; John R. Williams
185-192PREPARATION OF 5-IMINO-2-PYRROLIDINONE DERIVATIVES AND THEIR 5-ALKYLIMINO ANALOGSWłdzimierz Koberda; Jerzy Lange
193-196SYNTHESIS OF 4′-VINYLBENZOCROWN ETHERSJ. Smid; B. El Haj; T. Majewicz; A. Nonni; R. Sinta
197-199PREPARATION OF N,N′-DIALKYLUREASS. Wawzonek
200-201DIAZOPYRROLINE AS SYNTHETIC INTERMEDIATE. A SYNTHESIS OF PYRAZOLO[1,5-c]PYRIMIDINESR. Madhav
203-204BOOK REVIEW

Volume 8, Issue 3 (1976)

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103-106THE N-DEMETHYLATION OF MORPHINE AND CODEINE USING METHYL CHLOROFORMATEGeorge A. Brine; Karl G. Boldt; Carolyn King Hart; Frank I. Carroll
107-112SACCHARIDE 1,3,4-OXADIAZOLESM. Shaban; M. Nassr
113-118SUGAR 1,3,4-OXADIAZOLES. III. THE SYNTHESIS OF 1,2,3,4-TETRA-O-ACETYL-1,4-BIS(5-ARYL-1,3,4-OXADIAZOL-2-YL)-GALACTO-TETRITOLSM. Shaban; M. Nassr
119-124REDUCTION OF SULFOXIDES WITH METHANE- AND p-NITROBENZENESULFINYL CHLORIDE BY OXYGEN TRANSFER REACTIONTatsuo Numata; Katsuyata Ikura; Yasutaka Shimano; Shigeru Oae
125-132SYNTHESIS OF 2-(1-NAPHTHYLMETHYL)-3,4-DIHYDRONAPHTHALENE, 2-(1-NAPHTHYLMETHYL)-1,2,3,4-TETRAHYDRONAPHTHALENE, 7a, 8, 9, 13b-TETRAHYDRO-7H-DIBENZ [a, k L] ANTHRACENE, AND 5,6-DIHYDRO-4H-DIBENZ[a, k L]ANTHRACENEL. L. Ansell; T. E. Webb; J. W. Burnham; E. J. Eisenbraun; M. C. Hamming; G. W. Keen
133-140THE SYNTHESIS OF 1,2,3,7,8,9-HEXAHYDRODIBENZO[def, mno]CHRYSENE AND THE USE OF HYDRIODIC ACID-RED PHOSPHORUS IN THE DEOXYGENATION OF KETONESL. L. Ansell; T. Rangarajan; W. M. Burgess; E. J. Eisenbraun; G. W. Keen; M. C. Hamming
141-143A RAPID, CONVENIENT, HIGH YIELD PROCEDURE FOR THE REGENERATION OF 2,3-DICHLORO-5,6-DICYANOBENZOQUINONE (DDQ) FROM THE CORRESPONDING HYDROQUINONE (DDHQ)Ki Hwan Kim; Gary L. Grunewald
143-146A SIMPLIFIED PROCEDURE FOR THE SYNTHESIS OF THE 6,7-BENZOMORPHAN NUCLEUSE. Bellora; E. Cereda; A. Donetti
146-148SYNTHESIS OF NEW PHENYLQUINOXALINESJ. A. Harvey; M. A. Ogliaruso
148DIETHYL 2,5-DI [BENZYLOXY] TEREPHTHALATES. Wawzonek; J. E. Durham

Volume 8, Issue 2 (1976)

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51-74SELECTIVE ELECTROPHILIC AROMATIC SUBSTITUTIONS VIA POSITIONAL PROTECTIVE GROUPS: A REVIEWM. Tashiro; G. Fukata
75-80THE PREPARATION OF OLEFINIC DERIVATIVES OF PHTHALIMIDE AND THEIR USE AS THE PRECURSORS FOR HOMOALLYLIC AMINESE. D. Bergmann; Y. Migron
81-84AN EFFICIENT SYNTHESIS OF (±)-MUSCONEStephen H. Korzeniowski; David P. Vanderbilt; Lawrence B. Hendry
85-86A CONVENIENT PREPARATION OF 1-AROYLPIPERAZINESMahesh Desai; Jeffrey W. H. Watthey; Marie Zuckerman
87-90THE REACTION OF 3,5-DIMETHYLISOXAZOLE WITH NITRITES AND NITROSO COMPOUNDSChoji Kashima; Yoshimori Omote; Koji Kawada; Yoshihiko Tsuda
91-92A SYNTHESIS OF 1-METHYL-2-ALLYLPYRROLEJ. C. Chen
93-952,4,6-TRICHLORO-m-TOLUIDINEC. S. Giam; K. Ueno; M. G. Merkle
95-98THE SYNTHESIS OF SOME NEW 3-METHYL-2-PYRAZOLIN-5-ONESHari G. Garg; Raj K. Gupta
98-102SYNTHESIS OF OXY AND THIOARYLENE BISNAPHTHALIC ANHYDRIDESG. A. Loughran; F. E. Arnold

Volume 8, Issue 1 (1976)

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1-5SYNTHESIS OF 3- (CARBOXYMETHYL) BENZOTHIAZOLINE-2-THIONEC. H. Chen
7-11CONCERNING THE SYNTHESIS OF 4-METHOXYINDAN-1-ONEA. Barco; S. Benetti; G. P. Pollini
13-18SYNTHESIS OF t-BUTYLKETONES BY USE OF PHENYLTHIO (t-BUTYL) CUPRATE (POSNER'S REAGENT)G. B. Bennett; J. Nadelson; L. Alden; A. Jani
19-23SELECTIVE N-SUBSTITUTION OF 2,6-DIMETHYLPIPERAZINEJose E. Saavedra; Gloria G. Lyle; Robert E. Lyle
25-32PSEUDOHALOGENS XXI. N-CHLORO AMIDES WITH ELECTRON-WITHDRAWING GROUPS ON NITROGENSandra C. Cottrell; Cyril Abrams; Daniel Swern
33-36CARBONYL COMPOUNDS FROM THE OXIDATION OF BENZYLAMMONIUM BROMIDES WITH DIMETHYL SULFOXIDEP. A. Zoretic; P. Soja; M. Jodoin; R. Levine
37-40SYNTHESIS OF NEW BIS-DIPHENYLACETYLENESJ. A. Harvey; M. A. Ogliaruso
41-44CONVENIENT PREPARATION OF 2,3-DIALKYLINDOLESVinod Dave
45-49SYNTHESIS OF 3,4-DIHYDROXYCINNOLINE AND A CONVENIENT PREPARATION OF N-AMINOOXINDOLEM. Lora-Tamayo; B. Marco; P. Navarro

Volume 7, Issue 6 (1975)

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261-266INTERNALLY BRANCHED 1,5,9-TRIMETHYLALKANESPhilip E. Sonnet
267-270THE SYNTHESIS OF BENZ[α]ANTHRACENEFahim U. Ahmed; T. Rangarajan; E. J. Eisenbraun; G. W. Keen; M. C. Hamming
271-275A CONVENIENT METHOD FOR SYNTHESIS OF 4 (3H)-QUINAZOLINONESTakuzo Hisano; Kiyokatsu Shoji; Masataka Ichikawa
277-282THE UTILITY OF BENZYL SODIUM AS A REAGENT IN ALCOHOL SYNTHESISWalter T. Smith Jr.; David L. Nickel
283-290PREPARATION OF 3-t-BUTYL-1,5-PENTANEDIOIC ACID AND OF 3-t,-BUTYL-1,5-PENTANEDIOL DITOSYLATEW. R. Purdum; K. D. Berlin
291-296PREPARATION OF 1-ARYL-3-(TETRA-0-ACETYL-2-DEOXY-D-GLUCOS-2-YL)UREASNed D. Heindel; H. Donald Burns; Takashi Honda; Victor R. Risch; Luther W. Brady
297-303SYNTHESIS OF A PROSTANOIC ACID ANALOGB. Crammer; Z. Aizenshtat; R. Ikan
305-308SYNTHESIS OF METHYL-2-OXO-3-PENTYLCYCLOPENTYL-1-ACETATEJames A. Moore; Uzi Ravid; Raphael Ikan
309-310DI-ISOPROPYLPHOSPHINODITHIOIC ACIDJames L. Corbin; William E. Newton; John W. McDonald
311-312IMPROVED SYNTHESIS AND PURIFICATION OF p-METHOXYBENZAL-p-(n-BUTYL)ANILINE (MBBA)N. V. V. Raghavan; L. A. Paddock
313-325INDEXES

Volume 7, Issue 5 (1975)

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215-219THE SUCCESSFUL SYNTHESIS OF GLYCYL-GLYCINE PEPTIDE BONDS VIA THE EXCESS MIXED ANHYDRIDE METHODJ. A. Hoffman; M. A. Tilak
221-224SYNTHESIS OF TWO TOXIC 4-IPOMEANOL ANALOGSDominic T. C. Yang; S. W. Pelletier
225-229SYNTHESIS OF 2,3-DIHYDRO-3-METHYL-1-(2-NAPHTHYL)-1H-BENZ[E]INDENE AND 1,1,3-TRIMETHYL-3-PHENYLINDANW. P. Duncan; E. J. Eisenbraun; A. R. Taylor; G. W. Keen
231-236STUDIES ON POSITIONAL PROTECTIVE GROUPS. IV. A NEW PREPARATIVE METHOD FOR DIHYDROXYDIPHENYLMETHANES WITH THE T-BUTYL GROUP AS A PROTECTIVE GROUPM. Tashiro; G. Fukata; S. Mataka; K. Oe
237-242STUDIES ON POSITIONAL PROTECTIVE GROUPS. VII. A NEW PREPARATIVE METHOD FOR 2,2'-DIHYDROXYDIPHENYLMETHANES WITH THE CHLORO OR BROMO GROUPS AS A PROTECTIVE GROUPM. Tashiro; G. Fukata; K. Oe
243-250THE PREPARATION OF DIHYDROXYDIPHENYLMETHANES CONTAINING NITRO GROUPS. II. UNSYMMETRICALLY SUBSTITUTED COMPOUNDSV. Böhmer; W. Lotz
251-253A CONVENIENT PREPARATION OF 4-ARYL-1,2,4-TRIAZOLINE-3,5-DIONESHeinrich Wamhoff; Klemens Wald
255-259POSITIONAL PROTECTIVE GROUPS VIII. PREPARATION OF 2-HYDROXY-3,2′-DIMETHYLDIPHENYL ETHER WITH T-BUTYL GROUP AS A POSITIONAL PROTECTIVE GROUPM. Tashiro; H. Watanabe; K. Oe; O. Tsuge

Volume 7, Issue 4 (1975)

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155-158SYNTHESIS OF CHLOROCARBONYL KETENESSusumu Nakanishi; Kenneth Butler
159-162THIOCHROMONE 1-OXIDEIan W. J. Still; P. C. Arora; S. N. Sokolowsky
163-164FACILE REDUCTION OF SULFOXIDES WITH SODIUM BIS(2-METHOXYETHOXY) ALUMINUM HYDRIDETse-Lok Ho; C. M. Wong
165-172SYNTHESIS OF NITRONUCLEOSIDESTai-Shun Lin; Robert E. Harmon
173-177STUDIES OF ACENAPHTHENE DERIVATIVES. XXIX. THE REACTION OF CARBONYL-STABILIZED SULFONIUM AND PHOSPHONIUM YLIDES WITH 2-DIAZOACENAPHTHENONEOtohiko Tsuge; Masahiro Koga
179-181AN IMPROVED SYNTHESIS OF SUBSTITUTED 1,3,4-THIADIAZOLESE. V. P. Tao; C. F. Christie Jr.
183-188STUDIES ON POSITIONAL PROTECTIVE GROUPS. V. A NEW PREPARATIVE METHOD FOR 4,4′-DIHYDROXY DIPHENYLMETHANES WITH THE CHLORO OR BROMO GROUPS AS A PROTECTIVE GROUPM. Tashiro; G. Fukata; K. Oe
189-192STUDIES ON POSITIONAL PROTECTIVE GROUPS. VI. THE PREPARATION OF 2,6-DICHLORO- AND 2,6-DIBROMOPHENOL FROM THE CORRESPONDING TETRAHALOGEN SUBSTITUTED BISPHENOL AM. Tashiro; H. Watanabe; K. Oe
193-199THE SYNTHESIS OF SOME NEW DIARYL ETHERSR. E. Buhts; D. K. Chesney; J. R. Handley; F. D. Popp; D. C. Smith
201-206R,S-4-(4'-METHOXYBENZYLIDENEAMINO) PHENYLALANINE AND R,S-4-(2'-METHYL-4'-NITROPHENYLAZO) PHENYLALANINEJames A. Moore; C. A. Panetta; C. H. Yang
207-210THE CYCLIC OXALATE ESTERS OF CIS- AND TRANS-1.2-CYCLOHEXANEDIOLSWinston D. Lloyd; Barney J. Navarette; Michael F. Shaw
211-213SYNTHESIS OF STEROIDAL NITROIMIDAZOLESJ. E. Herz; Rafael Silva Torres

Volume 7, Issue 3 (1975)

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103-110AN EFFICIENT ROUTE TO XANTHOBILIRUBIC ACID, AN OXODIPYRRYLMETHENEJ. O. Grunewald; R. Cullen; J. Bredfeldt; E. R. Strope
111-115HETEROCYCLIC DERIVATIVES FROM SUGARS VIII. PREPARATION OF 1-(N-METHYL-N-PHENYL)-AMINO-1-DEOXY ALDITOLSR. Bogńar; P. Herczegh
117-122SYNTHESIS OF METABOLITES OF PHENOBARBITAL AND MEPHOBARBITALAbraham Philip; F. I. Carroll
123-127THE SYNTHESIS OF 2,3,7,8-TETRAAMINODIBENZOTHIOPHENE-5,5-DIOXIDEF. E. Arnold
129-136THE TOTAL SYNTHESIS OF DL-PHYLLODULCINY. Naoi; S. Higuchi; H. Ito; T. Nakano; K. Sakai; T. Matsui; S. Wagatsuma; A. Nishi; S. Sano
137-144PREPARATION OF ALKYNESJ. R. Sowa; E. J. Lamby; E. C. Calamai; D. A. Benko; A. Gordinier
145-1483- AND 4-(7-BENZ[A]ANTHRACENYL)PHENYL-2-IMIDAZOLINES, 3- AND 4-(9-ANTHRACENYL)PHENYL-2-IMIDAZOLINES, AND THEIR HYDROCHLORIDE SALTSF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
149-154BROMINATION OF UNSYMMETRICAL KETONES WITH CUPRIC BROMIDE. PRODUCT DEPENDENCE ON REACTION CONDITIONSJill H. Paul; Rubin Silverman; Leonard H. Schwartz

Volume 7, Issue 2 (1975)

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55-59SYNTHESIS OF SOME 1,2,4-THIADIAZOLO[2,3-a] PYRIDINE DERIVATIVES AND ITS AZA ANALOGUESB. Koren; B. Stanovnik; M. Tisler
61-655-METHYL- AND 5-PHENYL-1-AMINOTETRAZOLESK. Sakai; J. P. Anselme
67-70IMPROVED SYNTHESES OF PICRYLHYDRAZINE AND OF THE PICRYLHYDRAZONES OF ACETONE AND OF ACETALDEHYDETerence C. Morrill; Ann Ryer Bayley
71-74A CONVENIENT SYNTHESIS OF SUBSTITUTED PHENOLS BY THE YATES-HYRE PROCEDUREErnest A. Harrison Jr.
75-78A FACILE ROUTE TO BENZO[b]BICYCLO[3.2.2]NONENE DERIVATIVESIleana Dragutan; Ecaterina Cioranescu
79-83A SYNTHESIS OF TAIWANIN CRiaz Ahmed; Robert Stevenson
85-88A CONVENIENT PREPARATION OF MONOAROYLPIPERAZINE HYDROCHLORIDESBalram Dhawan; Philip L. Southwick
89-91AN IMPROVED SYNTHESIS OF L-γ-GLUTAMYL-4-NITROANILIDEJames A. Moore; Harold Lindsay; John F. Whitaker
92-973- AND 4-(7-BENZ[a]ANTHRACENYL)BENZAMIDES AND CYANOBENZENES AND 3- AND 4-(9-ANTHRACENYL)BENZAMIDES AND CYANOBENZENESP. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
98-101THE SYNTHESIS OF 5-METHYL- AND 5,5-DIMETHYL-5H-DIBENZO[a,d]CYCLOHEPTENEM. Vinatoru; M. Elian; Ecaterina Cioranescu

Volume 7, Issue 1 (1975)

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iNOTICE
iiPREFACEJ. P. Anselme
1-51-ACYL-4-SUBSTITUTED PIPERAZINESJames A. Moore; E. A. Steck
6-11SOME BENZIMIDAZOLE DERIVATIVESEdgar A. Steck; R. Pauline Brundage
11-14SYNTHESIS OF METHYL 2,3,4-TRI-0-ACETYL-6-DEOXY-6-IODO-α-D-GLUCOPYRANOSIDETai-Shun Lin; Robert E. Harmon
14-16AN IMPROVED SYNTHESIS OF 2-ETHYL-2-PHENYL-GLUTACONIMIDEHassan Y. Aboul-Enein
16-21THE SYNTHESIS OF STEROLS WITH MODIFIED SIDE CHAINS BY THE WITTIG REACTIONJ. E. Herz; S. M. Cruz
21-22THE SPECTRAL CHARACTERIZATION OF endo-4-OXATRICYCL[5,2,1,02,6]DEC-2-ENEBradford P. Mundy
23-26NEW MIXED KETENE DIALKYL ACETALSG. R. Cliff; D. J. Dunn
26-304H-BENZPYRANO [3,4-d]OXAZOL-4-ONES AND 3-[N,N-BIS(CARBOXYMETHYL)AMINO]-4-HYDROXYCOUMARIN DERIVATIVESM. Trkovnik; M. Kules; K. Krunic
31-34HYDROGENOLYSIS OF ARYL HALIDES IN THE PRESENCE OF RANEY NICKEL IN ALKALINE MEDIUMA. J. De Koning
35-37SYNTHESIS OF DIMETHYL 1,2-DIHYDROPYRIDAZINE-1,2-DICARBOXYLATEL. J. Altman; M. F. Semmelhack; R. B. Hornby; J. C. Vederas
39-42A NEW PORPHINOGEN TYPE COMPOUNDO. Tsuge; M. Tashiro; Y. Kiryu
43-46STUDIES ON POSITIONAL PROTECTIVE GROUPS III. A NEW PREPARATIVE METHOD FOR CHLOROPHENOLS WITH THE BROMO GROUP AS A PROTECTIVE GROUPM. Tashiro; H. Watanabe; O. Tsuge
47-50ELECTROCHEMICAL SYNTHESIS OF 3-AMINO-4-HYDROXYCOUMARINM. Trkovnik; M. Laćan; Z. Stunić; D. Nahmijaz
51-54ROBINSON ANNELATION WITH A β-HYDROXYKETAL IN THE PRESENCE OF AN ACIDP. A. Zoretic; B. Branchaud; T. Maestrone

Volume 6, Issue 6 (1974)

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259-263A SIMPLE, TWO STEP SYNTHESIS OF 1-(2-CHLOROETHYL)-1-NITROSO-3-(D-GLUCOS-2-YL) UREAH. Donald Burns; Ned D. Heindel
265-267PREPARATION OF 3, 6-EXO-OXO-HEXAHYDROPHTHALIDEHumberto Cervantes Cuevas; Federico García Jiménez
269-273cis-OLEFINS FROM THE WITTIG REACTIONP. E. Sonnet
275-280A CONVENIENT PREPARATION OF HOMOGENEOUS 2,3,6-TRICHLOROBENZOIC ACID AND ITS CONVERSION TO 2,2′,3,3′,6,6′-HEXACHLOROBIPHENYLLouis A. Levy
281-285N-BENZOYLBENZILIMINEPeter Yates; E. M. Levi
287-293SYNTHESIS OF 2-METHOXYDIBENZO [b,f] (1,4)-THIAZEPIN-11(10H)-ONE-5,5-DIOXIDEO. Francis Bennett; James Johnson; John Tramondozzi
295-298PREPARATION OF 1,2,3-TRIAZOLO[4,5-f]QUINOLINE N-OXIDES FROM 6-NITRO-5,8-DIMETHOXYQUINALDINEPaul C. Unangst; Ned D. Heindel
299-303REDUCTIVE ALKYLATION OF ACRYLONITRILES AND ACRYLATEST. Caronna; A. Citterio; A. Clerici; R. Galli
305-311HYDROXYL GROUP ELIMINATION IN THE MORPHINE SERIESR. Bognár; Gy. Gaál; P. Kerekes; G. Horváth; M. T. Kovács
313-324INDEXES

Volume 6, Issue 5 (1974)

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207-210SYNTHESIS OF OPTICALLY ACTIVE N-(p-TOLUENESULFONYL)-SULFOXIMINE BY SULFOXIDE AND CHLORAMINE T—COPPERM. Moriyama; T. Numata; S. Oae
211-214O-p-METHOXYBENZYL-L-TYROSINEB. Rzeszotarska; K. Weber
215-2161-ETHOXYMETHYLENEAZULENIUM PERCHLORATESE. C. Kirby
217-220SYNTHESIS OF cis-4-OCTENE-1,8-DIOIC ACID AND ITS ESTERSA. Barco; S. Benetti; G. P. Pollini; R. Taddia
221-230A CONVENIENT PREPARATION OF DISSYMMETRIC TERTIARY PHOSPHINES VIA ALKYLATION OF DISSYMMETRIC LITHIUM PHOSPHIDESTheodore E. Snider; Don L. Morris; W. Ronald Purdum; G. A. Dilbeck; K. D. Berlin
231-233A NEW SYNTHESIS OF 2,5-DI-t-BUTYL-5,6-DICHLORO-1,4-CYCLOHEXENEDIOINEMircea D. Gheorghiu; Margareta Avram
235-238AN IMPROVED SYNTHESIS OF GUANYLUREIDO ACIDSSusumu Nakanishi
239-242PREPARATION OF THE ISOMERIC BENZYLQUINOLINESEllis V. Brown; Andrew C. Plasz; Russell Isbrandt; Henry H. Bauer
243-250REACTION OF 3-SUBSTITUTED AND 3,5-DISUBSTITUTED PYRIDINE N-OXIDES WITH PHENYL ISOCYANATETakuzo Hisano; Toshikazu Matsuoka; Masataka Ichikawa
251-253AN IMPROVED PROCEDURE FOR THE META-BROMINATION OF AROMATIC CARBONYL COMPOUNDSRichard F. Eizember; A. S. Ammons
255-258AN IMPROVED SYNTHESIS OF 2,4-DIOXO-3,8-DIOXABICYCLO[3.2.1]OCTANEJ. A. Moore; James E. Kelly

Volume 6, Issue 4 (1974)

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161-167THE FORMATION OF 1H-DIBENZO[b,g][1,4,5]TRIAZAPENTALENE FROM 2-(o-NITROPHENYL)- AND 2-(o-AZIDOPHENYL)-2H-INDAZOLEOtohiko Tsuge; Hideo Samura
169-173SYNTHESIS OF SOME SUBSTITUTED BROMOANISOLESElizabeth A. Mawdsley; K. D. Berlin
175-178PREPARATION OF trans-2-OCTADECENOIC ACIDDavid R. Howton
179-182PREPARATION OF 2-HYDRAZINOBENZOTHIAZOLES BY EXCHANGE AMINATIONC. J. Barnett; J. C. Smirz
183-184AN IMPROVED METHOD FOR THE PREPARATION OF DIPHENYLACETYLENEJ. R. Sowa; E. G. Calamai
185-191SYNTHESIS OF THE PRECURSORS OF PHENANTHROINDOLIZIDINE ALKALOID ANALOGUESTai-Shun Lin; Robert E. Harmon; Wayne Pierantoni; Joseph C. W. Su
193-196IMPROVED TWO-STEP SYNTHESIS OF ETHYL CYCLOPROPANECARBOXYLATE AND CYCLOPROPANECARBOXYLIC ACIDStanley C. Bunce; Ronald A. Kent
197-2011,5-BENZOD IAZEP IN-2(1H)-ONESR. T. Blickenstaff; N. Wells
203-206REGIOSELECTIVE BECKMANN REARRANGEMENTN. Wakabayashi; Rolland M. Waters; M. W. Law

Volume 6, Issue 3 (1974)

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103-106CATALYTIC REDUCTION OF 1,1,1-TRIS(AZIDOMETHYL)ETHANE TO 1,1,1-TRIS(AMINOMETHYL)ETHANEL. J. Zompa; J. P. Anselme
107-115STUDIES ON POSITIONAL PROTECTIVE GROUPS ON AROMATIC RINGS I. A NEW PREPARATIVE METHOD FOR HALOPHENOLS WITH THE t-BUTYL OR BENZYL GROUP AS A PROTECTIVE GROUPM. Tashiro; H. Watanabe; O. Tsuge
117-122STUDIES ON POSITIONAL PROTECTIVE GROUPS ON AROMATIC RINGS II. A NEW PREPARATIVE METHOD FOR DIHYDROXYDI-PHENYLS WITH t-BUTYL GROUP AS A PROTECTIVE GROUPM. Tashiro; H. Watanabe; O. Tsuge
123-130THE PREPARATION OF DIHYDROXYDIPHENYLMETHANE DERIVATIVES CONTAINING NITRO GROUPS. I. SYMMETRICALLY SUBSTITUTED COMPOUNDSW. Lotz; V. Böhmer
131-1344-METHYLPENT-4-EN-2-ONE (iso-MESITYL OXIDE)R. D. Gillard; B. T. Heaton; M. P. Pilbrow
135-1391,5-DIMETHYLTETRAZOLEF. E. Condon; Robert Waldman; Nitya Kundu; J. P. Trivedi
141-144THE STUDIES ON DIHYDROISOCOUMARIN (III). THE SYNTHESIS OF 3-(3′-HYDROXY-4′-METHOXYPHENYL)-3,4-DIHYDROIROCOUMARINY. Naoi; K. Sakai; T. Nakano; H. Ito; S. Higuchi; T. Matsui; Y. Takahashi; S. Wagatsuma; A. Nishi; S. Sano
145-147NEW 2,4- AND 4,5-DIALKYLOXAZOLESJames A. Moore; P. B. Terentiev; A. N. Kost; N. P. Lomakina; V. G. Kartev
148-1494-(α,β-DIBROMOETHYL)PHENYLPHOSPHONIC ACIDM. A. Rea; T. L. Slapar; W. A. Trinler
149-1533,4-DIALKYLQUINOLINES BY AN EXTENSION OF THE BEYER SYNTHESISPaul A. Claret; A. G. Osborne
153-1562-CYCLOHEXYLIDENECYCLOPENTANONERichard D. Sands
156-1574-AMINO-3-HYDRAZINO-5-MERCAPTO-1,2,4-TRIAZOLER. G. Dickinson; N. W. Jacobsen
159CORRIGENDA

Volume 6, Issue 2 (1974)

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53-56BECKMANN REARRANGEMENTS USING THE CARBON TETRACHLORIDE-TRIPHENYLPHOSPHINE REAGENTRolland M. Waters; N. Wakabayashi; E. S. Fields
57-62REACTION OF 4-HOMOADAMANTENE WITH DICHLOROCARBENETadashi Sasaki; Shoji Eguchi; Masato Mizutani
63-66AN IMPROVED PROCEDURE FOR THE PREPARATION OF SOME METHYLENE CYCLOPROPENESTheophil Eicher; Theodor Pfister; Nils Krüger
67-68A CONVENIENT SYNTHESIS OF PHTHALAZINES. D. Carter; G. W. H. Cheeseman
69-72PREPARATION OF N,N-DIMETHYLHYDRAZIDESStanley Wawzonek
73-75DIRECT SYNTHESIS OF TRIOCTANOIN FROM GLYCEROL AND OCTANOIC ACIDArthur Furst; Jefferson W. Davis Jr.; Boleslaw L. Dunicz
77-102α-HALO SULFOXIDES. A REVIEWClifford G. Venier; Howard J. Barager III

Volume 6, Issue 1 (1974)

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1-3N-CARBOXYMETHYL-1,2-BENZISOTHIAZOLIN-3-ONE-1,1-DIOXIDEC. S. Giam; R. A. Lockhart
5-9FACILE SYNTHESIS OF α-SUBSTITUTED MALONATESGury Zvilichovsky; Upinder Fotadar
11-13A CONVENIENT SYNTHESIS OF THE PYRROLO[1,2-a]OUINOLINE RING SYSTEMEdward E. Garcia
15-18DIBENZO -[a,j] – XANTHYLIUM CHLORIDEG. Casiraghi; G. P. Gardini; G. Palla
19-24A SIMPLE SYNTHESIS OF ALICYCLIC Trans-GLYCOLS VIA HYDROBORATION OF SILYL ENOL ETHERSHiromichi Kono; Yoichiro Nagai
25-29THE SYNTHESIS OF ARYLAZOTRIPHENYLSILANESHamao Watanabe; Makoto Matsumoto; Yasuo Cho; Yoichiro Nagai
31-35A NEW SYNTHESIS OF Δ2-STEROIDSM. Fetizon; M. Jurion; A. Nguyen Trong
37-43A FACILE AND UNIFORM PROCEDURE FOR THE LARGE-SCALE PREPARATION OF SOME N-ALKYLRHODANINESF. E. Condon; D. Shapiro; P. Sulewski; I. Vasi; R. Waldman
45-47SIMPLE RE-USABLE “AMPULES” FOR MICRO-REACTIONSJefferson T. Eaton; Gordon W. Gribble
49-51A SIMPLIFIED PREPARATION OF CIS-1,3-CYCLOPENTANEDICARBOXYLIC ACIDRonald D. Clark

Volume 5, Issue 6 (1973)

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255-260FERROCENES FROM CYCLOPENTADIENES. 1,1′-DIMETHYLFERROCENEIlgvars J. Spilners; Robert J. Hartle
261-264SYNTHESIS OF 5-BENZOYL-6-PHENYL-1,3-0XAZINONES+ (SYNTHESES OF HETEROCYCLES, 179.)G. Kollenz; E. Ziegler; W. Ott
265-269SYNTHESIS OF α-AMINO-β-(p-HYDR0XYPHENOXY) PROPIONAMIDE HYDROCHLORIDES. Wawzonek; W. P. Gaffield Jr.
271-2732,4,6-TRINITRORESORCINOLB. A. Bydal
275-279AN IMPROVED STEREOSELECTIVE REDUCTION FOR THE PREPARATION OF endo-7-PHENYLNORCARANEPaul R. Morris; James D. Woodyard
281-284METHYLAMINOACETONE ETHYLENE KETAL HYDROCHLORIDEF. Benington; R. D. Morin
285-290THE SYNTHESIS OF 5-TERT-BUTYL-1,2,3,4-TETRAHYDRONAPHTHALENEJ. W. Burnham; W. P. Duncan; E. J. Eisenbraun; G. W. Keen; M. C. Hamming
291-298SYNTHESIS OF POLYMETHOXY-1-TETRALOUESTheodore E. Snider; Mohamed M. Hashem; K. D. Berlin; R. W. Chesnut; N. N. Durham
299-301AN IMPROVED SYNTHESIS OF 1,4-DIHYDRO-3-[2H]-ISOQUINOLONER. E. Lyle; D. A. Walsh
303-304exo-TRICYCLO[4.2.1.02,5] NON-7-EN-3-ONERoy C. De Selms
305-306AN IMPROVED SYNTHESIS OF 2-IODO-5-NITROPYRIDINEFrank L. Setliff
307-318INDEXES

Volume 5, Issue 5 (1973)

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203-207SYNTHESIS OF PURE ARYLKETONE CYANOHYDRINS AND ARYLKETONES FROM AROMATIC ALDEHYDESM. Makosza; T. Goetzen
209-213IMPROVED SYNTHESIS OF 2,4,4,6-TETRACHLORO-2,5-CYCLOHEXADIENONE AND OF 2,2,4,5,6,6-HEXACHLORO-3-CYCLOHEXENONEP. Švec; A. M. Sørensen; M. Zbirovský
215-217A NEW SYNTHESIS OF NORADAMANTANEJohn S. Wishnok; Paul v. R. Schleyer
219-224ETHYLHYDRAZINE. THE FISCHER SYNTHESIS REVISITEDF. E. Condon; D. C. Thakkar
225-232ETHYLMETHYLAMINE, ETHYLMETHYLNITROSAMINE AND 1-ETHYL-1-METHYLHYDRAZINEF. E. Condon; Daniel G. Shapiro
233-244THE TWENTY METHYL- AND ETHYL-SUBSTITUTED HYDRAZINESF. E. Condon; D. C. Thakkar; Tamara Briks Goldstein
245-249A SHORTER SYNTHESIS OF 5-THIO-α-D-GLUCOSE PENTAACETATEM. M. A. Abd El-Rahman; Roy L. Whistler
251-2532,3,6-TRI(ACETOXYMERCURI)-4-(TRIMETHYLAMMONIUM)ANILINIUM DIACETATE BY DIRECT TRIACETOXYMERCURATIONH. A. Friedman; G. B. Koelle

Volume 5, Issue 4 (1973)

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145-193RECENT STUDIES ON THE MODIFIED NIEMENTOWSKI 4-QUINAZOLONE SYNTHESIS. A REVIEWTakuzo Hisano
195-196OPPI BRIEFS: N-ISOHEXYL-N-METHYLAMINES. Wawzonek; S. M. Heilmann
197-1992,1-BenzisothiazolesM. Davis; E. Homfeld; T. Paproth
199-202ESTERS OF (±)HEXAHYDRO-5-HYDROXYMETHYL-2H-AZEPIN-2-ONEC. G. Overberger; J. H. Kozolwski

Volume 5, Issue 3 (1973)

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105-1073-(5)ALKYL PYRAZOLEST. Caronna; L. Filini
109-112tert-ALKYLATION OF PYRIDINE N-OXIDEF. Bertini; T. Caronna; M. Cecere
113-116A HIGH-DILUTION APPARATUS FOR THERMALLY UNSTABLE REACTANTSD. F�rcaşiu
117-124DANSYL AMINO ACIDSA. Chimiak; T. Połoński
125-128AN IMPROVED SYNTHESIS OF THE ISOMERIC AMINODIBENZOFURANSE. V. Brown; R. L. Coleman
129-132ORGANIC ELECTROSYNTHESES VII. CONVENIENT PREPARATION OF p-AMINOBENZYLCYANIDE BY CATHODIC REDUCTION OF p-NITROBENZYLCYANIDEPalle E. Iversen; J. H. P. Utley; S. O. Yeboah
133-134IMPROVED SYNTHESIS OF 6H,12H-DIBENZO[b,f][1,5]DITHIOCINAbdullatif K. Youssef; Michael A. Ogliaruso
135-139A CONVENIENT ROUTE TO AMINOSILANES USING HYDROSILANE-RHODIUM(I) COMPLEX COMBINATIONSHiromichi Kono; Iwao Ojima; Makoto Matsumoto; Yoichiro Nagai
141-143A HIGHLY EFFICIENT SYNTHESIS OF 3,4,5-TRIBROMO-N,N,α-TRIMETHYLPYRAZOLE-1-ACETMIDEG. Kornis; E. Nidy

Volume 5, Issue 2 (1973)

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49-54THE BECKMANN AND SCHMIDT REARRANGEMENTS OF 6-OXO-MORPHINE ALKALOIDSR. Bognár; S. Makleit; L. Radics; I. Seki
55-58ON THE PREPARATION OF α-KETOADIPIC ACIDRandall B. Nelson; Gordon W. Gribble
59-63PARTIAL SYNTHESIS OF GLOCHIDONEAntonio S. Samson; Robert Stevenson
65-70STUDIES ON DIHYDROISOCOUMARIN (I). A PRACTICAL SYNTHESIS OF 3-HYDROXYHOMOPHTHALIC ACIDS. Wagatsuma; S. Higuchi; H. Ito; T. Nakano; Y. Naoi; K. Sakai; T. Matsui; Y. Takahashi; A. Nishi; S. Sano
71-74IMPROVED SYNTHESIS OF tert-BUTYL 8-QUINOLYL CARBONATEBarbara Rzeszotarska; Stanislaw Wiejak; Krzysztof Pawelczak
75-80A HIGHLY SELECTIVE EPOXY CLEAVAGE OF 1-(5′-O-BENZOYL-2′,3′-EPOXY-β-D-LYXOSYL)URACIL WITH PYRIDINE HYDROCHLORIDETadashi Sasaki; Katsumaro Minamoto; Naoto Kidokoro
81-85STUDIES ON DIHYDROISOCOUMARIN (II). A NOVEL STOBBE-LIKE CONDENSATION CATALYZED BY 1,8-DIAZABICYCLO[5.4.0]-UNDECENE-7 (DBU)Y. Naoi; H. Ito; T. Nakano; S. Higuchi; K. Sakai; T. Matsui; S. Wagatsuma; Y. Takahashi; A. Nishi; S. Sano
87-93STRUCTURAL ASSIGNMENT OF CYCLIC PRODUCTS FROM 1,2-DICARBOXYLIC ANHYDRIDES AND HYDRAZINE. S,S-DIMETHYL SULFOXIMIDESB. Stanovnik; M. Tisler
95-103ISOLATION AND CHARACTERIZATION OF TWO PRIMARY CYCLOADDUCTS FROM THE REACTION OF PHENYLISOCYANATE WITH 3-PICOLINE-N-OXIDETakuzo Hisano; Shin Yoshikawa; Keiji Muraoka

Volume 5, Issue 1 (1973)

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1-41,5-DIBROMO- 3-tert-BUTYLPENTANEHideki Sakurai; Masashi Murakami
5-7AN IMPROVED SYNTHESIS OF L-HISTIDINOLK. W. Bentley; E. H. Creaser
9-12ALKYLATION OF LITHIUM ALUMINUM HYDRIDE REDUCTION PRODUCTS OF AMIDESS. Wawzonek; S. M. Heilmann
13-15SYNTHESIS OF 6,7-BENZO-2-AZABICYCLO[3.2.0]HEPTAN-3-ONEAilton de Sousa Gomes; A. M. Figueiredo
17-20A SIMPLE AND MILD PROCEDURE FOR THE REDUCTION OF 3-HYDROPEROXYINDOLENINES TO 3-HYDROXYINDOLENINESC. A. Mudry; A. R. Frasca
21-23SELECTIVE AIR OXIDATION OF ETHYLBENZENE TO ACETOPHENONEJozef Sliwiok; Leonard Ogierman
25-29DIETHYL CYCLOPROPANEMALONATERichard W. J. Carney; Janice Wojtkunski
31-35PREPARATION OF DL -threo - AND DL- erythro - 3,5 - DIAMINOHEXANOIC ACIDV. Krasnobajew; E. A. Rimerman; H. A. Barker
37-391,6 - BIS (HYDROXYMETHYL) PYRENE AND 1 - BROMO - 6 - HYDROXYMETHYLPYRENEGail D. Mulligan
41-43A SIMPLIFIED SYNTHESIS OF CIS-PENT-2-EN-4-YN-1-OLJ. A. Kepler; R. C. Strickland
45-48A NEW IMPROVED SYNTHESIS OF β-PHORONEJohn N. Marx

Volume 4, Issue 6 (1972)

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253-256SYNTHESIS OF 3,6-DIHYDROXY-4-PYRIMIDINONES (SYNTHESES OF HETEROCYCLES, 173.)W. Steiger; A. Argyrides; E. Ziegler
257-259DEHYDROABIETIC ACIDGoverdhan Mehta; Surinder K. Kapoor
261-263AN IMPROVED SYNTHESIS OF 1,4-DIISOPROPENYLBENZENE VIA 1,4-BIS (1-BROMO-1-METHYLETHYL) BENZENECharles F. Hobbs; Dudley E. McMackins
265-267A CONVENIENT SYNTHESIS OF 2-ACETYLDIHYDROBENZOFURANTse-Lok Ho; C. M. Wong
269-272A CONVENIENT PREPARATION OF DIPHENYLISOBENZOFURAN AND DIPHENYLISOBENZOTHIOPHENEK. T. Potts; A. J. Elliott
273-281STUDIES OF POLYAZAPENTALENES. II. THE PREPARATION OF 1,3a, 6a-TRIAZAPENTALENESO. Tsuge; H. Samura
283-288CHLOROMETHYLATION OF NITROPHENOLS WITH CHLOROMETHYL METHYL ETHERV. Böhmer; J. Deveaux
289-292AN IMPROVED HYDROGENATION FOR THE PREPARATION OF TETRAHYDROFURAN CIS-2, 5-DICARBOXYLIC ACIDJ. A. Moore; James E. Kelly
293-2962-NITROHOMOSYRINGIC ACIDR. M. Sotelo; D. Giacopello; M. J. Vernengo
297-2993-(2′-FORMYL-3′-METHOXYPHENYL)PROPIONIC ACIDT. -L. Ho; I. Chang; C. M. Wong
299-300ZINC ETHYL ACETOACETATEJ. Perz; J. Mehaffey
300-301NITRATION OF ALKYLPHENOLS WITH DINITROGEN TETROXIDEE. V. P. Tao; C. F. Christie Jr.
303-320INDEXES

Volume 4, Issue 5 (1972)

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211-213A CONVENIENT SYNTHESIS OF 2, 3, 6, 7-TETRAMETHYLANTHRACENEJ. C. Hinshaw
215-218A CONVENIENT LABORATORY NITRILE SYNTHESIS. THERMAL DECOMPOSITION OF O-(METHYLCARBAMOYL) ALDOXIMESJames A. Albright; Merry Lou Alexander
219-223ARYLBORON DICHLORIDESJohn Hooz; Jose G. Calzada
225-2262, 4, 5, 8-TETRAMETHYLOUINOLINE. A CLARIFICATIONP. A. Claret; A. G. Osborne
227-231IMPROVED SYNTHESIS OF 3-METHYL-2-NAPHTHOIC ACIDMelvin S. Newman; William M. Hung
233-236A new synthesis of the coumestan ring systemThomas Kappe; Heinrich Schmidt
237-245PHOSPHORINO [4, 3-d] PYRIMIDINES. II. SYNTHESIS UTILIZING METHYL 4-OXO-1-PHENYL-3-PHOSPHORINANECARBOXYLATE 1-SULFIDETheodore E. Snider; K. D. Berlin
247-252SYNTHESIS OF 1-AZIDO-1, 3-BUTADIENESKazuakl Isomura; Masato Okada; Hideaki Ogawa; Makoto Ichiki; Hiroshi Taniguchi

Volume 4, Issue 4 (1972)

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153-157COMPOUNDS RELATED TO ACRIDINE. IX. COPPER CATALYZED OXIDATION OF 9-ETHYNYLACRIDINE AND ITS REACTION WITH SECONDARY AMINESO. Tsuge; A. Torii
159-168STUDIES OF ACENAPHTHENE DERIVATIVES. XXV. PREPARATION OF ACENAPHTHENEQUINONEO. Tsuge; I. Shinkai
169-177STUDIES OF ACENAPHTHENE DERIVATIVES. XXVII. PREPARATION OF ACENAPHTHENEQUINONE MONOANIL N-OXIDES AND THEIR REACTIONS WITH ISOCYANATESO. Tsuge; I. Shinkai; M. Koga
179-209THE URUSHIBARA HYDROGENATION CATALYSTS A REVIEWKazuo Hata; Izumi Motoyama; Koji Sakai

Volume 4, Issue 3 (1972)

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105-111SELECTIVE CYCLIZATION IN THE MODIFIED WILLGERODT-KINDLER REACTIONTakuzo Hisano; Yuko Yabuta
113-118PREPARATION OF EPOXYOLEFINS EMPLOYING DIMETHYLOXOSULFONIUM METHYLIDEBenjamin C. Clark Jr.; David J. Goldsmith
119-121THE PREPARATION AND CHARACTERIZATION OF trans-1-METHYLENECYCLOPROPANE-2, 3-di-t-BUTYL PERESTERIra S. Krull
123-128THE PREPARATION OF STEROIDAL AMIDES I. TRIPHENYLPHOSPHITE METHODJ. E. Herz; Rosa Elena Mantecón
129-134THE PREPARATION OF STEROIDAL AMIDES II. IMIDAZOLIDE METHOD AND EEDQ METHODJ. E. Herz; Rosa Elena Mantecón
135-151SYNTHESIS OF N,N-DIALKYLHYDROXYLAMINES. A REVIEWStanley Wawzonek; J. Vern Kempf

Volume 4, Issue 2 (1972)

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51-53ESTERIFICATION OF 1-METHYLINDOLE-2-CARBOXYLIC ACID WITH TRIMETHYL PHOSPHITEJacob Szmuszkovicz
55-57PYRIDO(3,2-d)-v-TRIAZIN-4(3H)-ONEB. Stanovnik; M. Tišler
59-61TETRAHYDRO-4-PYRONERamesh M. Kanojia; Richard E. Adams
63-663-NITROPYRIDINEG. B. Barlin
67-72CHROMIC ACID OXIDATION OF INDANS AND HYDRINDACENES. SYNTHESIS OF 1,1-DIMETHYLINDENEW. M. Harms; E. J. Eisenbraun
73-74SYNTHESIS OF 4-ISOPROPYL-2,6-DINITROCHLOROBENZENEEddie V. P. Tao; C. F. Christie Jr.
75-77O-METHYLATION OF TROPOLONEDavid H. Evans; Richard B. Greenwald
79-81BIS(2,2,2-TRICHLOROETHYL) SULFITEY. Wiesel; Y. Liwschitz
83-87SOME NEW PYRIMIDINE DERIVATIVESMervyn Israel; Melvin M. Berman; Naseem Muhammad
89-96IMPROVED SYNTHESES OF 1-ETHOXYALKYNESMelvin S. Newman; Jay R. Geib; Wayne M. Stalick
97-104PREPARATION OF CALCIUM ELENOLATE FROM OLIVE PRESS JUICEJ. H. Ford; F. A. Mackellar; P. A. Meulman; R. J. Wnuk; G. C. Prescott

Volume 4, Issue 1 (1972)

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1-32,2-′AZOBIS(2-CYANO-n-PROPANOL). A NEW FREE RADICAL INITIATORP. O. McCoy
5-8A SYNTHESIS OF 2,3-DIMETHOXY-6-(3,4-DIMETHOXYPHENYLACETYL)TOLUENEJ. A. Bakker; H. C. Beyerman; L. Maat
9-114-NITROISOQUINOLINEJohn W. Bunting; William G. Meathrel
13-18PREPARATION OF HOMOMIRISTICINIC ACIDG. Y. Moltrasio; D. Giacopello; M. J. Vernengo
19-21INEXPENSIVE STEEL REACTION VESSELS AND ACCESSORIES FOR ORGANIC REACTIONSE. J. Eisenbraun; H. Hall
23-26HYDROLYSIS OF 2-OXOCYCLOPENTYL PHENYL KETIMINEStuart S. Kulp; Bartholomew Palenchar; Robert K. Sharer
27-303-METHYL-3-BUTEN-1-OL AND 3-BUTEN-1-OLR. B. Kinnel; B. B. Molloy; D. W. Graham; K. E. Harding
31-34AN IMPROVED PREPARATION OF DIETHYL 1,4-DIHYDROXY-CYCLOHEXA-1,4-DIENE-2,5-DICARBOXYLATEJ. A. Moore
35-42THE SYNTHESIS OF 1H, 3H-NAPHTHO[1,8-cd]PYRAN-1-ONE, 1,8-DIMETHYL-1, 2,3,4TETRAHYDRONAPHTHALENE, 1,3,3a,4,5,6-HEXAHYDRONAPHTHO[1,8-cd] PYRAN, AND 1,2,3,4-TETRAHYDRO-8-METHYL-1-NAPHTHALENEMETHANOLJ. W. Burnham; E. J. Eisenbraun; M. C. Hamming; G. W. Keen
43-474-(7-BENZ[a]ANTHRACENYL)-N-(2-SUBSTITUTED ETHYL)BENZAMIDESF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
492,4-DINITROPHENYLHYDRAZONESD. E. Pearson

Volume 3, Issue 6 (1971)

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271-273SYNTHESIS OF N-PHENYLTETRAMETHYLSUCCINIMIDEGeorge R. Newkome; L. C. Roach
275-278DEHALOGENATION OF 7,7-BIS(BROMOMETHYL) BICYCLO[4.1.0]HEPT-3-ENEMary D. Craig; Paul H. Mazzocchi
279-282A MODIFIED METHOD FOR PREPARING 2-(2-PHENETHYL)PHENYLACETIC ACIDJoseph G. Lombardino; N. W. Treadway
283-288STUDIES OF BENZOYLSULFENE. VI. THE CYCLOADDITION REACTION OF BENZOYLSULFENE WITH KETENIMINESO. Tsuge; S. Iwanami
289-293THE PREPARATION OF 1,4-DIBROMOMETHYL-1,4-DIPHENYL-AZINEMETHYLENE AND ITS REACTION WITH BENZYLAMINEO. Tsuge; M. Tashiro; K. Kamata; K. Hokama
295-297DIMETHYL-2,4-THIOPHENEDICARBOXYLATEM. Janda; J. Šrogl; M. Němec; I. Stibor
299-302SYNTHESIS OF 5,6-0-ALKYLIDENE DERIVATIVES OF L-ASCORBIC ACID BY THE ORTHOFORMATE METHODRalph W. Atchley; Bert M. Tolbert
303-3059-Alkyl-9-Fluorenols From 9-Fluorenone DianionJ. A. Campbell; J. F. Wolfe
305-306Convenient One-Step Dialkylation of Diethyl Malonate With Sodium HydrideEdwin M. Kaiser; Janet A. Fries; Walter J. Simonsen Jr.
307-328INDEXES

Volume 3, Issue 5 (1971)

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213-2153-(2-HYDROXYETHYL) TETRAHYDROFURAN. CYCUZATIONS IN LITHIUM ALUMINUM HYDRIDE REDUCTIONSLeonard O. Moore
217-222THE SYNTHESIS OF TWO NEW 2,3-DIHALO-5-METHYLPYRIDINESPrank L. Setliff
223-226DDQ DEHYDROGENATION OF DIHYDRODICTAMNINEF. Piozzi; P. Venturella; A. Bellino
227-230DIAZOACETALDEHYDEJohn Hooz; Geoffrey F. Morrison
231-233SYNTHESES WITH AMMONIUM PEROXYDISULPHATE. α,β-DIAZIDOETHYLBENZENE AND α-CHLORO-β-AZIDOETHYLBENZENER. Galli; V. Malatesta
235-2383- AND 4-(BENZ[a]ANTHRACENYL)PHENYL-2-THIAZ0LINES AND 3- AND 4-(9-ANTHRACENYL)PHENYL-2-THIAZ0LINES. A NEW METHOD OF PREPARATION OF THIAZOLINESF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
239-242AN IMPROVED SULFONIC ACID-RESIN CATALYZED CYCLIDEHYDRATION OF 2-METHYL-4-PHENYL-2-BUTANOL TO 1,1-DIMETHYLINDANW. M. Harms; E. J. Eisenbraun
243-248PREPARATION OF 4H-PYRAN-2,6-DICARBOXYLIC ACID AND 4-METHYL-4H-PYRAN-2,6-DICARBOXYLIC ACIDJ. C. Lewis; R. M. Seifert
249-254AN EFFICIENT TECHNIQUE FOR THE CLEAVAGE OF HYDROCARBON PICRATES. THE PURIFICATION OF 1,8-, 2,6-, and 2,7-DIMETHYLNAPHTHALENEE. J. Eisenbraun; T. E. Webb; J. W. Burnham; L. E. Harrisld
255-260DI-2-PYRIDYLMETHANOL AND 1,1-DI-2-PYRIDYLETHANOLJoe Murphy; John W. Bunting
261-2671-ETHYL-4-CARBOMETHOXYPYRIDINYL (Pyridinyl, 1-ethyl-4-carbomethoxy)E. M. Kosower; Harold P. Waits
269STYRYL CARBONATES FROM ARYLACETONES. A CORRECTIONJohn L. Wong; Calvin H. Savells Jr.

Volume 3, Issue 4 (1971)

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163-166DIPHENYLACETYLENE. THE NUCLEOPHILIC RING CLEAVAGE OF 1,2,3-THIADIAZOLESR. G. Micetich
167-169ARYLGLYOXYLIC ESTERS VIA ARYLLITHIUM COMPOUNDSR. G. Micetich; R. Raap
171-175AN IMPROVED SYNTHESIS OF 1-FERROCENYL-1,3-BUTADIENEB. W. Ponder; R. Craig Kneisel; Danny H. Lewis
177-1813-(p-METHOXYBENZOYL)PROPIONIC ACID. AN IMPROVED SUCCINOYLATION PROCEDUREY. Shyamsunder Rao; Richard A. Kretchmer
183-186MACROPOROUS POLYSTYRENE BEADS AS A NEW RIGID SUPPORT FOR SOLID PHASE PEPTIDE SYNTHESISManohar A. Tilak; C. Stephen Hollinden
187-1903- AND 4-(7-BENZ[a]ANTHRACENYL)-N-(2-CHLOROETHYL)BENZAMIDES AND 3- AND 4-(9-ANTHRACENYL)-N-(2-CHLOROETHYL)BENZAMIDESF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
191-195TRIMETHYLBOROXINED. W. Wester; L. Barton
197-200BENZOYLATION OF TETRALIN. PRODUCT DISTRIBUTION. PHENYL 5,6,7,8-TETRAHYDRO-2-NAPHTHYL KETONER. G. Melton; T. E. Webb; E. J. Eisenbraun
201-204DIPHENACYL ETHERR. J. Mayfield; Peter Yates
205-207THE REACTION OF 1,2-BIS(2-PIPERIDYL)ETHYLENE WITH PHOSGENEFrank D. Popp; A. Catala Casey; Dennis K. Chesney
209-211PYROLYSIS OF 1,1-DIMETHYL-1-PHENYLAMINE-2-BENZOYLIMIDES. Wawzonek; E. E. Paschke

Volume 3, Issue 3 (1971)

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109-112SYNTHESIS OF 4-ETHYL-2,6-DINITRO-N,N-DIPROPYLANILINE-A NEW PLANT-GROWTH REGULATOR AND SELECTIVE HERBICIDEC. S. Giam; R. C. Hall
113-116A NEW SYNTHESIS OF 10, 11 -DIHYDRO-5H-DIBENZO (a, d)CYCLOHEPTEN-5-ONEJasjit S. Bindra; Shiv N. Rastogi; Randhir S. Kapil; Nitya Anand
117-120OXIDATIVE PHOSPHORYIATION OF PHENOLS AND RELATED COMPOUNDSRoger P. Napier; S. T. D. Gough
121-1244-PYRIDYLETHYLENE OXIDEF. I. Carroll
125-1261-BROMOPHENANTHRIDINEJ. P. Casey; A. Catala Casey; F. D. Popp
127-1302,6-DIMETHYL-4-(MONO- AND DI-p-NITROBENZENESULFENYLMETHYLENE)-4H-PYRANR. A. Abramovitch; E. P. Kyba
131-1333,5-PYRIDINEDICARBOXYLIC ACID (Dinicotinic acid)Bruce E. Maryanoff; Robert O. Hutchins
135-138SYNTHESIS OF THIOKETONES AND OF TETRAARYLETHYLENESRiaz Ahmed; Walter Lwowski
139-142PREPARATION OF MONO, BIS, TRIS AND TETRAKIS(CHLOROMETHYL) DERIVATIVES BY PHOTOCHLORINATION OF HEXAMETHYLBENZENEE. Henzelmann; J. Schwarcz; A. R. Frasca
143-148SYNTHESES WITH BENZENEDIAZONIUM SALTS. DIPHENYLOCTADIENES AND TETBBPHENYLBUTANFSR. Galli; M. Perchinunno; A. Arnone
149-154DIRECT CHLORINATION OF SATURATED CYCLIC ETHERS USING TRICHLOROISOCYANURIC ACIDW. P. Duncan; G. D. Strate; B. G. Adcock
155-157A FACILE SYNTHESIS OF 4-ALKYL-2,6-DINITROCHLOROBENZENESC. S. Giam; R. C. Hall
159-162THE PREPARATION OF 1,3-DIBROMOADAMANTANET. M. Gorrie; P. v. R. Schleyer

Volume 3, Issue 2 (1971)

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iPREFACE
51-53AZIDOMETHYLDIPHENYLPHOSPHINE OXIDEDietmar Seyferth; Peter Hilbert
55-59POLYARYLPYRYLIUM HEXA CHLOROANTIM ONATESD. F�rcaŝiu; Irina Elian
61-70A VARIABLE TEMPERATURE PREPARATIVE SCALE PHOTOCHEMICAL REACTOR. CIS-DIMETHYL BICYCLO[3.2.0]HEPTANE-1,5-DICARBOXYLATEDennis C. Owsley; Jordan J. Bloomfield
71-76OPTICAL RESOLUTION OF 4,6,4′,6′-TETRACHLORODIPHENIC ACIDEdward R. Atkinson
77-81REACTION OF ENAMINES OF SOME BICYCLIC AND MONOCYCLIC KETONES WITH 2,4-DINITROCHLOROBENZENE AND 2-CHLORO-3,5-DINITROTHIOPHENELars H. Hellberg; Charles C. Adams; Robert J. Milligan; Robert N. Wilke
83-861,1,2,2-TETRAMETHYLCYCLOHEXANEA. J. M. Reuvers; J. A. Jongejan; J. Klomp; H. van Bekkum
87-91A SIMPLE PREPARATION OF 4-AMINO-2,3,5-TRICHLOROPYRIDINEC. S. Giam; S. D. Abbott; R. C. Hall
93-956,7-DIMETHOXYCARBOSTYRILGeorge R. Pettit; Benjamin Stevenson; Gabriel Gever
97-98CATALYTIC SYNTHESIS OF METAL-FREE PHTHALOCYANINEM. V. Twigg
99-102USE OF DIETHYL PHENYLMALONATE AS A NUCLEOPHILIC DONOR IN THE MICHAEL REACTIONWayland E. Noland; Richard B. Hart
103-1073- AND 4-(7-BENZ[a]ANTHRACENYL)PHENYL-2-OXAZOLINES AND 3- AND 4-(9-ANTHRACENYL)PHENYL-2-OXAZOLINES AND THEIR HYDROCHLORIDE SALTSF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso

Volume 3, Issue 1 (1971)

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1-4NOVEL METHODS OF PREPARATION OF 2-OXAZOLIDONESZ. Lukasiewicz; T. Urbanski
5-82-OXO-3-OXA-5-anti-6-syn-DIPHENYLBICYCLO[2.1.1]HEXANE. A gamma LACTONE FROM LEAD TETRAACETATE OXIDATION OF alpha-TRUXILLIC ACIDDonald G. Farnum; Abdol J. Mostashari
9-153- AND 4-(7-BENZ[a]ANTHRACENYL)-N-BENZOYLAZIRIDINES AND 3- AND 4-(9-ANTHRACENYL)-N-BENZOYLAZIRIDINESF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
17-20PREPARATION AND PROPERTIES OF N-α-CARBOBENZOXY-N-IMIDAZOLE ADAMANTYLOXYCARBONYL-L-HISTIDINEManohar A. Tilak; Ralph Russell; Mary L. Hendricks
21-251,3-DIALKYL-5,5-DIMETHYLHEXAHYDROPYRIMIDINESH. Piotrowska; T. Urbanski; W. Bednarska
27-321-THIA-3-AZACYCLOHEPTANE DERIVATIVESZ. Olszenko-Piontkowa; T. Urbanski
33-36AN IMPROVED SYNTHESIS OF 3,4-DIHYDRO-1H-2,1-BENZOTHIAZIN-4-ONE 2,2-DIOXIDEJ. G. Lombardino; N. W. Treadway Jr.
37-38HEXALOCYCLOPENTANTADIENES IV. SYNTHESIS AND PYROLYSIS OF OCTABROMO-3a,4,7,7a-TETRAHYDROMETHANOINDENE-1,8-DIONER. G. Pews
39-44THE (±)-p-MENTHANE-2,5-DIONES AND THE (±)-2-t-BUTYL-5-METHYL-1,4-CYCLOHEXANEDIONESRobert D. Stolow; Robert R. Krikorian
45-462-BENZYLQUINOXALINEK. C. Bass; P. Nababsing
47-50VINYLDIAZOMETHANEJohn Hooz; Hiromichi Kono

Volume 2, Issue 4 (1970)

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245-248IMPROVED PREPARATIONS OF CYCLONONEN-3-OL, CYCLONONEN-3-ONE, CYCLONONANONE AND CYCLONONANOLGoverdhan Mehta
249-252ARYLGLYOXYLIC ESTERS, FRIEDEL-CRAFTS REACTIONR. G. Micetich
253-254NOTICE TO AUTHORS
255-258AN IMPROVED SYNTHESIS OF L-HISTIDINE BENZYL ESTERA. M. Felix; D. P. Winter
259-263THE REACTION OF 2,3-DICHLORO-1,4-NAPHTHOQUINONE WITH p-NITROBENZHYDRAZIDE1F. I. Carroll; H. Wayne Miller
265-2694-(ISOPROPYLIDENE)-2-(2′-PHENYLETHYL)-5-OXAZOLONED. N. Reinhoudt; P. R. M. van der Kamp
271-2732,3-DIAZABICYCLO[2.2.1]-2-HEPTENE M-OXIDERobert C. Kerber; Thomas J. Ryan
275-2791-ACYL- AND 1,1-DIACYL-2,2-DIMETHYLHYDRAZINESE. A. Sedor; R. E. Freis; H. J. Richards
281-283CORYPALLINEA. Brossi; J. O'brien; S. Teitel
285-289SYNTHESIS OF METHOXYPYRIDYL PHENYL KETONES VIA PYRIDYLLITHIUM COMPOUNDSEllis V. Brown; M. B. Shambhu
291-2941-TERT-BUTYL-1,3-PROPANEDIOLR. O. Hutchins; Frank J. Dux
295-296METHYL γ-RESORCYLATEArthur Mendel
297-303AN IMPROVED SYNTHESIS OF INDOLE-3-CARBOXYLIC ACIDSA. S. Katner
305-3082,4-DIETHYLQUINOLINE - AN EXTENSION OF THE COMBES SYNTHESISP. A. Claret; A. G. Osborne
309-310CONVENIENT SYNTHESIS OF 4-NITROBENZOYL CHLORIDEPankaja K. Kadaba
313-315MICRO-DISTILLATION OF ORGANIC LIQUIDSKenn E. Harding; Robin B. Kinnel
317-319A SOLVENT PAIR RECRYSTALLIZATION APPARATUS FOR GROWING SINGLE CRYSTALSJ. N. Brown; L. M. Trefonas
321-325ANHYDRIDE FORMATION WITH THIONYL CHLORIDEJerry M. Adduci; Rene S. Ramirez
325-329MONO- AND DIKETONES FROM ALKYLTIN CARBOXYLATESBernard R. Laliberte; Helmut F. Reiff; Wenzel E. Davidsohn

Volume 2, Issue 3 (1970)

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157-159DIFERROCENYLPHENYLPHOSPHINE AND DIPHENYLFERROCENYLPHOSPHINECharles E. Sullivan; William E. McEwen
161-165THE THERMAL CYCLYZATION OF DIETHYL METHANETRICARBOXYLATE THIOANILIDEH. Junek; A. Metallidis; E. Ziegler
167-1691,1′-DIACETYLFERROCENE MONOTOSYLHYDRAZONE AND 1,1′-DIACETYLFERROCENE DITOSYLHYDRAZONEHoward Alper; Susan J. Brown; Kenneth P. Jaffe
171-173cis - AND trans - CYCLOTRIDECENED. S. Sethi; R. Vaidyanathaswamy; D. Devaprabhakara
175-1763-ACETYL-2,4,6-TRIMETHYLBENZOPHENONEP. H. Gore; J. A. Hoskins
177-184N-SULFENYL - AND N-SULFINYLSULFOXIMIDESHans Christian Buchholt
185-187AN IMPROVED SYNTHESIS OF 2′HYDROXYBIPHENYL-2-CARBOXYLIC ACID LACTONEAlex Gringauz; Eugene Tosk
189-191ARSENIC TRICHLORIDE AS HALOGENATING AGENT. THE TRANSFORMATION OF HYDROXYMETHYL TO METHYL GROUPHelena B. Land; Adolfo R. Frasca
193-195SYNTHESIS OF α-ARYL-β-KETOESTERSJohn L. Wong; Mohammad K. Ali
197-2057-(3- AND 4-CARBOXYPHENYL) BENZ [A] ANTHRACENES AND 9-(3- AND 4-CARBOXYPHENYL) ANTHRACENESF. A. Vingiello; M. P. Rorer; M. A. Ogliaruso
207-210THE SELECTIVE OXIDATION OF ETHYLBENZENESFrancis A. Daniher
211-220N,N′-DIALKYL-p-PHENYLENEDIAMINEST. Doornbos; G. Zuidema; J. Strating
221-2227-METHYLINDOLEK. C. Bass; P. Nababsing
223-2245-ETHYL-5-(1-METHYL-3-CARBOXYPROPYL)-BARBITURIC ACIDF. I. Carroll; Abraham Philip
225-2273-ARYL-5-CHLOROISOXAZOLESR. G. Micetich
229-2342′, 4′ AND 2′, 4′, 6′ -CYCLOHEXYL SUBSTITUTED PHENYL KETONESE. R. Lavagnino; L. A. White
235-244THE SYNTHESIS OF SULFINYL CHLORIDES. A REVIEWMoh-Lian Kee; Irwin B. Douglass

Volume 2, Issue 2 (1970)

CEditorial Board Page
79-81THE NITRATION OF DIPHENYLCYCLOPROPENONEC. W. Bird; A. F. Harmer
83-87THE PREPARATION OF 1,2:5,6-Di-O-Cyclohexylidene-α-D-GulofuranoseSusanne L. von Schuching; Glenn H. Frye
89-92REDUCTION OF 1,1-DICHLOROBENZOCYCLOBUTENESDavid J. Hart; Harold Hart
93-100THE RESOLUTION OF (±)-3-METHYLCYCLOHEXANONE AND (±)-3-tert-BUTYLCYCLOHEXANONEG. Adolphen; E. J. Eisenbraun; G. W. Keen; P. W. K. Flanagan
101-115N,N′-DIALKYLATION OF SULFONYLAMIDES OF p-PHENYLENEDIAMINEST. Doornbos; J. Strating
117-119SOME NITRO-1,2,3-TRIAZOLEST. E. Eagles; M. A. Khan; B. M. Lynch
121-124ARYL N, N-DIFLUOROSULFONAMIDES1Travis E. Stevens; Royland D. Shoults
125-1281,1-DIARYLHYDRAZINESJ. -P. Anselme; N. Koga
129-135cis- AND trans-N,N′-DIMETHYL-1,4-CYCLOHEXANEBIS (METHYLAMINE) BY METHYLATION OF THE BENZALDEHYDE IMINESJ. Richard Hall; Thomas A. Hollingworth Jr.
137-139ALKYLATION AND OXIDATION OF DIARYLACETONITRILESStuart S. Kulp
141-144KETALIZATION OF 5-KETO STEROID ESTERS1David M. Piatak; Eliahu Caspi
145-147PREPARATION OF N-BENZOYL-N-METHYLPHENYLGLYCINEDonald F. McLaen
149-156AN IMPROVED SYNTHESIS OF KETIMINESE. P. Kyba

Volume 2, Issue 1 (1970)

CEditorial Board Page
1-4UNSYMMETRICALLY ALKOXYLATED DISILAZANESR. E. Goldsberry; W. E. Weibrecht
5-10PREPARATION OF PHOSPHANILIC ACID (p-AMINOBENZENEPHOSPHONIC ACID)O. Grummitt; N. Vourlogianes; J. Mehaffey; R. Tebbe
11-17SOME DERIVATIVES OF 3-CARBOXYMETHYLSYDNONEF. H. C. Stewart
19-23THE SYNTHESIS OF TRICHLOROTRIS (4-BIPHENYLYL-1-NAPHTHYLPHENYL PHOSPHINE) RHODIUM(III). A NEW OCTAHEDRAL COMPLEXRobert E. Harmon; Jack L. Parsons; S. K. Gupta
25-27PROCEDURE FOR THE HOMOGENEOUS CATALYTIC HYDROGENATION OF α, β-UNSATURATED NITRO COMPOUNDS USING TRIARYLPHOSPHINE-RHODIUM COMPLEXESRobert E. Harmon; Jack L. Parsons; S. K. Gupta
29-31DIAZEPINES. VIII. 3,8-DINITRO-11H-DIBENZO[c, f] [1, 2]-DIAZEPINE-5-OXIDEA. Catala Casey; F. D. Popp
33-36THE PREPARATION OF A FORMALDEHYDE ADDUCT OF 3-DIMETHYLAMINO-2,2-DIMETHYLPROPIONALDEHYDELloyd D. Taylor; Paul McLaughlin; Martin Mach
37-43A CONVENIENT SYNTHESIS OF 2-BENZYLNAPHTHALENE AND 2-BENZYL-1,2,3,4-TETRAHYDRONAPHTHALENER. G. Melton; E. J. Eisenbraun; P. W. K. Flanagan; M. C. Hamming
45-50GRADIENT ELUTION CHROMATOGRAPHY OF S-PALMITYL COENZYME A*Steven S. Kuwahara
51-52DL-4-ACETAMIDO-4-HYDROXY-2-BUTENOIC ACID γ-LACTONEJoan A. Gratz; C. E. Cook; Monroe E. Wall
53-58PREPARATION OF 4,4-BIS(DIFLUORAMINO)CYCLOHEXANONE AND 5,5-BIS(DIFLUORAMINO)-2-AZACYCLOHEPTANONETravis E. Stevens
59-63ALKYLATION OF 2,6-DI-TERT-BUTYLPHENOL IN DIMETHYL SULFOXIDEEugene R. Wagner
65-672,5-BIS-(2-PYRROLYL)-1-PYRROLINESV. Bocchi; G. P. Gardini
69-70SYNTHESIS OF 4,4′-DIHYDROXY-3,3′,5,5′-TETRA-t-BUTYLBENZOPHENONEMary K. Conner; E. Legoff
71-745,6-DIHYDRO-4H-1,3-OXAZINES BY A MODIFICATION OF THE TILLMANNS-RITTER PROCEDURESamuel P. McManus; John T. Carroll
75-783-NITRO-1,3,5-HEXATRIENECharles W. Spangler; Ronald P. Hennis

Volume 1, Issue 4 (1969)

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221-224SANDMEYER TYPE REACTION IN DIMETHYL SULFOXIDEMichio Kobayashi; Eiichi Yamada; Mikio Matsui; Nobumasa Kobori
225-228PREPARATION OF TOSYLATES OF PHENOLS AND ACIDIC ALCOHOLSStanley E. Wentworth; Patrick L. Sciaraffa
229-2332-METHOXY-1,3-BUTADIENEL. J. Dolby; K. S. Marshall
235-2382,5,5-TRIMETHYL-2-OXAZOLINES. P. McManus; J. T. Carroll; P. M. Grohse; C. U. Pittman Jr.
239-241ACRYLYLOXYMETHYL METHYL SULFIDESR. L. Harville; Samuel F. Reed Jr.
243-248PREPARATION OF 3-PHENYL-1,2-CYCLOPROPANEDICARBOXYLIC ACIDSS. Wawzonek; A. R. Zigman
249-251α-ACETAMIDO-β-(1-AZULYL) PROPIONIC ACIDArthur G. Anderson Jr.; Robert C. Rhodes
253-254N-METHYL OCTAHYDROCARBAZOLEE. Schmitz; H. Fechner
255-2581,2,5-THIADIAZOLID-3,4-DIONE-1-OXIDEMarvin Carmack; Ian W. Stapleton; Richard Y. Wen
259-261cis-1,2-VINYLENEBIS (DIPHENYLPHOSPHINE)J. P. Mitchener; A. M. Aguiar
263-266PREPARATION OF 2-BENZYLPHTHALIMIDINE VIA INTRAMOLECULAR FRIEDEL-CRAFTS RING CLOSURE OF N,N-DIBENZYLCARBAMOYL CHLORIDED. E. Rivett; J. F. K. Wilshire
267-269β- AND δ-TRUXINIC ACIDSM. Freedman; Y. Mohadger; J. Rennert; S. Soloway; I. Waltcher
271-277γ-ARYL-γ-AMINO ACIDSV. Bocchi; G. P. Gardini
279-2813-NITRO-7-CHLOROQUINOLINENed D. Heindel; Stephen A. Fine
283-285AN IMPROVED SYNTHESIS OF METHYLENECYCLOPROPANEI. S. Krull; D. R. Arnold
287-303THE COMPLETE N-ALKYLATION OF 1,4-DIAMINO-2,5-DIBROMOBENZENE AND OF 1,4-DIAMINO-2,5-DIMETHOXYBENZENET. Doornbos; J. Strating

Volume 1, Issue 4 (1969)

305-324SYNTHESIS OF AZIRIDINES BY REDUCTION OF OXIMES WITH LITHIUM ALUMINUM HYDRIDE A REVIEWKatsumi Kotera; Keizo Kitahonoki
325-326Separation of cis- and trans-1,2-CyclohexanediaminesJames E. Douglass; Houng-Min Shin
326-328Diphenyllead DicarboxylatesBhuvan C. Pant; Gail D. Mulligan
329Adaptor for Rotary EvaporatorAnthony L. Disalvo
329-330Cleaning SolutionJohn J. Bardeleben
331-352INDEXES

Volume 1, Issue 3 (1969)

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147-156THE SYNTHESIS OF SUBSTITUTED PHENYLENE DIISOCYANATESElbert W. Crandall; Lawrence Harris
157-164SULFONIC-CARBOXYLIC ANHYDRIDESE. Sarlo; T. Lanigan
165-170SYNTHESIS OF 2,6-DIMETHYLANILINE-14CRobert E. Middlebrook; George R. Harvey
171-1724-DESMETHYLMESCALINEA. Brossi; S. Teitel
173-176PREPARATION OF ALKYLTIN POLYFLUOROCARBOXYLATES AND RELATED DISTANNOXANESBernard R. La Liberte; Helmut F. Reiff; Wenzel E. Davidsohn
177-182AMIDES OF (1-AZULYL)ACETIC AND (1-AZULYL)GLYOXYLIC ACIDSArthur G. Anderson Jr.; Robert D. Breazeale
183-1862-SUBSTITUTED-5-METHYL-2-OXAZOLINESS. P. McManus; J. T. Carroll; P. M. Grohse; C. U. Pittman Jr.
187-1912,3,5,6-TETRACHLORO-4-PYRIDYLCOPPER AND SOME DERIVATIVESS. S. Dua; A. E. Jukes; H. Gilman
193-199PREPARATIVE PROCEDURES FOR ALDEHYDES FROM DIHYDRO-1,3-OXAZINESJ. Michael Fitzpatrick; G. Ray Malone; Ieva Ruks Politzer; H. Wayne Adickes; A. I. Meyers
201-203FLUORENONE IMINEJ. -P. Anselme
205-208PREPARATION OF BIS(4-HYDROXYPHENYL) ETHERG. Koga; M. Yasaka; Y. Nakano
209-212THE PREPARATION OF 1-ARYL-2-(2-THIENYL)ETHYLENESThomas R. Pampalone
213-2152-METHYL-3-PHENYLPROPANAL. AN EXAMPLE OF A THREE CARBON CHAIN EXTENSION VIA THE OXAZINE-A LDEHYDE SYNTHESISA. C. Kovelesky; A. I. Meyers
217-219A CONVENIENT SYNTHESIS OF 5-OXAZOLONES. 2-PHENYL-5-OXAZOLONELloyd D. Taylor; Thomas E. Platt

Volume 1, Issue 2 (1969)

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77-79N-METHYLTETRAHYDROQUINOLINE AND N-METHYLINDOLINEF. Minisoi; R. Galli; M. Perchinunno
81-85PHENYLACETYLENE-1-13CJoseph Casanova Jr.; Manfred Geisel; Randall N. Morris
87-90N,N-DIALKYLAMINOPHENOLSF. Minisoi; R. Galli; M. Perchinunno
91-96THE PRODUCTS OF DEHYDRATION OF 2,4-DI-TERT-BUTYL-3,4-DIHYDROXYTETRAHYDROTHIOPHENE-1,1-DIOXIDE: A CORRECTIONJ. Strating; T. Doornbos
97-98DIETHYLVINYLPHOSPHATEH. Gross; B. Costisella
99-104SYNTHESIS OF DIAZOACETIC ESTERS AND AMIDES FROM CORRESPONDING ACETOACETIC ACID DERIVATIVESM. Regitz; J. Hocker; A. Liedhegener
105-1063,6-DIMETHOXY-9H- DIBENZO[a,c]CARBAZOLEJ. Szmuszkovicz
107-109THE PALLADIUM CATALYZED HYDROGENATION OF CHOLESTEROLR. L. Augustine; E. J. Reardon Jr.
111-116METHYL AND ETHYL (DIMETHYLSULFURANYLIDENE) ACETATEDavid A. Rutolo; Peter G. Truskier; Joseph Casanova Jr.; G. B. Payne
117-119POLY(2-VINYLPYRROLE)C. G. Overberger; A. Wartman; J. C. Salamone
121-126APPARATUS WITH UTILITY FOR ANHYDROUS HYDROGEN FLUORIDE TREATMENT OF PEPTIDES AND PEPTIDE-RESIN COMPLEXESLinda M. Pourchot (Mrs.); John J. Johnson
127-1294-HYDROXYCYCLOHEXANONED. Edward Emmert; Daniel Lednicer
131-136PREPARATION OF SOME FERROCENYLSILANESM. D. Rausch; G. C. Schloemer
137-142N-(2-PYRIMIDYL) GLYCINE HYDROCHLORIDEC. J. Thoman; J. M. Tien; J. -P. Anselme; I. M. Hunsberger
143-145o-HYDROXYMETHYLBENZHYDROLNed D. Heindel; E. William Sarver; P. D. Kennewell

Volume 1, Issue 1 (1969)

CEditorial Board Page
iPREFACEJ. -P. Anselme; J. L. Ferrari
iiAcknowledgmentJ. -P. Anselme
1-34(5)-METHYLIMIDAZOLIUM CHLORIDEC. G. Overberger; C. M. Shen
5-10PREPARATION AND REACTIVITY OF THE 2-NITROSO-2-NITROCYCLOHEXANONEF. Minisci; A. Quilico
11-19NEW SYNTHESES OF POLYFUNCTIONAL LONG-CHAIN COMPOUNDS BY ALTERNATING FREE RADICAL ADDITIONS TO CONJUGATED OLEFINSF. Minisci; M. Ceoere; R. Galli; A. Selva
21-23THE PREPARATION OF γ-THIOPYRANJ. Strating; E. Molenaar
25-27GLYCYLGLYCOLIC ACIDF. H. C. Stewart
29-32REACTIONS OF DIPHENYLLEAD OXIDE, SYNTHESIS OF DIPHENYLLEAD DIACYLATESBhuvan C. Pant; Wenzel E. Davidsohn; Malcolm C. Henry
33-349-BROMOANTHRACENENed M. Weinshenker
35-384-SUBSTITUTED-BICYCLO[5.2.1]DECAN-10-ONESC. David Gutsche; John W. Baum
39-413,3-DIMETHYLINDOLINER. A. Abramovitch; R. A. Brown
43-454-METHOXYBENZENETHIOLJ. Szmuszkovicz
47-55HEXAARYLVINYLFULVENESFrederick A. Varron; Ernest I. Becker
57-59TRIMETHYLBORONJ. Casanova Jr.; H. R. Kiefer; R. E. Williams
61-62A MODIFICATION OF THE PECHMANN REACTIONThomas Kappe; Erich Ziegler
63-662-ACETYL-3,5-DIMETHYLFURAN (3,5-Dimethyl-2-furyl methyl ketone)A. T. Balaban
67-72PREPARATION OF ISOMERIC 1-METHYL-2-PHENYLCYCLOPROPANESS. Wawzonek; B. J. Studnicka; A. R. Zigman
73-75trans-3,5-DIPHENYL-1-PYRAZOLINEJ. -P. Anselme